SE9600406L - Nya föreningar - Google Patents

Nya föreningar

Info

Publication number
SE9600406L
SE9600406L SE9600406A SE9600406A SE9600406L SE 9600406 L SE9600406 L SE 9600406L SE 9600406 A SE9600406 A SE 9600406A SE 9600406 A SE9600406 A SE 9600406A SE 9600406 L SE9600406 L SE 9600406L
Authority
SE
Sweden
Prior art keywords
preparing
new compounds
compounds
sufferer
administering
Prior art date
Application number
SE9600406A
Other languages
English (en)
Other versions
SE9600406D0 (sv
SE521084C2 (sv
Inventor
Victor Witold Jacewicz
Neal Ward
Original Assignee
Smithkline Beecham Plc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=27267578&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=SE9600406(L) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Priority claimed from GBGB9502297.6A external-priority patent/GB9502297D0/en
Priority claimed from GBGB9503112.6A external-priority patent/GB9503112D0/en
Priority claimed from GBGB9509807.5A external-priority patent/GB9509807D0/en
Application filed by Smithkline Beecham Plc filed Critical Smithkline Beecham Plc
Publication of SE9600406D0 publication Critical patent/SE9600406D0/sv
Publication of SE9600406L publication Critical patent/SE9600406L/sv
Publication of SE521084C2 publication Critical patent/SE521084C2/sv

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D405/00Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/12Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/04Centrally acting analgesics, e.g. opioids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/24Antidepressants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/26Psychostimulants, e.g. nicotine, cocaine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/28Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/04Anorexiants; Antiobesity agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P39/00General protective or antinoxious agents

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Psychiatry (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Diabetes (AREA)
  • Pain & Pain Management (AREA)
  • Toxicology (AREA)
  • Child & Adolescent Psychology (AREA)
  • Hospice & Palliative Care (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
SE9600406A 1995-02-06 1996-02-05 Förfarande för framställning av paroxetin-hydroklorid- anhydrat från ett paroxetin-hydroklorid-solvat SE521084C2 (sv)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GBGB9502297.6A GB9502297D0 (en) 1995-02-06 1995-02-06 Novel compound
GBGB9503112.6A GB9503112D0 (en) 1995-02-17 1995-02-17 Novel compound
GBGB9509807.5A GB9509807D0 (en) 1995-05-15 1995-05-15 Novel compounds

Publications (3)

Publication Number Publication Date
SE9600406D0 SE9600406D0 (sv) 1996-02-05
SE9600406L true SE9600406L (sv) 1996-08-07
SE521084C2 SE521084C2 (sv) 2003-09-30

Family

ID=27267578

Family Applications (1)

Application Number Title Priority Date Filing Date
SE9600406A SE521084C2 (sv) 1995-02-06 1996-02-05 Förfarande för framställning av paroxetin-hydroklorid- anhydrat från ett paroxetin-hydroklorid-solvat

Country Status (47)

