DK0854879T3 - Nye forbindelser afledt af 5-0-desosamiyl-6-0-methyl-erythronolid A, fremgangsmåde til deres fremstilling og deres anvendelse til fremstilling af biologisk aktive stoffer - Google Patents

Nye forbindelser afledt af 5-0-desosamiyl-6-0-methyl-erythronolid A, fremgangsmåde til deres fremstilling og deres anvendelse til fremstilling af biologisk aktive stoffer

Info

Publication number
DK0854879T3
DK0854879T3 DK96933501T DK96933501T DK0854879T3 DK 0854879 T3 DK0854879 T3 DK 0854879T3 DK 96933501 T DK96933501 T DK 96933501T DK 96933501 T DK96933501 T DK 96933501T DK 0854879 T3 DK0854879 T3 DK 0854879T3
Authority
DK
Denmark
Prior art keywords
preparation
desosamiyl
erythronolide
methyl
biologically active
Prior art date
Application number
DK96933501T
Other languages
English (en)
Inventor
Alain Bonnet
Bernadette Chappert
Jacques Lagouardat
Original Assignee
Aventis Pharma Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Aventis Pharma Sa filed Critical Aventis Pharma Sa
Application granted granted Critical
Publication of DK0854879T3 publication Critical patent/DK0854879T3/da

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • General Health & Medical Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
DK96933501T 1995-10-09 1996-10-08 Nye forbindelser afledt af 5-0-desosamiyl-6-0-methyl-erythronolid A, fremgangsmåde til deres fremstilling og deres anvendelse til fremstilling af biologisk aktive stoffer DK0854879T3 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR9511861A FR2739620B1 (fr) 1995-10-09 1995-10-09 Nouveaux derives de la 5-0-desosaminyl 6-o-methyl erythronolide a, leur procede de preparation et leur application a la preparation de produits biologiquement actifs
PCT/FR1996/001567 WO1997013774A2 (fr) 1995-10-09 1996-10-08 Nouveaux derives de la 5-o-desosaminyl 6-o-methyl erythronolide a, leur procede de preparation et leur application a la preparation de produits biologiquement actifs

Publications (1)

Publication Number Publication Date
DK0854879T3 true DK0854879T3 (da) 2002-05-06

Family

ID=9483377

Family Applications (1)

Application Number Title Priority Date Filing Date
DK96933501T DK0854879T3 (da) 1995-10-09 1996-10-08 Nye forbindelser afledt af 5-0-desosamiyl-6-0-methyl-erythronolid A, fremgangsmåde til deres fremstilling og deres anvendelse til fremstilling af biologisk aktive stoffer

Country Status (33)

Country Link
US (1) US6011142A (da)
EP (1) EP0854879B1 (da)
JP (1) JP4327248B2 (da)
KR (1) KR100451063B1 (da)
CN (1) CN1067401C (da)
AP (1) AP888A (da)
AR (1) AR004688A1 (da)
AT (1) ATE212034T1 (da)
AU (1) AU708351B2 (da)
BG (1) BG63752B1 (da)
BR (1) BR9610959A (da)
CA (1) CA2231562C (da)
CZ (1) CZ293430B6 (da)
DE (1) DE69618607T2 (da)
DK (1) DK0854879T3 (da)
EA (1) EA000765B1 (da)
EE (1) EE03878B1 (da)
ES (1) ES2171722T3 (da)
FR (1) FR2739620B1 (da)
GE (1) GEP20032899B (da)
HU (1) HUP9900136A3 (da)
IL (1) IL123613A0 (da)
MX (1) MX9802655A (da)
NO (1) NO312592B1 (da)
PL (1) PL183645B1 (da)
PT (1) PT854879E (da)
RO (1) RO118874B1 (da)
SI (1) SI0854879T1 (da)
SK (1) SK283619B6 (da)
TR (1) TR199800624T1 (da)
UA (1) UA52621C2 (da)
WO (1) WO1997013774A2 (da)
ZA (1) ZA966666B (da)

