SE7713341L - Sett att framstella grenade och cykloalifatiska estrar ur androstan- och ostranserierna - Google Patents

Sett att framstella grenade och cykloalifatiska estrar ur androstan- och ostranserierna

Info

Publication number: SE7713341L
Authority: SE; Sweden
Prior art keywords: esters; ostranseries; cycloalifatic; androstan; preparing branched
Prior art date: 1976-11-26

Application number

SE7713341A

Other languages

English (en)

Swedish (sv)

Inventor

L J W M Tax

Original Assignee

Akzo Nv

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1976-11-26

Filing date

1977-11-25

Publication date

1978-05-27

1977-11-25 Application filed by Akzo Nv filed Critical Akzo Nv

1978-05-27 Publication of SE7713341L publication Critical patent/SE7713341L/xx

Links

150000002148 esters Chemical class 0.000 title abstract 2
QZLYKIGBANMMBK-UGCZWRCOSA-N 5α-Androstane Chemical compound C([C@@H]1CC2)CCC[C@]1(C)[C@@H]1[C@@H]2[C@@H]2CCC[C@@]2(C)CC1 QZLYKIGBANMMBK-UGCZWRCOSA-N 0.000 title 1
-1 steroid esters Chemical class 0.000 abstract 2
230000001195 anabolic effect Effects 0.000 abstract 1
230000001548 androgenic effect Effects 0.000 abstract 1
230000001833 anti-estrogenic effect Effects 0.000 abstract 1
230000001076 estrogenic effect Effects 0.000 abstract 1
239000008194 pharmaceutical composition Substances 0.000 abstract 1
150000003431 steroids Chemical class 0.000 abstract 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J1/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane
- C07J1/0051—Estrane derivatives
- C07J1/0066—Estrane derivatives substituted in position 17 beta not substituted in position 17 alfa
- C07J1/007—Estrane derivatives substituted in position 17 beta not substituted in position 17 alfa the substituent being an OH group free esterified or etherified
- C07J1/0074—Esters
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J1/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane
- C07J1/0003—Androstane derivatives
- C07J1/0018—Androstane derivatives substituted in position 17 beta, not substituted in position 17 alfa
- C07J1/0022—Androstane derivatives substituted in position 17 beta, not substituted in position 17 alfa the substituent being an OH group free esterified or etherified
- C07J1/0025—Esters

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
General Health & Medical Sciences (AREA)
Steroid Compounds (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)

SE7713341A 1976-11-26 1977-11-25 Sett att framstella grenade och cykloalifatiska estrar ur androstan- och ostranserierna SE7713341L (sv)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
NL7613248A NL7613248A (nl)	1976-11-26	1976-11-26	Werkwijze voor het bereiden van nieuwe steroid- esters.

Publications (1)

Publication Number	Publication Date
SE7713341L true SE7713341L (sv)	1978-05-27

Family

ID=19827290

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
SE7713341A SE7713341L (sv)	1976-11-26	1977-11-25	Sett att framstella grenade och cykloalifatiska estrar ur androstan- och ostranserierna

Country Status (13)

Country	Link
US (5)	US4212864A (fr)
JP (1)	JPS5384957A (fr)
BE (1)	BE861224A (fr)
CA (1)	CA1095895A (fr)
CH (1)	CH637143A5 (fr)
DE (1)	DE2752695A1 (fr)
DK (1)	DK146221C (fr)
ES (1)	ES464504A1 (fr)
FR (1)	FR2373560A1 (fr)
GB (1)	GB1593515A (fr)
IE (1)	IE46092B1 (fr)
NL (1)	NL7613248A (fr)
SE (1)	SE7713341L (fr)

