SE438339B - Forfarande for framstellning av foreningar med analgetisk verkan - Google Patents

Forfarande for framstellning av foreningar med analgetisk verkan

Info

Publication number: SE438339B
Authority: SE; Sweden
Prior art keywords: mixture; methyl; added; mol; acid
Prior art date: 1976-09-27

Application number

SE7710755A

Other languages

English (en)

Swedish (sv)

Other versions

SE7710755L (sv

Inventor

Jr E L Smithwick

R C A Frederickson

R T Shuman

Original Assignee

Lilly Co Eli

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1976-09-27

Filing date

1977-09-26

Publication date

1985-04-15

1977-09-26 Application filed by Lilly Co Eli filed Critical Lilly Co Eli

1978-03-28 Publication of SE7710755L publication Critical patent/SE7710755L/xx

1985-04-15 Publication of SE438339B publication Critical patent/SE438339B/sv

Links

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- C07K14/435—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
- C07K14/665—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans derived from pro-opiomelanocortin, pro-enkephalin or pro-dynorphin
- C07K14/70—Enkephalins
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Public Health (AREA)
Veterinary Medicine (AREA)
Pharmacology & Pharmacy (AREA)
Biomedical Technology (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Animal Behavior & Ethology (AREA)
Bioinformatics & Cheminformatics (AREA)
General Chemical & Material Sciences (AREA)
Neurosurgery (AREA)
Chemical Kinetics & Catalysis (AREA)
Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Peptides Or Proteins (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)

SE7710755A 1976-09-27 1977-09-26 Forfarande for framstellning av foreningar med analgetisk verkan SE438339B (sv)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
US72672476A	1976-09-27	1976-09-27
US05/807,849 US4259234A (en)	1976-09-27	1977-06-20	Analgesic compounds

Publications (2)

Publication Number	Publication Date
SE7710755L SE7710755L (sv)	1978-03-28
SE438339B true SE438339B (sv)	1985-04-15

Family

ID=27111374

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
SE7710755A SE438339B (sv)	1976-09-27	1977-09-26	Forfarande for framstellning av foreningar med analgetisk verkan

Country Status (27)

Country	Link
US (1)	US4259234A (fr)
JP (1)	JPS5340736A (fr)
AR (1)	AR228937A1 (fr)
AT (1)	AT359219B (fr)
AU (1)	AU513702B2 (fr)
CA (1)	CA1201710A (fr)
CH (2)	CH636847A5 (fr)
CS (1)	CS204011B2 (fr)
DD (1)	DD132862A5 (fr)
DE (1)	DE2741393A1 (fr)
DK (1)	DK148904C (fr)
ES (1)	ES462658A1 (fr)
FR (1)	FR2365553A1 (fr)
GB (1)	GB1586521A (fr)
GR (1)	GR69224B (fr)
HK (1)	HK52681A (fr)
HU (1)	HU180723B (fr)
IE (1)	IE45576B1 (fr)
IL (1)	IL52872A (fr)
MY (1)	MY8200150A (fr)
NL (1)	NL7710502A (fr)
NZ (1)	NZ185084A (fr)
PL (1)	PL111136B1 (fr)
PT (1)	PT67026B (fr)
RO (1)	RO80379B (fr)
SE (1)	SE438339B (fr)
SU (1)	SU753358A3 (fr)