Country Link
EP (3) EP1136490B1 (sv)
JP (2) JP2915338B2 (sv)
KR (1) KR100289885B1 (sv)
CN (3) CN1090187C (sv)
AR (2) AR001982A1 (sv)
AT (1) AT407528B (sv)
AU (2) AU4786496A (sv)
BE (1) BE1009112A3 (sv)
BG (1) BG62967B1 (sv)
BR (1) BR9600534A (sv)
CA (3) CA2210022C (sv)
CH (3) CH689229A5 (sv)
CZ (1) CZ297171B6 (sv)
DE (3) DE69621777T2 (sv)
DK (2) DK11996A (sv)
DZ (1) DZ1989A1 (sv)
ES (1) ES2114471B1 (sv)
FI (3) FI111544B (sv)
FR (1) FR2730232B1 (sv)
GR (1) GR1002466B (sv)
HK (1) HK59397A (sv)
HU (1) HUP9600255A1 (sv)
IE (1) IE80500B1 (sv)
IL (1) IL117035A (sv)
IT (1) IT1289532B1 (sv)
LU (1) LU88711A1 (sv)
LV (1) LV11618B (sv)
MA (1) MA23802A1 (sv)
MC (1) MC2411A1 (sv)
MX (1) MX9600484A (sv)
MY (1) MY132529A (sv)
NL (1) NL1002248C2 (sv)
NO (3) NO301009B1 (sv)
NZ (1) NZ280943A (sv)
OA (1) OA10261A (sv)
PL (1) PL189247B1 (sv)
PT (1) PT101827B (sv)
RO (1) RO112426B1 (sv)
RU (1) RU2125052C1 (sv)
SE (1) SE521084C2 (sv)
SG (1) SG43787A1 (sv)
SI (2) SI9600036B (sv)
SK (1) SK283608B6 (sv)
TR (1) TR199600096A2 (sv)
TW (1) TW503238B (sv)
UA (1) UA49796C2 (sv)
WO (1) WO1996024595A1 (sv)

Families Citing this family (39)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP3882224B2 (ja) 1996-05-31 2007-02-14 旭硝子株式会社 パロキセチンの製造方法
EP1394160A1 (en) * 1996-06-13 2004-03-03 SUMIKA FINE CHEMICALS Co., Ltd. Process for preparing crystalline paroxetin hydrochloride
JP2000514653A (ja) * 1996-07-15 2000-11-07 スミスクライン・ビーチャム・パブリック・リミテッド・カンパニー 立体特異的分割のためのエステラーゼのスクリーニングおよびその使用
US6638948B1 (en) 1996-09-09 2003-10-28 Pentech Pharmaceuticals, Inc. Amorphous paroxetine composition
US5672612A (en) * 1996-09-09 1997-09-30 Pentech Pharmaceuticals, Inc. Amorphous paroxetine composition
EE03970B1 (et) 1997-06-10 2003-02-17 Synthon B.V. 4-fenüülpiperidiinühend, selle valmistamine ja kasutamine ning seda sisaldav ravim
DK0987256T3 (da) * 1997-08-08 2002-02-11 Aventis Pharma Gmbh Krystalform af N-(4-trifluormethylphenyl)-5-methylisoxazol-4-carboxylsyreamid
GB9726907D0 (en) * 1997-12-19 1998-02-18 Smithkline Beecham Plc Novel compounds
IL138390A0 (en) * 1998-03-16 2001-10-31 Smithkline Beecham Plc Crystalline form of paroxetine
GB9806312D0 (en) * 1998-03-24 1998-05-20 Smithkline Beecham Plc Novel formulations
AU2003200534B2 (en) * 1998-03-24 2004-12-02 Smithkline Beecham Plc Paroxetine compositions
US6699882B2 (en) 1998-03-24 2004-03-02 Smithkline Beecham P.L.C. Paroxetine compositions
JP3796351B2 (ja) 1998-04-13 2006-07-12 住友化学株式会社 パロキセチン塩酸塩無水和物の乾燥方法
GB9812941D0 (en) * 1998-06-16 1998-08-12 Smithkline Beecham Plc Method of treatment
CH689805A8 (fr) * 1998-07-02 2000-02-29 Smithkline Beecham Plc Méthanesulfonate de paroxétine, procédé pour sa préparation et compositions pharmaceutiques le contenant.
ES2138937B1 (es) 1998-07-07 2000-10-01 Medichem Sa Polimorfo de maleato de paroxetina y formulaciones farmaceuticas que lo contienen.
WO2000008017A1 (en) * 1998-08-07 2000-02-17 Smithkline Beecham Plc Process for the preparation of a non-crystalline anhydrate form of paroxetine hydrochloride
GB9824298D0 (en) * 1998-11-05 1998-12-30 Smithkline Beecham Plc Novel process
GB9826176D0 (en) * 1998-11-28 1999-01-20 Smithkline Beecham Plc Novel process
GB9826175D0 (en) * 1998-11-28 1999-01-20 Smithkline Beecham Plc Novel process
GB9826178D0 (en) * 1998-11-30 1999-01-20 Smithkline Beecham Plc Novel process
GB9826180D0 (en) * 1998-11-30 1999-01-20 Smithkline Beecham Plc Novel process
WO2000032594A1 (en) * 1998-11-30 2000-06-08 Smithkline Beecham Plc Mixed paroxetine propan-2-ol solvates
GB9826242D0 (en) * 1998-11-30 1999-01-20 Smithkline Beecham Plc Novel process
GB9826171D0 (en) * 1998-11-30 1999-01-20 Smithkline Beecham Plc Novel compounds
GB9828767D0 (en) * 1998-12-29 1999-02-17 Smithkline Beecham Plc Novel process
IT1308629B1 (it) * 1999-02-23 2002-01-09 Recordati Chem Pharm Processo per la produzione di paroxetina.
ATE311883T1 (de) * 1999-03-12 2005-12-15 Aesica Pharmaceuticals Ltd Stabile pharmazeutische anwendungsform für paroxetin-anhydrat
GB9914583D0 (en) * 1999-06-22 1999-08-25 Smithkline Beecham Plc Novel process
GB9914585D0 (en) * 1999-06-22 1999-08-25 Smithkline Beecham Plc Novel process
SE9902550D0 (sv) * 1999-07-02 1999-07-02 Astra Ab New crystalline forms
GB9919001D0 (en) * 1999-08-12 1999-10-13 Smithkline Beecham Plc Novel process
GB9923445D0 (en) * 1999-10-04 1999-12-08 Smithkline Beecham Plc Novel process
GB9923446D0 (en) * 1999-10-04 1999-12-08 Smithkline Beecham Plc Novel process
GB9923439D0 (en) * 1999-10-04 1999-12-08 Smithkline Beecham Plc Novel process
HU226912B1 (en) * 2000-04-07 2010-03-01 Richter Gedeon Nyrt New paroxetin salt and medicament containing it
AU2001286232A1 (en) * 2000-09-14 2002-03-26 Asahi Glass Company, Limited Process for producing paroxetine salt containing substantially no organic solvent
WO2003072104A1 (en) * 2002-02-22 2003-09-04 Teva Pharmaceutical Industries Ltd. Preparation of paroxetine involving novel intermediates
US7563930B2 (en) * 2005-11-22 2009-07-21 Teva Pharmaceutical Industries Ltd Crystal forms of Cinacalcet HCI and processes for their preparation