Families Citing this family (29)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
NL7613248A (nl) *	1976-11-26	1978-05-30	Akzo Nv	Werkwijze voor het bereiden van nieuwe steroid- esters.
US4705783A (en) *	1985-06-25	1987-11-10	Sri International	9α, 11β-substituted and 11β-substituted estranes
US4851402A (en) *	1987-02-27	1989-07-25	International Minerals & Chemical Corp.	Estriol growth promotant
US5137882A (en) *	1990-06-11	1992-08-11	Holt Dennis A	Steroidal 3-acetic acid derivatives as 5-alpha-reductase inhibitors
US5238929A (en) *	1991-10-22	1993-08-24	Development Products, Inc.	Correction of tribology of arthritis-affected joints and medicine for its implementation
US6908910B2 (en)	1993-08-06	2005-06-21	The Children's Medical Center Corporation	Estrogenic compounds as anti-mitotic agents
US5504074A (en) *	1993-08-06	1996-04-02	Children's Medical Center Corporation	Estrogenic compounds as anti-angiogenic agents
US20040214807A1 (en) *	1993-08-06	2004-10-28	D'amato Robert J.	Estrogenic compounds as anti-mitotic agents
US6346510B1 (en)	1995-10-23	2002-02-12	The Children's Medical Center Corporation	Therapeutic antiangiogenic endostatin compositions
US20020002294A1 (en) *	1997-09-24	2002-01-03	D' Amato Robert J.	Estrogenic compounds as antiangiogenic agents
EP1124545B1 (fr)	1998-08-11	2004-12-15	EntreMed, Inc.	Utilisation de 2-methoxyestradiol en tant qu'agents antifongiques
US20030083231A1 (en) *	1998-11-24	2003-05-01	Ahlem Clarence N.	Blood cell deficiency treatment method
DE19906159A1 (de) *	1999-02-09	2000-08-10	Schering Ag	16-Hydroxyestratriene als selektiv wirksame Estrogene
CN1250563C (zh)	1999-05-04	2006-04-12	斯特拉坎有限公司	雄激素糖苷及其产生雄性征的活性
US7087592B1 (en) *	1999-08-23	2006-08-08	Entre Med, Inc.	Compositions comprising purified 2-methoxyestradiol and methods of producing same
US20050192258A1 (en) *	2000-08-18	2005-09-01	Agoston Gregory E.	Antiangiogenic agents
US7135581B2 (en)	2000-08-18	2006-11-14	Entremed, Inc.	Antiangiogenic agents
US6995278B2 (en) *	2000-08-18	2006-02-07	Entre Med, Inc.	Antiangiogenic agents
WO2002022645A2 (fr) *	2000-09-14	2002-03-21	Accelerated Pharmaceuticals, Inc.	Procede de preparation de d'utilisation de 7alpha-methyl-11beta-methoxy estradiol
WO2003063787A2 (fr) *	2002-01-30	2003-08-07	Entremed, Inc.	Analogues non steroidiens de 2-methoxyestradiol
EP1633367A2 (fr) *	2003-05-28	2006-03-15	EntreMed, Inc.	Agents anti-angiogenese
CA2558014A1 (fr)	2004-03-12	2005-09-29	Entremed, Inc.	Agents anti-angiogeniques
US20070004689A1 (en) *	2004-03-12	2007-01-04	Agoston Gregory E	Antiangiogenic agents
JP2008521822A (ja) *	2004-11-29	2008-06-26	エントレメッドインコーポレイテッド	抗血管形成剤を投与する方法、およびそれを用いて疾病を治療する方法
WO2007059111A2 (fr) *	2005-11-14	2007-05-24	Entremed, Inc.	Activite antiangiogenese du 2-methoxyestradiol en combinaison avec des agents anticancereux
US20070176403A1 (en) *	2006-02-01	2007-08-02	Dennis Calderone	Air adjustable seat
CA2646065C (fr) *	2006-03-20	2014-01-14	Entremed, Inc.	2-methoxyestradiol presentant une activite anti-arthritique pouvant modifier l'evolution de la maladie
WO2008094665A1 (fr) *	2007-01-31	2008-08-07	Entremed, Inc.	Procédé de traitement des maladies associées à l'amylose
US20160060288A1 (en) *	2013-04-18	2016-03-03	Xi'anlibang Pharmaceutical Technology Co., Ltd.	Ester derivatives of 7-alpha-[9-(4,4,5,5,5-pentafluoropentylsulfinyl)nonyl)-estra-1,3,5(10)-triene-3,17beta-diol having anticancer activity and preparation method thereof

