SK19992000A3 - Použitie kyseliny 2-n-propyl-4-hexínovej na liečenie a prevenciu migrény a afektívneho ochorenia - Google Patents

Použitie kyseliny 2-n-propyl-4-hexínovej na liečenie a prevenciu migrény a afektívneho ochorenia Download PDF

Info

Publication number: SK19992000A3
Authority: SK; Slovakia
Prior art keywords: migraine; propyl; acid; valproic acid; compound
Prior art date: 1998-06-22

Application number

SK1999-2000A

Other languages

English (en)

Slovak (sk)

Inventor

Heinz Nau

Emer Leahy

Alan O'connell

Original Assignee

American Biogenetic Sciences, Inc.

Heinz Nau

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1998-06-22

Filing date

1999-06-22

Publication date

2001-08-06

1999-06-22 Application filed by American Biogenetic Sciences, Inc., Heinz Nau filed Critical American Biogenetic Sciences, Inc.

2001-08-06 Publication of SK19992000A3 publication Critical patent/SK19992000A3/sk

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HBAQYPYDRFILMT-UHFFFAOYSA-N 8-[3-(1-cyclopropylpyrazol-4-yl)-1H-pyrazolo[4,3-d]pyrimidin-5-yl]-3-methyl-3,8-diazabicyclo[3.2.1]octan-2-one Chemical class C1(CC1)N1N=CC(=C1)C1=NNC2=C1N=C(N=C2)N1C2C(N(CC1CC2)C)=O HBAQYPYDRFILMT-UHFFFAOYSA-N 0.000 claims description 4
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239000001593 sorbitan monooleate Substances 0.000 description 1
235000011069 sorbitan monooleate Nutrition 0.000 description 1
229940035049 sorbitan monooleate Drugs 0.000 description 1
230000001954 sterilising effect Effects 0.000 description 1
238000004659 sterilization and disinfection Methods 0.000 description 1
239000011550 stock solution Substances 0.000 description 1
150000008163 sugars Chemical class 0.000 description 1
239000000829 suppository Substances 0.000 description 1
239000004094 surface-active agent Substances 0.000 description 1
239000000375 suspending agent Substances 0.000 description 1
239000008399 tap water Substances 0.000 description 1
235000020679 tap water Nutrition 0.000 description 1
230000001225 therapeutic effect Effects 0.000 description 1
231100001274 therapeutic index Toxicity 0.000 description 1
231100000419 toxicity Toxicity 0.000 description 1
230000001988 toxicity Effects 0.000 description 1
239000000196 tragacanth Substances 0.000 description 1
235000010487 tragacanth Nutrition 0.000 description 1
229940116362 tragacanth Drugs 0.000 description 1
QORWJWZARLRLPR-UHFFFAOYSA-H tricalcium bis(phosphate) Chemical compound [Ca+2].[Ca+2].[Ca+2].[O-]P([O-])([O-])=O.[O-]P([O-])([O-])=O QORWJWZARLRLPR-UHFFFAOYSA-H 0.000 description 1
238000009827 uniform distribution Methods 0.000 description 1
239000005526 vasoconstrictor agent Substances 0.000 description 1
238000005303 weighing Methods 0.000 description 1

Classifications

- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/185—Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
- A61K31/19—Carboxylic acids, e.g. valproic acid
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/06—Antimigraine agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia

Landscapes

Health & Medical Sciences (AREA)
Pharmacology & Pharmacy (AREA)
Veterinary Medicine (AREA)
Public Health (AREA)
Chemical & Material Sciences (AREA)
General Health & Medical Sciences (AREA)
Animal Behavior & Ethology (AREA)
Medicinal Chemistry (AREA)
Life Sciences & Earth Sciences (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Epidemiology (AREA)
Neurosurgery (AREA)
Organic Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
General Chemical & Material Sciences (AREA)
Chemical Kinetics & Catalysis (AREA)
Neurology (AREA)
Biomedical Technology (AREA)
Pain & Pain Management (AREA)
Psychiatry (AREA)
Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

SK1999-2000A 1998-06-22 1999-06-22 Použitie kyseliny 2-n-propyl-4-hexínovej na liečenie a prevenciu migrény a afektívneho ochorenia SK19992000A3 (sk)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
US9028198P	1998-06-22	1998-06-22
PCT/US1999/014081 WO1999066920A1 (en)	1998-06-22	1999-06-22	The use of valproic acid analog for the treatment and prevention of migraine and affective illness

Publications (1)

Publication Number	Publication Date
SK19992000A3 true SK19992000A3 (sk)	2001-08-06

Family

ID=22222101

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
SK1999-2000A SK19992000A3 (sk)	1998-06-22	1999-06-22	Použitie kyseliny 2-n-propyl-4-hexínovej na liečenie a prevenciu migrény a afektívneho ochorenia

Country Status (19)

Country	Link
US (2)	US6268396B1 (cs)
EP (1)	EP1089725A1 (cs)
JP (1)	JP2002518442A (cs)
KR (1)	KR20010071572A (cs)
CN (1)	CN1310622A (cs)
AU (2)	AU752192B2 (cs)
BG (1)	BG63744B1 (cs)
BR (1)	BR9911421A (cs)
CA (1)	CA2335641A1 (cs)
CZ (1)	CZ20004833A3 (cs)
HU (1)	HUP0102456A3 (cs)
IL (1)	IL140415A0 (cs)
MX (1)	MXPA00012808A (cs)
NO (1)	NO20006506L (cs)
PL (1)	PL345364A1 (cs)
SK (1)	SK19992000A3 (cs)
TR (2)	TR200003800T2 (cs)
WO (1)	WO1999066920A1 (cs)
ZA (1)	ZA200007652B (cs)