Families Citing this family (22)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US4261888A (en) *	1976-04-12	1981-04-14	Sandoz Ltd.	Organic compounds
PT66982B (en) *	1976-09-01	1979-02-13	Coy David Howard	Process for preparing novel methionine enkephalin derivatives
HU178001B (en) *	1976-09-16	1982-02-28	Gyogyszekutato Intezet	Process for preparing new pentapeptides with morphine-like activity and derivatives thereof
US4322342A (en) *	1977-06-20	1982-03-30	Eli Lilly And Company	Analgesic compounds
JPS5424850A (en) *	1977-07-22	1979-02-24	Wellcome Found	Peptide compound
US4264491A (en) *	1977-10-03	1981-04-28	Eli Lilly And Company	Analgesic compounds
FR2424253A1 (fr) *	1978-04-27	1979-11-23	Brun Lab Sa Le	Nouveaux derives de peptides analogues des enkephalines, leur procede de preparation et leur application therapeutique
DE2933947A1 (de) *	1979-08-22	1981-03-12	Hoechst Ag, 6000 Frankfurt	Neue peptidamide und verfahren zu ihrer herstellung.
US4254024A (en) *	1979-10-16	1981-03-03	Pennwalt Corporation	Tetrapeptides and derivatives having opiate activity
US4283330A (en) *	1979-12-17	1981-08-11	Eli Lilly And Company	Pharmacologically active peptides
US4251439A (en) *	1979-12-17	1981-02-17	Eli Lilly And Company	Pharmacologically active peptides
US4283329A (en) *	1979-12-17	1981-08-11	Eli Lilly And Company	Pharmacologically active peptides
US4265808A (en) *	1979-12-17	1981-05-05	Eli Lilly And Company	Pharmacologically active peptides
US4351763A (en) *	1979-12-17	1982-09-28	Eli Lilly And Company	Pharmacologically active peptides
FR2488253A1 (fr) *	1980-08-08	1982-02-12	Roques Bernard	Nouveaux peptides et leur application en therapeutique
US4322339A (en) *	1980-10-20	1982-03-30	Eli Lilly And Company	Pharmacologically active peptides
ATE16495T1 (de) *	1981-06-22	1985-11-15	Ici Plc	Peptide und pseudopeptide, die zwei substituenten am n-terminus aufweisen.
US4430327A (en)	1982-05-18	1984-02-07	Eli Lilly And Company	Method for treating pregnant females for pain and anxiety
DE3915755A1 (de) *	1989-05-13	1990-11-29	Bayer Ag	Fungizide mittel sowie substituierte aminosaeureamid-derivate und deren herstellung
DE4102042A1 (de) *	1991-01-24	1992-07-30	Bayer Ag	Substituierte aminosaeureamid-derivate deren herstellung und verwendung als fungizide
JPH09173654A (ja) *	1995-12-21	1997-07-08	Ritsuwa Yo	積木
EP1297830A1 (fr) *	2001-09-28	2003-04-02	Flamma Fabbrica Lombarda Ammino Acidi S.p.a.	L'utilisation des acides aminés alpha ou bèta, leurs esters, ou de dipeptides de ces acides aminés avec des dérivés d'histidine, dans la prévention ou le traitement de lésions de la peau causées par l'ozone atmosphérique

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
FI770219A7 (fr) *	1976-02-02	1977-08-03	Sandoz Ag
GB1532181A (en) *	1976-02-02	1978-11-15	Beckman Instruments Inc	Pentapetides and a method of preparing them
NZ183712A (en) *	1976-04-08	1979-10-25	Ici Ltd	Polypeptide analogues of enkephalins, and pharmaceutical compositions
PT66982B (en) *	1976-09-01	1979-02-13	Coy David Howard	Process for preparing novel methionine enkephalin derivatives
HU178001B (en) *	1976-09-16	1982-02-28	Gyogyszekutato Intezet	Process for preparing new pentapeptides with morphine-like activity and derivatives thereof
US4178371A (en) *	1977-12-15	1979-12-11	Reckitt & Colman Products Limited	Tetrapeptide derivatives

1977
- 1977-06-20 US US05/807,849 patent/US4259234A/en not_active Expired - Lifetime
- 1977-08-30 IE IE1805/77A patent/IE45576B1/en unknown
- 1977-09-01 IL IL52872A patent/IL52872A/xx unknown
- 1977-09-01 GR GR54278A patent/GR69224B/el unknown
- 1977-09-02 NZ NZ185084A patent/NZ185084A/xx unknown
- 1977-09-09 AU AU28565/77A patent/AU513702B2/en not_active Expired
- 1977-09-12 CA CA000286528A patent/CA1201710A/fr not_active Expired
- 1977-09-13 PT PT67026A patent/PT67026B/pt unknown
- 1977-09-14 DE DE19772741393 patent/DE2741393A1/de active Granted
- 1977-09-16 CS CS776044A patent/CS204011B2/cs unknown
- 1977-09-22 AR AR269298A patent/AR228937A1/es active
- 1977-09-22 GB GB39459/77A patent/GB1586521A/en not_active Expired
- 1977-09-23 CH CH1165977A patent/CH636847A5/de not_active IP Right Cessation
- 1977-09-26 PL PL1977201049A patent/PL111136B1/pl unknown
- 1977-09-26 ES ES462658A patent/ES462658A1/es not_active Expired
- 1977-09-26 HU HU77EI763A patent/HU180723B/hu unknown
- 1977-09-26 DK DK424577A patent/DK148904C/da not_active IP Right Cessation
- 1977-09-26 FR FR7728939A patent/FR2365553A1/fr active Granted
- 1977-09-26 AT AT685977A patent/AT359219B/de not_active IP Right Cessation
- 1977-09-26 NL NL7710502A patent/NL7710502A/xx not_active Application Discontinuation
- 1977-09-26 DD DD7700201204A patent/DD132862A5/xx unknown
- 1977-09-26 SU SU772526421A patent/SU753358A3/ru active
- 1977-09-26 RO RO91664A patent/RO80379B/ro unknown
- 1977-09-26 SE SE7710755A patent/SE438339B/sv not_active IP Right Cessation
- 1977-09-27 JP JP11659077A patent/JPS5340736A/ja active Granted
1981
- 1981-10-29 HK HK526/81A patent/HK52681A/xx unknown
1982
- 1982-12-30 MY MY150/82A patent/MY8200150A/xx unknown
1983
- 1983-03-09 CH CH128183A patent/CH643533A5/de not_active IP Right Cessation

