SK14042003A3 - Kombinácia N-{5-[4-metylpiperazinometyl)benzoylamido]-2- metylfenyl}-4-(3-pyridyl)-2-pyrimidínamínu chemoterapeutického činidla a farmaceutický prostriedok, ktorý ju obsahuje - Google Patents

Kombinácia N-{5-[4-metylpiperazinometyl)benzoylamido]-2- metylfenyl}-4-(3-pyridyl)-2-pyrimidínamínu chemoterapeutického činidla a farmaceutický prostriedok, ktorý ju obsahuje Download PDF

Info

Publication number: SK14042003A3
Authority: SK; Slovakia
Prior art keywords: group; combination; compounds; administered; patients
Prior art date: 2001-05-16

Application number

SK1404-2003A

Other languages

English (en)

Slovak (sk)

Inventor

Christian Bruns

Elisabeth Buchdunger

Terence O'reilly

Sandra Leta Silberman

Markus Wartmann

Gisbert Weckbecker

Original Assignee

Novartis Ag

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2001-05-16

Filing date

2002-05-15

Publication date

2004-05-04

2002-05-15 Application filed by Novartis Ag filed Critical Novartis Ag

2004-05-04 Publication of SK14042003A3 publication Critical patent/SK14042003A3/sk

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Classifications

- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
- A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/506—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim not condensed and containing further heterocyclic rings
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A61P35/04—Antineoplastic agents specific for metastasis
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/02—Immunomodulators
- A61P37/06—Immunosuppressants, e.g. drugs for graft rejection
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

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Health & Medical Sciences (AREA)
Animal Behavior & Ethology (AREA)
Chemical & Material Sciences (AREA)
Veterinary Medicine (AREA)
Public Health (AREA)
Medicinal Chemistry (AREA)
General Health & Medical Sciences (AREA)
Pharmacology & Pharmacy (AREA)
Life Sciences & Earth Sciences (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Organic Chemistry (AREA)
General Chemical & Material Sciences (AREA)
Chemical Kinetics & Catalysis (AREA)
Epidemiology (AREA)
Immunology (AREA)
Bioinformatics & Cheminformatics (AREA)
Engineering & Computer Science (AREA)
Oncology (AREA)
Transplantation (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Pyridine Compounds (AREA)

SK1404-2003A 2001-05-16 2002-05-15 Kombinácia N-{5-[4-metylpiperazinometyl)benzoylamido]-2- metylfenyl}-4-(3-pyridyl)-2-pyrimidínamínu chemoterapeutického činidla a farmaceutický prostriedok, ktorý ju obsahuje SK14042003A3 (sk)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
US29142701P	2001-05-16	2001-05-16
PCT/EP2002/005362 WO2002092091A1 (en)	2001-05-16	2002-05-15	Combination comprising n-{5-[4-(4-methyl-piperazino-methyl)-benzoylamido]-2-methylphenyl}-4-(3-pyridyl)-2pyrimidine-amine and a chemotherapeutic agent

Publications (1)

Publication Number	Publication Date
SK14042003A3 true SK14042003A3 (sk)	2004-05-04

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Country Status (27)

Country	Link
US (3)	US20040167134A1 (es)
EP (2)	EP1392313B1 (es)
JP (2)	JP4477303B2 (es)
KR (2)	KR20030094415A (es)
CN (1)	CN1700917B (es)
AT (1)	ATE359790T1 (es)
AU (1)	AU2002342335B2 (es)
BR (1)	BR0209647A (es)
CA (1)	CA2444867C (es)
CO (1)	CO5540315A2 (es)
CZ (1)	CZ299756B6 (es)
DE (1)	DE60219617T2 (es)
DK (1)	DK1392313T3 (es)
EC (1)	ECSP034823A (es)
ES (1)	ES2283570T3 (es)
HU (1)	HUP0400038A3 (es)
IL (1)	IL158274A0 (es)
MX (1)	MXPA03010401A (es)
NO (2)	NO325453B1 (es)
NZ (1)	NZ529145A (es)
PL (2)	PL392652A1 (es)
PT (1)	PT1392313E (es)
RU (1)	RU2318517C2 (es)
SI (1)	SI1392313T1 (es)
SK (1)	SK14042003A3 (es)
WO (1)	WO2002092091A1 (es)
ZA (1)	ZA200307665B (es)

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2002
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Also Published As

Publication number	Publication date
CN1700917B (zh)	2010-04-28
HK1062895A1 (en)	2004-12-03
CA2444867A1 (en)	2002-11-21
US20040167134A1 (en)	2004-08-26
IL158274A0 (en)	2004-05-12
ATE359790T1 (de)	2007-05-15
CZ20033098A3 (cs)	2004-02-18
EP1392313A1 (en)	2004-03-03
RU2318517C2 (ru)	2008-03-10
ES2283570T3 (es)	2007-11-01
NO20034713D0 (no)	2003-10-21
WO2002092091A1 (en)	2002-11-21
CN1700917A (zh)	2005-11-23
CO5540315A2 (es)	2005-07-29
HUP0400038A2 (hu)	2004-04-28
US20120283206A1 (en)	2012-11-08
AU2002342335B2 (en)	2006-02-02
NO20034713L (no)	2003-10-21
PL368068A1 (en)	2005-03-21
KR20030094415A (ko)	2003-12-11
MXPA03010401A (es)	2004-03-09
SI1392313T1 (sl)	2007-08-31
NZ529145A (en)	2005-07-29
ZA200307665B (en)	2004-04-21
JP2004531549A (ja)	2004-10-14
DK1392313T3 (da)	2007-06-25
KR20080091866A (ko)	2008-10-14
HUP0400038A3 (en)	2007-05-29
US20090202541A1 (en)	2009-08-13
NO325453B1 (no)	2008-05-05
PT1392313E (pt)	2007-07-17
RU2003135786A (ru)	2005-02-27
EP2253319A1 (en)	2010-11-24
JP2010059202A (ja)	2010-03-18
PL392652A1 (pl)	2010-12-06
DE60219617T2 (de)	2008-01-03
NO20076323L (no)	2007-12-07
EP1392313B1 (en)	2007-04-18
ECSP034823A (es)	2003-12-24
JP4477303B2 (ja)	2010-06-09
CZ299756B6 (cs)	2008-11-12
DE60219617D1 (de)	2007-05-31
CA2444867C (en)	2010-08-17
BR0209647A (pt)	2004-07-27

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2010-05-07	FC9A	Refused patent application

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