RU2417077C2 - Способ лечения чрезмерной дневной сонливости (варианты) - Google Patents

Способ лечения чрезмерной дневной сонливости (варианты) Download PDF

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Publication number
RU2417077C2
RU2417077C2 RU2008100019/15A RU2008100019A RU2417077C2 RU 2417077 C2 RU2417077 C2 RU 2417077C2 RU 2008100019/15 A RU2008100019/15 A RU 2008100019/15A RU 2008100019 A RU2008100019 A RU 2008100019A RU 2417077 C2 RU2417077 C2 RU 2417077C2
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Russia
Prior art keywords
sleep
enantiomer
administration
dose
compounds
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RU2008100019/15A
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English (en)
Russian (ru)
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RU2008100019A (ru
Inventor
Абдаллах АХНАОУ (BE)
Абдаллах АХНАОУ
Вильгельмус Х. И. М. ДРИНКЕНБУРГ (NL)
Вильгельмус Х. И. М. ДРИНКЕНБУРГ
Джозеф ПАЛУМБО (US)
Джозеф ПАЛУМБО
Джонатан СПОРН (US)
Джонатан СПОРН
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Ск Холдингз Ко., Лтд.
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Application filed by Ск Холдингз Ко., Лтд. filed Critical Ск Холдингз Ко., Лтд.
Publication of RU2008100019A publication Critical patent/RU2008100019A/ru
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    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C271/00Derivatives of carbamic acids, i.e. compounds containing any of the groups, the nitrogen atom not being part of nitro or nitroso groups
    • C07C271/06Esters of carbamic acids
    • C07C271/08Esters of carbamic acids having oxygen atoms of carbamate groups bound to acyclic carbon atoms
    • C07C271/10Esters of carbamic acids having oxygen atoms of carbamate groups bound to acyclic carbon atoms with the nitrogen atoms of the carbamate groups bound to hydrogen atoms or to acyclic carbon atoms
    • C07C271/12Esters of carbamic acids having oxygen atoms of carbamate groups bound to acyclic carbon atoms with the nitrogen atoms of the carbamate groups bound to hydrogen atoms or to acyclic carbon atoms to hydrogen atoms or to carbon atoms of unsubstituted hydrocarbon radicals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/16Amides, e.g. hydroxamic acids
    • A61K31/165Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/21Esters, e.g. nitroglycerine, selenocyanates
    • A61K31/27Esters, e.g. nitroglycerine, selenocyanates of carbamic or thiocarbamic acids, meprobamate, carbachol, neostigmine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0053Mouth and digestive tract, i.e. intraoral and peroral administration
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/20Hypnotics; Sedatives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/26Psychostimulants, e.g. nicotine, cocaine

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Organic Chemistry (AREA)
  • Epidemiology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • General Chemical & Material Sciences (AREA)
  • Emergency Medicine (AREA)
  • Nutrition Science (AREA)
  • Physiology (AREA)
  • Psychiatry (AREA)
  • Anesthesiology (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
RU2008100019/15A 2005-06-08 2006-06-07 Способ лечения чрезмерной дневной сонливости (варианты) RU2417077C2 (ru)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US68863805P 2005-06-08 2005-06-08
US60/688,638 2005-06-08

Publications (2)

Publication Number Publication Date
RU2008100019A RU2008100019A (ru) 2009-07-20
RU2417077C2 true RU2417077C2 (ru) 2011-04-27

Family

ID=37085728

Family Applications (1)

Application Number Title Priority Date Filing Date
RU2008100019/15A RU2417077C2 (ru) 2005-06-08 2006-06-07 Способ лечения чрезмерной дневной сонливости (варианты)

Country Status (17)

Country Link
US (8) US8440715B2 (2)
EP (1) EP1890684B1 (2)
JP (1) JP5024635B2 (2)
KR (1) KR101335941B1 (2)
CN (1) CN101217949B (2)
AU (1) AU2006254899B2 (2)
BE (1) BE2020C004I2 (2)
BR (1) BRPI0613697A2 (2)
CA (1) CA2611713C (2)
DK (1) DK1890684T3 (2)
ES (1) ES2435403T3 (2)
FR (1) FR20C1014I2 (2)
NL (1) NL301037I2 (2)
PL (1) PL1890684T3 (2)
RU (1) RU2417077C2 (2)
TW (2) TW201328689A (2)
WO (1) WO2006133393A1 (2)

