ATE212034T1 - Derivate von 5-0-desosaminyl-6-0-methyl erythronolid a, ihre verfahren zur herstellung und verwendung zur herstellung von arzneimitteln - Google Patents

Derivate von 5-0-desosaminyl-6-0-methyl erythronolid a, ihre verfahren zur herstellung und verwendung zur herstellung von arzneimitteln

Info

Publication number: ATE212034T1
Authority: AT; Austria
Prior art keywords: production; desosaminyl; derivatives; medicinal products; methyl erythronolide
Prior art date: 1995-10-09

Application number

AT96933501T

Other languages

English (en)

Inventor

Alain Bonnet

Bernadette Chappert

Jacques Lagouardat

Original Assignee

Aventis Pharma Sa

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1995-10-09

Filing date

1996-10-08

Publication date

2002-02-15

1996-10-08 Application filed by Aventis Pharma Sa filed Critical Aventis Pharma Sa

2002-02-15 Application granted granted Critical

2002-02-15 Publication of ATE212034T1 publication Critical patent/ATE212034T1/de

Links

YVTFLQUPRIIRFE-QUMKBVJLSA-N erythronolide A Chemical compound CC[C@H]1OC(=O)[C@H](C)[C@@H](O)[C@H](C)[C@@H](O)[C@](C)(O)C[C@@H](C)C(=O)[C@H](C)[C@@H](O)[C@]1(C)O YVTFLQUPRIIRFE-QUMKBVJLSA-N 0.000 title 1
229940126601 medicinal product Drugs 0.000 title 1
238000000034 method Methods 0.000 title 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
- C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
- C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
Engineering & Computer Science (AREA)
Biochemistry (AREA)
Biotechnology (AREA)
General Health & Medical Sciences (AREA)
Genetics & Genomics (AREA)
Molecular Biology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Saccharide Compounds (AREA)

AT96933501T 1995-10-09 1996-10-08 Derivate von 5-0-desosaminyl-6-0-methyl erythronolid a, ihre verfahren zur herstellung und verwendung zur herstellung von arzneimitteln ATE212034T1 (de)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
FR9511861A FR2739620B1 (fr)	1995-10-09	1995-10-09	Nouveaux derives de la 5-0-desosaminyl 6-o-methyl erythronolide a, leur procede de preparation et leur application a la preparation de produits biologiquement actifs
PCT/FR1996/001567 WO1997013774A2 (fr)	1995-10-09	1996-10-08	Nouveaux derives de la 5-o-desosaminyl 6-o-methyl erythronolide a, leur procede de preparation et leur application a la preparation de produits biologiquement actifs

Publications (1)

Publication Number	Publication Date
ATE212034T1 true ATE212034T1 (de)	2002-02-15

Family

ID=9483377

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
AT96933501T ATE212034T1 (de)	1995-10-09	1996-10-08	Derivate von 5-0-desosaminyl-6-0-methyl erythronolid a, ihre verfahren zur herstellung und verwendung zur herstellung von arzneimitteln

Country Status (33)

Country	Link
US (1)	US6011142A (de)
EP (1)	EP0854879B1 (de)
JP (1)	JP4327248B2 (de)
KR (1)	KR100451063B1 (de)
CN (1)	CN1067401C (de)
AP (1)	AP888A (de)
AR (1)	AR004688A1 (de)
AT (1)	ATE212034T1 (de)
AU (1)	AU708351B2 (de)
BG (1)	BG63752B1 (de)
BR (1)	BR9610959A (de)
CA (1)	CA2231562C (de)
CZ (1)	CZ293430B6 (de)
DE (1)	DE69618607T2 (de)
DK (1)	DK0854879T3 (de)
EA (1)	EA000765B1 (de)
EE (1)	EE03878B1 (de)
ES (1)	ES2171722T3 (de)
FR (1)	FR2739620B1 (de)
GE (1)	GEP20032899B (de)
HU (1)	HUP9900136A3 (de)
IL (1)	IL123613A0 (de)
MX (1)	MX9802655A (de)
NO (1)	NO312592B1 (de)
PL (1)	PL183645B1 (de)
PT (1)	PT854879E (de)
RO (1)	RO118874B1 (de)
SI (1)	SI0854879T1 (de)
SK (1)	SK283619B6 (de)
TR (1)	TR199800624T1 (de)
UA (1)	UA52621C2 (de)
WO (1)	WO1997013774A2 (de)
ZA (1)	ZA966666B (de)

