SK283690B6 - Deriváty erytromycínu a spôsob ich prípravy - Google Patents

Deriváty erytromycínu a spôsob ich prípravy Download PDF

Info

Publication number: SK283690B6
Authority: SK; Slovakia
Prior art keywords: group; carbon atoms; formula; methyl; compound
Prior art date: 1995-09-11

Application number

SK294-98A

Other languages

English (en)

Slovak (sk)

Other versions

SK29498A3 (en

Inventor

Alain Bonnet

Michel Delthil

Alain Mazurie

Original Assignee

Aventis Pharma S. A.

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1995-09-11

Filing date

1996-09-10

Publication date

2003-12-02

Family has litigation

First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=9482423&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=SK283690(B6) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.

1996-09-10 Application filed by Aventis Pharma S. A. filed Critical Aventis Pharma S. A.

1998-12-02 Publication of SK29498A3 publication Critical patent/SK29498A3/sk

2003-12-02 Publication of SK283690B6 publication Critical patent/SK283690B6/sk

Links

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
- C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
- C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
- Y02P20/00—Technologies relating to chemical industry
- Y02P20/50—Improvements relating to the production of bulk chemicals
- Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Engineering & Computer Science (AREA)
Health & Medical Sciences (AREA)
Biochemistry (AREA)
Biotechnology (AREA)
General Health & Medical Sciences (AREA)
Genetics & Genomics (AREA)
Molecular Biology (AREA)
Life Sciences & Earth Sciences (AREA)
Saccharide Compounds (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)

SK294-98A 1995-09-11 1996-09-10 Deriváty erytromycínu a spôsob ich prípravy SK283690B6 (sk)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
FR9510601A FR2738571B1 (fr)	1995-09-11	1995-09-11	Nouveaux derives de la 5-0-desosaminyl 6-0-methyl- erythronolide a, leur procede de preparation et leur application a la preparation de produits biologiquement actifs
PCT/FR1996/001384 WO1997010251A1 (fr)	1995-09-11	1996-09-10	Nouveaux derives de la 5-0-desosaminyl 6-0-methyl erythronolide a, leur procede de preparation et leur application a la preparation de produits biologiquement actifs

Publications (2)

Publication Number	Publication Date
SK29498A3 SK29498A3 (en)	1998-12-02
SK283690B6 true SK283690B6 (sk)	2003-12-02

Family

ID=9482423

Family Applications (3)

Application Number	Title	Priority Date	Filing Date
SK294-98A SK283690B6 (sk)	1995-09-11	1996-09-10	Deriváty erytromycínu a spôsob ich prípravy
SK892-2003A SK285995B6 (sk)	1995-09-11	1996-09-10	Deriváty erytromycínu
SK893-2003A SK285853B6 (sk)	1995-09-11	1996-09-10	Spôsob prípravy derivátov erytromycínu

Family Applications After (2)

Application Number	Title	Priority Date	Filing Date
SK892-2003A SK285995B6 (sk)	1995-09-11	1996-09-10	Deriváty erytromycínu
SK893-2003A SK285853B6 (sk)	1995-09-11	1996-09-10	Spôsob prípravy derivátov erytromycínu

Country Status (34)

Country	Link
US (1)	US5969161A (de)
EP (1)	EP0854880B1 (de)
JP (1)	JP4332218B2 (de)
KR (1)	KR100457755B1 (de)
CN (2)	CN1237069C (de)
AP (1)	AP887A (de)
AR (1)	AR004195A1 (de)
AT (1)	ATE266035T1 (de)
AU (1)	AU708811B2 (de)
BG (1)	BG63822B1 (de)
BR (1)	BR9610503A (de)
CA (1)	CA2228670C (de)
CZ (3)	CZ289945B6 (de)
DE (1)	DE69632405T2 (de)
DK (1)	DK0854880T3 (de)
EA (1)	EA000575B1 (de)
EE (1)	EE03774B1 (de)
ES (1)	ES2219698T3 (de)
FR (1)	FR2738571B1 (de)
GE (1)	GEP20022838B (de)
HK (1)	HK1041489B (de)
HU (1)	HU227565B1 (de)
IL (1)	IL123550A (de)
MX (1)	MX9801859A (de)
NO (2)	NO312678B1 (de)
PL (1)	PL183652B1 (de)
PT (1)	PT854880E (de)
RO (1)	RO120137B1 (de)
SI (1)	SI0854880T1 (de)
SK (3)	SK283690B6 (de)
TR (1)	TR199800438T1 (de)
UA (1)	UA53628C2 (de)
WO (1)	WO1997010251A1 (de)
ZA (1)	ZA966837B (de)

