UA72039C2 - A method for the preparation of citalopram - Google Patents

A method for the preparation of citalopram Download PDF

Info

Publication number
UA72039C2
UA72039C2 UA2002118821A UA2002118821A UA72039C2 UA 72039 C2 UA72039 C2 UA 72039C2 UA 2002118821 A UA2002118821 A UA 2002118821A UA 2002118821 A UA2002118821 A UA 2002118821A UA 72039 C2 UA72039 C2 UA 72039C2
Authority
UA
Ukraine
Prior art keywords
formula
compound
differs
intermediate compound
interaction
Prior art date
Application number
UA2002118821A
Other languages
English (en)
Ukrainian (uk)
Original Assignee
Lundbeck & Co As H
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Lundbeck & Co As H filed Critical Lundbeck & Co As H
Publication of UA72039C2 publication Critical patent/UA72039C2/uk

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
    • C07D307/77—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom ortho- or peri-condensed with carbocyclic rings or ring systems
    • C07D307/87—Benzo [c] furans; Hydrogenated benzo [c] furans
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/24—Antidepressants
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
    • C07D307/77—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom ortho- or peri-condensed with carbocyclic rings or ring systems
    • C07D307/87—Benzo [c] furans; Hydrogenated benzo [c] furans
    • C07D307/88—Benzo [c] furans; Hydrogenated benzo [c] furans with one oxygen atom directly attached in position 1 or 3

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pain & Pain Management (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Psychiatry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Steroid Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Furan Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
UA2002118821A 2000-05-12 2001-10-05 A method for the preparation of citalopram UA72039C2 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DKPA200000783 2000-05-12
PCT/DK2001/000333 WO2001085712A1 (en) 2000-05-12 2001-05-10 Method for the preparation of citalopram

Publications (1)

Publication Number Publication Date
UA72039C2 true UA72039C2 (en) 2005-01-17

Family

ID=8159493

Family Applications (1)

Application Number Title Priority Date Filing Date
UA2002118821A UA72039C2 (en) 2000-05-12 2001-10-05 A method for the preparation of citalopram

Country Status (29)

Country Link
US (1) US6660873B2 (de)
EP (1) EP1296970B1 (de)
JP (1) JP2003532721A (de)
CN (1) CN100422166C (de)
AR (1) AR032455A1 (de)
AT (1) ATE389645T1 (de)
AU (2) AU5823901A (de)
BG (1) BG65820B1 (de)
BR (1) BR0110996A (de)
CA (1) CA2408292C (de)
CZ (1) CZ20024065A3 (de)
DE (1) DE60133280T2 (de)
DK (1) DK1296970T3 (de)
EA (1) EA005674B1 (de)
ES (1) ES2301541T3 (de)
HR (1) HRP20020881A2 (de)
HU (1) HUP0301942A2 (de)
IL (2) IL152645A0 (de)
IS (1) IS2586B (de)
MX (1) MXPA02011125A (de)
NO (1) NO327963B1 (de)
NZ (1) NZ522475A (de)
PL (1) PL358144A1 (de)
PT (1) PT1296970E (de)
SI (1) SI1296970T1 (de)
SK (1) SK287035B6 (de)
UA (1) UA72039C2 (de)
WO (1) WO2001085712A1 (de)
ZA (1) ZA200208973B (de)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TR200102957T2 (tr) 1999-04-14 2004-12-21 H. Lundbeck A/S Sitalopram hazırlanması için metod.
US6310222B1 (en) 1999-11-01 2001-10-30 Sumika Fine Chemicals Co., Ltd. Production method of 5-phthalancarbonitrile compound, intermediate therefor and production method of the intermediate
US6433196B1 (en) 2000-02-17 2002-08-13 Sumika Fine Chemicals Co., Ltd. Production method of citalopram, intermediate therefor and production method of the intermediate
NL1017417C1 (nl) 2000-03-03 2001-03-16 Lundbeck & Co As H Werkwijze voor de bereiding van Citalopram.
NL1017500C1 (nl) 2000-03-13 2001-04-26 Lundbeck & Co As H Werkwijze voor de bereiding van Citalopram.
BR0109364A (pt) * 2000-03-13 2002-12-24 Lundbeck & Co As H Métodos para fabricação de citalopram através de alquilação escalonada de 5-substituìda 1- (4-fluorofenil) - 1,3- diidroisobenzofuranos e citalopram
AR032455A1 (es) 2000-05-12 2003-11-12 Lundbeck & Co As H Metodo para la preparacion de citalopram, un intermediario empleado en el metodo, un metodo para la preparacion del intermediario empleado en el metodo y composicion farmaceutica antidepresiva
IN192057B (de) * 2001-07-19 2004-02-14 Ranbaxy Lab Ltd
WO2004085416A1 (en) * 2003-03-24 2004-10-07 Hetero Drugs Limited Novel crystalline forms of (s)-citalopram oxalate
CA2546422A1 (en) * 2003-10-28 2005-05-12 Wockhardt Limited Improved process for the manufacture of citalopram hydrobromide
US20050143350A1 (en) * 2003-11-19 2005-06-30 Seed John C. Combination drug therapy to treat obesity
WO2006021971A2 (en) 2004-08-23 2006-03-02 Sun Pharmaceutical Industries Limited 'process for preparation of citalopram and enantiomers'