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1422263A (en) * 1973-01-30 1976-01-21 Ferrosan As 4-phenyl-piperidine compounds
GB8430581D0 (en) * 1984-12-04 1985-01-09 Ferrosan As Treatment
EP0223403B1 (en) * 1985-10-25 1993-08-04 Beecham Group Plc Piperidine derivative, its preparation, and its use as medicament
US5017585A (en) * 1986-11-03 1991-05-21 Novo Nordisk A/S Method of treating calcium overload
GB8626936D0 (en) * 1986-11-11 1986-12-10 Ferrosan As Treatment
DK715988D0 (da) * 1988-12-22 1988-12-22 Ferrosan As Etherifikation og dealkylering af piperidin-derivater samt intermediater
DK716088D0 (da) * 1988-12-22 1988-12-22 Ferrosan As Reduktion af piperidin-dion-derivater samt intermediat
JPH06502854A (ja) * 1990-11-24 1994-03-31 ビーチャム・グループ・パブリック・リミテッド・カンパニー 老年痴呆、過食症、片頭痛または食欲不振の治療用のパロキセチンの使用
US5258517A (en) * 1992-08-06 1993-11-02 Sepracor, Inc. Method of preparing optically pure precursors of paroxetine
GB9325644D0 (en) * 1993-12-15 1994-02-16 Smithkline Beecham Plc Novel formulation