Families Citing this family (33)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
UA51730C2 (uk) *	1996-09-04	2002-12-16	Ебботт Лабораторіз	6-o-заміщені кетоліди з антибактеріальною активністю, спосіб їх одержання (варіанти), фармацевтична композиція та спосіб регулювання бактеріальної інфекції у ссавців
SK285534B6 (sk) *	1996-09-04	2007-03-01	Abbott Laboratories	6-O-substituované ketolidy s antibakteriálnou aktivitou, farmaceutická kompozícia s ich obsahom, ich použitie a spôsob ich prípravy
US6034069A (en) *	1997-09-30	2000-03-07	Abbott Laboratories	3-'N-modified 6-O-substituted erythromycin ketolide derivatives having antibacterial activity
US6124269A (en) *	1997-10-29	2000-09-26	Abbott Laboratories	2-Halo-6-O-substituted ketolide derivatives
US6046171A (en) *	1997-10-29	2000-04-04	Abbott Laboratories	6,11-bridged erythromycin derivatives
US6054435A (en) *	1999-03-19	2000-04-25	Abbott Laboratories	6-O-substituted macrolides having antibacterial activity
US6420535B1 (en)	1999-06-07	2002-07-16	Abbott Laboratories	6-O-carbamate ketolide derivatives
WO2003070174A2 (en) *	2002-02-15	2003-08-28	Sympore Gmbh	Conjugates of biologically active compounds, methods for their preparation and use, formulation and pharmaceutical applications thereof
EP1509538A1 (de) *	2002-05-13	2005-03-02	Enanta Pharmaceuticals, Inc.	6,11 bizyklische erythromycinderivate
US6764998B1 (en)	2003-06-18	2004-07-20	Enanta Pharmaceuticals, Inc.	6,11-4C-bicyclic 9a-azalide derivatives
US7910558B2 (en) *	2002-05-13	2011-03-22	Enanta Pharmaceuticals, Inc.	Bridged macrocyclic compounds and processes for the preparation thereof
US7135573B2 (en) *	2002-05-13	2006-11-14	Enanta Pharmaceuticals, Inc.	Processes for the preparation of O-(6-Pyrazol-1-yl-pyridin-3-ylmethyl)-hydroxylamine
US6878691B2 (en) *	2002-05-13	2005-04-12	Enanta Pharmaceuticals, Inc.	6-11 bicyclic ketolide derivatives
US7064110B2 (en) *	2002-05-13	2006-06-20	Enanta Pharmaceuticals, Inc.	6-11 bicycle ketolide derivatives
WO2005070918A1 (en) *	2002-05-13	2005-08-04	Enanta Pharmaceuticals, Inc.	Process for the preparation of t-11 bicyclic erythromycin derivatives
US7273853B2 (en) *	2002-05-13	2007-09-25	Enanta Pharmaceuticals, Inc.	6-11 bicyclic ketolide derivatives
US6753318B1 (en) *	2002-07-25	2004-06-22	Enanta Pharmaceuticals, Inc.	6,11-4-carbon bridged erythromycin derivatives
US6841664B2 (en)	2002-07-25	2005-01-11	Enanra Pharmaceuticals, Inc.	6,11-4-carbon bridged ketolides
ITMI20021726A1 (it) *	2002-08-01	2004-02-02	Zambon Spa	Macrolidi ad attivita' antiinfiammatoria.
US6645941B1 (en)	2003-03-26	2003-11-11	Enanta Pharmaceuticals, Inc.	6,11-3C-bicyclic 9a-azalide derivatives
WO2005030227A1 (en) *	2003-09-23	2005-04-07	Enanta Pharmaceuticals, Inc.	9a, 11-3C-BICYCLIC 9a-AZALIDE DERIVATIVES
WO2005067564A2 (en) *	2004-01-07	2005-07-28	Enanta Pharmaceuticals, Inc.	6-11 bicyclic erythromycin derivatives
US7265094B2 (en) *	2004-01-09	2007-09-04	Enanta Pharmaceuticals, Inc.	9N-substituted 6-11 bicyclic erythromycin derivatives
US7229972B2 (en)	2004-12-07	2007-06-12	Enanta Pharmaceuticals, Inc.	3,6-Bicyclolides
US7419962B2 (en)	2004-12-07	2008-09-02	Enanta Pharmaceuticals, Inc.	3,6-bicyclolides
WO2006065721A2 (en)	2004-12-13	2006-06-22	Enanta Pharmaceuticals, Inc.	11, 12-lactone bicyclolides
WO2006065743A2 (en)	2004-12-13	2006-06-22	Enanta Pharmaceuticals, Inc.	Tetracylic bicyclolides
US7384922B2 (en) *	2005-05-04	2008-06-10	Enanta Pharmaceuticals, Inc.	6-11 bridged oxime erythromycin derivatives
CA2615581A1 (en) *	2005-07-26	2007-02-01	Merckle Gmbh	Macrolide conjugates of pyrrolizine and indolizine compounds as inhibitors of 5-lipooxygenase and cyclooxygenase
US8273720B2 (en) *	2007-09-17	2012-09-25	Enanta Pharmaceuticals, Inc.	6,11-bicyclolides: bridged biaryl macrolide derivatives
US8354383B2 (en) *	2007-09-17	2013-01-15	Enanta Pharmaceuticals, Inc.	6,11-bridged biaryl macrolides
KR101223158B1 (ko) *	2007-09-17	2013-01-17	이난타 파마슈티칼스, 인코포레이티드	6,11-다리걸친 바이아릴 매크로라이드
CN103232501A (zh) *	2013-04-11	2013-08-07	宜昌东阳光药业股份有限公司	阿奇霉素或阿奇霉素的中间体脱去克拉定糖化合物的制备工艺

