ATE100798T1 - Pyridinyl-derivate von 2-aminoacetamid. - Google Patents

Pyridinyl-derivate von 2-aminoacetamid.

Info

Publication number: ATE100798T1
Authority: AT; Austria
Prior art keywords: pyridinyl; aminoacetamide; pyridinyl derivatives; phenyl; independently selected
Prior art date: 1987-02-06

Application number

AT87118509T

Other languages

English (en)

Inventor

Ronald C Griffith

James J Napier

Original Assignee

Fisons Corp

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1987-02-06

Filing date

1987-12-14

Publication date

1994-02-15

1987-12-14 Application filed by Fisons Corp filed Critical Fisons Corp

1994-02-15 Application granted granted Critical

1994-02-15 Publication of ATE100798T1 publication Critical patent/ATE100798T1/de

Links

-1 PYRIDINYL DERIVATIVES OF 2-AMINOACETAMIDE Chemical class 0.000 title abstract 3
125000001997 phenyl group Chemical group [H]C1=C([H])C([H])=C(*)C([H])=C1[H] 0.000 abstract 2
125000004214 1-pyrrolidinyl group Chemical group [H]C1([H])N(*)C([H])([H])C([H])([H])C1([H])[H] 0.000 abstract 1
KPCZJLGGXRGYIE-UHFFFAOYSA-N [C]1=CC=CN=C1 Chemical group [C]1=CC=CN=C1 KPCZJLGGXRGYIE-UHFFFAOYSA-N 0.000 abstract 1
150000001875 compounds Chemical class 0.000 abstract 1
125000006317 cyclopropyl amino group Chemical group 0.000 abstract 1
125000004663 dialkyl amino group Chemical group 0.000 abstract 1
229910052739 hydrogen Inorganic materials 0.000 abstract 1
239000001257 hydrogen Substances 0.000 abstract 1
125000004435 hydrogen atom Chemical group [H]* 0.000 abstract 1
125000002496 methyl group Chemical group [H]C([H])([H])* 0.000 abstract 1
125000004573 morpholin-4-yl group Chemical group N1(CCOCC1)* 0.000 abstract 1
125000000587 piperidin-1-yl group Chemical group [H]C1([H])N(*)C([H])([H])C([H])([H])C([H])([H])C1([H])[H] 0.000 abstract 1
125000002924 primary amino group Chemical group [H]N([H])* 0.000 abstract 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/24—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with substituted hydrocarbon radicals attached to ring carbon atoms
- C07D213/36—Radicals substituted by singly-bound nitrogen atoms
- C07D213/40—Acylated substituent nitrogen atom
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/08—Antiepileptics; Anticonvulsants
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/20—Hypnotics; Sedatives

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Medicinal Chemistry (AREA)
General Health & Medical Sciences (AREA)
Neurology (AREA)
Neurosurgery (AREA)
Bioinformatics & Cheminformatics (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Engineering & Computer Science (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Veterinary Medicine (AREA)
Pharmacology & Pharmacy (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
Biomedical Technology (AREA)
Public Health (AREA)
Pain & Pain Management (AREA)
Anesthesiology (AREA)
Pyridine Compounds (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

AT87118509T 1987-02-06 1987-12-14 Pyridinyl-derivate von 2-aminoacetamid. ATE100798T1 (de)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
US07/011,983 US4769466A (en)	1987-02-06	1987-02-06	2-aminoacetamide pyridinyl derivatives
EP87118509A EP0278090B1 (de)	1987-02-06	1987-12-14	Pyridinyl-Derivate von 2-Aminoacetamid

Publications (1)

Publication Number	Publication Date
ATE100798T1 true ATE100798T1 (de)	1994-02-15

Family

ID=21752815

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
AT87118509T ATE100798T1 (de)	1987-02-06	1987-12-14	Pyridinyl-derivate von 2-aminoacetamid.

Country Status (8)

Country	Link
US (1)	US4769466A (de)
EP (1)	EP0278090B1 (de)
JP (1)	JPH0825998B2 (de)
AT (1)	ATE100798T1 (de)
CA (1)	CA1299571C (de)
DE (1)	DE3788955T2 (de)
IE (1)	IE61880B1 (de)
PT (1)	PT86251B (de)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US5430044A (en) *	1987-02-06	1995-07-04	Fisons Corporation	Arylalkyl-amines and -amides having anticonvulsant and neuroprotective properties
EP0356035B1 (de) *	1988-08-12	1996-03-13	Astra Aktiebolag	Arylalkylamine und -amide mit krampflösender und nervenschützender Wirkung
EP0540318A1 (de) *	1991-10-30	1993-05-05	Fisons Corporation	2-Heterozyklische Ethylaminderivate und ihre Verwendung als Arzneimittel
US5541213A (en) *	1993-06-24	1996-07-30	Eisai Co., Ltd.	Propenoic acid derivatives diazole propenoic acid compounds which have useful pharmaceutical utility
DK3066091T3 (da) *	2013-11-05	2019-07-15	Astrazeneca Ab	Nmda-antagonist-prodrugs
WO2018098344A1 (en) *	2016-11-28	2018-05-31	Biohaven Pharmaceutical Holding Company Ltd.	Prodrugs of lanicemine and their method of use

