BRPI0512420A - novos derivados de piperidina como moduladores do receptor de quimocina ccr5 - Google Patents

novos derivados de piperidina como moduladores do receptor de quimocina ccr5

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Publication number
BRPI0512420A
BRPI0512420A BRPI0512420-4A BRPI0512420A BRPI0512420A BR PI0512420 A BRPI0512420 A BR PI0512420A BR PI0512420 A BRPI0512420 A BR PI0512420A BR PI0512420 A BRPI0512420 A BR PI0512420A
Authority
BR
Brazil
Prior art keywords
chemokine receptor
receptor modulators
piperidine derivatives
ccr5 chemokine
new piperidine
Prior art date
Application number
BRPI0512420-4A
Other languages
English (en)
Portuguese (pt)
Inventor
Howard Tucker
Original Assignee
Astrazeneca Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=32733687&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=BRPI0512420(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Astrazeneca Ab filed Critical Astrazeneca Ab
Publication of BRPI0512420A publication Critical patent/BRPI0512420A/pt

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    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/06Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
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    • C07D211/56Nitrogen atoms
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  • Animal Behavior & Ethology (AREA)
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  • Pain & Pain Management (AREA)
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  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
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BRPI0512420-4A 2004-06-24 2005-06-20 novos derivados de piperidina como moduladores do receptor de quimocina ccr5 BRPI0512420A (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
SE0401657A SE0401657D0 (sv) 2004-06-24 2004-06-24 Chemical compounds
PCT/SE2005/000952 WO2006001751A1 (en) 2004-06-24 2005-06-20 Chemical compounds i

Publications (1)

Publication Number Publication Date
BRPI0512420A true BRPI0512420A (pt) 2008-03-04

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ID=32733687

Family Applications (1)

Application Number Title Priority Date Filing Date
BRPI0512420-4A BRPI0512420A (pt) 2004-06-24 2005-06-20 novos derivados de piperidina como moduladores do receptor de quimocina ccr5

Country Status (22)

Country Link
US (1) US20070259914A1 (es)
EP (1) EP1761494B1 (es)
JP (1) JP5147393B2 (es)
CN (1) CN101006058A (es)
AR (1) AR049830A1 (es)
AT (1) ATE465148T1 (es)
AU (1) AU2005257707B2 (es)
BR (1) BRPI0512420A (es)
CA (1) CA2571087A1 (es)
DE (1) DE602005020787D1 (es)
ES (1) ES2342181T3 (es)
IL (1) IL179729A0 (es)
MX (1) MXPA06014413A (es)
MY (1) MY139268A (es)
NO (1) NO20070431L (es)
RU (1) RU2381216C2 (es)
SE (1) SE0401657D0 (es)
TW (1) TW200610759A (es)
UA (1) UA88303C2 (es)
UY (1) UY28974A1 (es)
WO (1) WO2006001751A1 (es)
ZA (1) ZA200610526B (es)

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TW200610761A (en) * 2004-04-23 2006-04-01 Astrazeneca Ab Chemical compounds
EP2066674B1 (en) 2006-09-18 2010-06-30 F.Hoffmann-La Roche Ag Octahydropyrrolo [3, 4-c] pyrrole derivatives and their use as antiviral agents
EP2173715A2 (en) * 2007-07-13 2010-04-14 Euroscreen S.A. Use of piperidine derivatives as agonists of chemokine receptor activity
WO2009151910A2 (en) * 2008-05-25 2009-12-17 Wyeth Combination product of receptor tyrosine kinase inhibitor and fatty acid synthase inhibitor for treating cancer
WO2012113103A1 (en) 2011-02-25 2012-08-30 Helsinn Healthcare S.A. Asymmetric ureas and medical uses thereof
GB201321746D0 (en) * 2013-12-09 2014-01-22 Ucb Pharma Sa Therapeutic agents
NO2699580T3 (es) 2014-01-24 2018-02-24
CA3017048C (en) 2016-03-22 2023-11-07 Helsinn Healthcare Sa Benzenesulfonyl-asymmetric ureas and medical uses thereof
US20220072013A1 (en) * 2018-12-21 2022-03-10 Ca*Tx, Inc. Pharmaceutical Combinations for the Treatment of Cancer

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GB9624482D0 (en) 1995-12-18 1997-01-15 Zeneca Phaema S A Chemical compounds
WO1997030035A1 (en) 1996-02-13 1997-08-21 Zeneca Limited Quinazoline derivatives as vegf inhibitors
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DE602005020787D1 (de) 2010-06-02
WO2006001751A1 (en) 2006-01-05
US20070259914A1 (en) 2007-11-08
MXPA06014413A (es) 2007-02-19
JP5147393B2 (ja) 2013-02-20
EP1761494B1 (en) 2010-04-21
NO20070431L (no) 2007-03-26
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ES2342181T3 (es) 2010-07-02
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ZA200610526B (en) 2008-08-27
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RU2006146877A (ru) 2008-07-27
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EP1761494A1 (en) 2007-03-14
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