UA117253C2 - ПОХІДНІ ТІЄНО[3,2-d]ПІРИМІДИНІВ ДЛЯ ЛІКУВАННЯ ВІРУСНИХ ІНФЕКЦІЙ - Google Patents

ПОХІДНІ ТІЄНО[3,2-d]ПІРИМІДИНІВ ДЛЯ ЛІКУВАННЯ ВІРУСНИХ ІНФЕКЦІЙ

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Publication number
UA117253C2
UA117253C2 UAA201601818A UAA201601818A UA117253C2 UA 117253 C2 UA117253 C2 UA 117253C2 UA A201601818 A UAA201601818 A UA A201601818A UA A201601818 A UAA201601818 A UA A201601818A UA 117253 C2 UA117253 C2 UA 117253C2
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UA
Ukraine
Prior art keywords
thieno
viral infections
treatment
pyrimidines derivatives
pyrimidines
Prior art date
Application number
UAA201601818A
Other languages
English (en)
Inventor
Гоуен Девід Крейг Мак
П'єр Жан-Марі Бернар Рабуассон
Original Assignee
ЯНССЕН САЙЄНСЕЗ АЙРЛЕНД ЮСі
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
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Application filed by ЯНССЕН САЙЄНСЕЗ АЙРЛЕНД ЮСі filed Critical ЯНССЕН САЙЄНСЕЗ АЙРЛЕНД ЮСі
Publication of UA117253C2 publication Critical patent/UA117253C2/uk

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D495/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/02—Immunomodulators
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/02—Immunomodulators
    • A61P37/04—Immunostimulants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Immunology (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Communicable Diseases (AREA)
  • Virology (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Oncology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)

Abstract

Даний винахід належить до похідних тієно[3,2-d]піримідинів, способів їх отримання, фармацевтичних композицій та їх застосування в лікуванні вірусних інфекцій.
UAA201601818A 2013-07-30 2014-07-29 ПОХІДНІ ТІЄНО[3,2-d]ПІРИМІДИНІВ ДЛЯ ЛІКУВАННЯ ВІРУСНИХ ІНФЕКЦІЙ UA117253C2 (uk)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP13178534 2013-07-30
PCT/EP2014/066219 WO2015014815A1 (en) 2013-07-30 2014-07-29 THIENO[3,2-d]PYRIMIDINES DERIVATIVES FOR THE TREATMENT OF VIRAL INFECTIONS

Publications (1)

Publication Number Publication Date
UA117253C2 true UA117253C2 (uk) 2018-07-10

Family

ID=48874951

Family Applications (1)

Application Number Title Priority Date Filing Date
UAA201601818A UA117253C2 (uk) 2013-07-30 2014-07-29 ПОХІДНІ ТІЄНО[3,2-d]ПІРИМІДИНІВ ДЛЯ ЛІКУВАННЯ ВІРУСНИХ ІНФЕКЦІЙ

Country Status (20)

Country Link
US (3) US9556199B2 (uk)
EP (2) EP3027624B1 (uk)
JP (1) JP6401788B2 (uk)
KR (1) KR102322425B1 (uk)
CN (2) CN105492446B (uk)
AU (2) AU2014298540B2 (uk)
BR (1) BR112016001570B1 (uk)
CA (1) CA2913691C (uk)
CL (1) CL2015003767A1 (uk)
DK (2) DK3027624T3 (uk)
EA (1) EA036162B1 (uk)
ES (2) ES2836881T3 (uk)
IL (2) IL242872B (uk)
MX (1) MX368625B (uk)
MY (1) MY179503A (uk)
PH (1) PH12015502797B1 (uk)
SG (2) SG11201510736PA (uk)
UA (1) UA117253C2 (uk)
WO (1) WO2015014815A1 (uk)
ZA (1) ZA201600655B (uk)

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