Also Published As

Publication number Publication date
CN1289496C (zh) 2006-12-13
AU4332896A (en) 1996-08-15
OA10261A (en) 1997-09-19
CA2211522C (en) 1999-12-07
AU701518C (en) 2006-12-07
FI960519L (sv) 1996-08-07
IL117035A (en) 2000-02-29
SI21923B (sl) 2006-12-31
EP0808314B1 (en) 2002-06-12
NO311519B1 (no) 2001-12-03
FR2730232B1 (fr) 1997-08-01
HUP9600255A1 (en) 1997-03-28
EP0808314A1 (en) 1997-11-26
MY132529A (en) 2007-10-31
NO301009B1 (no) 1997-09-01
CH688353A5 (de) 1997-08-15
IE960104A1 (en) 1996-08-07
CN1090187C (zh) 2002-09-04
DK11996A (da) 1996-08-07
DZ1989A1 (fr) 2002-10-15
IT1289532B1 (it) 1998-10-15
MX9600484A (es) 1997-01-31
PT101827A (pt) 1996-09-30
DE19603797C2 (de) 1998-11-12
CZ32096A3 (en) 1996-08-14
DE69621777T2 (de) 2003-01-02
ES2114471B1 (es) 1999-08-16
NZ280943A (en) 1997-01-29
JPH11228571A (ja) 1999-08-24
EP1136490A1 (en) 2001-09-26
CN1636993A (zh) 2005-07-13
AR001982A1 (es) 1998-01-07
CA2211522A1 (en) 1996-08-07
SI9600036B (sl) 2006-12-31
FI20030370L (sv) 2003-03-12
CN1143643A (zh) 1997-02-26
CA2168829C (en) 1997-12-16
MC2411A1 (fr) 1996-12-02
NO20015070D0 (no) 2001-10-18
CH689229A5 (de) 1998-12-31
AT407528B (de) 2001-04-25
ATA21096A (de) 2000-08-15
TW503238B (en) 2002-09-21
DK200100223A (sv) 2001-02-12
AU701518B2 (en) 1999-01-28
RU2125052C1 (ru) 1999-01-20
NL1002248C2 (nl) 1996-09-11
CA2210023A1 (en) 1996-08-07
NO301009B3 (sv) 2003-01-06
SK14396A3 (en) 1996-11-06
CN1310180A (zh) 2001-08-29
FI960519A0 (sv) 1996-02-05
LV11618A (lv) 1996-12-20
PL312646A1 (en) 1996-08-19
JP2915338B2 (ja) 1999-07-05
DE69621777D1 (de) 2002-07-18
SI9600036A (en) 1996-10-31
CA2210023C (en) 1999-02-09
BR9600534A (pt) 1997-05-13
CA2210022A1 (en) 1996-08-07
KR960031409A (ko) 1996-09-17
KR100289885B1 (ko) 2001-05-15
FR2730232A1 (fr) 1996-08-09
LV11618B (en) 1997-04-20
AU4786496A (en) 1996-08-27
BG100333A (bg) 1996-08-30
SK283608B6 (sk) 2003-10-07
NO960472L (no) 1996-08-07
FI111544B (sv) 2003-08-15
FI20030370A7 (sv) 2003-03-12
SE9600406D0 (sv) 1996-02-05
MA23802A1 (fr) 1996-10-01
DE19603797A1 (de) 1996-08-14
BG62967B1 (bg) 2000-12-29
DE69631298D1 (de) 2004-02-12
IL117035A0 (en) 1996-09-12
ES2114471A1 (es) 1998-05-16
ITMI960203A1 (it) 1997-08-05
NL1002248A1 (nl) 1996-08-06
FI20030162A7 (sv) 2003-02-03
CA2168829A1 (en) 1996-08-07
NO20015070L (no) 1996-08-07
NO960472D0 (no) 1996-02-05
SI21923A (sl) 2006-06-30
SG43787A1 (en) 1997-11-14
GR1002466B (el) 1996-11-06
CZ297171B6 (cs) 2006-09-13
NO970939D0 (no) 1997-02-28
PL189247B1 (pl) 2005-07-29
FI20030162L (sv) 2003-02-03
TR199600096A2 (tr) 1996-08-21
JPH08245620A (ja) 1996-09-24
IE80500B1 (en) 1998-08-12
SE521084C2 (sv) 2003-09-30
UA49796C2 (uk) 2002-10-15
HU9600255D0 (en) 1996-03-28
DE69631298T2 (de) 2004-11-18
EP1136490B1 (en) 2004-01-07
WO1996024595A1 (en) 1996-08-15
LU88711A1 (fr) 1996-08-23
ITMI960203A0 (sv) 1996-02-05
BE1009112A3 (fr) 1996-11-05
CN1216055C (zh) 2005-08-24
NO970939L (no) 1996-08-07
PT101827B (pt) 1997-08-29
RO112426B1 (ro) 1997-09-30
AR036856A2 (es) 2004-10-06
MX198371B (sv) 2000-08-29
HK59397A (en) 1997-05-16
EP1378508A1 (en) 2004-01-07
CA2210022C (en) 2005-09-13
CH689804A5 (de) 1999-11-30

