TR200103237T2 - İmidazodiazepin türevi - Google Patents

İmidazodiazepin türevi

Info

Publication number
TR200103237T2
TR200103237T2 TR2001/03237T TR200103237T TR200103237T2 TR 200103237 T2 TR200103237 T2 TR 200103237T2 TR 2001/03237 T TR2001/03237 T TR 2001/03237T TR 200103237 T TR200103237 T TR 200103237T TR 200103237 T2 TR200103237 T2 TR 200103237T2
Authority
TR
Turkey
Prior art keywords
imidazodiazepine
derivative
drugs
imidazodiazepine derivative
axiolytic
Prior art date
Application number
TR2001/03237T
Other languages
English (en)
Inventor
Jenck Fran�Ois
Hoffmann-Emery Fabienne
Hunkeler Walker
Richard Martin James
Sleight Andrew
Original Assignee
F. Hoffmann-La Roche Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by F. Hoffmann-La Roche Ag filed Critical F. Hoffmann-La Roche Ag
Publication of TR200103237T2 publication Critical patent/TR200103237T2/tr

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/06—Peri-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/08—Antiepileptics; Anticonvulsants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/20—Hypnotics; Sedatives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/22—Anxiolytics

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Biomedical Technology (AREA)
  • Public Health (AREA)
  • Pain & Pain Management (AREA)
  • Anesthesiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)

Abstract

Mevcut bulus, 7-klor-3-(5-dimetilaminometil- [1,2,4]oksadiazol-3-il)-5-metil-4, 5-dihidro-imidazo[1,5-a] [1,4]benzodiazepin-6-on-(I) bilesimiyle ve formül (I) bilesiminin aksiolitik ve/veya antikonvulsan ve/veya sedatif olmayan uyku indükleyici ilaçlar olarak kullanilacak olan ilaçlarin yapiminda kullanilmasiyla ilgilidir.
TR2001/03237T 1999-05-12 2000-05-05 İmidazodiazepin türevi TR200103237T2 (tr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP99109513 1999-05-12

Publications (1)

Publication Number Publication Date
TR200103237T2 true TR200103237T2 (tr) 2002-04-22

Family

ID=8238165

Family Applications (1)

Application Number Title Priority Date Filing Date
TR2001/03237T TR200103237T2 (tr) 1999-05-12 2000-05-05 İmidazodiazepin türevi

Country Status (17)

Country Link
US (1) US6391873B1 (tr)
EP (1) EP1178990B1 (tr)
JP (1) JP3706307B2 (tr)
KR (1) KR100451610B1 (tr)
CN (1) CN1164590C (tr)
AR (1) AR023884A1 (tr)
AT (1) ATE231865T1 (tr)
AU (1) AU769666B2 (tr)
BR (1) BR0010495A (tr)
CA (1) CA2372040C (tr)
DE (1) DE60001313T2 (tr)
DK (1) DK1178990T3 (tr)
ES (1) ES2189759T3 (tr)
MX (1) MXPA01011449A (tr)
TR (1) TR200103237T2 (tr)
WO (1) WO2000069858A1 (tr)
ZA (1) ZA200108913B (tr)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP5180077B2 (ja) 2006-08-11 2013-04-10 パナソニック株式会社 複数ドライブ装置の遅延対策と省電力制御を行う記録再生装置
US20090054412A1 (en) * 2007-08-20 2009-02-26 John Alan Kemp Treatment of Sleep Disorders
WO2009024324A2 (en) * 2007-08-20 2009-02-26 Evotec Neurosciences Gmbh Treatment of sleep disorders
WO2009024325A2 (en) * 2007-08-20 2009-02-26 Evotec Neurosciences Gmbh Treatment of sleep disorders
JP5345637B2 (ja) * 2008-01-22 2013-11-20 イーライ リリー アンド カンパニー κ選択的オピオイド受容体アンタゴニスト
CN107007559B (zh) * 2017-04-21 2020-05-15 浙江京新药业股份有限公司 一种稳定的口服药物组合物及其制备方法
CN109134471B (zh) * 2017-06-27 2020-05-15 浙江京新药业股份有限公司 一种苯并二氮杂*化合物的固态形式及其制备方法和应用
CN112778220B (zh) * 2019-11-02 2024-06-07 浙江京新药业股份有限公司 一种苯并二氮杂䓬二酮化合物d的制备方法及其中间体
CN113045574B (zh) * 2019-12-26 2024-06-07 浙江京新药业股份有限公司 二氮杂䓬衍生物的制备方法及其中间体
US12161622B2 (en) 2021-05-04 2024-12-10 Janssen Pharmaceuticals, Inc. Compositions and methods for the treatment of depression
WO2023170554A1 (en) 2022-03-07 2023-09-14 Janssen Pharmaceuticals, Inc. Compositions comprising aticaprant
WO2023170550A1 (en) 2022-03-07 2023-09-14 Janssen Pharmaceuticals, Inc. Polymorph forms of aticaprant for use in treating major depressive disorder

