TR200200183T2 - 2- Aminometil-4-siyanotiyazolün hazırlanması. - Google Patents

2- Aminometil-4-siyanotiyazolün hazırlanması.

Info

Publication number
TR200200183T2
TR200200183T2 TR2002/00183T TR200200183T TR200200183T2 TR 200200183 T2 TR200200183 T2 TR 200200183T2 TR 2002/00183 T TR2002/00183 T TR 2002/00183T TR 200200183 T TR200200183 T TR 200200183T TR 200200183 T2 TR200200183 T2 TR 200200183T2
Authority
TR
Turkey
Prior art keywords
alkyl
formula
cyanothiazole
aminomethyl
thioamidine
Prior art date
Application number
TR2002/00183T
Other languages
English (en)
Inventor
Pfeiffer Thomas
Original Assignee
Basf Aktiengesellshaft
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Basf Aktiengesellshaft filed Critical Basf Aktiengesellshaft
Publication of TR200200183T2 publication Critical patent/TR200200183T2/tr

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
    • C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D277/32—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D277/56—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/06—Dipeptides
    • C07K5/06008—Dipeptides with the first amino acid being neutral
    • C07K5/06078—Dipeptides with the first amino acid being neutral and aromatic or cycloaliphatic

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Biochemistry (AREA)
  • Biophysics (AREA)
  • General Health & Medical Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Medicinal Chemistry (AREA)
  • Molecular Biology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

Mevcut bulus, 2-aminometil-4-siyanotiyazolün ve bunun genel formül (Ia) ve (Ib)' ye tuzlarinin üretilmesi için bir islem ile ilgilidir, burada n, 1 veya 2' dir; n, 1 oldugunda, X, klorit, bromit, triflat ve hidrojen sülfattir ve n, 2 oldugunda, X, sülfattir. Yöntem, formül IV' e ait tiyoamidin, formül V' e ait bir bromopiruvik asit esteri ile karistirilmasini içerir, ki buradaki R1, bir R2OH alkolü içinde dalli veya lineer C1-4 alkildir, ki buradaki R2, dalli veya lineer C1-8 alkil, HO-CH2-CH2-, HO-CH2-CH2-CH2- veya C1-4-alkil-O-CH2-CH2' dir. Adi geçen karistirma islemi, -5 C ila 40 C arasinda, formül (IV)' e ait tiyoamidin resksiyonu pratikte tamamlanana kadar gerçeklestirilir. Bu bulus ayrica formül (Ia) ve (Ib)' ye ait bilesikler ile ilgilidir.
TR2002/00183T 1999-07-23 2000-07-11 2- Aminometil-4-siyanotiyazolün hazırlanması. TR200200183T2 (tr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE19933861A DE19933861A1 (de) 1999-07-23 1999-07-23 Verfahren zur Herstellung von 2-Aminomethyl-4-cyano-thiazol

Publications (1)

Publication Number Publication Date
TR200200183T2 true TR200200183T2 (tr) 2002-08-21

Family

ID=7915334

Family Applications (1)

Application Number Title Priority Date Filing Date
TR2002/00183T TR200200183T2 (tr) 1999-07-23 2000-07-11 2- Aminometil-4-siyanotiyazolün hazırlanması.

Country Status (19)

Country Link
US (1) US6642388B1 (tr)
EP (1) EP1196401A1 (tr)
JP (2) JP4027092B2 (tr)
KR (1) KR20020022781A (tr)
CN (1) CN1364163A (tr)
AU (1) AU6157900A (tr)
BG (1) BG106333A (tr)
BR (1) BR0012651A (tr)
CA (1) CA2380084C (tr)
DE (1) DE19933861A1 (tr)
HK (1) HK1048470A1 (tr)
HU (1) HUP0202109A2 (tr)
IL (1) IL147769A0 (tr)
MX (1) MXPA02000716A (tr)
NO (1) NO20020327L (tr)
PL (1) PL355110A1 (tr)
SK (1) SK1052002A3 (tr)
TR (1) TR200200183T2 (tr)
WO (1) WO2001007425A1 (tr)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE19934066A1 (de) * 1999-07-23 2001-01-25 Basf Ag Verfahren zur Herstellung von 4-Cyano-2-aminomethylthiazol
JP7148792B2 (ja) 2018-09-27 2022-10-06 日亜化学工業株式会社 光半導体装置用金属材料、及びその製造方法、及びそれを用いた光半導体装置

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE19632773A1 (de) * 1996-08-14 1998-02-19 Basf Ag Neue Thrombininhibitoren
EP0928790B1 (en) 1998-01-02 2003-03-05 F. Hoffmann-La Roche Ag Thiazole derivatives
KR20000047461A (ko) * 1998-12-29 2000-07-25 성재갑 트롬빈 억제제
DE19934066A1 (de) * 1999-07-23 2001-01-25 Basf Ag Verfahren zur Herstellung von 4-Cyano-2-aminomethylthiazol

Also Published As

Publication number Publication date
JP2003505454A (ja) 2003-02-12
WO2001007425A1 (de) 2001-02-01
BR0012651A (pt) 2002-04-09
CA2380084C (en) 2007-01-09
DE19933861A1 (de) 2001-01-25
JP4027092B2 (ja) 2007-12-26
MXPA02000716A (es) 2002-07-22
BG106333A (bg) 2002-08-30
IL147769A0 (en) 2002-08-14
NO20020327L (no) 2002-03-21
NO20020327D0 (no) 2002-01-22
EP1196401A1 (de) 2002-04-17
JP2006219498A (ja) 2006-08-24
HK1048470A1 (zh) 2003-04-04
US6642388B1 (en) 2003-11-04
CN1364163A (zh) 2002-08-14
CA2380084A1 (en) 2001-02-01
HUP0202109A2 (en) 2002-09-28
KR20020022781A (ko) 2002-03-27
PL355110A1 (en) 2004-04-05
SK1052002A3 (en) 2002-07-02
AU6157900A (en) 2001-02-13

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