DK0872478T3 - Mellemprodukter til fremstilling af 1-substituerede, 2-substituerede 1H-imidazo[4,5-c]quinolin-4-aminer - Google Patents

Mellemprodukter til fremstilling af 1-substituerede, 2-substituerede 1H-imidazo[4,5-c]quinolin-4-aminer

Info

Publication number
DK0872478T3
DK0872478T3 DK98105754T DK98105754T DK0872478T3 DK 0872478 T3 DK0872478 T3 DK 0872478T3 DK 98105754 T DK98105754 T DK 98105754T DK 98105754 T DK98105754 T DK 98105754T DK 0872478 T3 DK0872478 T3 DK 0872478T3
Authority
DK
Denmark
Prior art keywords
substituted
imidazo
intermediates
amines
quinoline
Prior art date
Application number
DK98105754T
Other languages
English (en)
Inventor
John F Gerster
Stephen L Crooks
Kyle J Lindstrom
Original Assignee
Minnesota Mining & Mfg
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Minnesota Mining & Mfg filed Critical Minnesota Mining & Mfg
Application granted granted Critical
Publication of DK0872478T3 publication Critical patent/DK0872478T3/da

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
    • C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
    • C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D215/38—Nitrogen atoms
    • C07D215/42—Nitrogen atoms attached in position 4

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Virology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Quinoline Compounds (AREA)
  • Lubricants (AREA)
  • Emulsifying, Dispersing, Foam-Producing Or Wetting Agents (AREA)
DK98105754T 1991-03-01 1992-02-20 Mellemprodukter til fremstilling af 1-substituerede, 2-substituerede 1H-imidazo[4,5-c]quinolin-4-aminer DK0872478T3 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US66292691A 1991-03-01 1991-03-01
US68732691A 1991-04-18 1991-04-18

Publications (1)

Publication Number Publication Date
DK0872478T3 true DK0872478T3 (da) 2003-03-31

Family

ID=27098631

Family Applications (2)

Application Number Title Priority Date Filing Date
DK92906763T DK0582581T3 (da) 1991-03-01 1992-02-20 1,2-substituerede 1H-imidazo[4,5-c]quinolin-4-aminer
DK98105754T DK0872478T3 (da) 1991-03-01 1992-02-20 Mellemprodukter til fremstilling af 1-substituerede, 2-substituerede 1H-imidazo[4,5-c]quinolin-4-aminer

Family Applications Before (1)

Application Number Title Priority Date Filing Date
DK92906763T DK0582581T3 (da) 1991-03-01 1992-02-20 1,2-substituerede 1H-imidazo[4,5-c]quinolin-4-aminer

Country Status (18)

Country Link
EP (2) EP0582581B1 (da)
JP (1) JP2955019B2 (da)
AT (2) ATE229943T1 (da)
AU (2) AU658621B2 (da)
CA (2) CA2289219C (da)
CZ (1) CZ285050B6 (da)
DE (2) DE69232878T2 (da)
DK (2) DK0582581T3 (da)
ES (2) ES2186034T3 (da)
HU (5) HU222111B1 (da)
IE (1) IE920605A1 (da)
IL (2) IL114570A (da)
NO (1) NO303729B1 (da)
NZ (1) NZ241784A (da)
PH (1) PH31614A (da)
SG (2) SG46492A1 (da)
UA (1) UA32546C2 (da)
WO (1) WO1992015582A1 (da)

Families Citing this family (88)

* Cited by examiner, † Cited by third party
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US5266575A (en) * 1991-11-06 1993-11-30 Minnesota Mining And Manufacturing Company 2-ethyl 1H-imidazo[4,5-ciquinolin-4-amines
US5395937A (en) * 1993-01-29 1995-03-07 Minnesota Mining And Manufacturing Company Process for preparing quinoline amines
US5352784A (en) * 1993-07-15 1994-10-04 Minnesota Mining And Manufacturing Company Fused cycloalkylimidazopyridines
EP0708772B1 (en) * 1993-07-15 2000-08-23 Minnesota Mining And Manufacturing Company IMIDAZO [4,5-c]PYRIDIN-4-AMINES
US5648516A (en) * 1994-07-20 1997-07-15 Minnesota Mining And Manufacturing Company Fused cycloalkylimidazopyridines
US5482936A (en) * 1995-01-12 1996-01-09 Minnesota Mining And Manufacturing Company Imidazo[4,5-C]quinoline amines
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IL73534A (en) 1983-11-18 1990-12-23 Riker Laboratories Inc 1h-imidazo(4,5-c)quinoline-4-amines,their preparation and pharmaceutical compositions containing certain such compounds
CA1271477A (en) * 1983-11-18 1990-07-10 John F. Gerster 1h-imidazo[4,5-c]quinolin-4-amines
EP0385630B1 (en) * 1989-02-27 1996-11-27 Riker Laboratories, Inc. 1H-imidazo(4,5-c)Quinolin-4-amines as antivirals

Also Published As

Publication number Publication date
DE69229114T2 (de) 1999-11-04
AU658621B2 (en) 1995-04-27
HUT67026A (en) 1995-01-30
EP0872478A3 (en) 1998-11-04
NZ241784A (en) 1995-06-27
CA2104782A1 (en) 1992-09-02
ES2131070T3 (es) 1999-07-16
ATE229943T1 (de) 2003-01-15
CZ178893A3 (en) 1995-10-18
HU9701083D0 (en) 1997-08-28
HU222250B1 (hu) 2003-05-28
IL114570A0 (en) 1995-11-27
EP0872478A2 (en) 1998-10-21
WO1992015582A1 (en) 1992-09-17
NO933069L (no) 1993-11-01
JPH06504789A (ja) 1994-06-02
IE990988A1 (en) 2000-12-13
ATE179711T1 (de) 1999-05-15
DK0582581T3 (da) 1999-11-08
AU673309B2 (en) 1996-10-31
HU222111B1 (hu) 2003-04-28
EP0872478B1 (en) 2002-12-18
HU9701084D0 (en) 1997-08-28
CZ285050B6 (cs) 1999-05-12
PH31614A (en) 1999-01-12
UA32546C2 (uk) 2001-02-15
AU1566992A (en) 1992-10-06
DE69232878D1 (de) 2003-01-30
CA2289219C (en) 2003-05-20
EP0582581A1 (en) 1994-02-16
HU222247B1 (hu) 2003-05-28
HU211242A9 (en) 1995-11-28
IL101110A0 (en) 1992-11-15
AU2715795A (en) 1995-09-21
HU222251B1 (hu) 2003-05-28
HU9701089D0 (en) 1997-08-28
NO303729B1 (no) 1998-08-24
EP0582581B1 (en) 1999-05-06
JP2955019B2 (ja) 1999-10-04
IE920605A1 (en) 1992-09-09
HU9302457D0 (en) 1993-11-29
IL101110A (en) 1995-12-08
CA2289219A1 (en) 1992-09-02
IL114570A (en) 1996-10-31
NO933069D0 (no) 1993-08-27
DE69229114D1 (de) 1999-06-10
CA2104782C (en) 2001-08-07
SG70625A1 (en) 2000-02-22
ES2186034T3 (es) 2003-05-01
DE69232878T2 (de) 2003-11-20
SG46492A1 (en) 1998-02-20

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