Family Cites Families (40)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1143703A (de) 1965-03-18
GB1526331A (en) * 1976-01-14 1978-09-27 Kefalas As Phthalanes
GB8419963D0 (en) 1984-08-06 1984-09-12 Lundbeck & Co As H Intermediate compound and method
GB8814057D0 (en) 1988-06-14 1988-07-20 Lundbeck & Co As H New enantiomers & their isolation
US5296507A (en) 1990-09-06 1994-03-22 H.Lundbeck A/S Treatment of cerbrovascular disorders
DE19626659A1 (de) 1996-07-03 1998-01-08 Basf Ag Verfahren zur Herstellung von Phthaliden
DE19627697A1 (de) 1996-07-10 1998-01-15 Basf Ag Verfahren zur Herstellung von Phthaliden
CN1206207C (zh) 1997-07-08 2005-06-15 H.隆德贝克有限公司 氰酞氟苯胺的制备方法
UA62985C2 (en) 1997-11-10 2004-01-15 Lunnbeck As H A method for the preparation of citalopram
HUP0002953A3 (en) * 1997-11-11 2002-12-28 Lundbeck & Co As H Method for preparation of citalopram and intermediates used for them
DE69904853T2 (de) 1998-10-20 2003-09-04 Lundbeck As Valby H Verfahren zur herstellung von citalopram
SI1140886T1 (en) 1998-12-23 2003-08-31 H. Lundbeck A/S Method for the preparation of 5-cyanophthalide
AR022329A1 (es) 1999-01-29 2002-09-04 Lundbeck & Co As H Metodo para la preparacion de 5-cianoftalida
TR200102957T2 (tr) 1999-04-14 2004-12-21 H. Lundbeck A/S Sitalopram hazırlanması için metod.
ITMI991579A1 (it) 1999-06-25 2001-01-15 Lundbeck & Co As H Metodo per la preparazione di citalopram
ITMI991581A1 (it) 1999-06-25 2001-01-15 Lundbeck & Co As H Metodo per la preparazione di citalopram
ITMI991486A1 (it) 1999-07-06 2001-01-06 Vis Farmaceutici S P A Processo per la sintesi di citalopram
EP1228056B1 (de) 1999-10-25 2004-09-22 H. Lundbeck A/S Verfahren zur herstellung von citalopram
AR026063A1 (es) 1999-11-01 2002-12-26 Lundbeck & Co As H Metodo para la preparacion de 5-carboxiftalida.
US6310222B1 (en) 1999-11-01 2001-10-30 Sumika Fine Chemicals Co., Ltd. Production method of 5-phthalancarbonitrile compound, intermediate therefor and production method of the intermediate
EP1246812B1 (de) 1999-12-28 2004-03-17 H. Lundbeck A/S Verfahren zur herstellung von citalopram
SI1246813T1 (en) 1999-12-30 2004-08-31 H. Lundbeck A/S Method for the preparation of citalopram
PL197821B1 (pl) 2000-01-14 2008-04-30 Lundbeck & Co As H Sposób wytwarzania 5-cyjanoftalidu
IT1317729B1 (it) 2000-01-18 2003-07-15 Norpharma S P A Procedimento per la preparazione della 5-carbossiftalide.
US6433196B1 (en) 2000-02-17 2002-08-13 Sumika Fine Chemicals Co., Ltd. Production method of citalopram, intermediate therefor and production method of the intermediate
FR2805812A1 (fr) 2000-02-24 2001-09-07 Lundbeck & Co As H Procede de preparation du citalopram
IES20010143A2 (en) 2000-02-24 2001-07-25 Lundbeck & Co As H Method for the preparation of citalopram
NL1017417C1 (nl) 2000-03-03 2001-03-16 Lundbeck & Co As H Werkwijze voor de bereiding van Citalopram.
GB0005477D0 (en) 2000-03-07 2000-04-26 Resolution Chemicals Limited Process for the preparation of citalopram
BR0109364A (pt) 2000-03-13 2002-12-24 Lundbeck & Co As H Métodos para fabricação de citalopram através de alquilação escalonada de 5-substituìda 1- (4-fluorofenil) - 1,3- diidroisobenzofuranos e citalopram
PL360110A1 (en) 2000-03-13 2004-09-06 H.Lundbeck A/S Method for the preparation of citalopram
NL1017500C1 (nl) 2000-03-13 2001-04-26 Lundbeck & Co As H Werkwijze voor de bereiding van Citalopram.
GB2357762B (en) 2000-03-13 2002-01-30 Lundbeck & Co As H Crystalline base of citalopram
JP2003527386A (ja) 2000-03-14 2003-09-16 ハー・ルンドベック・アクチエゼルスカベット シタロプラムの製造方法
CH692148A5 (de) 2000-03-16 2002-02-28 Lundbeck & Co As H Verfahren zur Herstellung von Citalopram.
AR032455A1 (es) 2000-05-12 2003-11-12 Lundbeck & Co As H Metodo para la preparacion de citalopram, un intermediario empleado en el metodo, un metodo para la preparacion del intermediario empleado en el metodo y composicion farmaceutica antidepresiva
IL148525A0 (en) 2000-07-06 2002-09-12 Lundbeck & Co As H Method for the preparation of citalopram
CA2354877C (en) 2000-08-18 2006-05-02 H. Lundbeck A/S Method for the preparation of citalopram
EA003581B1 (ru) 2000-12-22 2003-06-26 Х.Лундбекк А/С Способ получения чистого циталопрама
AU2001100399B4 (en) 2000-12-28 2002-03-21 H Lundbeck As Process for the preparation of pure citalopram

