SU1614763A3 - Способ получени карбапенемовых производных - Google Patents

Способ получени карбапенемовых производных Download PDF

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Publication number
SU1614763A3
SU1614763A3 SU864028623A SU4028623A SU1614763A3 SU 1614763 A3 SU1614763 A3 SU 1614763A3 SU 864028623 A SU864028623 A SU 864028623A SU 4028623 A SU4028623 A SU 4028623A SU 1614763 A3 SU1614763 A3 SU 1614763A3
Authority
SU
USSR - Soviet Union
Prior art keywords
group
general formula
carbapenem derivatives
compound
cycloaliphatic
Prior art date
Application number
SU864028623A
Other languages
English (en)
Russian (ru)
Inventor
Декстрейз Пьер
Original Assignee
Бристоль Мейерз Сквибб Компани (Фирма)
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Бристоль Мейерз Сквибб Компани (Фирма) filed Critical Бристоль Мейерз Сквибб Компани (Фирма)
Application granted granted Critical
Publication of SU1614763A3 publication Critical patent/SU1614763A3/ru

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D477/00—Heterocyclic compounds containing 1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. carbapenicillins, thienamycins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulphur-containing hetero ring
    • C07D477/10—Heterocyclic compounds containing 1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. carbapenicillins, thienamycins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulphur-containing hetero ring with hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached in position 4, and with a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2
    • C07D477/12—Heterocyclic compounds containing 1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. carbapenicillins, thienamycins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulphur-containing hetero ring with hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached in position 4, and with a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2 with hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, attached in position 6
    • C07D477/16—Heterocyclic compounds containing 1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. carbapenicillins, thienamycins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulphur-containing hetero ring with hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached in position 4, and with a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2 with hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, attached in position 6 with hetero atoms or carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 3
    • C07D477/20—Sulfur atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Oncology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Communicable Diseases (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
SU864028623A 1985-11-22 1986-11-21 Способ получени карбапенемовых производных SU1614763A3 (ru)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US06/800,867 US4880922A (en) 1985-11-22 1985-11-22 Carbapenems with quaternized heterothioalkylthio substitution at position 2

Publications (1)

Publication Number Publication Date
SU1614763A3 true SU1614763A3 (ru) 1990-12-15

Family

ID=25179586

Family Applications (1)

Application Number Title Priority Date Filing Date
SU864028623A SU1614763A3 (ru) 1985-11-22 1986-11-21 Способ получени карбапенемовых производных

Country Status (35)

Country Link
US (1) US4880922A (2)
JP (1) JPS62195382A (2)
KR (1) KR870004985A (2)
CN (1) CN86107742A (2)
AR (1) AR242209A1 (2)
AT (1) AT397090B (2)
AU (1) AU598767B2 (2)
BE (1) BE905801A (2)
CA (1) CA1273015A (2)
CH (1) CH671020A5 (2)
CS (1) CS259895B2 (2)
DD (1) DD250710A5 (2)
DE (1) DE3639762A1 (2)
DK (1) DK560886A (2)
EG (1) EG18111A (2)
ES (1) ES2002914A6 (2)
FI (1) FI83323C (2)
FR (1) FR2590574B1 (2)
GB (1) GB2183237B (2)
GR (1) GR862786B (2)
HU (1) HU197748B (2)
IL (1) IL80694A0 (2)
IT (1) IT1199669B (2)
LU (1) LU86678A1 (2)
MY (1) MY102954A (2)
NL (1) NL8602964A (2)
NO (1) NO164239C (2)
NZ (1) NZ218296A (2)
OA (1) OA08488A (2)
PT (1) PT83797B (2)
SE (1) SE469631B (2)
SU (1) SU1614763A3 (2)
YU (1) YU46030B (2)
ZA (1) ZA868829B (2)
ZW (1) ZW23486A1 (2)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NZ219892A (en) * 1986-04-15 1991-02-26 Merck & Co Inc N-amino quaternised heteroarylium carbapenem derivatives and pharmaceutical compositions thereof
US5116833A (en) * 1990-10-19 1992-05-26 Bristol-Myers Squibb Company Antibiotic c-3 dithioacetal-substituted carbapenem compounds, compositions, and methods of use thereof
KR920019791A (ko) * 1991-04-05 1992-11-20 우메모또 요시마사 다환성 카르바페넴 화합물, 그의 제조방법 및 용도
FR2920778B1 (fr) 2007-09-11 2009-10-30 Oreal Composes quinoliniums azoiques a motif disulfure/thiol, compositions les comprenant, procede de coloration de fibres keratiniques et dispositif.
FR2921382B1 (fr) 2007-09-21 2009-10-30 Oreal Colorant derive de phenyl-pyridol[1,2-a]indolium thiol-disulfure, composition tinctoriale comprenant ce colorant, procede d'eclaircissement des matieres keratiniques a partir de ce colorant
FR2921258A1 (fr) 2007-09-24 2009-03-27 Oreal Composition tinctoriale comprenant au moins un precurseur incolore disulfures/thiol, proced de coloration a partir de la composition

