ATE286058T1 - Thiazolpyrimidin-verbindungen, verfahren zu ihrer herstellung und ihre anwendung - Google Patents

Thiazolpyrimidin-verbindungen, verfahren zu ihrer herstellung und ihre anwendung

Info

Publication number: ATE286058T1
Authority: AT; Austria
Prior art keywords: compounds; thiazolpyrimidine; production; application; optionally substituted
Prior art date: 1999-01-28

Application number

AT00901914T

Other languages

English (en)

Inventor

Shigenori Ohkawa

Naoyuki Kanzaki

Seiji Miwatashi

Original Assignee

Takeda Pharmaceutical

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1999-01-28

Filing date

2000-01-27

Publication date

2005-01-15

2000-01-27 Application filed by Takeda Pharmaceutical filed Critical Takeda Pharmaceutical

2005-01-15 Application granted granted Critical

2005-01-15 Publication of ATE286058T1 publication Critical patent/ATE286058T1/de

Links

150000001875 compounds Chemical class 0.000 title abstract 2
102000008161 Adenosine A3 Receptor Human genes 0.000 abstract 1
108010060261 Adenosine A3 Receptor Proteins 0.000 abstract 1
230000008485 antagonism Effects 0.000 abstract 1
230000001747 exhibiting effect Effects 0.000 abstract 1
125000001997 phenyl group Chemical group [H]C1=C([H])C([H])=C(*)C([H])=C1[H] 0.000 abstract 1
150000003839 salts Chemical class 0.000 abstract 1
125000005750 substituted cyclic group Chemical group 0.000 abstract 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
- C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
- C07D513/04—Ortho-condensed systems
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/06—Antiasthmatics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Veterinary Medicine (AREA)
Medicinal Chemistry (AREA)
Pharmacology & Pharmacy (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
Bioinformatics & Cheminformatics (AREA)
Engineering & Computer Science (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Pulmonology (AREA)
Neurology (AREA)
Biomedical Technology (AREA)
Epidemiology (AREA)
Neurosurgery (AREA)
Cardiology (AREA)
Heart & Thoracic Surgery (AREA)
Hospice & Palliative Care (AREA)
Vascular Medicine (AREA)
Psychiatry (AREA)
Immunology (AREA)
Pain & Pain Management (AREA)
Rheumatology (AREA)
Urology & Nephrology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Plural Heterocyclic Compounds (AREA)
Thiazole And Isothizaole Compounds (AREA)

AT00901914T 1999-01-28 2000-01-27 Thiazolpyrimidin-verbindungen, verfahren zu ihrer herstellung und ihre anwendung ATE286058T1 (de)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
JP1982899		1999-01-28
PCT/JP2000/000395 WO2000044756A1 (en)	1999-01-28	2000-01-27	Thiazolopyrimidine compounds, process for the preparation of the same and uses thereof

Publications (1)

Publication Number	Publication Date
ATE286058T1 true ATE286058T1 (de)	2005-01-15

Family

ID=12010167

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
AT00901914T ATE286058T1 (de)	1999-01-28	2000-01-27	Thiazolpyrimidin-verbindungen, verfahren zu ihrer herstellung und ihre anwendung

Country Status (7)

Country	Link
US (1)	US6583146B1 (de)
EP (1)	EP1148059B1 (de)
AT (1)	ATE286058T1 (de)
AU (1)	AU2319000A (de)
CA (1)	CA2359011A1 (de)
DE (1)	DE60017084T2 (de)
WO (1)	WO2000044756A1 (de)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
AU2001290243A1 (en) *	2000-09-20	2002-04-02	Nikken Chemicals Co., Ltd.	Novel thiazole bicyclic compounds
WO2005026166A1 (en) *	2003-09-16	2005-03-24	'chemical Diversity Research Institute', Ltd.	Physiologically active composition, pharmaceutical composition, substituted 1,2-dihydro[2,7] naphthyridines, method for the production and use thereof

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US3919201A (en) *	1970-09-30	1975-11-11	Lilly Industries Ltd	2-({62 -Aminoacryloyl)iminobenzothiazolines
GB1582744A (en)	1976-06-04	1981-01-14	Gruenenthal Gmbh	7h-thiazolo (and 1,3,4-thiadiazolo-)(3,2-a) pyrimidin-7-one-5-carboxylic acids derivatives and medicaments therof
WO1997033879A1 (en) *	1996-03-15	1997-09-18	Merck & Co., Inc.	Compounds and methods for selectively inhibiting activation of the human a3 adenosine receptor

2000
- 2000-01-27 AT AT00901914T patent/ATE286058T1/de not_active IP Right Cessation
- 2000-01-27 CA CA002359011A patent/CA2359011A1/en not_active Abandoned
- 2000-01-27 WO PCT/JP2000/000395 patent/WO2000044756A1/ja not_active Ceased
- 2000-01-27 DE DE60017084T patent/DE60017084T2/de not_active Expired - Fee Related
- 2000-01-27 EP EP00901914A patent/EP1148059B1/de not_active Expired - Lifetime
- 2000-01-27 AU AU23190/00A patent/AU2319000A/en not_active Abandoned
- 2000-01-27 US US09/889,139 patent/US6583146B1/en not_active Expired - Fee Related

Also Published As

Publication number	Publication date
US6583146B1 (en)	2003-06-24
EP1148059B1 (de)	2004-12-29
EP1148059A1 (de)	2001-10-24
WO2000044756A1 (en)	2000-08-03
EP1148059A4 (de)	2002-04-10
AU2319000A (en)	2000-08-18
CA2359011A1 (en)	2000-08-03
DE60017084D1 (de)	2005-02-03
DE60017084T2 (de)	2005-12-22

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Legal Events

Date	Code	Title	Description
2005-06-15	RER	Ceased as to paragraph 5 lit. 3 law introducing patent treaties