ATE229943T1 - Zwischenprodukte zur herstellung von 1- substituierten, 2-substituierten-1h-imidazo(4,5- c)chinolin-4-aminen - Google Patents

Zwischenprodukte zur herstellung von 1- substituierten, 2-substituierten-1h-imidazo(4,5- c)chinolin-4-aminen

Info

Publication number
ATE229943T1
ATE229943T1 AT98105754T AT98105754T ATE229943T1 AT E229943 T1 ATE229943 T1 AT E229943T1 AT 98105754 T AT98105754 T AT 98105754T AT 98105754 T AT98105754 T AT 98105754T AT E229943 T1 ATE229943 T1 AT E229943T1
Authority
AT
Austria
Prior art keywords
substituted
imidazo
amines
quinoline
production
Prior art date
Application number
AT98105754T
Other languages
English (en)
Inventor
John F Gerster
Stephen L Crooks
Kyle J Lindstrom
Original Assignee
Minnesota Mining & Mfg
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Minnesota Mining & Mfg filed Critical Minnesota Mining & Mfg
Application granted granted Critical
Publication of ATE229943T1 publication Critical patent/ATE229943T1/de

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D215/00Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
    • C07D215/02Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
    • C07D215/16Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D215/38Nitrogen atoms
    • C07D215/42Nitrogen atoms attached in position 4

Landscapes

  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Virology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Quinoline Compounds (AREA)
  • Emulsifying, Dispersing, Foam-Producing Or Wetting Agents (AREA)
  • Lubricants (AREA)
AT98105754T 1991-03-01 1992-02-20 Zwischenprodukte zur herstellung von 1- substituierten, 2-substituierten-1h-imidazo(4,5- c)chinolin-4-aminen ATE229943T1 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US66292691A 1991-03-01 1991-03-01
US68732691A 1991-04-18 1991-04-18

Publications (1)

Publication Number Publication Date
ATE229943T1 true ATE229943T1 (de) 2003-01-15

Family

ID=27098631

Family Applications (2)

Application Number Title Priority Date Filing Date
AT92906763T ATE179711T1 (de) 1991-03-01 1992-02-20 1,2-substituierte 1h-imidazo(4,5-c>chinolin-4- amine
AT98105754T ATE229943T1 (de) 1991-03-01 1992-02-20 Zwischenprodukte zur herstellung von 1- substituierten, 2-substituierten-1h-imidazo(4,5- c)chinolin-4-aminen

Family Applications Before (1)

Application Number Title Priority Date Filing Date
AT92906763T ATE179711T1 (de) 1991-03-01 1992-02-20 1,2-substituierte 1h-imidazo(4,5-c>chinolin-4- amine

Country Status (18)

Country Link
EP (2) EP0872478B1 (de)
JP (1) JP2955019B2 (de)
AT (2) ATE179711T1 (de)
AU (2) AU658621B2 (de)
CA (2) CA2289219C (de)
CZ (1) CZ285050B6 (de)
DE (2) DE69229114T2 (de)
DK (2) DK0872478T3 (de)
ES (2) ES2131070T3 (de)
HU (5) HU222251B1 (de)
IE (1) IE920605A1 (de)
IL (2) IL101110A (de)
NO (1) NO303729B1 (de)
NZ (1) NZ241784A (de)
PH (1) PH31614A (de)
SG (2) SG70625A1 (de)
UA (1) UA32546C2 (de)
WO (1) WO1992015582A1 (de)

Families Citing this family (88)

* Cited by examiner, † Cited by third party
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US5648516A (en) * 1994-07-20 1997-07-15 Minnesota Mining And Manufacturing Company Fused cycloalkylimidazopyridines
US5352784A (en) * 1993-07-15 1994-10-04 Minnesota Mining And Manufacturing Company Fused cycloalkylimidazopyridines
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CN108137586B (zh) * 2015-09-14 2021-04-13 辉瑞大药厂 作为LRRK2抑制剂的新颖咪唑并[4,5-c]喹啉和咪唑并[4,5-c][1,5]萘啶衍生物
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JP7012668B2 (ja) 2016-06-12 2022-02-14 エフ・ホフマン-ラ・ロシュ・アクチェンゲゼルシャフト ジヒドロピリミジニルベンズアゼピンジカルボキサミド化合物
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CA1271477A (en) * 1983-11-18 1990-07-10 John F. Gerster 1h-imidazo[4,5-c]quinolin-4-amines
IL73534A (en) 1983-11-18 1990-12-23 Riker Laboratories Inc 1h-imidazo(4,5-c)quinoline-4-amines,their preparation and pharmaceutical compositions containing certain such compounds
DK0385630T3 (da) * 1989-02-27 1997-05-12 Riker Laboratories Inc 1H-imidazo(4,5-c)quinolin-4-aminer som antivirale midler

Also Published As

Publication number Publication date
CA2289219A1 (en) 1992-09-02
CZ178893A3 (en) 1995-10-18
AU673309B2 (en) 1996-10-31
EP0872478B1 (de) 2002-12-18
DK0872478T3 (da) 2003-03-31
WO1992015582A1 (en) 1992-09-17
EP0582581B1 (de) 1999-05-06
JPH06504789A (ja) 1994-06-02
IL114570A (en) 1996-10-31
SG70625A1 (en) 2000-02-22
NO933069D0 (no) 1993-08-27
NO933069L (no) 1993-11-01
DE69229114T2 (de) 1999-11-04
IL114570A0 (en) 1995-11-27
CA2289219C (en) 2003-05-20
ATE179711T1 (de) 1999-05-15
HU222111B1 (hu) 2003-04-28
HUT67026A (en) 1995-01-30
NO303729B1 (no) 1998-08-24
EP0872478A2 (de) 1998-10-21
EP0582581A1 (de) 1994-02-16
JP2955019B2 (ja) 1999-10-04
IL101110A0 (en) 1992-11-15
HU222250B1 (hu) 2003-05-28
AU658621B2 (en) 1995-04-27
HU9302457D0 (en) 1993-11-29
IE990988A1 (en) 2000-12-13
CA2104782A1 (en) 1992-09-02
PH31614A (en) 1999-01-12
UA32546C2 (uk) 2001-02-15
CA2104782C (en) 2001-08-07
DE69232878T2 (de) 2003-11-20
DE69229114D1 (de) 1999-06-10
SG46492A1 (en) 1998-02-20
HU211242A9 (en) 1995-11-28
EP0872478A3 (de) 1998-11-04
DK0582581T3 (da) 1999-11-08
IE920605A1 (en) 1992-09-09
AU2715795A (en) 1995-09-21
HU222247B1 (hu) 2003-05-28
AU1566992A (en) 1992-10-06
NZ241784A (en) 1995-06-27
ES2131070T3 (es) 1999-07-16
ES2186034T3 (es) 2003-05-01
HU9701083D0 (en) 1997-08-28
HU9701089D0 (en) 1997-08-28
HU222251B1 (hu) 2003-05-28
CZ285050B6 (cs) 1999-05-12
DE69232878D1 (de) 2003-01-30
HU9701084D0 (en) 1997-08-28
IL101110A (en) 1995-12-08

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