SE0401657D0 - Chemical compounds - Google Patents

Chemical compounds

Info

Publication number
SE0401657D0
SE0401657D0 SE0401657A SE0401657A SE0401657D0 SE 0401657 D0 SE0401657 D0 SE 0401657D0 SE 0401657 A SE0401657 A SE 0401657A SE 0401657 A SE0401657 A SE 0401657A SE 0401657 D0 SE0401657 D0 SE 0401657D0
Authority
SE
Sweden
Prior art keywords
chemical compounds
compounds
compositions
preparing
processes
Prior art date
Application number
SE0401657A
Other languages
English (en)
Swedish (sv)
Inventor
Howard Tucker
Original Assignee
Astrazeneca Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=32733687&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=SE0401657(D0) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Astrazeneca Ab filed Critical Astrazeneca Ab
Priority to SE0401657A priority Critical patent/SE0401657D0/xx
Publication of SE0401657D0 publication Critical patent/SE0401657D0/xx
Priority to TW094119533A priority patent/TW200610759A/zh
Priority to ES05753676T priority patent/ES2342181T3/es
Priority to CNA2005800284341A priority patent/CN101006058A/zh
Priority to PCT/SE2005/000952 priority patent/WO2006001751A1/en
Priority to RU2006146877/04A priority patent/RU2381216C2/ru
Priority to AU2005257707A priority patent/AU2005257707B2/en
Priority to JP2007518001A priority patent/JP5147393B2/ja
Priority to CA002571087A priority patent/CA2571087A1/en
Priority to US11/628,724 priority patent/US20070259914A1/en
Priority to UAA200613008A priority patent/UA88303C2/ru
Priority to EP05753676A priority patent/EP1761494B1/en
Priority to AT05753676T priority patent/ATE465148T1/de
Priority to BRPI0512420-4A priority patent/BRPI0512420A/pt
Priority to DE602005020787T priority patent/DE602005020787D1/de
Priority to MXPA06014413A priority patent/MXPA06014413A/es
Priority to UY28974A priority patent/UY28974A1/es
Priority to ARP050102573A priority patent/AR049830A1/es
Priority to MYPI20052861A priority patent/MY139268A/en
Priority to IL179729A priority patent/IL179729A0/en
Priority to ZA200610526A priority patent/ZA200610526B/xx
Priority to NO20070431A priority patent/NO20070431L/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D211/36—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D211/56—Nitrogen atoms
    • C07D211/58—Nitrogen atoms attached in position 4

Landscapes

  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Virology (AREA)
  • Pulmonology (AREA)
  • Biomedical Technology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Dermatology (AREA)
  • Oncology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Immunology (AREA)
  • Communicable Diseases (AREA)
  • Urology & Nephrology (AREA)
  • Rheumatology (AREA)
  • Pain & Pain Management (AREA)
  • Reproductive Health (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Molecular Biology (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Endocrinology (AREA)
  • Ophthalmology & Optometry (AREA)
  • Diabetes (AREA)
  • Gynecology & Obstetrics (AREA)
  • Hematology (AREA)
  • Biotechnology (AREA)
  • Psychiatry (AREA)
SE0401657A 2004-06-24 2004-06-24 Chemical compounds SE0401657D0 (sv)

Priority Applications (22)

