ATE289812T1 - Azolylcarbynol-derivative von aryl (oder heteroaryl) zur behandlung von atemwegserkrankungen - Google Patents

Azolylcarbynol-derivative von aryl (oder heteroaryl) zur behandlung von atemwegserkrankungen

Info

Publication number: ATE289812T1
Authority: AT; Austria
Prior art keywords: heteroaryl; aryl; treatment; derivatives; azolylcarbynol
Prior art date: 2001-04-06

Application number

AT02714232T

Other languages

English (en)

Inventor

Ramon Merce-Vidal

Blas Andaluz-Matero

Jordi Frigola-Constansa

Original Assignee

Esteve Labor Dr

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2001-04-06

Filing date

2002-03-21

Publication date

2005-03-15

2002-03-21 Application filed by Esteve Labor Dr filed Critical Esteve Labor Dr

2005-03-15 Application granted granted Critical

2005-03-15 Publication of ATE289812T1 publication Critical patent/ATE289812T1/de

Links

201000010099 disease Diseases 0.000 title 1
208000037265 diseases, disorders, signs and symptoms Diseases 0.000 title 1
230000000241 respiratory effect Effects 0.000 title 1
239000003814 drug Substances 0.000 abstract 2
KAESVJOAVNADME-UHFFFAOYSA-N 1H-pyrrole Natural products C=1C=CNC=1 KAESVJOAVNADME-UHFFFAOYSA-N 0.000 abstract 1
208000006545 Chronic Obstructive Pulmonary Disease Diseases 0.000 abstract 1
206010011224 Cough Diseases 0.000 abstract 1
206010039085 Rhinitis allergic Diseases 0.000 abstract 1
CIUQDSCDWFSTQR-UHFFFAOYSA-N [C]1=CC=CC=C1 Chemical group [C]1=CC=CC=C1 CIUQDSCDWFSTQR-UHFFFAOYSA-N 0.000 abstract 1
125000000217 alkyl group Chemical group 0.000 abstract 1
201000009961 allergic asthma Diseases 0.000 abstract 1
201000010105 allergic rhinitis Diseases 0.000 abstract 1
125000003118 aryl group Chemical group 0.000 abstract 1
208000006673 asthma Diseases 0.000 abstract 1
150000003851 azoles Chemical class 0.000 abstract 1
206010006451 bronchitis Diseases 0.000 abstract 1
125000004985 dialkyl amino alkyl group Chemical group 0.000 abstract 1
229940079593 drug Drugs 0.000 abstract 1
125000001072 heteroaryl group Chemical group 0.000 abstract 1
125000004435 hydrogen atom Chemical group [H]* 0.000 abstract 1
150000003839 salts Chemical class 0.000 abstract 1
125000001424 substituent group Chemical group 0.000 abstract 1

Classifications

- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/415—1,2-Diazoles
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/38—Heterocyclic compounds having sulfur as a ring hetero atom
- A61K31/381—Heterocyclic compounds having sulfur as a ring hetero atom having five-membered rings
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/02—Nasal agents, e.g. decongestants
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/06—Antiasthmatics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/08—Bronchodilators
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/14—Antitussive agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents

Landscapes

Health & Medical Sciences (AREA)
Public Health (AREA)
Animal Behavior & Ethology (AREA)
Veterinary Medicine (AREA)
General Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Pharmacology & Pharmacy (AREA)
Life Sciences & Earth Sciences (AREA)
Medicinal Chemistry (AREA)
Chemical Kinetics & Catalysis (AREA)
Engineering & Computer Science (AREA)
Organic Chemistry (AREA)
General Chemical & Material Sciences (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Pulmonology (AREA)
Bioinformatics & Cheminformatics (AREA)
Epidemiology (AREA)
Immunology (AREA)
Otolaryngology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

