ATE150963T1 - Kugelförmige granula mit kern sowie deren herstellung - Google Patents

Kugelförmige granula mit kern sowie deren herstellung

Info

Publication number
ATE150963T1
ATE150963T1 AT91202685T AT91202685T ATE150963T1 AT E150963 T1 ATE150963 T1 AT E150963T1 AT 91202685 T AT91202685 T AT 91202685T AT 91202685 T AT91202685 T AT 91202685T AT E150963 T1 ATE150963 T1 AT E150963T1
Authority
AT
Austria
Prior art keywords
core
sphere
production
shaped granules
granules
Prior art date
Application number
AT91202685T
Other languages
English (en)
Inventor
Tadashi Makino
Tetsuro Tabata
Shin-Ichiro Hirai
Original Assignee
Takeda Chemical Industries Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=11992094&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=ATE150963(T1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Takeda Chemical Industries Ltd filed Critical Takeda Chemical Industries Ltd
Application granted granted Critical
Publication of ATE150963T1 publication Critical patent/ATE150963T1/de

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/50—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
    • A61K9/5073—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals having two or more different coatings optionally including drug-containing subcoatings
    • A61K9/5078—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals having two or more different coatings optionally including drug-containing subcoatings with drug-free core
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • A61K9/167—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction with an outer layer or coating comprising drug; with chemically bound drugs or non-active substances on their surface
    • A61K9/1676—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction with an outer layer or coating comprising drug; with chemically bound drugs or non-active substances on their surface having a drug-free core with discrete complete coating layer containing drug

Landscapes

  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Manufacturing Of Micro-Capsules (AREA)
  • Cereal-Derived Products (AREA)
AT91202685T 1987-01-29 1988-01-25 Kugelförmige granula mit kern sowie deren herstellung ATE150963T1 (de)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP1917887 1987-01-29

Publications (1)

Publication Number Publication Date
ATE150963T1 true ATE150963T1 (de) 1997-04-15

Family

ID=11992094

Family Applications (1)

Application Number Title Priority Date Filing Date
AT91202685T ATE150963T1 (de) 1987-01-29 1988-01-25 Kugelförmige granula mit kern sowie deren herstellung

Country Status (9)

Country Link
US (2) US5026560A (de)
EP (2) EP0475536B1 (de)
KR (1) KR960005138B1 (de)
AT (1) ATE150963T1 (de)
CA (1) CA1312548C (de)
DE (2) DE3874360T2 (de)
ES (2) ES2052697T3 (de)
GR (1) GR3006170T3 (de)
HU (1) HU198396B (de)

Families Citing this family (242)

* Cited by examiner, † Cited by third party
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KR960005138B1 (ko) 1996-04-22
CA1312548C (en) 1993-01-12
US5516531A (en) 1996-05-14
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DE3874360T2 (de) 1993-01-14
US5026560A (en) 1991-06-25
KR880008803A (ko) 1988-09-13
HU198396B (en) 1989-10-30
GR3006170T3 (de) 1993-06-21
DE3874360D1 (de) 1992-10-15
ES2052697T3 (es) 1994-07-16
HUT46238A (en) 1988-10-28
ES2099130T3 (es) 1997-05-16
DE3855852D1 (de) 1997-05-07
EP0277741A1 (de) 1988-08-10
DE3855852T2 (de) 1997-07-17
EP0475536A1 (de) 1992-03-18

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