Application Number Priority Date Filing Date Title
SE0401657A SE0401657D0 (sv) 2004-06-24 2004-06-24 Chemical compounds
TW094119533A TW200610759A (en) 2004-06-24 2005-06-13 Chemical compounds
DE602005020787T DE602005020787D1 (de) 2004-06-24 2005-06-20 Chemische verbindungen i
MXPA06014413A MXPA06014413A (es) 2004-06-24 2005-06-20 Compuestos quimicos de derivados heterociclicos.
US11/628,724 US20070259914A1 (en) 2004-06-24 2005-06-20 Novel Piperidine Derivates as Modulators of Chemokine Receptor Ccr5.
EP05753676A EP1761494B1 (en) 2004-06-24 2005-06-20 Chemical compounds i
PCT/SE2005/000952 WO2006001751A1 (en) 2004-06-24 2005-06-20 Chemical compounds i
RU2006146877/04A RU2381216C2 (ru) 2004-06-24 2005-06-20 Химические соединения i
AU2005257707A AU2005257707B2 (en) 2004-06-24 2005-06-20 Chemical compounds I
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CA002571087A CA2571087A1 (en) 2004-06-24 2005-06-20 Novel piperidine derivates as modulators of chemokine receptor ccr5
ES05753676T ES2342181T3 (es) 2004-06-24 2005-06-20 Compuestos quimicos i.
UAA200613008A UA88303C2 (ru) 2004-06-24 2005-06-20 Производные пиперидина, которые имеют активность по отношению к ccr5 (хемокинового рецептора 5)
CNA2005800284341A CN101006058A (zh) 2004-06-24 2005-06-20 化合物ⅰ
AT05753676T ATE465148T1 (de) 2004-06-24 2005-06-20 Chemische verbindungen i
BRPI0512420-4A BRPI0512420A (pt) 2004-06-24 2005-06-20 novos derivados de piperidina como moduladores do receptor de quimocina ccr5
UY28974A UY28974A1 (es) 2004-06-24 2005-06-21 Derivados heterocíclicos de piperidina, composiciones que los contienen y procedimiento de preparación
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ARP050102573A AR049830A1 (es) 2004-06-24 2005-06-22 Derivados de piperidina
IL179729A IL179729A0 (en) 2004-06-24 2006-11-30 Novel piperidine derivates as modulators of chemokine receptor ccr5
ZA200610526A ZA200610526B (en) 2004-06-24 2006-12-14 Chemical compounds I
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TW200610761A (en) * 2004-04-23 2006-04-01 Astrazeneca Ab Chemical compounds
EP2066674B1 (en) 2006-09-18 2010-06-30 F.Hoffmann-La Roche Ag Octahydropyrrolo [3, 4-c] pyrrole derivatives and their use as antiviral agents
EP2173715A2 (en) * 2007-07-13 2010-04-14 Euroscreen S.A. Use of piperidine derivatives as agonists of chemokine receptor activity
WO2009151910A2 (en) * 2008-05-25 2009-12-17 Wyeth Combination product of receptor tyrosine kinase inhibitor and fatty acid synthase inhibitor for treating cancer
WO2012113103A1 (en) 2011-02-25 2012-08-30 Helsinn Healthcare S.A. Asymmetric ureas and medical uses thereof
GB201321746D0 (en) * 2013-12-09 2014-01-22 Ucb Pharma Sa Therapeutic agents
NO2699580T3 (es) 2014-01-24 2018-02-24
CA3017048C (en) 2016-03-22 2023-11-07 Helsinn Healthcare Sa Benzenesulfonyl-asymmetric ureas and medical uses thereof
US20220072013A1 (en) * 2018-12-21 2022-03-10 Ca*Tx, Inc. Pharmaceutical Combinations for the Treatment of Cancer

Family Cites Families (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB9624482D0 (en) 1995-12-18 1997-01-15 Zeneca Phaema S A Chemical compounds
WO1997030035A1 (en) 1996-02-13 1997-08-21 Zeneca Limited Quinazoline derivatives as vegf inhibitors
ES2169355T3 (es) 1996-03-05 2002-07-01 Astrazeneca Ab Derivados de 4-anilinoquinazolina.
GB9718972D0 (en) 1996-09-25 1997-11-12 Zeneca Ltd Chemical compounds
GB9714249D0 (en) 1997-07-08 1997-09-10 Angiogene Pharm Ltd Vascular damaging agents
PL192083B1 (pl) * 1997-11-18 2006-08-31 Dupont Pharmaceuticals Res Lab Pochodne amin cyklicznych i ich zastosowanie
EP1013276A1 (en) * 1998-12-23 2000-06-28 Pfizer Inc. Aminoazacycloalkanes as CCR5 modulators
GB9900334D0 (en) 1999-01-07 1999-02-24 Angiogene Pharm Ltd Tricylic vascular damaging agents
GB9900752D0 (en) 1999-01-15 1999-03-03 Angiogene Pharm Ltd Benzimidazole vascular damaging agents
SE9902987D0 (sv) * 1999-08-24 1999-08-24 Astra Pharma Prod Novel compounds
IL152682A0 (en) 2000-05-31 2003-06-24 Astrazeneca Ab Indole derivatives with vascular damaging activity
HUP0301742A3 (en) 2000-07-07 2005-08-29 Angiogene Pharm Ltd Colchinol derivatives as angiogenesis inhibitors, process for producing them, pharmaceutical compositions containing them and their use
BR0112224A (pt) 2000-07-07 2003-06-10 Angiogene Pharm Ltd Composto, composição farmacêutica, uso de um composto ou de um sal, solvato ou pró-droga farmaceuticamente aceitável do mesmo, e, processo para preparar um composto
SE0103818D0 (sv) * 2001-11-15 2001-11-15 Astrazeneca Ab Chemical compounds
SE0103819D0 (sv) * 2001-11-15 2001-11-15 Astrazeneca Ab Chemical compounds
RU2005118407A (ru) * 2002-12-13 2006-03-10 СмитКлайн Бичем Корпорейшн (US) Производные пиперидина в качестве антагонистов ccr5
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US20070259914A1 (en) 2007-11-08
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EP1761494B1 (en) 2010-04-21
BRPI0512420A (pt) 2008-03-04
NO20070431L (no) 2007-03-26
TW200610759A (en) 2006-04-01
ES2342181T3 (es) 2010-07-02
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IL179729A0 (en) 2007-05-15
AU2005257707B2 (en) 2009-03-26
RU2006146877A (ru) 2008-07-27
CN101006058A (zh) 2007-07-25
JP2008503572A (ja) 2008-02-07
AR049830A1 (es) 2006-09-06
RU2381216C2 (ru) 2010-02-10
EP1761494A1 (en) 2007-03-14
UY28974A1 (es) 2006-01-31

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