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
KR960000434B1 (ko) *	1986-12-17	1996-01-06	다이쇼 세이야꾸 가부시끼가이샤	에리스로마이신 a유도체 및 그의 제조 방법
US5523399A (en) *	1991-12-27	1996-06-04	Taisho Pharmaceutical Co., Ltd.	5-O-desosaminylerythronolide derivatives

1995
- 1995-09-11 FR FR9510601A patent/FR2738571B1/fr not_active Expired - Lifetime
1996
- 1996-08-13 ZA ZA9606837A patent/ZA966837B/xx unknown
- 1996-09-05 AR ARP960104239A patent/AR004195A1/es unknown
- 1996-09-10 BR BR9610503A patent/BR9610503A/pt not_active IP Right Cessation
- 1996-09-10 US US09/043,044 patent/US5969161A/en not_active Expired - Lifetime
- 1996-09-10 SK SK294-98A patent/SK283690B6/sk not_active IP Right Cessation
- 1996-09-10 CN CNB001309064A patent/CN1237069C/zh not_active Expired - Lifetime
- 1996-09-10 EE EE9800065A patent/EE03774B1/xx unknown
- 1996-09-10 DE DE69632405T patent/DE69632405T2/de not_active Expired - Lifetime
- 1996-09-10 HU HU9802930A patent/HU227565B1/hu unknown
- 1996-09-10 AT AT96931098T patent/ATE266035T1/de active
- 1996-09-10 SK SK892-2003A patent/SK285995B6/sk not_active IP Right Cessation
- 1996-09-10 DK DK96931098T patent/DK0854880T3/da active
- 1996-09-10 IL IL12355096A patent/IL123550A/en not_active IP Right Cessation
- 1996-09-10 PL PL96326274A patent/PL183652B1/pl unknown
- 1996-09-10 CZ CZ1998717A patent/CZ289945B6/cs not_active IP Right Cessation
- 1996-09-10 PT PT96931098T patent/PT854880E/pt unknown
- 1996-09-10 CA CA002228670A patent/CA2228670C/fr not_active Expired - Lifetime
- 1996-09-10 KR KR10-1998-0701791A patent/KR100457755B1/ko not_active Expired - Lifetime
- 1996-09-10 SK SK893-2003A patent/SK285853B6/sk not_active IP Right Cessation
- 1996-09-10 CZ CZ20012389A patent/CZ294865B6/cs not_active IP Right Cessation
- 1996-09-10 WO PCT/FR1996/001384 patent/WO1997010251A1/fr not_active Ceased
- 1996-09-10 EP EP96931098A patent/EP0854880B1/de not_active Expired - Lifetime
- 1996-09-10 AP APAP/P/1998/001210A patent/AP887A/en active
- 1996-09-10 CN CN96198171A patent/CN1070498C/zh not_active Expired - Lifetime
- 1996-09-10 RO RO98-00685A patent/RO120137B1/ro unknown
- 1996-09-10 CZ CZ20012390A patent/CZ294866B6/cs not_active IP Right Cessation
- 1996-09-10 TR TR1998/00438T patent/TR199800438T1/xx unknown
- 1996-09-10 SI SI9630684T patent/SI0854880T1/xx unknown
- 1996-09-10 ES ES96931098T patent/ES2219698T3/es not_active Expired - Lifetime
- 1996-09-10 EA EA199800288A patent/EA000575B1/ru not_active IP Right Cessation
