ATE208791T1 - Chemisches verfahren zur herstellung von amidderivaten von a 40926 antibiotikum - Google Patents

Chemisches verfahren zur herstellung von amidderivaten von a 40926 antibiotikum

Info

Publication number
ATE208791T1
ATE208791T1 AT97919359T AT97919359T ATE208791T1 AT E208791 T1 ATE208791 T1 AT E208791T1 AT 97919359 T AT97919359 T AT 97919359T AT 97919359 T AT97919359 T AT 97919359T AT E208791 T1 ATE208791 T1 AT E208791T1
Authority
AT
Austria
Prior art keywords
formula
compound
alk3
alk2
alk1
Prior art date
Application number
AT97919359T
Other languages
English (en)
Inventor
Gianbattista Panzone
Alessandra Maria Marazzi
Ermenegildo Restelli
Anacleto Gianantonio
Original Assignee
Biosearch Italia Spa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Biosearch Italia Spa filed Critical Biosearch Italia Spa
Application granted granted Critical
Publication of ATE208791T1 publication Critical patent/ATE208791T1/de

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K9/00—Peptides having up to 20 amino acids, containing saccharide radicals and having a fully defined sequence; Derivatives thereof
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K9/00—Peptides having up to 20 amino acids, containing saccharide radicals and having a fully defined sequence; Derivatives thereof
    • C07K9/006—Peptides having up to 20 amino acids, containing saccharide radicals and having a fully defined sequence; Derivatives thereof the peptide sequence being part of a ring structure
    • C07K9/008—Peptides having up to 20 amino acids, containing saccharide radicals and having a fully defined sequence; Derivatives thereof the peptide sequence being part of a ring structure directly attached to a hetero atom of the saccharide radical, e.g. actaplanin, avoparcin, ristomycin, vancomycin

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Genetics & Genomics (AREA)
  • Biochemistry (AREA)
  • Biophysics (AREA)
  • General Health & Medical Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Molecular Biology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Cephalosporin Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Peptides Or Proteins (AREA)
AT97919359T 1996-04-23 1997-04-15 Chemisches verfahren zur herstellung von amidderivaten von a 40926 antibiotikum ATE208791T1 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP96106341 1996-04-23
PCT/EP1997/001874 WO1997040067A1 (en) 1996-04-23 1997-04-15 Improved chemical process for preparing amide derivatives of antibiotic a 40926

Publications (1)

Publication Number Publication Date
ATE208791T1 true ATE208791T1 (de) 2001-11-15

Family

ID=8222699

Family Applications (1)

Application Number Title Priority Date Filing Date
AT97919359T ATE208791T1 (de) 1996-04-23 1997-04-15 Chemisches verfahren zur herstellung von amidderivaten von a 40926 antibiotikum

Country Status (13)

Country Link
US (1) US6218505B1 (de)
EP (1) EP0912604B1 (de)
JP (1) JP2000508671A (de)
KR (1) KR20000010589A (de)
AT (1) ATE208791T1 (de)
AU (1) AU719947B2 (de)
CA (1) CA2250578C (de)
DE (1) DE69708293T2 (de)
DK (1) DK0912604T3 (de)
ES (1) ES2165047T3 (de)
IL (1) IL126430A0 (de)
PT (1) PT912604E (de)
WO (1) WO1997040067A1 (de)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DK1140993T3 (da) 1998-12-23 2003-10-06 Theravance Inc Glycopeptidderivater og farmaceutiske præparater indeholdende dem
US7119061B2 (en) * 2002-11-18 2006-10-10 Vicuron Pharmaceuticals, Inc. Dalbavancin compositions for treatment of bacterial infections
US20060074014A1 (en) * 2002-11-18 2006-04-06 Vicuron Pharmaceuticals Inc. Dalbavancin compositions for treatment of bacterial infections
US20050090433A1 (en) * 2002-11-18 2005-04-28 Vicuron Pharmaceuticals, Inc Dalbavancin compositions for treatment of bacterial infections