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ES2344469T3 (es) * 2005-06-22 2010-08-27 Sk Holdings Co., Ltd. Tratamiento de disfuncion sexual.
KR20120098578A (ko) 2009-06-22 2012-09-05 에스케이바이오팜 주식회사 피로의 치료 또는 예방 방법
US8232315B2 (en) * 2009-06-26 2012-07-31 Sk Biopharmaceuticals Co., Ltd. Methods for treating drug addiction and improving addiction-related behavior
BR112012010670A2 (pt) 2009-11-06 2016-04-12 Sk Biopharmaceuticals Co Ltd métodos para tratamento de distúrbio de défict de atenção/hiperatividade
EP2496227B1 (en) * 2009-11-06 2019-05-22 SK Biopharmaceuticals Co., Ltd. Methods for treating fibromyalgia syndrome
US9610274B2 (en) * 2010-06-30 2017-04-04 Sk Biopharmaceuticals Co., Ltd. Methods for treating bipolar disorder
US8623913B2 (en) * 2010-06-30 2014-01-07 Sk Biopharmaceuticals Co., Ltd. Methods for treating restless legs syndrome
CA2905457A1 (en) * 2013-03-13 2014-10-09 Aerial Biopharma, Llc Treatment of cataplexy
CA2917702A1 (en) 2013-07-18 2015-01-22 Jazz Pharmaceuticals International Iii Limited Treatment for obesity
US10888542B2 (en) 2014-02-28 2021-01-12 Sk Biopharmaceuticals Co., Ltd. Aminocarbonylcarbamate compounds
TWI698415B (zh) * 2014-02-28 2020-07-11 南韓商愛思開生物製藥股份有限公司 胺基羰基胺基甲酸酯化合物
WO2016061488A1 (en) * 2014-10-17 2016-04-21 Concert Pharmaceuticals, Inc. Amine reuptake inhibitors
JP6466792B2 (ja) * 2015-07-03 2019-02-06 エスケー バイオファーマスティカルズ カンパニー リミテッド 注意欠陥/多動性障害(adhd)の治療方法
TWI637765B (zh) * 2016-05-10 2018-10-11 台灣共振波研發股份有限公司 Soothing device for attention deficit hyperactivity disorder
US10195151B2 (en) 2016-09-06 2019-02-05 Jazz Pharmaceuticals International Iii Limited Formulations of (R)-2-amino-3-phenylpropyl carbamate
MY197630A (en) 2016-09-06 2023-06-29 Sk Biopharmaceuticals Co Ltd Solvate form of (r)-2-amino-3-phenylpropyl carbamate
ES2964943T3 (es) 2016-10-06 2024-04-10 Axsome Malta Ltd Compuestos de carbamoilfenilalaninol para uso médico
BR112019025286A2 (pt) 2017-06-02 2020-06-23 Jazz Pharmaceuticals Ireland Limited Métodos e composições para tratamento de sonolência excessiva
JP7366002B2 (ja) * 2017-07-31 2023-10-20 ジャズ ファーマシューティカルズ アイルランド リミテッド カルバモイルフェニルアラニノール類縁体およびその使用
US10940133B1 (en) 2020-03-19 2021-03-09 Jazz Pharmaceuticals Ireland Limited Methods of providing solriamfetol therapy to subjects with impaired renal function
US11033214B1 (en) * 2020-05-19 2021-06-15 United Arab Emirates University Wearable eye tracking system
KR102390194B1 (ko) * 2020-08-03 2022-04-25 셀라이온바이오메드 주식회사 페닐알킬 카바메이트 화합물을 포함하는 Kca3.1채널 매개질환 치료용 조성물
AU2023375326A1 (en) * 2022-11-07 2025-05-22 Axsome Therapeutics Compositions and methods for treating insomnia
EP4626417A1 (en) * 2022-11-30 2025-10-08 Axsome Therapeutics Methods and compositions for improving driving performance
KR20260033050A (ko) 2023-06-29 2026-03-10 액섬 테라퓨틱스, 인크. 수유 여성에게 솔리암페톨을 투여하는 방법
WO2025165760A1 (en) * 2024-01-29 2025-08-07 Axsome Therapeutics, Inc. Phenylalkylamino carbamates for use in the treatment of attention deficit/hyperactivity disorder

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US8232315B2 (en) 2009-06-26 2012-07-31 Sk Biopharmaceuticals Co., Ltd. Methods for treating drug addiction and improving addiction-related behavior
EP2496227B1 (en) 2009-11-06 2019-05-22 SK Biopharmaceuticals Co., Ltd. Methods for treating fibromyalgia syndrome
BR112012010670A2 (pt) 2009-11-06 2016-04-12 Sk Biopharmaceuticals Co Ltd métodos para tratamento de distúrbio de défict de atenção/hiperatividade
US8623913B2 (en) 2010-06-30 2014-01-07 Sk Biopharmaceuticals Co., Ltd. Methods for treating restless legs syndrome
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Also Published As

Publication number Publication date
TW200716084A (en) 2007-05-01
US20090312416A1 (en) 2009-12-17
BE2020C004I2 (2) 2026-01-06
US20240239740A1 (en) 2024-07-18
NL301037I2 (nl) 2020-05-12
RU2008100019A (ru) 2009-07-20
EP1890684B1 (en) 2013-08-14
FR20C1014I2 (fr) 2021-04-23
DK1890684T3 (da) 2013-10-14
JP5024635B2 (ja) 2012-09-12
US20130137764A1 (en) 2013-05-30
CA2611713C (en) 2013-10-01
AU2006254899B2 (en) 2011-11-24
EP1890684A1 (en) 2008-02-27
CN101217949B (zh) 2012-10-17
AU2006254899A1 (en) 2006-12-14
US20250109099A1 (en) 2025-04-03
CN101217949A (zh) 2008-07-09
KR20080035565A (ko) 2008-04-23
TW201328689A (zh) 2013-07-16
US9604917B2 (en) 2017-03-28
BRPI0613697A2 (pt) 2011-01-25
NL301037I1 (2) 2020-04-01
TWI419681B (zh) 2013-12-21
US11753368B2 (en) 2023-09-12
PL1890684T3 (pl) 2014-05-30
US12209059B2 (en) 2025-01-28
ES2435403T3 (es) 2013-12-19
US8877806B2 (en) 2014-11-04
US10351517B2 (en) 2019-07-16
US20140350098A1 (en) 2014-11-27
JP2008545795A (ja) 2008-12-18
US8440715B2 (en) 2013-05-14
US20210078943A1 (en) 2021-03-18
FR20C1014I1 (2) 2020-06-12
US20190367448A1 (en) 2019-12-05
CA2611713A1 (en) 2006-12-14
US20170158622A1 (en) 2017-06-08
WO2006133393A1 (en) 2006-12-14
KR101335941B1 (ko) 2013-12-04

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