- 1996-09-10 GE GEAP19964228A patent/GEP20022838B/en unknown
- 1996-09-10 AU AU69910/96A patent/AU708811B2/en not_active Expired
- 1996-09-10 JP JP51169697A patent/JP4332218B2/ja not_active Expired - Lifetime
- 1996-10-09 UA UA98041835A patent/UA53628C2/uk unknown
1998
- 1998-03-09 MX MX9801859A patent/MX9801859A/es unknown
- 1998-03-10 BG BG102312A patent/BG63822B1/bg unknown
- 1998-03-10 NO NO19981053A patent/NO312678B1/no not_active IP Right Cessation
2002
- 2002-03-06 NO NO20021111A patent/NO315048B1/no not_active IP Right Cessation
- 2002-04-19 HK HK02103101.8A patent/HK1041489B/zh not_active IP Right Cessation

Also Published As

Publication number	Publication date
JPH11512416A (ja)	1999-10-26
CZ71798A3 (cs)	1998-07-15
AU6991096A (en)	1997-04-01
NO20021111D0 (no)	2002-03-06
HK1041489A1 (en)	2002-07-12
SI0854880T1 (en)	2004-12-31
DE69632405D1 (de)	2004-06-09
BR9610503A (pt)	1999-07-06
HUP9802930A3 (en)	1999-12-28
CA2228670A1 (fr)	1997-03-20
FR2738571B1 (fr)	1997-10-17
AP9801210A0 (en)	1998-03-31
PT854880E (pt)	2004-09-30
HK1016187A1 (en)	1999-10-29
EA000575B1 (ru)	1999-12-29
CN1237069C (zh)	2006-01-18
EE03774B1 (et)	2002-06-17
ZA966837B (en)	1997-08-13
CZ289945B6 (cs)	2002-04-17
PL326274A1 (en)	1998-08-31
BG63822B1 (bg)	2003-02-28
EE9800065A (et)	1998-08-17
IL123550A0 (en)	1998-10-30
PL183652B1 (pl)	2002-06-28
AP887A (en)	2000-11-10
EA199800288A1 (ru)	1998-08-27
ATE266035T1 (de)	2004-05-15
UA53628C2 (uk)	2003-02-17
CN1070498C (zh)	2001-09-05
CA2228670C (fr)	2005-04-12
NO315048B1 (no)	2003-06-30
SK29498A3 (en)	1998-12-02
BG102312A (bg)	1998-09-30
KR19990044543A (ko)	1999-06-25
AU708811B2 (en)	1999-08-12
CZ294865B6 (cs)	2005-04-13
NO981053D0 (no)	1998-03-10
CN1201462A (zh)	1998-12-09
EP0854880A1 (de)	1998-07-29
RO120137B1 (ro)	2005-09-30
IL123550A (en)	2002-09-12
DK0854880T3 (da)	2004-08-16
WO1997010251A1 (fr)	1997-03-20
HUP9802930A1 (hu)	1999-04-28
ES2219698T3 (es)	2004-12-01
HU227565B1 (en)	2011-08-29
FR2738571A1 (fr)	1997-03-14
US5969161A (en)	1999-10-19
DE69632405T2 (de)	2005-05-19
NO312678B1 (no)	2002-06-17
KR100457755B1 (ko)	2005-02-28
SK285853B6 (sk)	2007-09-06
AR004195A1 (es)	1998-11-04
TR199800438T1 (xx)	1998-05-21
NO981053L (no)	1998-03-10
NO20021111L (no)	1998-03-10
CZ294866B6 (cs)	2005-04-13
GEP20022838B (en)	2002-11-25
EP0854880B1 (de)	2004-05-06
SK285995B6 (sk)	2008-01-07
JP4332218B2 (ja)	2009-09-16
CN1319602A (zh)	2001-10-31
HK1041489B (zh)	2006-09-08
MX9801859A (es)	1998-11-30

