ATE124039T1 - Durch azetidine substituierte derivate von pyridon-carboxylsäure, ihre herstellung und verwendung als arzneimittel. - Google Patents

Durch azetidine substituierte derivate von pyridon-carboxylsäure, ihre herstellung und verwendung als arzneimittel.

Info

Publication number
ATE124039T1
ATE124039T1 AT90400684T AT90400684T ATE124039T1 AT E124039 T1 ATE124039 T1 AT E124039T1 AT 90400684 T AT90400684 T AT 90400684T AT 90400684 T AT90400684 T AT 90400684T AT E124039 T1 ATE124039 T1 AT E124039T1
Authority
AT
Austria
Prior art keywords
derivatives
azetidines
pyridone
production
carboxylic acid
Prior art date
Application number
AT90400684T
Other languages
English (en)
Inventor
Corominas Juan Pares
Pinol Augusto Colombo
Constansa Jordi Frigola
Original Assignee
Esteve Labor Dr
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from FR8903459A external-priority patent/FR2644455B1/fr
Priority claimed from FR8908695A external-priority patent/FR2649106A2/fr
Priority claimed from FR8915178A external-priority patent/FR2654728B2/fr
Application filed by Esteve Labor Dr filed Critical Esteve Labor Dr
Application granted granted Critical
Publication of ATE124039T1 publication Critical patent/ATE124039T1/de

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Oncology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Communicable Diseases (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pyridine Compounds (AREA)
AT90400684T 1989-03-16 1990-03-14 Durch azetidine substituierte derivate von pyridon-carboxylsäure, ihre herstellung und verwendung als arzneimittel. ATE124039T1 (de)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
FR8903459A FR2644455B1 (fr) 1989-03-16 1989-03-16 Derives d'acides pyridone carboxyliques azetidinyl substitues, leur preparation et leur application en tant que medicaments
FR8908695A FR2649106A2 (fr) 1989-06-29 1989-06-29 Derives d'acides pyridone carboxyliques azetidinyl substitues, leur preparation et leur application en tant que medicament
FR8915178A FR2654728B2 (fr) 1989-03-16 1989-11-20 Derives d'acides pyridone carboxyliques azetidinyl substitues, leur preparation et leur application en tant que medicament.

Publications (1)

Publication Number Publication Date
ATE124039T1 true ATE124039T1 (de) 1995-07-15

Family

ID=27251837

Family Applications (1)

Application Number Title Priority Date Filing Date
AT90400684T ATE124039T1 (de) 1989-03-16 1990-03-14 Durch azetidine substituierte derivate von pyridon-carboxylsäure, ihre herstellung und verwendung als arzneimittel.

Country Status (16)

Country Link
US (1) US5393758A (de)
EP (1) EP0388298B1 (de)
JP (1) JPH075586B2 (de)
KR (1) KR940006595B1 (de)
AT (1) ATE124039T1 (de)
AU (2) AU638437B2 (de)
CA (1) CA2012223A1 (de)
DE (1) DE69020199T2 (de)
DK (1) DK0388298T3 (de)
ES (1) ES2022006A6 (de)
GR (1) GR3017304T3 (de)
HU (1) HU206702B (de)
NO (1) NO177302C (de)
PT (1) PT93450B (de)
RU (1) RU2044735C1 (de)
YU (1) YU47430B (de)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ATE194612T1 (de) * 1990-12-05 2000-07-15 Naeja Pharmaceutical Inc 7-substituierte-6-fluor-1,4-dihydro-4-oxo- chinolin-3-carbonsäurederivate als antibakterielle wirkstoffe
US5342846A (en) * 1990-12-05 1994-08-30 Synphar Laboratories, Inc. 7-substituted-6-fluoro-1,4-dihydro-4-oxo-quinoline-3-carboxylic acid compounds and 7-(substituted triazolyl pyrrolidin-1-yl) 4-oxoquinoline-3-carboxylic acid derivatives useful as antibacterial agents
FR2676445B1 (fr) * 1991-05-16 1995-02-03 Esteve Labor Dr Derives de pyridone amino acide azetidinyl substitues, leur preparation et leur application en tant que medicaments.
FR2681865B1 (fr) * 1991-10-01 1993-11-19 Bel Laboratoire Roger Nouveaux derives de la benzonaphtyridine-1,8 leur preparation et les compositions qui les contiennent.
US5221676A (en) * 1992-02-06 1993-06-22 Warner-Lambert Company 7-substituted quinolones and naphthyridones as antibacterial agents
FR2690161B1 (fr) * 1992-04-16 1995-06-30 Esteve Labor Dr Derives de pyridone azetidinyl substitues avec activite antimicrobienne.
JPH0999195A (ja) * 1995-10-02 1997-04-15 Eiji Maruko 高能率電子洗濯法
MY119816A (en) * 1997-05-30 2005-07-29 Daiichi Seiyaku Co Substituted cyclobutylamine derivatives
MXPA02000103A (es) * 1999-07-01 2003-07-21 Wakunaga Pharma Co Ltd Derivado de acido quinolin carboxilico o sales del mismo.
RU2298006C2 (ru) * 2000-11-20 2007-04-27 Дайити Фармасьютикал Ко., Лтд. Дегалогенированные соединения, антибактериальное средство и терапевтическое средство на их основе, способ получения антибактериального или лекарственного средства, применение дегалогенированных соединений для получения антибактериального или лекарственного средства
WO2005026146A1 (en) * 2003-09-12 2005-03-24 Warner-Lambert Company Llc Azetidinyl quinolones as antibacterial agents