Also Published As

Publication number Publication date
JP2003532721A (ja) 2003-11-05
ES2301541T3 (es) 2008-07-01
PL358144A1 (en) 2004-08-09
ATE389645T1 (de) 2008-04-15
AR032455A1 (es) 2003-11-12
ZA200208973B (en) 2003-11-05
DE60133280D1 (de) 2008-04-30
CN100422166C (zh) 2008-10-01
NO20025423L (no) 2002-11-12
PT1296970E (pt) 2008-06-11
CZ20024065A3 (cs) 2003-03-12
HRP20020881A2 (en) 2004-12-31
AU5823901A (en) 2001-11-20
IL152645A0 (en) 2003-06-24
HUP0301942A2 (hu) 2003-09-29
SI1296970T1 (sl) 2008-08-31
CA2408292C (en) 2009-11-10
IS2586B (is) 2010-02-15
EP1296970A1 (de) 2003-04-02
SK287035B6 (sk) 2009-10-07
DK1296970T3 (da) 2008-07-14
US20030134895A1 (en) 2003-07-17
DE60133280T2 (de) 2009-04-16
SK17542002A3 (sk) 2003-04-01
CN1441795A (zh) 2003-09-10
BR0110996A (pt) 2003-03-18
IS6605A (is) 2002-10-31
EA200201211A1 (ru) 2003-04-24
IL152645A (en) 2009-12-24
WO2001085712A1 (en) 2001-11-15
EA005674B1 (ru) 2005-04-28
AU2001258239B2 (en) 2005-12-08
NO20025423D0 (no) 2002-11-12
CA2408292A1 (en) 2001-11-15
NZ522475A (en) 2004-09-24
NO327963B1 (no) 2009-10-26
EP1296970B1 (de) 2008-03-19
BG107349A (bg) 2003-09-30
BG65820B1 (bg) 2010-01-29
MXPA02011125A (es) 2003-03-10
HK1056171A1 (zh) 2004-02-06
US6660873B2 (en) 2003-12-09

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