ATE157647T1 - Verfahren zur herstellung von alpha- ketoamidderivaten - Google Patents

Verfahren zur herstellung von alpha- ketoamidderivaten

Info

Publication number
ATE157647T1
ATE157647T1 AT92311175T AT92311175T ATE157647T1 AT E157647 T1 ATE157647 T1 AT E157647T1 AT 92311175 T AT92311175 T AT 92311175T AT 92311175 T AT92311175 T AT 92311175T AT E157647 T1 ATE157647 T1 AT E157647T1
Authority
AT
Austria
Prior art keywords
producing
alphaketoamide
derivatives
ketoacetamide
alpha
Prior art date
Application number
AT92311175T
Other languages
English (en)
Inventor
Akira Murabayashi
Hideyuki Takenaka
Hiroyuki Kai
Original Assignee
Shionogi & Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Shionogi & Co filed Critical Shionogi & Co
Application granted granted Critical
Publication of ATE157647T1 publication Critical patent/ATE157647T1/de

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C231/00Preparation of carboxylic acid amides
    • C07C231/10Preparation of carboxylic acid amides from compounds not provided for in groups C07C231/02 - C07C231/08

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
AT92311175T 1991-12-18 1992-12-08 Verfahren zur herstellung von alpha- ketoamidderivaten ATE157647T1 (de)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP33485891 1991-12-18

Publications (1)

Publication Number Publication Date
ATE157647T1 true ATE157647T1 (de) 1997-09-15

Family

ID=18282010

Family Applications (1)

Application Number Title Priority Date Filing Date
AT92311175T ATE157647T1 (de) 1991-12-18 1992-12-08 Verfahren zur herstellung von alpha- ketoamidderivaten

Country Status (8)

Country Link
US (2) US5258551A (de)
EP (1) EP0547825B1 (de)
JP (1) JPH05331124A (de)
AT (1) ATE157647T1 (de)
DE (1) DE69222012T2 (de)
DK (1) DK0547825T3 (de)
ES (1) ES2106835T3 (de)
GR (1) GR3024653T3 (de)

Families Citing this family (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5258551A (en) * 1991-12-18 1993-11-02 Shionogi & Co., Ltd. Process for producing α-ketoamide derivative
DK0801054T3 (da) * 1994-12-26 2000-08-07 Shionogi & Co Fremgangsmåde til fremstilling af 2-(2-hydroxymethylphenyl)acetamidderivater og mellemprodukter til fremstilling deraf
GB9602623D0 (en) 1996-02-09 1996-04-10 Zeneca Ltd Fungicides
DE19645313A1 (de) 1996-11-04 1998-05-07 Basf Ag Substituierte 3-Benzylpyrazole
RU2167852C1 (ru) * 2000-07-04 2001-05-27 Санкт-Петербургская Государственная Химико-Фармацевтическая Академия Способ получения этилового эфира 4-карбоксифениламида малоновой кислоты
EP1406867B1 (de) * 2001-05-30 2008-12-31 Guilford Pharmaceuticals Inc. Thiolalkylbezoesäurederivate
US6727277B1 (en) 2002-11-12 2004-04-27 Kansas State University Research Foundation Compounds affecting cholesterol absorption
US20070027067A1 (en) * 2005-05-13 2007-02-01 Felicia Etzkorn Transition-state Inhibitors of Pin1, alpha-Ketoamide-containing peptidomimetics, and synthesis thereof
EP2545964A1 (de) 2011-07-13 2013-01-16 Phenex Pharmaceuticals AG Neuartige FXR- (NR1H4)-Binde- und -Aktivitätsmodulationsverbindungen
CN102603563B (zh) * 2012-01-16 2014-03-12 山东康乔生物科技有限公司 苯氧菌胺的制备方法
CA3252823A1 (en) 2016-06-13 2025-02-25 Gilead Sciences, Inc. Substituted tert-butyl-3-(2-chloro-phenyl)-3-hydroxyazetidine-1-carboxylate compounds
BR112018075734A2 (pt) 2016-06-13 2019-04-02 Gilead Sciences, Inc. composto, composição farmacêutica, método para tratar um paciente com uma doença ou condição mediada pelo menos em parte por fxr, e, uso de um composto.
CN110461328A (zh) 2017-03-28 2019-11-15 吉利德科学公司 治疗肝疾病的治疗组合
EP4360632B1 (de) 2019-01-15 2025-10-29 Gilead Sciences, Inc. Fxr (nr1h4) modulierende verbindungen
US11524005B2 (en) 2019-02-19 2022-12-13 Gilead Sciences, Inc. Solid forms of FXR agonists

Family Cites Families (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2428027A1 (fr) * 1978-06-08 1980-01-04 Anvar Nouveaux intermediaires de synthese perfluores et leur preparation
JPS58152846A (ja) * 1982-03-05 1983-09-10 Akio Yamamoto α−ケトアミド類の製造方法
US4657579A (en) * 1982-09-13 1987-04-14 Sandoz Ltd. Novel N-(5-pyrimidinyl)-chloroacetamides
JPS59172448A (ja) * 1983-07-29 1984-09-29 Nippon Nohyaku Co Ltd 安息香酸アニリド類の製造法
US4820872A (en) * 1984-07-17 1989-04-11 Allied Colloids Ltd. Process for hydrolyzing nitriles
NZ213630A (en) * 1984-10-19 1990-02-26 Ici Plc Acrylic acid derivatives and fungicidal compositions
JPH0657684B2 (ja) * 1986-03-28 1994-08-03 宇部興産株式会社 N―ベンジル2―(4―フルオル―3―トリフルオルメチルフェノキシ)ブタン酸アミド及びそれを含有する除草剤
DE3623921A1 (de) * 1986-07-16 1988-01-21 Basf Ag Oximether und diese enthaltende fungizide
DE69029334T2 (de) * 1989-05-17 1997-04-30 Shionogi Seiyaku Kk Verfahren zur Herstellung von Alkoxyiminoacetamid-Derivaten und ein Zwischenproduckt dafür
DE4030038A1 (de) * 1990-09-22 1992-03-26 Basf Ag Ortho-substituierte phenylessigsaeureamide
EP0712833B1 (de) * 1990-12-31 1997-09-03 Basf Aktiengesellschaft Verfahren zur Herstellung von 2-Phenoxymethylbenzoesäuren
US5258551A (en) * 1991-12-18 1993-11-02 Shionogi & Co., Ltd. Process for producing α-ketoamide derivative

Also Published As

Publication number Publication date
US5258551A (en) 1993-11-02
DE69222012T2 (de) 1998-01-29
JPH05331124A (ja) 1993-12-14
DE69222012D1 (de) 1997-10-09
EP0547825A2 (de) 1993-06-23
DK0547825T3 (da) 1997-10-06
EP0547825B1 (de) 1997-09-03
EP0547825A3 (en) 1993-09-08
GR3024653T3 (en) 1997-12-31
US5414122A (en) 1995-05-09
ES2106835T3 (es) 1997-11-16

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Legal Events

Date Code Title Description
UEP Publication of translation of european patent specification
REN Ceased due to non-payment of the annual fee