Family Cites Families (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3998808A (en) * 1968-05-22 1976-12-21 Velsicol Chemical Corporation Compositions of matter D-hetero-1,1-(α-thiocyanoacetyl) compounds
US4183923A (en) * 1977-11-07 1980-01-15 Schering Corporation Antipsoriatic compositions
JPS5746986A (en) * 1980-09-02 1982-03-17 Dai Ichi Seiyaku Co Ltd Pyrido(1,2,3-de)(1,4)benzoxazine derivative
IE55898B1 (en) * 1982-09-09 1991-02-14 Warner Lambert Co Antibacterial agents
US4777175A (en) * 1982-09-09 1988-10-11 Warner-Lambert Company Antibacterial agents
US4665079A (en) * 1984-02-17 1987-05-12 Warner-Lambert Company Antibacterial agents
JPS6089480A (ja) * 1983-10-21 1985-05-20 Dainippon Pharmaceut Co Ltd ピリドンカルボン酸誘導体
JPS60126284A (ja) * 1983-12-09 1985-07-05 Dainippon Pharmaceut Co Ltd ピリドンカルボン酸誘導体およびその塩
FR2560194B1 (fr) * 1984-02-27 1987-08-07 Midy Spa 3-aminoazetidine, ses sels, procede pour leur preparation et intermediaires de synthese
JPS61137885A (ja) * 1984-12-08 1986-06-25 Dainippon Pharmaceut Co Ltd １，８−ナフチリジン誘導体、そのエステルおよびその塩
JPS61143383A (ja) * 1985-10-28 1986-07-01 Toyama Chem Co Ltd １，４−ジヒドロ−４−オキソナフチリジン誘導体またはその塩を含有する抗菌剤
EP0241206A3 (de) * 1986-03-31 1989-05-10 Sankyo Company Limited Chinolin-3-carbonsäurederivate, ihre Herstellung und Verwendung
JPS63198664A (ja) * 1986-03-31 1988-08-17 Sankyo Co Ltd キノロンカルボン酸誘導体
JPH0633262B2 (ja) * 1987-10-12 1994-05-02 富山化学工業株式会社 １，４−ジヒドロ−４−オキソナフチリジン誘導体およびその塩
HU205105B (en) * 1987-10-26 1992-03-30 Pfizer Process for producing azetidinyl quinoline carboxylic acids and pharmaceutical compositions comprising same
FR2634483B2 (fr) * 1987-12-29 1994-03-04 Esteve Labor Dr Derives des acides 7-(1-azetidinyl)-1,4-dihydro-4-oxoquinoleine-3-carboxyliques, leur preparation et leur application en tant que medicaments

Also Published As

Publication number Publication date
JPH02279683A (ja) 1990-11-15
HU206702B (en) 1992-12-28
NO901171L (no) 1990-09-17
AU4746993A (en) 1993-12-02
HUT53643A (en) 1990-11-28
HU901570D0 (en) 1990-06-28
AU648212B2 (en) 1994-04-14
AU638437B2 (en) 1993-07-01
AU5137590A (en) 1990-09-20
EP0388298A3 (de) 1991-07-31
DE69020199T2 (de) 1995-12-14
EP0388298A2 (de) 1990-09-19
DK0388298T3 (da) 1995-08-14
US5393758A (en) 1995-02-28
KR940006595B1 (ko) 1994-07-23
KR900014380A (ko) 1990-10-23
GR3017304T3 (en) 1995-12-31
PT93450A (pt) 1990-11-07
NO177302B (no) 1995-05-15
JPH075586B2 (ja) 1995-01-25
RU2044735C1 (ru) 1995-09-27
PT93450B (pt) 1996-07-31
DE69020199D1 (de) 1995-07-27
ES2022006A6 (es) 1991-11-16
NO901171D0 (no) 1990-03-13
YU50590A (sh) 1993-05-28
NO177302C (no) 1995-08-23
CA2012223A1 (en) 1990-09-16
EP0388298B1 (de) 1995-06-21
YU47430B (sh) 1995-03-27

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Legal Events

Date Code Title Description
UEP Publication of translation of european patent specification
REN Ceased due to non-payment of the annual fee