UA53788C2 - Рідкі полімерні композиції для регульованого виділення біоактивних речовин - Google Patents

Рідкі полімерні композиції для регульованого виділення біоактивних речовин Download PDF

Info

Publication number: UA53788C2
Authority: UA; Ukraine
Prior art keywords: lactide; glycolide; copolymer; bioactive substance; hydrophilic
Prior art date: 1998-03-19

Application number

UA2000105893A

Other languages

English (en)

Russian (ru)

Ukrainian (uk)

Inventor

Рей Т. Черн

Джоел Р. Зінгерман

Original Assignee

Мерк Енд Ко., Інк.

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1998-03-19

Filing date

1999-03-18

Publication date

2003-02-17

1999-03-18 Application filed by Мерк Енд Ко., Інк. filed Critical Мерк Енд Ко., Інк.

1999-03-18 Priority claimed from PCT/US1999/005938 external-priority patent/WO1999047073A1/en

2003-02-17 Publication of UA53788C2 publication Critical patent/UA53788C2/uk

Links

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URAYPUMNDPQOKB-UHFFFAOYSA-N triacetin Chemical compound CC(=O)OCC(OC(C)=O)COC(C)=O URAYPUMNDPQOKB-UHFFFAOYSA-N 0.000 claims description 26
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JJTUDXZGHPGLLC-UHFFFAOYSA-N lactide Chemical compound CC1OC(=O)C(C)OC1=O JJTUDXZGHPGLLC-UHFFFAOYSA-N 0.000 claims description 23
238000000034 method Methods 0.000 claims description 15
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Classifications

- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
- A61K47/08—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
- A61K47/14—Esters of carboxylic acids, e.g. fatty acid monoglycerides, medium-chain triglycerides, parabens or PEG fatty acid esters
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/30—Macromolecular organic or inorganic compounds, e.g. inorganic polyphosphates
- A61K47/34—Macromolecular compounds obtained otherwise than by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyesters, polyamino acids, polysiloxanes, polyphosphazines, copolymers of polyalkylene glycol or poloxamers
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0019—Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0019—Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
- A61K9/0024—Solid, semi-solid or solidifying implants, which are implanted or injected in body tissue

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
Veterinary Medicine (AREA)
Pharmacology & Pharmacy (AREA)
Epidemiology (AREA)
Medicinal Chemistry (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
Dermatology (AREA)
Engineering & Computer Science (AREA)
Inorganic Chemistry (AREA)
Proteomics, Peptides & Aminoacids (AREA)
Biomedical Technology (AREA)
Neurosurgery (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Oil, Petroleum & Natural Gas (AREA)
Medicinal Preparation (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Agricultural Chemicals And Associated Chemicals (AREA)
Compositions Of Macromolecular Compounds (AREA)

UA2000105893A 1998-03-19 1999-03-18 Рідкі полімерні композиції для регульованого виділення біоактивних речовин UA53788C2 (uk)

Applications Claiming Priority (3)

Application Number	Priority Date	Filing Date	Title
US7957498P	1998-03-19	1998-03-19
GBGB9815801.7A GB9815801D0 (en)	1998-07-21	1998-07-21	Liquid polymeric compositions for controlled released bioactive substances
PCT/US1999/005938 WO1999047073A1 (en)	1998-03-19	1999-03-18	Liquid polymeric compositions for controlled release of bioactive substances

Publications (1)

Publication Number	Publication Date
UA53788C2 true UA53788C2 (uk)	2003-02-17

Family

ID=10835852

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
UA2000105893A UA53788C2 (uk)	1998-03-19	1999-03-18	Рідкі полімерні композиції для регульованого виділення біоактивних речовин

Country Status (10)

Country	Link
JP (1)	JP4829405B2 (sr)
AT (1)	ATE499069T1 (sr)
DE (1)	DE69943225D1 (sr)
DK (1)	DK1484033T3 (sr)
GB (1)	GB9815801D0 (sr)
GE (1)	GEP20033012B (sr)
PT (1)	PT1484033E (sr)
RS (1)	RS49840B (sr)
SI (1)	SI1484033T1 (sr)
UA (1)	UA53788C2 (sr)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US8362086B2 (en) *	2005-08-19	2013-01-29	Merial Limited	Long acting injectable formulations
EP2825154A4 (en) *	2012-03-13	2015-11-11	Bayer New Zealand Ltd	LONG ACTIVE COMPOSITIONS
KR20210153745A (ko) *	2013-09-16	2021-12-17	머크 샤프 앤드 돔 코포레이션	Cgrp 수용체 길항제를 위한 제제
KR102101969B1 (ko) *	2017-09-06	2020-04-22	(주)인벤티지랩	목시덱틴을 포함하는 마이크로 입자 및 이의 제조 방법

1998
- 1998-07-21 GB GBGB9815801.7A patent/GB9815801D0/en not_active Ceased
1999
- 1999-03-18 PT PT04076699T patent/PT1484033E/pt unknown
- 1999-03-18 UA UA2000105893A patent/UA53788C2/uk unknown
- 1999-03-18 DE DE69943225T patent/DE69943225D1/de not_active Expired - Lifetime
- 1999-03-18 AT AT04076699T patent/ATE499069T1/de active
- 1999-03-18 GE GEAP19995598A patent/GEP20033012B/en unknown
- 1999-03-18 SI SI9931052T patent/SI1484033T1/sl unknown
- 1999-03-18 JP JP2000536316A patent/JP4829405B2/ja not_active Expired - Lifetime
- 1999-03-18 RS YUP-541/00A patent/RS49840B/sr unknown
- 1999-03-18 DK DK04076699.0T patent/DK1484033T3/da active

Also Published As

Publication number	Publication date
DE69943225D1 (de)	2011-04-07
SI1484033T1 (sl)	2011-06-30
JP4829405B2 (ja)	2011-12-07
PT1484033E (pt)	2011-04-21
JP2002506797A (ja)	2002-03-05
YU54100A (sh)	2002-11-15
ATE499069T1 (de)	2011-03-15
DK1484033T3 (da)	2011-06-14
GEP20033012B (en)	2003-07-25
GB9815801D0 (en)	1998-09-16
RS49840B (sr)	2008-08-07

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MXPA00009143A (en)	2001-07-09	Liquid polymeric compositions for controlled release of bioactive substances
HK1031990B (en)	2005-02-25	Liquid polymeric compositions for controlled release of bioactive substances
HK1036579B (en)	2007-02-09	Liquid polymeric compositions for controlled release of bioactive substances
AU2002366248A1 (en)	2003-06-30	Radioopaque sustained release pharmaceutical system
MXPA00005552A (en)	2001-07-03	Long acting injectable formulations containing hydrogenated castor oil