AT02714232T 2001-04-06 2002-03-21 Azolylcarbynol-derivative von aryl (oder heteroaryl) zur behandlung von atemwegserkrankungen ATE289812T1 (de)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
ES200100817A ES2174756B2 (es)	2001-04-06	2001-04-06	Derivados de aril (o heteroaril) azolilcarbinoles para el tratamiento de enfermedades respiratorias.
PCT/ES2002/000136 WO2002080908A1 (es)	2001-04-06	2002-03-21	Derivados de aril (o heteroaril) azolilcarbinoles para el tratamiento de enfermedades respiratorias

Publications (1)

Publication Number	Publication Date
ATE289812T1 true ATE289812T1 (de)	2005-03-15

Family

ID=8497368

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
AT02714232T ATE289812T1 (de)	2001-04-06	2002-03-21	Azolylcarbynol-derivative von aryl (oder heteroaryl) zur behandlung von atemwegserkrankungen

Country Status (22)

Country	Link
US (1)	US20040142994A1 (de)
EP (1)	EP1384476B1 (de)
JP (1)	JP2004531511A (de)
KR (1)	KR20040025913A (de)
CN (1)	CN1230165C (de)
AT (1)	ATE289812T1 (de)
AU (1)	AU2002246151B2 (de)
BR (1)	BR0208807A (de)
CA (1)	CA2443015A1 (de)
DE (1)	DE60203106T2 (de)
DK (1)	DK1384476T3 (de)
ES (2)	ES2174756B2 (de)
HU (1)	HUP0400925A3 (de)
IL (1)	IL158268A0 (de)
MX (1)	MXPA03009125A (de)
NO (1)	NO20034471L (de)
NZ (1)	NZ529303A (de)
PL (1)	PL365251A1 (de)
PT (1)	PT1384476E (de)
RU (1)	RU2294198C2 (de)
WO (1)	WO2002080908A1 (de)
ZA (1)	ZA200308630B (de)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
DE10335566A1 (de) *	2003-07-31	2005-02-24	Grünenthal GmbH	Arzneimittel enthaltend Derivate von Aryl( oder Heteroaryl)azolylcarbinolen
EP1584335A3 (de) *	2004-04-05	2006-02-22	Laboratorios Del Dr. Esteve, S.A.	Zusammensetzung aus Aktiva mit einer Carbinolverbindung und einem Opioid
ES2244326B1 (es) *	2004-04-05	2007-02-16	Laboratorios Del Dr. Esteve, S.A.	Combinacion de substancias activas.
WO2006010627A1 (en) *	2004-07-30	2006-02-02	Laboratorios Del Dr. Esteve, S.A.	Aryl (or heteroaryl) azolylcarbinols
EP1632227A1 (de) *	2004-09-07	2006-03-08	Laboratorios del Dr. Esteve S.A.	Aryl- (oder Heteroaryl-) Azolcarbinole (insbesondere Cizolirtin Citrate) für die Behandlung von Opioid Abhängigkeit
EP1820502A1 (de) *	2006-02-10	2007-08-22	Laboratorios Del Dr. Esteve, S.A.	Wirkstoffzusammensetzungen enthaltend Azolycarbinolderivate
US20100291151A1 (en) *	2009-04-21	2010-11-18	Auspex Pharmaceuticals, Inc.	1-methylpyrazole modulators of substance p, calcitonin gene-related peptide, adrenergic receptor, and/or 5-ht receptor

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
ES2150353B1 (es) *	1998-04-15	2001-07-01	Esteve Labor Dr	Tienilazolilalcoxietanaminas, su preparacion y su aplicacion como medicamentos.
ES2137136B1 (es) *	1998-05-18	2000-07-01	Esteve Labor Dr	Empleo de derivados de aril (o heteroaril) azolilcarbinoles en la elaboracion de un medicamento para el tratamiento de la inflamacion neurogenica.
ES2150378B1 (es) *	1998-08-07	2001-07-01	Esteve Labor Dr	Empleo de derivados de aril(o heteroaril)azolilcarbinoles en la elaboracion de un medicamento para el tratamiento de los trastornos mediados por un exceso de substancia p.