Family Cites Families (52)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1496386A (en) 1975-03-05 1977-12-30 Lepetit Spa Antibiotics
FI73697C (fi) 1982-06-08 1987-11-09 Lepetit Spa Foerfarande foer framstaellning av individuella faktorer 1, 2, 3, 4 och 5 av teikomysin a2.
GB8307847D0 (en) 1983-03-22 1983-04-27 Lepetit Spa Antibiotics l 17054 and l 17046
GB8311136D0 (en) 1983-04-25 1983-06-02 Lepetit Spa Immobilised oligopeptides
AU579120B2 (en) 1983-12-16 1988-11-17 Gruppo Lepetit S.P.A. Chemical process for preparing antibiotic L 17392 (deglucoteicoplanin) and its salts
GB8333624D0 (en) 1983-12-16 1984-01-25 Lepetit Spa Antibiotics l 17054 and l 17392
GB8415092D0 (en) 1984-06-13 1984-07-18 Lepetit Spa Ester derivatives
GB8415093D0 (en) 1984-06-13 1984-07-18 Lepetit Spa Antibiotic l 17392
GB8420405D0 (en) 1984-08-10 1984-09-12 Lepetit Spa Preparing antibiotic l 17046
GB8425685D0 (en) 1984-10-11 1984-11-14 Lepetit Spa Antibiotic a 40926 complex
US4914187A (en) 1984-11-13 1990-04-03 Gruppo Lepetit S.P.A Ester derivatives of antibiotic L 17046
DE3577733C5 (de) 1984-12-03 2010-12-30 Maschinenfabrik Rieter Ag Garnbehandlungsdüse.
GB8512795D0 (en) 1985-05-21 1985-06-26 Lepetit Spa Increasing ratio of components of teicoplanin a2 complex
GB8522574D0 (en) 1985-09-12 1985-10-16 Lepetit Spa Amides of teicoplanin compounds
GB8529272D0 (en) 1985-11-28 1986-01-02 Lepetit Spa Teicoplanin derivatives
GB8531846D0 (en) 1985-12-30 1986-02-05 Lepetit Spa Antibiotic a 40926 mannosyl aglycon
GB8608798D0 (en) 1986-04-11 1986-05-14 Lepetit Spa Recovery of glycopeptide antibiotics from aqueous solutions
GB8608809D0 (en) 1986-04-11 1986-05-14 Lepetit Spa Antibiotic
CA1282725C (en) 1986-04-18 1991-04-09 Brian A. Naughton Process for replicating bone marrow in vitro and using the same
GR871488B (en) 1986-10-10 1987-11-12 Lepetit Spa New antibiotics
GB8701872D0 (en) 1987-01-28 1987-03-04 Lepetit Spa N15-alkyl & n15,n15-dialkyl derivatives
GB8704847D0 (en) 1987-03-02 1987-04-08 Lepetit Spa Substituted alkylamides of teicoplanin compounds
GB8711066D0 (en) 1987-05-11 1987-06-17 Lepetit Spa Teicoplanin derivatives
GB8715735D0 (en) 1987-07-03 1987-08-12 Lepetit Spa De-mannosyl teicoplanin derivatives
GB8720980D0 (en) 1987-09-07 1987-10-14 Lepetit Spa Derivatives
US4816706A (en) 1987-09-10 1989-03-28 International Business Machines Corporation Sense amplifier with improved bitline precharging for dynamic random access memory
GB8729989D0 (en) 1987-12-23 1988-02-03 Lepetit Spa Novel hydrogenated derivatives of antibiotic a/16686
GB8802211D0 (en) 1988-02-02 1988-03-02 Lepetit Spa Teicoplanin hydrazides
GB8808658D0 (en) 1988-04-13 1988-05-18 Lepetit Spa Aglycons of a/16686 antibiotics
GB8817053D0 (en) 1988-07-18 1988-08-24 Lepetit Spa Process for preparing n15 n15-dialkyl derivatives of teicoplanin compounds
GB8817052D0 (en) 1988-07-18 1988-08-24 Lepetit Spa Process for preparing n15-alkyl derivatives of teicoplanin compounds
GB8817397D0 (en) 1988-07-21 1988-08-24 Lepetit Spa N15-alkyl & n15 n15-di-alkyl derivatives of teicoplanin antibiotics carrying functional groups on alkyl side chain
