SMT201700314T1 - Processo per la preparazione di modulatori del recettore di istammina h3 - Google Patents
Processo per la preparazione di modulatori del recettore di istammina h3Info
- Publication number
- SMT201700314T1 SMT201700314T1 SM20170314T SMT201700314T SMT201700314T1 SM T201700314 T1 SMT201700314 T1 SM T201700314T1 SM 20170314 T SM20170314 T SM 20170314T SM T201700314 T SMT201700314 T SM T201700314T SM T201700314 T1 SMT201700314 T1 SM T201700314T1
- Authority
- SM
- San Marino
- Prior art keywords
- histamine
- preparation
- receptor modulators
- modulators
- receptor
- Prior art date
Links
- 102000004384 Histamine H3 receptors Human genes 0.000 title 1
- 108090000981 Histamine H3 receptors Proteins 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D213/78—Carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, e.g. ester or nitrile radicals
- C07D213/81—Amides; Imides
- C07D213/82—Amides; Imides in position 3
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
- C07B2200/00—Indexing scheme relating to specific properties of organic compounds
- C07B2200/13—Crystalline forms, e.g. polymorphs
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Medicines Containing Plant Substances (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US16117709P | 2009-03-18 | 2009-03-18 | |
| EP10722449.5A EP2429996B1 (en) | 2009-03-18 | 2010-03-17 | Process for the preparation of histamine h3 receptor modulators |
| PCT/US2010/027638 WO2010107897A2 (en) | 2009-03-18 | 2010-03-17 | Process for the preparation of histamine h3 receptor modulators |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| SMT201700314T1 true SMT201700314T1 (it) | 2017-07-18 |
Family
ID=42315639
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| SM20190217T SMT201900217T1 (it) | 2009-03-18 | 2010-03-17 | Processo per la preparazione di modulatori del recettore di istammina h3 |
| SM20170314T SMT201700314T1 (it) | 2009-03-18 | 2010-03-17 | Processo per la preparazione di modulatori del recettore di istammina h3 |
Family Applications Before (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| SM20190217T SMT201900217T1 (it) | 2009-03-18 | 2010-03-17 | Processo per la preparazione di modulatori del recettore di istammina h3 |
Country Status (19)
| Country | Link |
|---|---|
| US (4) | US8748596B2 (it) |
| EP (3) | EP3492451B1 (it) |
| JP (1) | JP5642149B2 (it) |
| CN (1) | CN102428070B (it) |
| AU (1) | AU2010226711B2 (it) |
| CA (2) | CA2755335C (it) |
| CY (2) | CY1119437T1 (it) |
| DK (2) | DK3216784T3 (it) |
| ES (2) | ES2625261T3 (it) |
| HR (2) | HRP20170776T1 (it) |
| HU (2) | HUE032345T2 (it) |
| LT (2) | LT2429996T (it) |
| MX (3) | MX347775B (it) |
| PL (2) | PL2429996T3 (it) |
| PT (2) | PT3216784T (it) |
| SI (2) | SI3216784T1 (it) |
| SM (2) | SMT201900217T1 (it) |
| TR (1) | TR201902858T4 (it) |
| WO (1) | WO2010107897A2 (it) |
Families Citing this family (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| PT3216784T (pt) | 2009-03-18 | 2019-04-01 | Janssen Pharmaceutica Nv | Processo para a preparação de moduladores do recetor h3 de histamina |
| KR101427221B1 (ko) * | 2012-08-29 | 2014-08-13 | 주식회사 에스텍파마 | 플루복사민 자유 염기의 정제방법 및 이를 이용한 고순도 플루복사민 말레이트의 제조방법 |
| CN104447867B (zh) * | 2013-09-17 | 2017-12-26 | 江苏天士力帝益药业有限公司 | 一种噻吩并哌啶衍生物、制备方法及其应用 |