2001
- 2001-04-06 ES ES200100817A patent/ES2174756B2/es not_active Expired - Fee Related
2002
- 2002-03-21 CN CNB028098943A patent/CN1230165C/zh not_active Expired - Fee Related
- 2002-03-21 NZ NZ529303A patent/NZ529303A/en unknown
- 2002-03-21 DE DE60203106T patent/DE60203106T2/de not_active Expired - Fee Related
- 2002-03-21 MX MXPA03009125A patent/MXPA03009125A/es active IP Right Grant
- 2002-03-21 DK DK02714232T patent/DK1384476T3/da active
- 2002-03-21 US US10/474,232 patent/US20040142994A1/en not_active Abandoned
- 2002-03-21 AT AT02714232T patent/ATE289812T1/de not_active IP Right Cessation
- 2002-03-21 PL PL02365251A patent/PL365251A1/xx not_active Application Discontinuation
- 2002-03-21 ES ES02714232T patent/ES2236497T3/es not_active Expired - Lifetime
- 2002-03-21 WO PCT/ES2002/000136 patent/WO2002080908A1/es not_active Ceased
- 2002-03-21 AU AU2002246151A patent/AU2002246151B2/en not_active Ceased
- 2002-03-21 RU RU2003132456/15A patent/RU2294198C2/ru not_active IP Right Cessation
- 2002-03-21 BR BR0208807-0A patent/BR0208807A/pt not_active IP Right Cessation
- 2002-03-21 JP JP2002578947A patent/JP2004531511A/ja not_active Withdrawn
- 2002-03-21 CA CA002443015A patent/CA2443015A1/en not_active Abandoned
- 2002-03-21 HU HU0400925A patent/HUP0400925A3/hu unknown
- 2002-03-21 IL IL15826802A patent/IL158268A0/xx unknown
- 2002-03-21 KR KR10-2003-7013063A patent/KR20040025913A/ko not_active Ceased
- 2002-03-21 PT PT02714232T patent/PT1384476E/pt unknown
- 2002-03-21 EP EP02714232A patent/EP1384476B1/de not_active Expired - Lifetime
2003
- 2003-10-06 NO NO20034471A patent/NO20034471L/no not_active Application Discontinuation
- 2003-11-05 ZA ZA200308630A patent/ZA200308630B/en unknown

Also Published As

Publication number	Publication date
WO2002080908A1 (es)	2002-10-17
ZA200308630B (en)	2004-11-05
US20040142994A1 (en)	2004-07-22
NO20034471L (no)	2003-12-03
IL158268A0 (en)	2004-05-12
DE60203106D1 (de)	2005-04-07
ES2174756A1 (es)	2002-11-01
NO20034471D0 (no)	2003-10-06
RU2003132456A (ru)	2005-04-10
CN1535147A (zh)	2004-10-06
KR20040025913A (ko)	2004-03-26
PT1384476E (pt)	2005-05-31
BR0208807A (pt)	2004-07-13
ES2174756B2 (es)	2003-11-16
EP1384476B1 (de)	2005-03-02
DK1384476T3 (da)	2005-05-30
HUP0400925A2 (hu)	2004-07-28
CA2443015A1 (en)	2002-10-17
HUP0400925A3 (en)	2004-10-28
RU2294198C2 (ru)	2007-02-27
EP1384476A1 (de)	2004-01-28
CN1230165C (zh)	2005-12-07
AU2002246151B2 (en)	2007-05-31
DE60203106T2 (de)	2006-04-13
ES2236497T3 (es)	2005-07-16
NZ529303A (en)	2005-06-24
PL365251A1 (en)	2004-12-27
AU2002246151C1 (en)	2002-10-21
JP2004531511A (ja)	2004-10-14
MXPA03009125A (es)	2005-04-11

Legal Events

Date

Code

Title

Description

2005-09-15

UEP

Publication of translation of european patent specification

Ref document number: 1384476

Country of ref document: EP

2008-12-15

REN

Ceased due to non-payment of the annual fee

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