ATE247656T1 - Pyrazolo(1,5-a)triazine als crf antagonisten - Google Patents
Pyrazolo(1,5-a)triazine als crf antagonistenInfo
- Publication number
- ATE247656T1 ATE247656T1 AT99930438T AT99930438T ATE247656T1 AT E247656 T1 ATE247656 T1 AT E247656T1 AT 99930438 T AT99930438 T AT 99930438T AT 99930438 T AT99930438 T AT 99930438T AT E247656 T1 ATE247656 T1 AT E247656T1
- Authority
- AT
- Austria
- Prior art keywords
- pyrazolo
- triazine
- crf antagonists
- crf
- antagonists
- Prior art date
Links
- 239000005557 antagonist Substances 0.000 title abstract 2
- JYEUMXHLPRZUAT-UHFFFAOYSA-N 1,2,3-triazine Chemical compound C1=CN=NN=C1 JYEUMXHLPRZUAT-UHFFFAOYSA-N 0.000 title 1
- 125000003342 alkenyl group Chemical group 0.000 abstract 1
- 125000000217 alkyl group Chemical group 0.000 abstract 1
- 125000000304 alkynyl group Chemical group 0.000 abstract 1
- 125000000753 cycloalkyl group Chemical group 0.000 abstract 1
- 150000003839 salts Chemical group 0.000 abstract 1
- 150000003918 triazines Chemical class 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US9020798P | 1998-06-22 | 1998-06-22 | |
| PCT/US1999/013870 WO1999067247A1 (en) | 1998-06-22 | 1999-06-18 | PYRAZOLO[1,5-a]TRIAZINE CORTICOTROPIN RELEASING FACTOR ANTAGONISTS |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ATE247656T1 true ATE247656T1 (de) | 2003-09-15 |
Family
ID=22221780
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AT99930438T ATE247656T1 (de) | 1998-06-22 | 1999-06-18 | Pyrazolo(1,5-a)triazine als crf antagonisten |
Country Status (8)
| Country | Link |
|---|---|
| US (1) | US6509338B1 (de) |
| EP (1) | EP1090005B1 (de) |
| AT (1) | ATE247656T1 (de) |
| AU (1) | AU4698199A (de) |
| CA (1) | CA2333633A1 (de) |
| DE (1) | DE69910574T2 (de) |
| ES (1) | ES2203152T3 (de) |
| WO (1) | WO1999067247A1 (de) |
Families Citing this family (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP1345941A1 (de) * | 2000-12-20 | 2003-09-24 | Societe De Conseils De Recherches Et D'applications Scientifiques (S.C.R.A.S.) | Cyclin-abhängige kinase (cdk) und glycogen synthase kinase-3 inhibitoren |
| KR20040034594A (ko) | 2001-01-26 | 2004-04-28 | 브리스톨-마이어스스퀴브컴파니 | 코르티코트로핀 방출 인자 억제제로서의 이미다졸릴 유도체 |
| FR2842809A1 (fr) * | 2002-07-26 | 2004-01-30 | Greenpharma Sas | NOUVELLES PYRAZOLO[1,5-a]-1,3,5-TRIAZINES SUBSTITUEES ET LEURS ANALOGUES, COMPOSITIONS PHARMACEUTIQUES LES CONTENANT, UTILISATION A TITRE DE MEDICAMENT ET PROCEDES POUR LEUR PREPARATION |
| FR2850653A1 (fr) * | 2003-02-04 | 2004-08-06 | Univ Pasteur | Derives de pyrazolotriazine, procede de preparation et utilisations |
| US7329658B2 (en) * | 2003-02-06 | 2008-02-12 | Pfizer Inc | Cannabinoid receptor ligands and uses thereof |
| AR047969A1 (es) | 2004-02-25 | 2006-03-15 | Schering Corp | Pirazolotriazinas como inhibidores de quinasa |
| US7723336B2 (en) * | 2005-09-22 | 2010-05-25 | Bristol-Myers Squibb Company | Fused heterocyclic compounds useful as kinase modulators |
| WO2011153359A1 (en) | 2010-06-04 | 2011-12-08 | Albany Molecular Research, Inc. | Glycine transporter-1 inhibitors, methods of making them, and uses thereof |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| PT778277E (pt) | 1995-12-08 | 2003-11-28 | Pfizer | Derivados heterociclicos substituidos como antagonistas do crf |
| HU229024B1 (en) | 1996-07-24 | 2013-07-29 | Bristol Myers Squibb Pharma Co | Azolo-pyridimidines, pharmaceutical compositions containing the same and use thereof |
| JP3621706B2 (ja) | 1996-08-28 | 2005-02-16 | ファイザー・インク | 置換された６，５―ヘテロ―二環式誘導体 |
-
1999
- 1999-06-14 US US09/333,160 patent/US6509338B1/en not_active Expired - Lifetime
- 1999-06-18 AT AT99930438T patent/ATE247656T1/de not_active IP Right Cessation
- 1999-06-18 ES ES99930438T patent/ES2203152T3/es not_active Expired - Lifetime
- 1999-06-18 CA CA002333633A patent/CA2333633A1/en not_active Abandoned
- 1999-06-18 DE DE69910574T patent/DE69910574T2/de not_active Expired - Fee Related
- 1999-06-18 EP EP99930438A patent/EP1090005B1/de not_active Expired - Lifetime
- 1999-06-18 AU AU46981/99A patent/AU4698199A/en not_active Abandoned
- 1999-06-18 WO PCT/US1999/013870 patent/WO1999067247A1/en not_active Ceased
Also Published As
| Publication number | Publication date |
|---|---|
| EP1090005B1 (de) | 2003-08-20 |
| WO1999067247A1 (en) | 1999-12-29 |
| ES2203152T3 (es) | 2004-04-01 |
| DE69910574T2 (de) | 2004-03-04 |
| DE69910574D1 (de) | 2003-09-25 |
| CA2333633A1 (en) | 1999-12-29 |
| AU4698199A (en) | 2000-01-10 |
| US6509338B1 (en) | 2003-01-21 |
| EP1090005A1 (de) | 2001-04-11 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| RER | Ceased as to paragraph 5 lit. 3 law introducing patent treaties |