ATE116545T1 - Pyridopyrazinderivate zur behandlung von drogenmissbrauch und -sucht. - Google Patents

Pyridopyrazinderivate zur behandlung von drogenmissbrauch und -sucht.

Info

Publication number
ATE116545T1
ATE116545T1 AT91910566T AT91910566T ATE116545T1 AT E116545 T1 ATE116545 T1 AT E116545T1 AT 91910566 T AT91910566 T AT 91910566T AT 91910566 T AT91910566 T AT 91910566T AT E116545 T1 ATE116545 T1 AT E116545T1
Authority
AT
Austria
Prior art keywords
addiction
treatment
drug abuse
pyridopyrazine derivatives
derivatives
Prior art date
Application number
AT91910566T
Other languages
English (en)
Inventor
Gene Michael Bright
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Application granted granted Critical
Publication of ATE116545T1 publication Critical patent/ATE116545T1/de

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Addiction (AREA)
  • Psychiatry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
AT91910566T 1990-06-29 1991-05-28 Pyridopyrazinderivate zur behandlung von drogenmissbrauch und -sucht. ATE116545T1 (de)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
PCT/US1990/003708 WO1992000075A1 (en) 1990-06-29 1990-06-29 Pyridopyrazine derivatives for treating substance abuse and addiction

Publications (1)

Publication Number Publication Date
ATE116545T1 true ATE116545T1 (de) 1995-01-15

Family

ID=22220931

Family Applications (1)

Application Number Title Priority Date Filing Date
AT91910566T ATE116545T1 (de) 1990-06-29 1991-05-28 Pyridopyrazinderivate zur behandlung von drogenmissbrauch und -sucht.

Country Status (17)

Country Link
US (1) US5616585A (de)
EP (1) EP0536173B1 (de)
JP (1) JPH05507274A (de)
KR (1) KR930701171A (de)
AT (1) ATE116545T1 (de)
AU (1) AU651977B2 (de)
CA (1) CA2086335C (de)
DE (1) DE69106516T2 (de)
DK (1) DK0536173T3 (de)
ES (1) ES2066447T3 (de)
HU (1) HUT62797A (de)
IE (1) IE64467B1 (de)
IL (1) IL98588A (de)
MY (1) MY106553A (de)
NZ (1) NZ238750A (de)
WO (2) WO1992000075A1 (de)
ZA (1) ZA915012B (de)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6231833B1 (en) 1999-08-05 2001-05-15 Pfizer Inc 2,7-substituted octahydro-1H-pyrido[1,2-A]pyrazine derivatives as ligands for serotonin receptors
HN1999000146A (es) * 1998-09-21 2000-11-11 Pfizer Prod Inc Agentes farmaceuticos para el tratamiento de la enfermedad de parkinson, adhd y microadenomas.
EP1177792A3 (de) * 2000-07-27 2002-10-23 Pfizer Products Inc. Dopamin-d4-ligande zur behandlung von gaudi-suchenden krankheiten
UA110688C2 (uk) 2012-09-21 2016-01-25 Пфайзер Інк. Біциклічні піридинони
MX368391B (es) 2015-02-03 2019-09-30 Pfizer Ciclopropabenzofuranil-piridopirazindionas novedosas.

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DK144213C (da) * 1979-06-20 1982-06-21 H B Nielsen Hylster til garnspole
US4777173A (en) * 1987-03-25 1988-10-11 Bristol-Myers Company Method for treatment of alcohol abuse
DE3727879A1 (de) * 1987-08-21 1989-03-02 Troponwerke Gmbh & Co Kg Verwendung von 2-pyrimidinyl-1-piperazin-derivaten
DE3736974A1 (de) * 1987-10-31 1989-05-11 Troponwerke Gmbh & Co Kg Verwendung von 2-pyrimidinyl-1-piperazin-derivaten
IL91451A0 (en) * 1988-08-30 1990-04-29 Bristol Myers Co Pharmaceutical compositions comprising azapiron compounds and their use in the treatment of addiction
WO1990008148A1 (en) * 1989-01-23 1990-07-26 Pfizer Inc. Bis-aza-bicyclic anxiolytic agents

Also Published As

Publication number Publication date
WO1992000074A3 (en) 1992-03-05
AU651977B2 (en) 1994-08-11
IE912259A1 (en) 1992-01-01
CA2086335A1 (en) 1991-12-30
KR930701171A (ko) 1993-06-11
EP0536173B1 (de) 1995-01-04
JPH05507274A (ja) 1993-10-21
NZ238750A (en) 1999-09-29
IE64467B1 (en) 1995-08-09
DE69106516D1 (de) 1995-02-16
IL98588A0 (en) 1992-07-15
CA2086335C (en) 1996-01-02
ZA915012B (en) 1993-02-24
MY106553A (en) 1995-06-30
US5616585A (en) 1997-04-01
IL98588A (en) 1995-06-29
DE69106516T2 (de) 1995-05-11
HUT62797A (en) 1993-06-28
DK0536173T3 (da) 1995-05-01
WO1992000075A1 (en) 1992-01-09
EP0536173A1 (de) 1993-04-14
WO1992000074A2 (en) 1992-01-09
AU7909491A (en) 1992-01-23
HU9204138D0 (en) 1993-04-28
ES2066447T3 (es) 1995-03-01

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Legal Events

Date Code Title Description
UEP Publication of translation of european patent specification
REN Ceased due to non-payment of the annual fee