Legal Events

Date	Code	Title	Description
2016-11-02	MK4A	Patent expired	Expiry date: 20160910

Publication	Publication Date	Title
SK285995B6 (sk)	2008-01-07	Deriváty erytromycínu
Ogilvie et al.	1977	Synthesis of oligoribonucleotides
Chow et al.	1990	Stereospecific Vorbrueggen-like reactions of 1, 2-anhydro sugars. An alternative route to the synthesis of nucleosides
Hodge et al.	1991	Synthesis of 1-and 1, 2, 2'-deuteriated deoxyribose and incorporation into deoxyribonucleosides
EP0214708A2 (de)	1987-03-18	Griseolinsäurederivate, ihre Herstellung und ihre Verwendung
GB2100721A (en)	1983-01-06	Neplanocin a derivatives with antitumor activity
Knapp et al.	1984	Synthesis of protected aminocyclohexanediols
US4816575A (en)	1989-03-28	2'-(R)-substituted-2'-deoxyneplanocin A derivatives
EP0328345A2 (de)	1989-08-16	Verfahren zur Herstellung von beta-2',2'-Difluornukleosiden
Mao et al.	1984	Synthesis of 3-hydroxy-2-and-4-pyridone nucleosides as potential antitumor agents
RU2346948C2 (ru)	2009-02-20	ПРОИЗВОДНЫЕ 1-α-ГАЛОГЕН-2,2-ДИФТОР-2-ДЕЗОКСИ-D-РИБОФУРАНОЗЫ И СПОСОБ ИХ ПОЛУЧЕНИЯ
CA2022061A1 (en)	1991-01-28	Piperidine compounds
US4166849A (en)	1979-09-04	Peruvoside derivatives and processes for their preparation
EP4524145A1 (de)	2025-03-19	Verfahren zur herstellung von 4?-thio-5-aza-2?-deoxycytidin
MacCulloch et al.	1999	Stereoselective synthesis of novel 1′-substituted 2′-deoxy-4-thionucleosides
US5621086A (en)	1997-04-15	Sialic acid derivative and method of manufacturing it
SU828671A1 (ru)	1981-05-07	Способ удалени тритильных защитныхгРупп C пРОизВОдНыХ НуКлЕОзидОВ,НуКлЕОТидОВ и ОлигОНуКлЕОТидОВ
Alzerreca	2003	New approach to l'C‐modified riboside scaffold via stereoselective functionalization of D‐(+)‐ribonic‐y‐lactone
EP0535083A1 (de)	1993-04-07	Verfahren zur herstellung von 2-deoxyglucosiden
HK1016187B (en)	2002-03-01	Novel 5-o-deoaminyl 6-o-methyl erythronolide a derivatives, method for preparing the same