Also Published As

Publication number	Publication date
CA1201710A (fr)	1986-03-11
DK424577A (da)	1978-03-28
DK148904B (da)	1985-11-11
AU513702B2 (en)	1980-12-18
AT359219B (de)	1980-10-27
NZ185084A (en)	1980-11-14
PT67026A (en)	1977-10-01
RO80379A (fr)	1983-04-29
RO80379B (ro)	1983-04-30
IL52872A (en)	1983-07-31
SU753358A3 (ru)	1980-07-30
AR228937A1 (es)	1983-05-13
CS204011B2 (en)	1981-03-31
DE2741393A1 (de)	1978-03-30
MY8200150A (en)	1982-12-31
IE45576L (en)	1978-03-27
SE7710755L (sv)	1978-03-28
DK148904C (da)	1986-04-14
PT67026B (en)	1979-02-14
AU2856577A (en)	1979-03-15
NL7710502A (nl)	1978-03-29
ATA685977A (de)	1980-03-15
CH643533A5 (de)	1984-06-15
FR2365553B1 (fr)	1980-11-14
ES462658A1 (es)	1978-11-01
GR69224B (fr)	1982-05-10
PL201049A1 (pl)	1979-01-29
DE2741393C2 (fr)	1988-03-10
GB1586521A (en)	1981-03-18
CH636847A5 (de)	1983-06-30
HU180723B (en)	1983-04-29
JPS5340736A (en)	1978-04-13
PL111136B1 (en)	1980-08-30
US4259234A (en)	1981-03-31
DD132862A5 (de)	1978-11-15
HK52681A (en)	1981-11-06
FR2365553A1 (fr)	1978-04-21
JPS6254800B2 (fr)	1987-11-17
IE45576B1 (en)	1982-10-06

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1995-01-31

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Publication	Publication Date	Title
SE438339B (sv)	1985-04-15	Forfarande for framstellning av foreningar med analgetisk verkan
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Taylor	1985	Ynthesis of
GB2120256A (en)	1983-11-30	Novel peptides
NO166532B (no)	1991-04-29	Fremgangsmaate for fremstilling av peptidet h-arg-x-z-y-tyr-r.
EP0050503B1 (fr)	1984-07-04	Dérivés des pentapeptides avec activité pharmacologique
CS235072B2 (en)	1985-04-16	Method of l-tyrosyl-d-alanyl-glycyl-l-phenylalanylamide's new derivatives production
GB2058077A (en)	1981-04-08	Enkephalin analogues
US4322342A (en)	1982-03-30	Analgesic compounds
JPH0665291A (ja)	1994-03-08	環状ペプチドの合成方法
EP0018182B1 (fr)	1982-10-20	Peptides possédant une activité analogue à celle de la thymopoiétine, compositions pharmaceutiques qui les contiennent, et procédé pour les préparer
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US3364193A (en)	1968-01-16	Undeca- and dodecapeptides related to methionyl-lysyl-bradykinin
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PL91030B1 (fr)	1977-02-28
GB1584669A (en)	1981-02-18	Process for synthesising peptides containing a sulphated tyrosine residue
CN105418737A (zh)	2016-03-23	一种短瓣花环肽a的固相合成方法和应用
USRE29732E (en)	1978-08-15	Tripeptide
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US3780015A (en)	1973-12-18	Process for preparing lysine containing peptides
EP0311391B1 (fr)	1993-12-29	Procédé de préparation d'un octapeptide