RS20060049A - Novi n-supstituisani amidi indolil-3-glioksilne kiseline, njihova upotreba kao leka i postupak za njihovo dobijanje - Google Patents

Novi n-supstituisani amidi indolil-3-glioksilne kiseline, njihova upotreba kao leka i postupak za njihovo dobijanje

Info

Publication number
RS20060049A
RS20060049A YUP-2006/0049A YUP20060049A RS20060049A RS 20060049 A RS20060049 A RS 20060049A YU P20060049 A YUP20060049 A YU P20060049A RS 20060049 A RS20060049 A RS 20060049A
Authority
RS
Serbia
Prior art keywords
substituted
unsubstituted
alkyl
general formula
aryl
Prior art date
Application number
YUP-2006/0049A
Other languages
English (en)
Serbian (sr)
Inventor
Eckhard Gunther
Silke Baasner
Matthias Gerlach
Tilmann Schuster
Peter Schmidt
Original Assignee
Zentaris Gmbh.,
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Zentaris Gmbh., filed Critical Zentaris Gmbh.,
Publication of RS20060049A publication Critical patent/RS20060049A/sr

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
YUP-2006/0049A 2003-07-25 2004-07-09 Novi n-supstituisani amidi indolil-3-glioksilne kiseline, njihova upotreba kao leka i postupak za njihovo dobijanje RS20060049A (sr)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE10334040A DE10334040A1 (de) 2003-07-25 2003-07-25 Neue N-substituierte Indolyl-3-glyoxylsäureamide, deren Verwendung als Arzneimittel und Verfahren zu deren Herstellung
PCT/EP2004/007573 WO2005014542A2 (de) 2003-07-25 2004-07-09 Neue n-substituierte indolyl-3-glyoxylsäureamide, deren verwendung als arzneimittel gegen krebs und verfahren zu deren herstellung

Publications (1)

Publication Number Publication Date
RS20060049A true RS20060049A (sr) 2008-08-07

Family

ID=34129467

Family Applications (1)

Application Number Title Priority Date Filing Date
YUP-2006/0049A RS20060049A (sr) 2003-07-25 2004-07-09 Novi n-supstituisani amidi indolil-3-glioksilne kiseline, njihova upotreba kao leka i postupak za njihovo dobijanje

Country Status (18)

Country Link
EP (1) EP1651600A2 (pt)
JP (1) JP2007503376A (pt)
KR (1) KR20060037398A (pt)
CN (1) CN1839129A (pt)
AR (1) AR045928A1 (pt)
AU (1) AU2004263238A1 (pt)
BR (1) BRPI0412898A (pt)
CA (1) CA2533433A1 (pt)
DE (1) DE10334040A1 (pt)
IL (1) IL173335A0 (pt)
MX (1) MXPA06000995A (pt)
NO (1) NO20060697L (pt)
RS (1) RS20060049A (pt)
RU (1) RU2317293C9 (pt)
TW (1) TW200524863A (pt)
UA (1) UA83498C2 (pt)
WO (1) WO2005014542A2 (pt)
ZA (1) ZA200601300B (pt)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP2049520A4 (en) 2006-08-07 2011-01-05 Ironwood Pharmaceuticals Inc indole compounds
AR084433A1 (es) 2010-12-22 2013-05-15 Ironwood Pharmaceuticals Inc Inhibidores de la faah y composiciones farmaceuticas que los contienen

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE19636150A1 (de) * 1996-09-06 1998-03-12 Asta Medica Ag N-substituierte Indol-3-glyoxylamide mit antiasthmatischer, antiallergischer und immunsuppressiver/immunmodulierender Wirkung
AU2002324591A1 (en) * 2001-08-01 2003-02-17 The Ohio State University Clinical refractive instruments
AU2002323474B2 (en) * 2001-09-13 2006-10-05 Synta Pharmaceuticals Corp 3-glyoxlylamideindoles for treating cancer

Also Published As

Publication number Publication date
AU2004263238A1 (en) 2005-02-17
CA2533433A1 (en) 2005-02-17
DE10334040A1 (de) 2005-03-10
MXPA06000995A (es) 2006-04-11
JP2007503376A (ja) 2007-02-22
CN1839129A (zh) 2006-09-27
RU2317293C2 (ru) 2008-02-20
NO20060697L (no) 2006-02-14
WO2005014542A2 (de) 2005-02-17
IL173335A0 (en) 2006-06-11
TW200524863A (en) 2005-08-01
WO2005014542A3 (de) 2006-10-19
RU2317293C9 (ru) 2008-05-10
ZA200601300B (en) 2007-03-28
BRPI0412898A (pt) 2006-10-03
AR045928A1 (es) 2005-11-16
EP1651600A2 (de) 2006-05-03
RU2006105708A (ru) 2006-06-27
KR20060037398A (ko) 2006-05-03
UA83498C2 (uk) 2008-07-25

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