Families Citing this family (16)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
FR2777282B1 (fr) *	1998-04-08	2001-04-20	Hoechst Marion Roussel Inc	Nouveaux derives de la 2-fluoro 3-de((2,6-dideoxy 3-c-methyl 3-0-methyl-alpha-l-ribohexopyranosyl) oxyl) 6-o-methyl 3-oxo erythromycine, leur procede de preparation et leur application a la synthese de principes actifs de medicaments
US6590083B1 (en)	1999-04-16	2003-07-08	Ortho-Mcneil Pharmaceutical, Inc.	Ketolide antibacterials
AU775637B2 (en) *	1999-04-16	2004-08-12	Kosan Biosciences, Inc.	Macrolide antiinfective agents
JP2002542197A (ja)	1999-04-16	2002-12-10	オーソ−マクニール・フアーマシユーチカル・インコーポレーテツド	ケトライド抗菌剤
GB0031312D0 (en) *	2000-12-21	2001-02-07	Glaxo Group Ltd	Macrolides
EP3738591A3 (de) *	2003-03-10	2021-03-24	Merck Sharp & Dohme Corp.	Neuartige antibakterielle wirkstoffe
CN101917850B (zh)	2007-10-25	2016-01-13	森普拉制药公司	大环内酯类抗菌剂的制备方法
DK2358379T3 (en) *	2008-10-24	2016-03-07	Cempra Pharmaceuticals Inc	BIOFORSVAR USING TRIAZOLHOLDIGE macrolides
US9937194B1 (en)	2009-06-12	2018-04-10	Cempra Pharmaceuticals, Inc.	Compounds and methods for treating inflammatory diseases
EP2475253B1 (de)	2009-09-10	2016-10-26	Cempra Pharmaceuticals, Inc.	Verfahren zur behandlung von malaria, tuberkulose und mac-erkrankungen
BR112012023950A2 (pt)	2010-03-22	2016-07-05	Cempra Pharmaceuticals Inc	formas cristalinas de um macrolídeo, e usos dos mesmos
PL2571506T3 (pl)	2010-05-20	2017-10-31	Cempra Pharmaceuticals Inc	Sposoby sporządzania makrolidów i ketolidów oraz ich produktów pośrednich
US9815863B2 (en)	2010-09-10	2017-11-14	Cempra Pharmaceuticals, Inc.	Hydrogen bond forming fluoro ketolides for treating diseases
MX2014011537A (es)	2012-03-27	2015-02-10	Cempra Pharmaceuticals Inc	Formulaciones parenterales para la administracion de antibioticos macrolidos.
WO2014152326A1 (en)	2013-03-14	2014-09-25	Cempra Pharmaceuticals, Inc.	Methods for treating respiratory diseases and formulations therefor
BR112015023670A2 (pt)	2013-03-15	2017-07-18	Cempra Pharmaceuticals Inc	processo para preparar um composto

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US3923784A (en) *	1973-09-10	1975-12-02	Hoffmann La Roche	Erythromycin a derivatives
US4518590A (en) *	1984-04-13	1985-05-21	Pfizer Inc.	9α-Aza-9α-homoerythromycin compounds, pharmaceutical compositions and therapeutic method
US4742049A (en) *	1986-06-04	1988-05-03	Abbott Laboratories	Semisynthetic erythromycin antibiotics
PT86800B (pt) *	1987-02-24	1992-05-29	Beecham Group Plc	Processo para a preparacao de derivados de eritromicina
US5523399A (en) *	1991-12-27	1996-06-04	Taisho Pharmaceutical Co., Ltd.	5-O-desosaminylerythronolide derivatives
DE69301916T2 (de) *	1992-04-22	1996-08-08	Taisho Pharmaceutical Co., Ltd., Tokio/Tokyo	5-0-desosaminylerythronolid a derivate
FR2692579B1 (fr) *	1992-06-19	1995-06-02	Roussel Uclaf	Nouveaux dérivés de la picromycine, leur procédé de préparation et leur application comme médicaments.
US5602239A (en) *	1993-01-26	1997-02-11	Taisho Pharmaceutical Co., Ltd.	5-O-desosaminylerythronolide derivatives