Family Cites Families (12)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
GB826790A (en) *	1957-05-07	1960-01-20	British Drug Houses Ltd	Improvements in or relating to the preparation of cyclopentanophenanthrene compounds
DE1117113B (de) *	1959-12-05	1961-11-16	Schering Ag	Verfahren zur Herstellung ªú¼ ª-ungesaettigter Ketosteroide, die am ª-staendigen Kohlenstoffatom eine Methylgruppe tragen
US3018297A (en) *	1960-02-29	1962-01-23	Searle & Co	1, 3- and 1, 4-bisoxygenated estra-1, 3, 5(10)-trienes and intermediates
CH399447A (de) *	1961-04-14	1965-09-30	Ciba Geigy	Verfahren zur Herstellung eines neuen Steroid-Hormon-Esters
US3226991A (en) *	1962-12-17	1966-01-04	United Carr Fastener Corp	Indexing device for a rotary snap switch
FR5519M (fr) *	1966-06-07	1967-11-06
US4098802A (en) *	1975-02-18	1978-07-04	Akzona Incorporated	Oral pharmaceutical preparation having androgenic activity
NL189235C (nl) *	1974-02-28	1993-02-16	Akzo Nv	Werkwijze voor de bereiding van een oraal toe te dienen farmaceutisch preparaat met androgene werking.
US4147783A (en) *	1974-02-28	1979-04-03	Akzona Incorporated	Oral pharmaceutical preparation
NL7506407A (nl) *	1975-05-30	1976-12-02	Akzo Nv	Werkwijze ter bereiding van een oraal werkzaam far- maceutisch preparaat.
DE2558076C2 (de) *	1975-12-19	1983-12-15	Schering AG, 1000 Berlin und 4709 Bergkamen	Depot-Steroidester, Verfahren zu ihrer Herstellung und diese enthaltende pharmazeutische Präparate
NL7613248A (nl) *	1976-11-26	1978-05-30	Akzo Nv	Werkwijze voor het bereiden van nieuwe steroid- esters.

1976
- 1976-11-26 NL NL7613248A patent/NL7613248A/xx not_active Application Discontinuation
1977
- 1977-11-17 GB GB47888/77A patent/GB1593515A/en not_active Expired
- 1977-11-17 IE IE2341/77A patent/IE46092B1/en unknown
- 1977-11-17 US US05/852,326 patent/US4212864A/en not_active Expired - Lifetime
- 1977-11-23 CH CH1436277A patent/CH637143A5/de not_active IP Right Cessation
- 1977-11-24 JP JP14106677A patent/JPS5384957A/ja active Pending
- 1977-11-24 DK DK522277A patent/DK146221C/da not_active IP Right Cessation
- 1977-11-25 FR FR7735633A patent/FR2373560A1/fr active Granted
- 1977-11-25 BE BE182946A patent/BE861224A/fr not_active IP Right Cessation
- 1977-11-25 DE DE19772752695 patent/DE2752695A1/de not_active Withdrawn
- 1977-11-25 ES ES464504A patent/ES464504A1/es not_active Expired
- 1977-11-25 SE SE7713341A patent/SE7713341L/xx not_active Application Discontinuation
- 1977-11-28 CA CA291,885A patent/CA1095895A/fr not_active Expired
1980
- 1980-02-12 US US06/120,598 patent/US4312864A/en not_active Expired - Lifetime
- 1980-02-12 US US06/120,608 patent/US4329296A/en not_active Expired - Lifetime
- 1980-02-12 US US06/120,607 patent/US4307086A/en not_active Expired - Lifetime
- 1980-02-12 US US06/120,609 patent/US4307087A/en not_active Expired - Lifetime

