SE8105452L - Forfarande for framstellning av cefalosporiner - Google Patents

Forfarande for framstellning av cefalosporiner

Info

Publication number: SE8105452L
Authority: SE; Sweden
Prior art keywords: group; acid; displaces; image; cephalosporines
Prior art date: 1980-09-15

Application number

SE8105452A

Other languages

English (en)

Other versions

SE452619B (sv

Inventor

S Iimura

J Naito

J Okumura

Original Assignee

Bristol Myers Co

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1980-09-15

Filing date

1981-09-14

Publication date

1982-03-16

1981-09-14 Application filed by Bristol Myers Co filed Critical Bristol Myers Co

1982-03-16 Publication of SE8105452L publication Critical patent/SE8105452L/sv

1987-12-07 Publication of SE452619B publication Critical patent/SE452619B/sv

Links

239000002253 acid Substances 0.000 abstract 3
125000003277 amino group Chemical group 0.000 abstract 2
229930186147 Cephalosporin Natural products 0.000 abstract 1
UFHFLCQGNIYNRP-UHFFFAOYSA-N Hydrogen Chemical compound [H][H] UFHFLCQGNIYNRP-UHFFFAOYSA-N 0.000 abstract 1
125000002252 acyl group Chemical group 0.000 abstract 1
GCFBRXLSHGKWDP-XCGNWRKASA-N cefoperazone Chemical compound O=C1C(=O)N(CC)CCN1C(=O)N[C@H](C=1C=CC(O)=CC=1)C(=O)N[C@@H]1C(=O)N2C(C(O)=O)=C(CSC=3N(N=NN=3)C)CS[C@@H]21 GCFBRXLSHGKWDP-XCGNWRKASA-N 0.000 abstract 1
229960004682 cefoperazone Drugs 0.000 abstract 1
229940124587 cephalosporin Drugs 0.000 abstract 1
150000001780 cephalosporins Chemical class 0.000 abstract 1
229910052739 hydrogen Inorganic materials 0.000 abstract 1
239000001257 hydrogen Substances 0.000 abstract 1
150000007970 thio esters Chemical class 0.000 abstract 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Communicable Diseases (AREA)
Oncology (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Pharmacology & Pharmacy (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Cephalosporin Compounds (AREA)
Plural Heterocyclic Compounds (AREA)
Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)

SE8105452A 1980-09-15 1981-09-14 Nytt forfarande for framstellning av cefalosporiner SE452619B (sv)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
US06/187,273 US4316024A (en)	1980-09-15	1980-09-15	Dioxo piperazine compounds

Publications (2)

Publication Number	Publication Date
SE8105452L true SE8105452L (sv)	1982-03-16
SE452619B SE452619B (sv)	1987-12-07

Family

ID=22688303

Family Applications (2)

Application Number	Title	Priority Date	Filing Date
SE8105452A SE452619B (sv)	1980-09-15	1981-09-14	Nytt forfarande for framstellning av cefalosporiner
SE8505891A SE458607B (sv)	1980-09-15	1985-12-12	1-metyltetrazol-5-yl-(4-etyl-2,3-dioxopierazin-1-yl)-karbonyltiolat och tetrazolo-(1,5-b)pyridazin-6-yl-(4-etyl-2,3-dioxopiperazin-l-yl) karbonyltiolat

Family Applications After (1)

Application Number	Title	Priority Date	Filing Date
SE8505891A SE458607B (sv)	1980-09-15	1985-12-12	1-metyltetrazol-5-yl-(4-etyl-2,3-dioxopierazin-1-yl)-karbonyltiolat och tetrazolo-(1,5-b)pyridazin-6-yl-(4-etyl-2,3-dioxopiperazin-l-yl) karbonyltiolat

Country Status (10)