GB8817736D0 (en) 1988-07-26 1988-09-01 Lepetit Spa New teicoplanin antibiotics
GB8827202D0 (en) 1988-11-22 1988-12-29 Lepetit Spa Process for preparing 63-carboxyamides of teicoplanin antibiotics
US5194424A (en) 1988-12-27 1993-03-16 Gruppo Lepetit Spa C63 -amide derivatives of 34-de(acetylglucosaminyl)-34-deoxy-teicoplanin and their use as medicaments against bacteria resistant to glycopeptide antibiotics
ATE135369T1 (de) 1988-12-27 1996-03-15 Lepetit Spa Chemisches verfahren zur herstellung des antibiotikums l 17392 (deglukoteicoplanin) und dessen salze
US5500410A (en) 1989-03-29 1996-03-19 Gruppo Lepetit S.P.A. Substituted alkylamide derivatives of teicoplanin
US5185320A (en) 1989-04-03 1993-02-09 Gruppo Lepetit S.P.A. O56 -alkyl derivatives of aglycone and pseudo aglycones of teicoplanin
DK0409045T3 (da) 1989-07-18 1997-12-22 Biosearch Italia Spa Pentapeptidantibiotika afledt fra dalbaheptider.
EP0427142B1 (de) 1989-11-07 1995-05-17 GRUPPO LEPETIT S.p.A. Verfahren zur Rückgewinnung von Antibiotikum A/16686
ATE158306T1 (de) 1990-03-28 1997-10-15 Lepetit Spa Verfahren zur herstellung von mannosylteicoplaninderivaten und mannosylteicoplaninaglykon
DK0479086T3 (da) 1990-10-01 1995-10-23 Lepetit Spa Fremgangsmåde til indvinding af teicoplanin
HUT63860A (en) * 1990-12-05 1993-10-28 Lepetit Spa Process for producing 39-decarboxy-38-(hydroxymethyl) derivatives of teikoplanin antibiotics
US5644025A (en) 1990-12-10 1997-07-01 Gruppo Lepetit Spa Tetrapeptides deriving from dalbaheptide antibiotics
US5438117A (en) 1990-12-20 1995-08-01 Gruppo Lepetit S.P.A. Hexapeptides deriving from aglucoteicoplanin and a process for preparing them
US5606036A (en) 1991-03-27 1997-02-25 Gruppo Lepetit Spa Antibiotic A 40926 ester derivatives
DE69215665T2 (de) * 1991-03-27 1997-06-12 Gruppo Lepetit S.P.A., Lainate Esterderivate von antibiotikum-a 40926
US5750509A (en) 1991-07-29 1998-05-12 Gruppo Lepetit S.P.A. Amide derivatives of antibiotic A 40926
ATE125551T1 (de) * 1991-07-29 1995-08-15 Lepetit Spa Amidderivate vom antibiotikum a 40926.
RU2126419C1 (ru) 1993-05-19 1999-02-20 Группо Лепетит С.П.А. Аглюкодальбагептиды и/или их соли с кислотами или основаниями, или их внутренние соли, способ получения, фармацевтическая композиция
JP2888741B2 (ja) * 1993-09-27 1999-05-10 日本ペイント株式会社 薄膜パターン形成法
WO1997002288A1 (en) * 1995-07-05 1997-01-23 Gruppo Lepetit S.P.A. Purification of dalbaheptide antibiotics by isoelectric focusing

Also Published As

Publication number Publication date
DK0912604T3 (da) 2002-03-25
KR20000010589A (ko) 2000-02-15
DE69708293T2 (de) 2002-05-02
AU2386197A (en) 1997-11-12
WO1997040067A1 (en) 1997-10-30
DE69708293D1 (de) 2001-12-20
JP2000508671A (ja) 2000-07-11
EP0912604B1 (de) 2001-11-14
ES2165047T3 (es) 2002-03-01
IL126430A0 (en) 1999-08-17
CA2250578C (en) 2003-06-24
US6218505B1 (en) 2001-04-17
CA2250578A1 (en) 1997-10-30
AU719947B2 (en) 2000-05-18
PT912604E (pt) 2002-05-31
EP0912604A1 (de) 1999-05-06

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Legal Events

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EEIH Change in the person of patent owner
REN Ceased due to non-payment of the annual fee