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
DE955508C (de) *	1954-07-28	1957-01-03	Cilag Ag	Verfahren zur Herstellung von antikonvulsivisch wirkenden Carbonsaeureamiden
CH343388A (de) *	1956-03-09	1959-12-31	Cilag Chemie Aktiengesellschaf	Verfahren zur Herstellung neuer Amide
US4500714A (en) *	1981-10-15	1985-02-19	Chugai Seiyaku Kabushiki Kaisha	3-Substituted-ureido-N-pyridyl benzamides

1987
- 1987-02-06 US US07/011,983 patent/US4769466A/en not_active Expired - Fee Related
- 1987-10-30 IE IE293187A patent/IE61880B1/en not_active IP Right Cessation
- 1987-11-10 CA CA000551551A patent/CA1299571C/en not_active Expired - Lifetime
- 1987-11-30 PT PT86251A patent/PT86251B/pt not_active IP Right Cessation
- 1987-12-14 AT AT87118509T patent/ATE100798T1/de not_active IP Right Cessation
- 1987-12-14 DE DE87118509T patent/DE3788955T2/de not_active Expired - Fee Related
- 1987-12-14 EP EP87118509A patent/EP0278090B1/de not_active Expired - Lifetime
1988
- 1988-02-04 JP JP63022958A patent/JPH0825998B2/ja not_active Expired - Lifetime

Also Published As

Publication number	Publication date
PT86251A (en)	1987-12-01
DE3788955D1 (de)	1994-03-10
PT86251B (pt)	1991-02-08
JPS63201169A (ja)	1988-08-19
EP0278090A3 (en)	1990-04-11
JPH0825998B2 (ja)	1996-03-13
US4769466A (en)	1988-09-06
DE3788955T2 (de)	1994-05-11
EP0278090B1 (de)	1994-01-26
IE61880B1 (en)	1994-11-30
CA1299571C (en)	1992-04-28
IE872931L (en)	1988-08-06
EP0278090A2 (de)	1988-08-17

Legal Events

Date	Code	Title	Description
1994-07-15	RER	Ceased as to paragraph 5 lit. 3 law introducing patent treaties

Publication	Publication Date	Title
DK0646115T3 (da)	2003-04-22	Heterocykliske/cykliske aminderivater
AU4929690A (en)	1990-08-16	Phenyl pyradazine-3(2H)one, thiadizin-2(3H)one, triazin-3(2H) one and oxadiazin-5(4H)one derivatives for the treatment of congestive heart failure
DE3468878D1 (en)	1988-02-25	7-amino-azoloû1,5-a¨pyrimidines and fungicides containing them
PL315747A1 (en)	1996-11-25	Fungicidal cyclic amides
DK0564409T3 (da)	2000-06-19	Pyrimidinderivater og fremgangsmåde til fremstilling deraf
DE69106388D1 (de)	1995-02-09	Antipsychotische 4-(1,2-benzisoazolyl)piperidinderivate.
DE3788955D1 (de)	1994-03-10	Pyridinyl-Derivate von 2-Aminoacetamid.
MY106474A (en)	1995-05-30	Guanidine derivatives.
DK0852580T3 (da)	2000-11-20	Fremgangsmåde til fremstilling af dihydroxypyrimidin-derivater
DK0579968T3 (da)	2000-03-27	4-Iminoquinoliner, fremgangsmåde til deres fremstilling og deres anvendelse
ES8802499A1 (es)	1988-07-01	Procedimiento para la obtencion de 1-aril-4-nitropirazoles
GB1530415A (en)	1978-11-01	Pyridinylpyrimidine derivatives
NO941084L (no)	1994-03-24	Neuroleptiske 2-substituerte perhydro-1-H-pyrido[1,2-aÅpyraziner
IL87042A (en)	1992-03-29	Process for the preparation of amino pyridylalkyl ketones,intermediates therefor and their preparation
DK436181A (da)	1982-04-03	Substituerede 6-halogen-tert. butyl1,2,4-triazin-5-oner deres fremstilling og anvendelse
NO914942L (no)	1992-06-15	Kjemiske mellomprodukter
DE3779190D1 (de)	1992-06-25	T-butyl ergolinderivate.
NO954764L (no)	1996-01-25	Psoralen-derivater, deres fremstilling og anvendelse
IE870556L (en)	1987-09-05	4-(2-pyrimidinyl)-1-piperazinyl heterocyclic carbonyl¹derivatives