TW200524863A - Novel N-substituted indolyl-3-glyoxylamides, their use as medicaments and process for their preparation - Google Patents
Novel N-substituted indolyl-3-glyoxylamides, their use as medicaments and process for their preparation Download PDFInfo
- Publication number
- TW200524863A TW200524863A TW093121509A TW93121509A TW200524863A TW 200524863 A TW200524863 A TW 200524863A TW 093121509 A TW093121509 A TW 093121509A TW 93121509 A TW93121509 A TW 93121509A TW 200524863 A TW200524863 A TW 200524863A
- Authority
- TW
- Taiwan
- Prior art keywords
- substituted
- unsubstituted
- aryl
- alkyl
- group
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
- C07D403/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE10334040A DE10334040A1 (de) | 2003-07-25 | 2003-07-25 | Neue N-substituierte Indolyl-3-glyoxylsäureamide, deren Verwendung als Arzneimittel und Verfahren zu deren Herstellung |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| TW200524863A true TW200524863A (en) | 2005-08-01 |
Family
ID=34129467
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| TW093121509A TW200524863A (en) | 2003-07-25 | 2004-07-19 | Novel N-substituted indolyl-3-glyoxylamides, their use as medicaments and process for their preparation |
Country Status (18)
| Country | Link |
|---|---|
| EP (1) | EP1651600A2 (pt) |
| JP (1) | JP2007503376A (pt) |
| KR (1) | KR20060037398A (pt) |
| CN (1) | CN1839129A (pt) |
| AR (1) | AR045928A1 (pt) |
| AU (1) | AU2004263238A1 (pt) |
| BR (1) | BRPI0412898A (pt) |
| CA (1) | CA2533433A1 (pt) |
| DE (1) | DE10334040A1 (pt) |
| IL (1) | IL173335A0 (pt) |
| MX (1) | MXPA06000995A (pt) |
| NO (1) | NO20060697L (pt) |
| RS (1) | RS20060049A (pt) |
| RU (1) | RU2317293C9 (pt) |
| TW (1) | TW200524863A (pt) |
| UA (1) | UA83498C2 (pt) |
| WO (1) | WO2005014542A2 (pt) |
| ZA (1) | ZA200601300B (pt) |
Families Citing this family (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| SG176477A1 (en) | 2006-08-07 | 2011-12-29 | Ironwood Pharmaceuticals Inc | Indole compounds |
| AR084433A1 (es) | 2010-12-22 | 2013-05-15 | Ironwood Pharmaceuticals Inc | Inhibidores de la faah y composiciones farmaceuticas que los contienen |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE19636150A1 (de) * | 1996-09-06 | 1998-03-12 | Asta Medica Ag | N-substituierte Indol-3-glyoxylamide mit antiasthmatischer, antiallergischer und immunsuppressiver/immunmodulierender Wirkung |
| WO2003011180A2 (en) * | 2001-08-01 | 2003-02-13 | The Ohio State University | Clinical refractive instruments |
| CA2460347A1 (en) * | 2001-09-13 | 2003-03-20 | Synta Pharmaceuticals Corp. | 3-glyoxlylamideindoles for treating cancer |
-
2003
- 2003-07-25 DE DE10334040A patent/DE10334040A1/de not_active Withdrawn
-
2004
- 2004-07-09 CA CA002533433A patent/CA2533433A1/en not_active Abandoned
- 2004-07-09 RS YUP-2006/0049A patent/RS20060049A/sr unknown
- 2004-07-09 WO PCT/EP2004/007573 patent/WO2005014542A2/de not_active Ceased
- 2004-07-09 BR BRPI0412898-2A patent/BRPI0412898A/pt not_active IP Right Cessation
- 2004-07-09 JP JP2006521430A patent/JP2007503376A/ja not_active Withdrawn
- 2004-07-09 RU RU2006105708/04A patent/RU2317293C9/ru not_active IP Right Cessation
- 2004-07-09 AU AU2004263238A patent/AU2004263238A1/en not_active Abandoned
- 2004-07-09 KR KR1020067001636A patent/KR20060037398A/ko not_active Ceased
- 2004-07-09 MX MXPA06000995A patent/MXPA06000995A/es unknown
- 2004-07-09 EP EP04740854A patent/EP1651600A2/de not_active Withdrawn
- 2004-07-09 CN CNA2004800240832A patent/CN1839129A/zh active Pending
- 2004-07-19 TW TW093121509A patent/TW200524863A/zh unknown
- 2004-07-23 AR ARP040102632A patent/AR045928A1/es not_active Application Discontinuation
- 2004-09-07 UA UAA200601216A patent/UA83498C2/uk unknown
-
2006
- 2006-01-24 IL IL173335A patent/IL173335A0/en unknown
- 2006-02-13 ZA ZA200601300A patent/ZA200601300B/xx unknown
- 2006-02-14 NO NO20060697A patent/NO20060697L/no not_active Application Discontinuation
Also Published As
| Publication number | Publication date |
|---|---|
| WO2005014542A3 (de) | 2006-10-19 |
| RU2317293C9 (ru) | 2008-05-10 |
| AU2004263238A1 (en) | 2005-02-17 |
| WO2005014542A2 (de) | 2005-02-17 |
| CA2533433A1 (en) | 2005-02-17 |
| CN1839129A (zh) | 2006-09-27 |
| MXPA06000995A (es) | 2006-04-11 |
| RU2006105708A (ru) | 2006-06-27 |
| NO20060697L (no) | 2006-02-14 |
| KR20060037398A (ko) | 2006-05-03 |
| RU2317293C2 (ru) | 2008-02-20 |
| UA83498C2 (uk) | 2008-07-25 |
| BRPI0412898A (pt) | 2006-10-03 |
| RS20060049A (sr) | 2008-08-07 |
| AR045928A1 (es) | 2005-11-16 |
| DE10334040A1 (de) | 2005-03-10 |
| IL173335A0 (en) | 2006-06-11 |
| JP2007503376A (ja) | 2007-02-22 |
| EP1651600A2 (de) | 2006-05-03 |
| ZA200601300B (en) | 2007-03-28 |
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