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2143246C (en) * 1994-03-16 2000-08-22 Thierry Godel Imidazodiazepines
PT801651E (pt) * 1995-01-06 2001-12-28 Hoffmann La Roche Hidroximetil-imidazodiazepinas e seus esteres

Also Published As

Publication number Publication date
DE60001313T2 (de) 2004-01-22
EP1178990A1 (en) 2002-02-13
CA2372040A1 (en) 2000-11-23
ATE231865T1 (de) 2003-02-15
BR0010495A (pt) 2002-02-13
AU769666B2 (en) 2004-01-29
CN1350538A (zh) 2002-05-22
CN1164590C (zh) 2004-09-01
JP3706307B2 (ja) 2005-10-12
KR20010112487A (ko) 2001-12-20
EP1178990B1 (en) 2003-01-29
KR100451610B1 (ko) 2004-10-06
WO2000069858A1 (en) 2000-11-23
AU5211400A (en) 2000-12-05
ES2189759T3 (es) 2003-07-16
ZA200108913B (en) 2003-03-26
DE60001313D1 (en) 2003-03-06
JP2002544277A (ja) 2002-12-24
DK1178990T3 (da) 2003-05-26
MXPA01011449A (es) 2002-06-04
US6391873B1 (en) 2002-05-21
AR023884A1 (es) 2002-09-04
CA2372040C (en) 2008-12-02

Similar Documents

Publication Publication Date Title
BG103251A (bg) Оксадиазоли, методи за получаването им и приложението им като лекарствени средства
TR200000197T2 (tr) Yeni bileşimler
NO20014728L (no) Derivater av pyrimido[6,1-a]isokinolin-4-on
ATE320436T1 (de) Dimere pyrrolobenzodiazepine
TR200000151T2 (tr) Yeni bileşimler.
WO1992007830A3 (en) Oxindole peptide antagonists
TR199800012T1 (tr) Piroloprimidinler ve preparasyon için tatbikler.
ATE218581T1 (de) Cyclosporinderivat, dessen herstellung und pharmazeutische zusammensetzung
DK0970095T3 (da) Hidtil ukendte benzimidazolinhibitorer for fructose-1,6-bisphosphase
DE69622031D1 (de) INDOLDERIVATE ALS cGMP-PDE INHIBITOREN
TR199902538T2 (tr) Yeni bilesimler.
EP1445317A3 (en) Compositions and methods for the diagnosis and treatment of tumor
MX9702307A (es) Pirrolo (2,3-d)pirimidinas y su uso.
ATE521353T1 (de) Neues trisubstitutiertes 8h-pyridoä2,3- düpyrimidin-7-onderivat zur behandlung von durch csbp/p38kinase vermittelten krankheiten
PL338339A1 (en) Novel derivatives of tetrazole
TR200103237T2 (tr) İmidazodiazepin türevi
SE9904129D0 (sv) Novel compounds
DE69924292D1 (de) Pyrazol verbindungen und ihre verwendung
WO2000040583A3 (de) Imidazo[4,5-c]-pyridin-4-on-derivate
ID29790A (id) PENGGUNAAN IMIDAZO(1,5-a)-PIRIDO(3,2-e)-PIRAZINON SEBAGAI OBAT
TR200000907T2 (tr) Nötrofil elastaz inhibitörleri olarak pirolopirolon türevleri.
MXPA03003923A (es) Compuestos de n-([1,2,4]triazoloazinil)tiofensulfonamida como herbicidas.
EE200200337A (et) Uued ühendid ning nende kasutamine
DE60008400D1 (de) Triazolopyrimidinderivate
TR200001102T2 (tr) İkameli tetrahidropirimidinen türevleri, üretimleri ve kullanımları.