ZA988923B - Polymeric derivatives of camptothecin - Google Patents

Polymeric derivatives of camptothecin

Info

Publication number
ZA988923B
ZA988923B ZA988923A ZA988923A ZA988923B ZA 988923 B ZA988923 B ZA 988923B ZA 988923 A ZA988923 A ZA 988923A ZA 988923 A ZA988923 A ZA 988923A ZA 988923 B ZA988923 B ZA 988923B
Authority
ZA
South Africa
Prior art keywords
camptothecin
polymeric derivatives
polymeric
derivatives
Prior art date
Application number
ZA988923A
Other languages
English (en)
Inventor
Francesco Angelucci
Fabrizio Orzi
Gabriele Fachin
Valeria Rosaria Caiolfa
Moreno Zamai
Antonio Suarato
Original Assignee
Pharmacia & Upjohn Spa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pharmacia & Upjohn Spa filed Critical Pharmacia & Upjohn Spa
Publication of ZA988923B publication Critical patent/ZA988923B/xx

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/50—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/50—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates
    • A61K47/51—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent
    • A61K47/56—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent the modifying agent being an organic macromolecular compound, e.g. an oligomeric, polymeric or dendrimeric molecule
    • A61K47/58—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent the modifying agent being an organic macromolecular compound, e.g. an oligomeric, polymeric or dendrimeric molecule obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. poly[meth]acrylate, polyacrylamide, polystyrene, polyvinylpyrrolidone, polyvinylalcohol or polystyrene sulfonic acid resin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents

Landscapes

  • Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Addition Polymer Or Copolymer, Post-Treatments, Or Chemical Modifications (AREA)
ZA988923A 1997-10-03 1998-09-30 Polymeric derivatives of camptothecin ZA988923B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GBGB9721069.4A GB9721069D0 (en) 1997-10-03 1997-10-03 Polymeric derivatives of camptothecin

Publications (1)

Publication Number Publication Date
ZA988923B true ZA988923B (en) 1999-04-12

Family

ID=10820048

Family Applications (1)

Application Number Title Priority Date Filing Date
ZA988923A ZA988923B (en) 1997-10-03 1998-09-30 Polymeric derivatives of camptothecin

Country Status (27)

Country Link
US (1) US6328953B1 (pt)
EP (1) EP1019090B1 (pt)
JP (1) JP2001518521A (pt)
KR (1) KR100559068B1 (pt)
CN (1) CN1154512C (pt)
AR (1) AR013535A1 (pt)
AT (1) ATE259662T1 (pt)
AU (1) AU749321B2 (pt)
BG (1) BG64894B1 (pt)
BR (1) BR9815236A (pt)
CA (1) CA2303097A1 (pt)
DE (1) DE69821783T2 (pt)
DK (1) DK1019090T3 (pt)
EA (1) EA002030B1 (pt)
ES (1) ES2216317T3 (pt)
GB (1) GB9721069D0 (pt)
HU (1) HUP0003690A3 (pt)
IL (1) IL134871A (pt)
MY (1) MY116287A (pt)
NO (1) NO20001628D0 (pt)
NZ (1) NZ503879A (pt)
PL (1) PL191609B1 (pt)
PT (1) PT1019090E (pt)
TW (1) TW564178B (pt)
UA (1) UA70930C2 (pt)
WO (1) WO1999017804A1 (pt)
ZA (1) ZA988923B (pt)

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Also Published As

Publication number Publication date
HUP0003690A2 (hu) 2001-09-28
PT1019090E (pt) 2004-05-31
IL134871A (en) 2005-11-20
EP1019090B1 (en) 2004-02-18
BG104355A (en) 2001-01-31
EA002030B1 (ru) 2001-12-24
US6328953B1 (en) 2001-12-11
WO1999017804A1 (en) 1999-04-15
NZ503879A (en) 2002-03-28
MY116287A (en) 2003-12-31
IL134871A0 (en) 2001-05-20
CN1272796A (zh) 2000-11-08
UA70930C2 (uk) 2004-11-15
CA2303097A1 (en) 1999-04-15
HUP0003690A3 (en) 2003-08-28
DE69821783T2 (de) 2004-12-30
DK1019090T3 (da) 2004-04-26
KR100559068B1 (ko) 2006-03-10
BR9815236A (pt) 2002-07-23
JP2001518521A (ja) 2001-10-16
CN1154512C (zh) 2004-06-23
PL339574A1 (en) 2000-12-18
AR013535A1 (es) 2000-12-27
HK1032005A1 (en) 2001-07-06
DE69821783D1 (de) 2004-03-25
NO20001628L (no) 2000-03-29
PL191609B1 (pl) 2006-06-30
ES2216317T3 (es) 2004-10-16
GB9721069D0 (en) 1997-12-03
AU9627398A (en) 1999-04-27
AU749321B2 (en) 2002-06-20
KR20010015687A (ko) 2001-02-26
EP1019090A1 (en) 2000-07-19
NO20001628D0 (no) 2000-03-29
TW564178B (en) 2003-12-01
BG64894B1 (bg) 2006-08-31
EA200000376A1 (ru) 2000-10-30
ATE259662T1 (de) 2004-03-15

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