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4376774A (en) * 1979-05-29 1983-03-15 Merck & Co., Inc. Antibiotic N-heterocyclyl thienamycin
US4552696A (en) * 1982-04-09 1985-11-12 Bristol-Myers Company Carbapenem antibiotics
US4536335A (en) * 1982-06-18 1985-08-20 Bristol-Myers Company Carbapenem antibiotics
CA1269978A (en) * 1982-09-28 1990-06-05 Choung U. Kim Carbapenem antibiotics
AR241016A1 (es) * 1983-03-08 1991-04-30 Bristol Myeres Squibb Company "derivados de aminotiol cuaternario, procedimiento para prepararlos y procedimiento para preparar compuestos de carbapenem a partir de dichos derivados".
CA1273012A (en) * 1984-07-02 1990-08-21 Burton G. Christensen 1-methylcarbapenems having an externally alkylated mono- of bicyclic 2-quarternary heteroarylalkylthio substituent
CA1273011A (en) * 1984-07-02 1990-08-21 Susan M. Schmitt Carbapenems having an externally alkylated mono- or bicyclic 2-quaternary heteroarylalkylthio substituent
NZ219892A (en) * 1986-04-15 1991-02-26 Merck & Co Inc N-amino quaternised heteroarylium carbapenem derivatives and pharmaceutical compositions thereof

Non-Patent Citations (1)

* Cited by examiner, † Cited by third party
Title
Европейский патент № 0006639, кл. С 07 D 487/04, 1984. *

Also Published As

Publication number Publication date
AU6534386A (en) 1987-05-28
AT397090B (de) 1994-01-25
KR870004985A (ko) 1987-06-04
JPS62195382A (ja) 1987-08-28
IL80694A0 (en) 1987-02-27
AR242209A1 (es) 1993-03-31
CH671020A5 (2) 1989-07-31
FR2590574A1 (fr) 1987-05-29
OA08488A (fr) 1988-07-29
PT83797A (en) 1986-12-01
IT8622426A0 (it) 1986-11-21
CN86107742A (zh) 1987-08-12
EG18111A (en) 1992-09-30
ES2002914A6 (es) 1988-10-01
YU46030B (sh) 1992-12-21
FI864714A7 (fi) 1987-05-23
ATA313686A (de) 1993-06-15
AU598767B2 (en) 1990-07-05
BE905801A (fr) 1987-05-21
DE3639762A1 (de) 1987-06-04
ZA868829B (en) 1987-08-26
GB2183237B (en) 1989-11-08
IT8622426A1 (it) 1988-05-21
NL8602964A (nl) 1987-06-16
IT1199669B (it) 1988-12-30
CS259895B2 (en) 1988-11-15
SE8604990D0 (sv) 1986-11-21
GR862786B (en) 1987-03-24
DD250710A5 (de) 1987-10-21
US4880922A (en) 1989-11-14
NO164239C (no) 1990-09-12
NZ218296A (en) 1990-04-26
ZW23486A1 (en) 1987-04-29
CA1273015A (en) 1990-08-21
PT83797B (pt) 1989-06-30
CS843186A2 (en) 1988-03-15
FI83323B (fi) 1991-03-15
NO864669D0 (no) 1986-11-21
GB8627913D0 (en) 1986-12-31
SE8604990L (sv) 1987-05-23
DK560886A (da) 1987-05-23
NO864669L (no) 1987-05-25
YU199486A (en) 1988-02-29
HUT42486A (en) 1987-07-28
SE469631B (sv) 1993-08-09
FR2590574B1 (fr) 1989-07-28
DK560886D0 (da) 1986-11-21
MY102954A (en) 1993-03-31
NO164239B (no) 1990-06-05
LU86678A1 (fr) 1987-06-26
FI864714A0 (fi) 1986-11-19
GB2183237A (en) 1987-06-03
HU197748B (en) 1989-05-29
FI83323C (fi) 1991-06-25

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