1995
- 1995-10-09 FR FR9511861A patent/FR2739620B1/fr not_active Expired - Fee Related
1996
- 1996-08-06 ZA ZA9606666A patent/ZA966666B/xx unknown
- 1996-08-10 UA UA98041836A patent/UA52621C2/uk unknown
- 1996-10-07 AR ARP960104634A patent/AR004688A1/es not_active Application Discontinuation
- 1996-10-08 SK SK431-98A patent/SK283619B6/sk unknown
- 1996-10-08 US US09/051,378 patent/US6011142A/en not_active Ceased
- 1996-10-08 AU AU72208/96A patent/AU708351B2/en not_active Expired
- 1996-10-08 RO RO98-00826A patent/RO118874B1/ro unknown
- 1996-10-08 PT PT96933501T patent/PT854879E/pt unknown
- 1996-10-08 EA EA199800280A patent/EA000765B1/ru not_active IP Right Cessation
- 1996-10-08 ES ES96933501T patent/ES2171722T3/es not_active Expired - Lifetime
- 1996-10-08 DE DE69618607T patent/DE69618607T2/de not_active Expired - Lifetime
- 1996-10-08 GE GEAP19964227A patent/GEP20032899B/en unknown
- 1996-10-08 EP EP96933501A patent/EP0854879B1/de not_active Expired - Lifetime
- 1996-10-08 IL IL12361396A patent/IL123613A0/xx not_active IP Right Cessation
- 1996-10-08 AP APAP/P/1998/001216A patent/AP888A/en active
- 1996-10-08 HU HU9900136A patent/HUP9900136A3/hu unknown
- 1996-10-08 BR BR9610959A patent/BR9610959A/pt not_active Application Discontinuation
- 1996-10-08 PL PL96326001A patent/PL183645B1/pl not_active IP Right Cessation
- 1996-10-08 WO PCT/FR1996/001567 patent/WO1997013774A2/fr not_active Ceased
- 1996-10-08 JP JP51476697A patent/JP4327248B2/ja not_active Expired - Lifetime
- 1996-10-08 AT AT96933501T patent/ATE212034T1/de active
- 1996-10-08 DK DK96933501T patent/DK0854879T3/da active
- 1996-10-08 CA CA002231562A patent/CA2231562C/fr not_active Expired - Lifetime
- 1996-10-08 SI SI9630452T patent/SI0854879T1/xx unknown
- 1996-10-08 TR TR1998/00624T patent/TR199800624T1/xx unknown
- 1996-10-08 KR KR10-1998-0702581A patent/KR100451063B1/ko not_active Expired - Lifetime
- 1996-10-08 EE EE9800109A patent/EE03878B1/xx not_active IP Right Cessation
- 1996-10-08 CZ CZ19981055A patent/CZ293430B6/cs not_active IP Right Cessation
- 1996-10-08 CN CN96197514A patent/CN1067401C/zh not_active Expired - Lifetime
1998
- 1998-03-25 BG BG102350A patent/BG63752B1/bg unknown
- 1998-04-03 MX MX9802655A patent/MX9802655A/es unknown
- 1998-04-08 NO NO19981630A patent/NO312592B1/no not_active IP Right Cessation

Also Published As

Publication number	Publication date
EP0854879B1 (de)	2002-01-16
EA199800280A1 (ru)	1998-10-29
NO981630D0 (no)	1998-04-08
DE69618607D1 (de)	2002-02-21
SK43198A3 (en)	1998-11-04
AU708351B2 (en)	1999-08-05
KR19990064100A (ko)	1999-07-26
DE69618607T2 (de)	2002-08-14
UA52621C2 (uk)	2003-01-15
CN1067401C (zh)	2001-06-20
IL123613A0 (en)	1998-10-30
BR9610959A (pt)	1999-03-02
EA000765B1 (ru)	2000-04-24
MX9802655A (es)	1998-11-30
SK283619B6 (sk)	2003-10-07
AP888A (en)	2000-11-10
PL326001A1 (en)	1998-08-17
CZ105598A3 (cs)	1998-07-15
AR004688A1 (es)	1999-03-10
HUP9900136A1 (hu)	1999-05-28
AU7220896A (en)	1997-04-30
FR2739620A1 (fr)	1997-04-11
BG102350A (en)	1999-03-31
EP0854879A2 (de)	1998-07-29
NO312592B1 (no)	2002-06-03
GEP20032899B (en)	2003-02-25
PL183645B1 (pl)	2002-06-28
NO981630L (no)	1998-04-08
EE03878B1 (et)	2002-10-15
CZ293430B6 (cs)	2004-04-14
TR199800624T1 (xx)	1998-06-22
WO1997013774A3 (fr)	1997-05-29
RO118874B1 (ro)	2003-12-30
EE9800109A (et)	1998-10-15
US6011142A (en)	2000-01-04
WO1997013774A2 (fr)	1997-04-17
SI0854879T1 (en)	2002-08-31
PT854879E (pt)	2002-07-31
DK0854879T3 (da)	2002-05-06
HUP9900136A3 (en)	2000-04-28
ES2171722T3 (es)	2002-09-16
ZA966666B (en)	1997-08-06
CA2231562C (fr)	2006-11-28
CN1199403A (zh)	1998-11-18
JPH11513401A (ja)	1999-11-16
JP4327248B2 (ja)	2009-09-09
BG63752B1 (bg)	2002-11-29
CA2231562A1 (fr)	1997-04-17
KR100451063B1 (ko)	2004-12-17
FR2739620B1 (fr)	1997-12-19

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Legal Events

Date	Code	Title	Description
2002-06-15	UEP	Publication of translation of european patent specification