Country	Link
US (1)	US4316024A (sv)
JP (2)	JPS5781490A (sv)
DK (2)	DK161521C (sv)
ES (1)	ES8301238A1 (sv)
FI (1)	FI76349C (sv)
GR (1)	GR74670B (sv)
HU (1)	HU184882B (sv)
IT (1)	IT1209898B (sv)
SE (2)	SE452619B (sv)
YU (2)	YU44963B (sv)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
EP0047014B1 (en) *	1980-09-02	1986-01-15	Asahi Kasei Kogyo Kabushiki Kaisha	Novel thioesters and process for the preparation of the same
CH648038A5 (de) *	1981-01-19	1985-02-28	Sandoz Ag	7-((carboxymethoxyimino)-1h-pyrazol-3-yl-acetyl)amino-3-desacetoxy-3-(1-methyl-1h-tetrazol-5-yl-thio)cephalosporansaeure und salze, verfahren zur herstellung und verwendung.
JPS60142987A (ja) *	1983-12-29	1985-07-29	Mochida Pharmaceut Co Ltd	セフアロスポリン誘導体
EP0150507B1 (en) *	1983-12-29	1992-08-05	Mochida Pharmaceutical Co., Ltd.	Cephalosporin derivatives, processes for producing the same and compositions containing them
US4840945A (en) *	1985-04-01	1989-06-20	Mochida Pharmaceutical Co., Ltd.	Cephalosporin derivatives
JPS63132893A (ja) *	1986-11-25	1988-06-04	Mochida Pharmaceut Co Ltd	新規セフアロスポリン誘導体、その製法およびそれらを有効成分とする抗菌剤
US4880798A (en) *	1986-11-25	1989-11-14	Mochida Pharmaceutical Co., Ltd.	Cephalosporin derivatives
SI8711089A8 (en) *	1987-06-11	1996-08-31	Krka Tovarna Zdravil	Process for preparation of 6-/d(-)-alpha-(4-ethyl-2,3-dioxo-1- piperazine-carboxyamido)-phenylacetamido/-penicillanic acid
CN102372728B (zh) *	2011-11-28	2013-12-11	齐鲁安替制药有限公司	一种头孢菌素类化合物的合成方法
CN102372729B (zh) *	2011-12-14	2014-09-24	哈药集团制药总厂	一种合成头孢哌酮钠化合物的新方法
CN103641847B (zh) *	2013-11-28	2016-04-20	山东鑫泉医药有限公司	头孢哌酮酸的制备方法

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US4087424A (en) *	1974-05-09	1978-05-02	Toyama Chemical Co., Ltd.	Novel penicillins and cephalosporins and process for producing the same
JPS51115491A (en) *	1975-04-03	1976-10-12	Sumitomo Chem Co Ltd	Method for preparing 77* 44hydroxyy15 naphthyridinee33carboxyamino ** phenylacetamido*cephalosporins
JPS5520711A (en) *	1978-08-01	1980-02-14	Asahi Chem Ind Co Ltd	New 1,3,4-thiadiazol-5-ylthiol esters and their preparation
JPS6052711B2 (ja) *	1978-03-09	1985-11-20	旭化成株式会社	セフアロスポリン化合物の製法
US4198504A (en) *	1978-11-02	1980-04-15	Bristol-Myers Company	[3-(Pyridinium)-7-(naphthyiridinyl carbonylamino)acetamido]cephalosporanic acid derivatives

1980
- 1980-09-15 US US06/187,273 patent/US4316024A/en not_active Expired - Lifetime
1981
- 1981-08-28 GR GR65890A patent/GR74670B/el unknown
- 1981-09-04 YU YU2131/81A patent/YU44963B/xx unknown
- 1981-09-10 FI FI812821A patent/FI76349C/sv not_active IP Right Cessation
- 1981-09-11 DK DK404181A patent/DK161521C/da not_active IP Right Cessation
- 1981-09-14 SE SE8105452A patent/SE452619B/sv not_active IP Right Cessation
- 1981-09-14 HU HU812652A patent/HU184882B/hu not_active IP Right Cessation
- 1981-09-14 ES ES505465A patent/ES8301238A1/es not_active Expired
- 1981-09-15 IT IT8149296A patent/IT1209898B/it active
- 1981-09-16 JP JP56144790A patent/JPS5781490A/ja active Granted
1983
- 1983-10-31 YU YU2174/83A patent/YU44754B/xx unknown
1985
- 1985-12-12 SE SE8505891A patent/SE458607B/sv not_active IP Right Cessation
1989
- 1989-08-24 JP JP1216008A patent/JPH0285278A/ja active Granted
1991
- 1991-01-18 DK DK008991A patent/DK164505C/da not_active IP Right Cessation

Also Published As

Publication number	Publication date
YU213181A (en)	1984-06-30
DK8991A (da)	1991-01-18
HU184882B (en)	1984-10-29
GR74670B (sv)	1984-07-02
YU217483A (en)	1985-10-31
ES505465A0 (es)	1982-12-01
YU44754B (en)	1991-02-28
DK164505B (da)	1992-07-06
FI76349C (sv)	1988-10-10
DK161521B (da)	1991-07-15
IT8149296A0 (it)	1981-09-15
JPH0245636B2 (sv)	1990-10-11
JPS5781490A (en)	1982-05-21
YU44963B (en)	1991-06-30
SE8505891D0 (sv)	1985-12-12
JPH0285278A (ja)	1990-03-26
SE452619B (sv)	1987-12-07
SE458607B (sv)	1989-04-17
ES8301238A1 (es)	1982-12-01
DK8991D0 (da)	1991-01-18
US4316024A (en)	1982-02-16
DK164505C (da)	1992-11-23
FI812821L (fi)	1982-03-16
JPH0246587B2 (sv)	1990-10-16
IT1209898B (it)	1989-08-30
FI76349B (fi)	1988-06-30
DK404181A (da)	1982-03-16
DK161521C (da)	1991-12-23
SE8505891L (sv)	1985-12-12

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Legal Events

Date

Code

Title

Description

1995-01-31

NUG

Patent has lapsed

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Effective date: 19940410

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