Families Citing this family (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2777282B1 (fr) * 1998-04-08 2001-04-20 Hoechst Marion Roussel Inc Nouveaux derives de la 2-fluoro 3-de((2,6-dideoxy 3-c-methyl 3-0-methyl-alpha-l-ribohexopyranosyl) oxyl) 6-o-methyl 3-oxo erythromycine, leur procede de preparation et leur application a la synthese de principes actifs de medicaments
IL145976A0 (en) 1999-04-16 2002-07-25 Ortho Mcneil Pharm Inc Ketolide antibacterials
US6590083B1 (en) 1999-04-16 2003-07-08 Ortho-Mcneil Pharmaceutical, Inc. Ketolide antibacterials
US6395710B1 (en) * 1999-04-16 2002-05-28 Kosan Biosciences, Inc. Macrolide antiinfective agents
GB0031312D0 (en) * 2000-12-21 2001-02-07 Glaxo Group Ltd Macrolides
EP1638549A4 (en) 2003-03-10 2011-06-15 Optimer Pharmaceuticals Inc NEW ANTIBACTERIAL AGENTS
CA2703475A1 (en) * 2007-10-25 2009-04-30 Cempra Pharmaceuticals, Inc. Process for the preparation of macrolide antibacterial agents
US8796232B2 (en) * 2008-10-24 2014-08-05 Cempra Pharmaceuticals, Inc. Methods for treating resistant diseases using triazole containing macrolides
US9937194B1 (en) 2009-06-12 2018-04-10 Cempra Pharmaceuticals, Inc. Compounds and methods for treating inflammatory diseases
JP5914335B2 (ja) 2009-09-10 2016-05-11 センプラ ファーマシューティカルズ，インコーポレイテッド マラリア、結核、及びｍａｃ病の治療方法
CN103080122A (zh) 2010-03-22 2013-05-01 森普拉制药公司 大环内脂的结晶形式及其用途
WO2011146829A1 (en) 2010-05-20 2011-11-24 Cempra Pharmaceuticals, Inc. Processes for preparing macrolides and ketolides and intermediates therefor
JP6042334B2 (ja) 2010-09-10 2016-12-14 センプラ ファーマシューティカルズ，インコーポレイテッド 疾患治療のための水素結合形成フルオロケトライド
CN104470527B (zh) 2012-03-27 2019-05-28 森普拉制药公司 用于施用大环内酯抗生素的肠胃外制剂
RU2015138796A (ru) 2013-03-14 2017-04-19 Семпра Фармасьютикалс, Инк. Способы и составы для лечения респираторных заболеваний
WO2014145210A1 (en) 2013-03-15 2014-09-18 Cempra Pharmaceuticals, Inc. Convergent processes for preparing macrolide antibacterial agents

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3923784A (en) * 1973-09-10 1975-12-02 Hoffmann La Roche Erythromycin a derivatives
US4518590A (en) * 1984-04-13 1985-05-21 Pfizer Inc. 9α-Aza-9α-homoerythromycin compounds, pharmaceutical compositions and therapeutic method
US4742049A (en) * 1986-06-04 1988-05-03 Abbott Laboratories Semisynthetic erythromycin antibiotics
KR880009960A (ko) * 1987-02-24 1988-10-06 데이빗 로버츠 화학적 화합물
US5523399A (en) * 1991-12-27 1996-06-04 Taisho Pharmaceutical Co., Ltd. 5-O-desosaminylerythronolide derivatives
US5631355A (en) * 1992-04-22 1997-05-20 Taisho Pharmaceutical Co., Ltd. 5-O-desosaminylerythronolide a derivatives
FR2692579B1 (fr) * 1992-06-19 1995-06-02 Roussel Uclaf Nouveaux dérivés de la picromycine, leur procédé de préparation et leur application comme médicaments.
KR960700258A (ko) * 1993-01-26 1996-01-19 우에하라 아키라 5-0-데소사미닐에리쓰로노라이드 유도체

Also Published As

Publication number Publication date
HUP9900136A3 (en) 2000-04-28
NO981630D0 (no) 1998-04-08
GEP20032899B (en) 2003-02-25
AR004688A1 (es) 1999-03-10
TR199800624T1 (xx) 1998-06-22
CZ105598A3 (cs) 1998-07-15
HUP9900136A1 (hu) 1999-05-28
AU7220896A (en) 1997-04-30
WO1997013774A3 (fr) 1997-05-29
WO1997013774A2 (fr) 1997-04-17
RO118874B1 (ro) 2003-12-30
FR2739620B1 (fr) 1997-12-19
PL326001A1 (en) 1998-08-17
NO981630L (no) 1998-04-08
ZA966666B (en) 1997-08-06
BG102350A (en) 1999-03-31
CZ293430B6 (cs) 2004-04-14
CN1067401C (zh) 2001-06-20
IL123613A0 (en) 1998-10-30
KR19990064100A (ko) 1999-07-26
SK43198A3 (en) 1998-11-04
EP0854879A2 (fr) 1998-07-29
JPH11513401A (ja) 1999-11-16
EE9800109A (et) 1998-10-15
SI0854879T1 (en) 2002-08-31
AP888A (en) 2000-11-10
SK283619B6 (sk) 2003-10-07
CA2231562A1 (fr) 1997-04-17
ES2171722T3 (es) 2002-09-16
FR2739620A1 (fr) 1997-04-11
MX9802655A (es) 1998-11-30
CN1199403A (zh) 1998-11-18
ATE212034T1 (de) 2002-02-15
BG63752B1 (bg) 2002-11-29
UA52621C2 (uk) 2003-01-15
EE03878B1 (et) 2002-10-15
PL183645B1 (pl) 2002-06-28
BR9610959A (pt) 1999-03-02
DE69618607D1 (de) 2002-02-21
KR100451063B1 (ko) 2004-12-17
AU708351B2 (en) 1999-08-05
NO312592B1 (no) 2002-06-03
US6011142A (en) 2000-01-04
EA199800280A1 (ru) 1998-10-29
CA2231562C (fr) 2006-11-28
DE69618607T2 (de) 2002-08-14
PT854879E (pt) 2002-07-31
JP4327248B2 (ja) 2009-09-09
EP0854879B1 (fr) 2002-01-16
EA000765B1 (ru) 2000-04-24

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