Also Published As

Publication number	Publication date
CH637143A5 (de)	1983-07-15
GB1593515A (en)	1981-07-15
US4329296A (en)	1982-05-11
US4212864A (en)	1980-07-15
FR2373560A1 (fr)	1978-07-07
ES464504A1 (es)	1978-09-01
IE46092B1 (en)	1983-02-23
BE861224A (fr)	1978-05-25
DK146221B (da)	1983-08-01
FR2373560B1 (fr)	1980-08-22
DK146221C (da)	1984-01-09
JPS5384957A (en)	1978-07-26
CA1095895A (fr)	1981-02-17
US4307086A (en)	1981-12-22
IE46092L (en)	1978-05-26
US4312864A (en)	1982-01-26
DK522277A (da)	1978-05-27
DE2752695A1 (de)	1978-06-01
NL7613248A (nl)	1978-05-30
US4307087A (en)	1981-12-22

Legal Events

Date

Code

Title

Description

1995-02-28

NAV

Patent application has lapsed

Ref document number: 7713341-1

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Publication	Publication Date	Title
SE7713341L (sv)	1978-05-27	Sett att framstella grenade och cykloalifatiska estrar ur androstan- och ostranserierna
MX9304541A (es)	1994-05-31	Esteriodes de 17-espirometileno.
CA2114630A1 (fr)	1993-03-18	Inhibiteurs de la steroide sulfatase
IL57728A (en)	1983-06-15	Hemiesters of steryl glycosides,their preparation and pharmaceutical compositions containing them
NL7611073A (nl)	1977-04-13	Werkwijze voor het bereiden van delta15-steroiden, alsmede werkwijze voor het bereiden van een ge- neesmiddel met gestagene werking.
IL56076A0 (en)	1979-01-31	Novel steroids of the androstane series,their preparation compositions containing them
SE7608092L (sv)	1977-01-17	Nya steroider
GB1104462A (en)	1968-02-28	7ª-methyl-steroids of the oestrane series
GB2000137A (en)	1979-01-04	7,8-Dihydro-14-hydroxy-normorphine
NZ188755A (en)	1981-02-11	Formulations of steroids of estrane,androstane and 19-nor-pregnane series and tocol or a derivative thereof
IL49132A0 (en)	1976-05-31	New steroids of the androstane series,their preparation and pharmaceutical compositions containing them
ES2071939T3 (es)	1995-07-01	Nuevos productos esteroides que comprenden un radical espiro en posicion 17, su procedimiento de preparacion y los productos intermedios de este procedimiento, su aplicacion como medicamentos y composiciones farmaceuticas que los contienen.
FR2384794A1 (fr)	1978-10-20	Methylene-1a,2a steroides et medicaments qui en contiennent
FR2422689A1 (fr)	1979-11-09	Steroides de la serie du pregnane a groupe hydroxy etherifie en position 17 et medicaments qui en contiennent
DK208780A (da)	1980-11-18	16alfa-alkylsteroider fremgangsmaade til deres fremstilling og farmaceutiske praeparater indeholdende dem
DE2962721D1 (en)	1982-06-24	Hydrocortisone esters, pharmaceutical compositions containing them and process for their preparation
GB1100444A (en)	1968-01-24	13-alkyl 17-halogenoalkynyl steroid 3-alcohols and their esters
SE336789B (fr)	1971-07-19
GB1469223A (en)	1977-04-06	Azidocarbonic acid esters of steroids
GB1089237A (en)	1967-11-01	Improvements in or relating to tetrahydrofuranyl ethers of 17ª‰-hydroxy-androstane compounds
JPS5236654A (en)	1977-03-22	Process for preparation of steroid derivatives
DK103018C (da)	1965-11-08	Fremgangsmåde til fremstilling af 3-keto-Δ<4,6>-steroider af androstan- eller pregnanrækken.
FI793027A7 (fi)	1981-01-01	Uusia androstaani-, estraani- ja pregnaani-sarjan 3 -amino-2 -hydroksi-steroideja, menetelmiä niiden vavalmistamiseksi sekä farmaseuttisia yhdistelmiä.
GB1244143A (en)	1971-08-25	Trialkyl-silyloxy-steroids
JPS5283446A (en)	1977-07-12	Preparation of hydrocortisone derivatives