ZA200200057B - Compounds for the modulation of PPARγ activity. - Google Patents

Compounds for the modulation of PPARγ activity. Download PDF

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Publication number
ZA200200057B
ZA200200057B ZA200200057A ZA200200057A ZA200200057B ZA 200200057 B ZA200200057 B ZA 200200057B ZA 200200057 A ZA200200057 A ZA 200200057A ZA 200200057 A ZA200200057 A ZA 200200057A ZA 200200057 B ZA200200057 B ZA 200200057B
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South Africa
Prior art keywords
alkyl
group
compound
halogen
aryl
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ZA200200057A
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English (en)
Inventor
Lawrence R Mcgee
Jonathan B Houze
Steven M Rubenstein
Atsushi Hagiwara
Noboru Furukawa
Hisashi Shinkai
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Tularik Inc
Japan Tobacco Inc
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Application filed by Tularik Inc, Japan Tobacco Inc filed Critical Tularik Inc
Publication of ZA200200057B publication Critical patent/ZA200200057B/en

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    • C07D213/02Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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ZA200200057A 1999-06-30 2002-01-03 Compounds for the modulation of PPARγ activity. ZA200200057B (en)

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ZA200200057A ZA200200057B (en) 1999-06-30 2002-01-03 Compounds for the modulation of PPARγ activity.

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EP (1) EP1192137B1 (fr)
JP (1) JP4295458B2 (fr)
CN (1) CN1171872C (fr)
CA (1) CA2377309C (fr)
DK (1) DK1192137T3 (fr)
EA (1) EA004887B1 (fr)
ES (1) ES2437103T3 (fr)
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IL (2) IL147308A0 (fr)
MX (2) MXPA01013199A (fr)
NZ (2) NZ516455A (fr)
SG (1) SG148834A1 (fr)
WO (1) WO2001000579A1 (fr)
ZA (1) ZA200200057B (fr)

Families Citing this family (68)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6583157B2 (en) 1998-01-29 2003-06-24 Tularik Inc. Quinolinyl and benzothiazolyl modulators
US7041691B1 (en) 1999-06-30 2006-05-09 Amgen Inc. Compounds for the modulation of PPARγ activity
AU6118001A (en) 2000-05-03 2001-11-12 Tularik Inc Combination therapeutic compositions and methods of use
US20030171399A1 (en) 2000-06-28 2003-09-11 Tularik Inc. Quinolinyl and benzothiazolyl modulators
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