Similar Documents

Publication Publication Date Title
SE9600406D0 (sv) Novel coompounds
DE69427017D1 (de) Herstellung von 3,4,4-trisubstituiertem Piperidinyl-n-alkylcarboxylaten und Zwischenverbindungen, verwendbar als opioid Antagonisten
HU9600834D0 (en) Quinazoline derivatives
PT923554E (pt) N-benzilpiperidina e derivados tetrahidropiridina
DE69527072D1 (de) Endothelin antagoniste
DE69716810D1 (de) 2,3-Disubstituierte-(5,6)-heteroarylkondensierte-pyrimidin-4-one
BR9506835A (pt) Acido micofenólico substituído em 6 e derivados
DK1109817T3 (da) Phosphohalogenhydriner, deres fremstilling og anvendelse
DE69613705D1 (de) Piperinderivate als neurokininantagoniste
FI914927A0 (fi) Fungicida oxazolidinoner.
NO921182L (no) Piperidinderivater
ATE127693T1 (de) Zusammensetzung und verfahren zum schutz gegen durch mikroorganismen verursachte krankheiten.
DE69816731D1 (de) Benzofuranon-derivate und verfahren zu ihrer herstellung
DE69431035D1 (de) 2-Phenyl-3-Azoylbenzothiophene zur Erhöhung der Thrombomodulin Expression
ATE303362T1 (de) Chalcon-derivate mit antiproliferativer aktivität
DE69805305D1 (de) Verwendung von phanquinon zur behandlung von alzheimer's krankheit
BR9612074A (pt) Novos 4-(1h-benzimidazol-2-il)(1,4) diazepanos substituidos úteis para o tratamento de doenças alérgicas
EA199800102A1 (ru) Получение производных бициклогексана
TR199901395T2 (xx) Yeni karboksi ikameli siklik karboksamid t�revleri.
PT96422A (pt) Processo para a preparacao de derivados de piperidina e de pirrolidina uteis como agentes anticolinergicos
PT889044E (pt) Derivados do 5-(heteroaril)alquil-3-oxo-pirido-(1,2-a)benzimidazole-4-carboxamida (pbi) uteis no tratamento de perturbacoes do sistema nervoso central
SE9404438D0 (sv) New process
NO995132L (no) Fremgangsmåte for reduksjon av fibrinogen

Legal Events

Date Code Title Description
CANC Patent cancelled, revoked after opposition
NUG Patent has lapsed