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AU2003278565A1 (en) *	2002-10-25	2004-05-13	Yissum Research Development Company Of The Hebrew University Of Jerusalem	Steroid compounds comprising superoxide dismutase mimic groups and nitric oxide donor groups, and their use in the preparation of medicaments
US20060166894A1 (en) *	2002-11-29	2006-07-27	Yissum Research Development Company Of The Hebrew University Of Jerusalem	Ace-inhibitors having antioxidant and no-donor activity
AU2003289782A1 (en) *	2002-12-16	2004-07-09	The University Of British Columbia	Valproic acid analogues and pharmaceutical compositions thereof
EP1543831A1 (en) *	2003-12-18	2005-06-22	Pfizer GmbH Arzneimittelwerk Gödecke	Pregabalin composition
US20060025477A1 (en) *	2004-07-22	2006-02-02	Artman Linda D	Analogs of isovaleramide, a pharmaceutical composition including the same, and a method of treating central nervous system conditions or diseases
US20080234213A1 (en) *	2005-09-02	2008-09-25	Matthias Wabl	Oncogenic regulatory RNAs for diagnostics and therapeutics
US7459280B2 (en) *	2006-02-27	2008-12-02	Picobella, Llc	Methods for diagnosing and treating kidney cancer
US20080267977A1 (en) *	2007-04-26	2008-10-30	Friedrich-Alexander University Of Erlangen-Nuremberg	Combined immunological agent and sensitizing agent for the treatment of cancer
AU2013257710B2 (en) *	2012-05-08	2016-10-20	Cellixbio Private Limited	Compositions and methods for the treatment of neurological disorders

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1999
- 1999-06-22 MX MXPA00012808A patent/MXPA00012808A/es unknown
- 1999-06-22 US US09/337,986 patent/US6268396B1/en not_active Expired - Fee Related
- 1999-06-22 JP JP2000555606A patent/JP2002518442A/ja active Pending
- 1999-06-22 CN CN99808955A patent/CN1310622A/zh active Pending
- 1999-06-22 CA CA002335641A patent/CA2335641A1/en not_active Abandoned
- 1999-06-22 EP EP99930555A patent/EP1089725A1/en not_active Withdrawn
- 1999-06-22 HU HU0102456A patent/HUP0102456A3/hu unknown
- 1999-06-22 WO PCT/US1999/014081 patent/WO1999066920A1/en not_active Ceased
- 1999-06-22 PL PL99345364A patent/PL345364A1/xx not_active Application Discontinuation
- 1999-06-22 BR BR9911421-6A patent/BR9911421A/pt not_active IP Right Cessation
- 1999-06-22 AU AU47071/99A patent/AU752192B2/en not_active Ceased
- 1999-06-22 IL IL14041599A patent/IL140415A0/xx unknown
- 1999-06-22 SK SK1999-2000A patent/SK19992000A3/sk unknown
- 1999-06-22 CZ CZ20004833A patent/CZ20004833A3/cs unknown
- 1999-06-22 KR KR1020007014630A patent/KR20010071572A/ko not_active Withdrawn
- 1999-06-22 TR TR2000/03800T patent/TR200003800T2/xx unknown
- 1999-06-27 TR TR2001/03249T patent/TR200103249T2/xx unknown
- 1999-06-28 AU AU52071/99A patent/AU5207199A/en not_active Abandoned
2000
- 2000-12-19 ZA ZA200007652A patent/ZA200007652B/en unknown
- 2000-12-20 NO NO20006506A patent/NO20006506L/no not_active Application Discontinuation
2001
- 2001-01-17 BG BG105163A patent/BG63744B1/bg unknown
- 2001-04-23 US US09/840,376 patent/US6458840B2/en not_active Expired - Fee Related

Also Published As

Publication number	Publication date
US20010031789A1 (en)	2001-10-18
KR20010071572A (ko)	2001-07-28
PL345364A1 (en)	2001-12-17
HUP0102456A3 (en)	2003-07-28
BG105163A (bg)	2002-03-29
HUP0102456A2 (hu)	2001-10-28
EP1089725A1 (en)	2001-04-11
TR200103249T2 (tr)	2002-05-21
WO1999066920A1 (en)	1999-12-29
AU5207199A (en)	2000-01-24
IL140415A0 (en)	2002-02-10
CZ20004833A3 (cs)	2002-01-16
TR200003800T2 (tr)	2001-06-21
BR9911421A (pt)	2001-03-27
CA2335641A1 (en)	1999-12-29
AU752192B2 (en)	2002-09-12
AU4707199A (en)	2000-01-10
CN1310622A (zh)	2001-08-29
MXPA00012808A (es)	2002-04-24
US6458840B2 (en)	2002-10-01
JP2002518442A (ja)	2002-06-25
ZA200007652B (en)	2002-03-19
NO20006506D0 (no)	2000-12-20
NO20006506L (no)	2001-02-21
US6268396B1 (en)	2001-07-31
BG63744B1 (bg)	2002-11-29

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