ATE207742T1 - Heterodisperse hydrogelsysteme zur verzögerten freisetzung unlöslicher arzneistoffe - Google Patents

Heterodisperse hydrogelsysteme zur verzögerten freisetzung unlöslicher arzneistoffe

Info

Publication number
ATE207742T1
ATE207742T1 AT94401925T AT94401925T ATE207742T1 AT E207742 T1 ATE207742 T1 AT E207742T1 AT 94401925 T AT94401925 T AT 94401925T AT 94401925 T AT94401925 T AT 94401925T AT E207742 T1 ATE207742 T1 AT E207742T1
Authority
AT
Austria
Prior art keywords
delayed release
sustained release
medicinal substances
hydrogel systems
insoluble medicinal
Prior art date
Application number
AT94401925T
Other languages
English (en)
Inventor
Anand R Baichwal
Original Assignee
Mendell Co Inc Edward
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Mendell Co Inc Edward filed Critical Mendell Co Inc Edward
Application granted granted Critical
Publication of ATE207742T1 publication Critical patent/ATE207742T1/de

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2095—Tabletting processes
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2009—Inorganic compounds
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2013—Organic compounds, e.g. phospholipids, fats
    • A61K9/2018—Sugars, or sugar alcohols, e.g. lactose, mannitol; Derivatives thereof, e.g. polysorbates
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2022—Organic macromolecular compounds
    • A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2022—Organic macromolecular compounds
    • A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2054—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A61K9/2806—Coating materials
    • A61K9/2833—Organic macromolecular compounds
    • A61K9/286—Polysaccharides, e.g. gums; Cyclodextrin
    • A61K9/2866—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
    • C—CHEMISTRY; METALLURGY
    • C08—ORGANIC MACROMOLECULAR COMPOUNDS; THEIR PREPARATION OR CHEMICAL WORKING-UP; COMPOSITIONS BASED THEREON
    • C08J—WORKING-UP; GENERAL PROCESSES OF COMPOUNDING; AFTER-TREATMENT NOT COVERED BY SUBCLASSES C08B, C08C, C08F, C08G or C08H
    • C08J3/00—Processes of treating or compounding macromolecular substances
    • C08J3/02—Making solutions, dispersions, lattices or gels by other methods than by solution, emulsion or suspension polymerisation techniques
    • C08J3/03—Making solutions, dispersions, lattices or gels by other methods than by solution, emulsion or suspension polymerisation techniques in aqueous media
    • C08J3/075—Macromolecular gels

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Dispersion Chemistry (AREA)
  • Inorganic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Biophysics (AREA)
  • Molecular Biology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Polymers & Plastics (AREA)
  • Organic Chemistry (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
AT94401925T 1993-09-09 1994-08-30 Heterodisperse hydrogelsysteme zur verzögerten freisetzung unlöslicher arzneistoffe ATE207742T1 (de)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US08/118,924 US5455046A (en) 1993-09-09 1993-09-09 Sustained release heterodisperse hydrogel systems for insoluble drugs

Publications (1)

Publication Number Publication Date
ATE207742T1 true ATE207742T1 (de) 2001-11-15

Family

ID=22381584

Family Applications (2)

Application Number Title Priority Date Filing Date
AT94401925T ATE207742T1 (de) 1993-09-09 1994-08-30 Heterodisperse hydrogelsysteme zur verzögerten freisetzung unlöslicher arzneistoffe
AT01104276T ATE318586T1 (de) 1993-09-09 1994-08-30 Heterodisperse hydrogelsysteme zur verzögerten freisetzung unlöslicher arzneistoffe

Family Applications After (1)

Application Number Title Priority Date Filing Date
AT01104276T ATE318586T1 (de) 1993-09-09 1994-08-30 Heterodisperse hydrogelsysteme zur verzögerten freisetzung unlöslicher arzneistoffe

Country Status (11)

Country Link
US (6) US5455046A (de)
EP (2) EP1101489B1 (de)
JP (1) JP4077886B2 (de)
AT (2) ATE207742T1 (de)
CA (1) CA2131647C (de)
DE (3) DE69428853T2 (de)
DK (1) DK0642785T3 (de)
ES (2) ES2070810T3 (de)
GR (1) GR950300035T1 (de)
IL (1) IL110744A (de)
PT (2) PT642785E (de)

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DK0642785T3 (da) 2001-12-31
JPH07165615A (ja) 1995-06-27
DE69434640D1 (de) 2006-04-27
EP0642785B1 (de) 2001-10-31
EP1101489A3 (de) 2001-09-19
PT642785E (pt) 2002-02-28
DE642785T1 (de) 1995-09-28
ATE318586T1 (de) 2006-03-15
EP1101489A2 (de) 2001-05-23
EP0642785A3 (de) 1996-11-06
ES2254274T3 (es) 2006-06-16
ES2070810T3 (es) 2001-12-16
DE69434640T2 (de) 2006-08-10
US5455046A (en) 1995-10-03
US5667801A (en) 1997-09-16
US5554387A (en) 1996-09-10
CA2131647C (en) 1999-08-10
JP4077886B2 (ja) 2008-04-23
IL110744A0 (en) 1994-08-22
PT1101489E (pt) 2006-05-31
DE69428853T2 (de) 2002-04-11
US6136343A (en) 2000-10-24
ES2070810T1 (es) 1995-06-16
GR950300035T1 (en) 1995-07-31
US5846563A (en) 1998-12-08
US5512297A (en) 1996-04-30
IL110744A (en) 1998-12-27
CA2131647A1 (en) 1995-03-10
EP0642785A2 (de) 1995-03-15
EP1101489B1 (de) 2006-03-01
DE69428853D1 (de) 2001-12-06

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