| IL295338A (en) * | 2020-02-06 | 2022-10-01 | London Pharmaceuticals And Res Corporation | Cannabinoid sulfate esters, their salts and uses thereof |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPS5724346B2 (it) * | 1973-06-22 | 1982-05-24 | ||
| SI1558595T1 (sl) * | 2002-10-23 | 2010-03-31 | Janssen Pharmaceutica Nv | Piperazinilni in diazapanilni benzamidi in benztioamidi |
| EA015555B1 (ru) | 2006-05-30 | 2011-08-30 | Янссен Фармацевтика Н.В. | Замещенные пиридиламидные соединения в качестве модуляторов гистаминового h-рецептора |
| EA018582B1 (ru) * | 2007-11-20 | 2013-09-30 | Янссен Фармацевтика Н.В. | Соединения циклоалкилокси- и гетероциклоалкилоксипиридина как модуляторы гистаминового рецептора н |
| PT3216784T (pt) | 2009-03-18 | 2019-04-01 | Janssen Pharmaceutica Nv | Processo para a preparação de moduladores do recetor h3 de histamina |
-
2010
- 2010-03-17 PT PT17151754T patent/PT3216784T/pt unknown
- 2010-03-17 US US13/257,224 patent/US8748596B2/en active Active
- 2010-03-17 MX MX2014015305A patent/MX347775B/es unknown
- 2010-03-17 HU HUE10722449A patent/HUE032345T2/en unknown
- 2010-03-17 MX MX2016007228A patent/MX349489B/es unknown
- 2010-03-17 PL PL10722449T patent/PL2429996T3/pl unknown
- 2010-03-17 AU AU2010226711A patent/AU2010226711B2/en not_active Ceased
- 2010-03-17 MX MX2011009784A patent/MX2011009784A/es active IP Right Grant
- 2010-03-17 CA CA2755335A patent/CA2755335C/en active Active
- 2010-03-17 ES ES10722449.5T patent/ES2625261T3/es active Active
- 2010-03-17 DK DK17151754.3T patent/DK3216784T3/en active
- 2010-03-17 EP EP18194673.2A patent/EP3492451B1/en active Active
- 2010-03-17 WO PCT/US2010/027638 patent/WO2010107897A2/en not_active Ceased
- 2010-03-17 PT PT107224495T patent/PT2429996T/pt unknown
- 2010-03-17 TR TR2019/02858T patent/TR201902858T4/tr unknown
- 2010-03-17 SM SM20190217T patent/SMT201900217T1/it unknown
- 2010-03-17 LT LTEP10722449.5T patent/LT2429996T/lt unknown
- 2010-03-17 CN CN201080022339.1A patent/CN102428070B/zh active Active
- 2010-03-17 CA CA2965059A patent/CA2965059C/en active Active
- 2010-03-17 JP JP2012500921A patent/JP5642149B2/ja active Active
- 2010-03-17 LT LTEP17151754.3T patent/LT3216784T/lt unknown
- 2010-03-17 DK DK10722449.5T patent/DK2429996T3/da active
- 2010-03-17 PL PL17151754T patent/PL3216784T3/pl unknown
- 2010-03-17 HU HUE17151754 patent/HUE044837T2/hu unknown
- 2010-03-17 HR HRP20170776TT patent/HRP20170776T1/hr unknown
- 2010-03-17 ES ES17151754T patent/ES2714852T3/es active Active
- 2010-03-17 SI SI201031867T patent/SI3216784T1/sl unknown
- 2010-03-17 EP EP17151754.3A patent/EP3216784B1/en active Active
- 2010-03-17 EP EP10722449.5A patent/EP2429996B1/en active Active
- 2010-03-17 SI SI201031474T patent/SI2429996T1/sl unknown
- 2010-03-17 SM SM20170314T patent/SMT201700314T1/it unknown
-
2014
- 2014-04-25 US US14/261,713 patent/US9518021B2/en active Active
-
2016
- 2016-11-11 US US15/349,521 patent/US9809547B2/en not_active Expired - Fee Related
-
2017
- 2017-05-26 CY CY20171100547T patent/CY1119437T1/el unknown
- 2017-10-04 US US15/724,711 patent/US10323002B2/en active Active
-
2019
- 2019-03-11 HR HRP20190476TT patent/HRP20190476T1/hr unknown
- 2019-03-12 CY CY20191100292T patent/CY1121556T1/el unknown
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