WO2012000608A3 - Beta -aminoaldehyd- derivate, verfahren zu ihrer herstellung und ihre chemische verwendung als reaktive intermediate - Google Patents

Beta -aminoaldehyd- derivate, verfahren zu ihrer herstellung und ihre chemische verwendung als reaktive intermediate Download PDF

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WO2012000608A3
WO2012000608A3 PCT/EP2011/002923 EP2011002923W WO2012000608A3 WO 2012000608 A3 WO2012000608 A3 WO 2012000608A3 EP 2011002923 W EP2011002923 W EP 2011002923W WO 2012000608 A3 WO2012000608 A3 WO 2012000608A3
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preparation
novel beta
reactive intermediates
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aminoaldehyde derivatives
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WO2012000608A2 (de
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Karl-Heinz GLÜSENKAMP
Christian Mengede
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Abstract

Die vorliegende Erfindung beschreibt neue beta-Aminoaldehyd-Derivate der Formeln (I), (II) und (III),in welchen die Substituenten R1 bis R5 und A die in der Beschreibung angegebene Bedeutung haben, ein neues Verfahren zur deren Herstellung, dessen Zwischenprodukte, sowie Verwendungen dieser neuen beta-Aminoaldehyd-Derivate, z.B. zur (chemischen) Verwendung als reaktive Intermediate, zur Verwendung in der Medizin, z.B. als Peptidomimetikum, als Kopplungsagens, etc.
PCT/EP2011/002923 2010-06-30 2011-06-14 Neue beta-aminoaldehyd-derivate, verfahren zu ihrer herstellung und ihre chemische verwendung als reaktive intermediate Ceased WO2012000608A2 (de)

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DE102010025663A DE102010025663A1 (de) 2010-06-30 2010-06-30 Neue beta-Aminoaldehyd-Derivate, Verfahren zu ihrer Herstellung und ihre chemische Verwendung als reaktive Intermediate
DE102010025663.3 2010-06-30

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WO2012000608A2 WO2012000608A2 (de) 2012-01-05
WO2012000608A3 true WO2012000608A3 (de) 2012-03-08

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