ATE29215T1 - Diaethylpropionpraeparate mit verzoegerter wirkung. - Google Patents

Diaethylpropionpraeparate mit verzoegerter wirkung.

Info

Publication number: ATE29215T1
Authority: AT; Austria
Prior art keywords: diaethylpropionic; preparations; delayed; acting; capsules
Prior art date: 1982-05-20

Application number

AT83104832T

Other languages

English (en)

Inventor

Eugene L Walters

Original Assignee

Merrell Dow Pharma

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1982-05-20

Filing date

1983-05-17

Publication date

1987-09-15

1983-05-17 Application filed by Merrell Dow Pharma filed Critical Merrell Dow Pharma

1987-09-15 Application granted granted Critical

1987-09-15 Publication of ATE29215T1 publication Critical patent/ATE29215T1/de

Links

238000002360 preparation method Methods 0.000 title 1
XHZFHAGIQPYPAM-UHFFFAOYSA-N 3-hydroxy-1-[(4-methoxyphenyl)methyl]piperidin-2-one Chemical compound C1=CC(OC)=CC=C1CN1C(=O)C(O)CCC1 XHZFHAGIQPYPAM-UHFFFAOYSA-N 0.000 abstract 1
229940125709 anorectic agent Drugs 0.000 abstract 1
239000002830 appetite depressant Substances 0.000 abstract 1
239000002775 capsule Substances 0.000 abstract 1
229960005259 diethylpropion hydrochloride Drugs 0.000 abstract 1
238000009472 formulation Methods 0.000 abstract 1
239000000203 mixture Substances 0.000 abstract 1
238000013268 sustained release Methods 0.000 abstract 1
239000012730 sustained-release form Substances 0.000 abstract 1

Classifications

- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/13—Amines
- A61K31/135—Amines having aromatic rings, e.g. ketamine, nortriptyline
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
- A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
- A61K9/1605—Excipients; Inactive ingredients
- A61K9/1617—Organic compounds, e.g. phospholipids, fats
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
- A61K9/4841—Filling excipients; Inactive ingredients
- A61K9/4858—Organic compounds
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
- A61K9/4841—Filling excipients; Inactive ingredients
- A61K9/4866—Organic macromolecular compounds
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/04—Anorexiants; Antiobesity agents

Landscapes

Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
Public Health (AREA)
Chemical & Material Sciences (AREA)
Veterinary Medicine (AREA)
Medicinal Chemistry (AREA)
General Health & Medical Sciences (AREA)
Animal Behavior & Ethology (AREA)
Pharmacology & Pharmacy (AREA)
Epidemiology (AREA)
Bioinformatics & Cheminformatics (AREA)
Engineering & Computer Science (AREA)
Biophysics (AREA)
Molecular Biology (AREA)
Obesity (AREA)
Organic Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
General Chemical & Material Sciences (AREA)
Chemical Kinetics & Catalysis (AREA)
Hematology (AREA)
Diabetes (AREA)
Child & Adolescent Psychology (AREA)
Medicinal Preparation (AREA)
Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)

AT83104832T 1982-05-20 1983-05-17 Diaethylpropionpraeparate mit verzoegerter wirkung. ATE29215T1 (de)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
US06/379,848 US4421736A (en)	1982-05-20	1982-05-20	Sustained release diethylpropion compositions
EP83104832A EP0095123B1 (de)	1982-05-20	1983-05-17	Diäthylpropionpräparate mit verzögerter Wirkung

Publications (1)

Publication Number	Publication Date
ATE29215T1 true ATE29215T1 (de)	1987-09-15

Family

ID=23498964

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
AT83104832T ATE29215T1 (de)	1982-05-20	1983-05-17	Diaethylpropionpraeparate mit verzoegerter wirkung.

Country Status (11)

Country	Link
US (1)	US4421736A (de)
EP (1)	EP0095123B1 (de)
JP (1)	JPS58210008A (de)
AT (1)	ATE29215T1 (de)
AU (1)	AU550992B2 (de)
DE (1)	DE3373272D1 (de)
IE (1)	IE55115B1 (de)
IL (1)	IL68703A (de)
NZ (1)	NZ204263A (de)
PH (1)	PH19295A (de)
ZA (1)	ZA833489B (de)

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US20040162351A1 (en) *	2002-12-11	2004-08-19	Gallop Mark A.	Orally administered dosage forms of fused GABA analog prodrugs having reduced toxicity
KR20050119676A (ko) *	2003-03-31	2005-12-21	제노포트 인코포레이티드	가바 유사체의 프로드러그를 사용한 열성 홍조의 치료 또는예방
EP2354120A1 (de)	2003-08-20	2011-08-10	XenoPort, Inc.	Synthese von Acyloxyalkylcarbamat-Prodrugs und Zwischenprodukten davon
BRPI0413756A (pt) *	2003-08-20	2006-10-31	Xenoport Inc	composto, métodos para tratar ou evitar espasticidade ou um sintoma de espasticidade, doença de refluxo gastro-esofágico, vìcio em droga, vìcio em ou abuso de álcool, ou vìcio em ou abuso de nicotina, e tosse ou êmese em um paciente, e, composição farmacêutica
KR20060119971A (ko) *	2003-09-11	2006-11-24	제노포트 인코포레이티드	Ｇａｂａ 유사체의 전구약물을 이용한 요실금의 치료및/또는 예방
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US20060128676A1 (en) *	2004-07-13	2006-06-15	Pharmacofore, Inc.	Compositions of nicotinic agonists and therapeutic agents and methods for treating or preventing diseases or pain
US7566738B2 (en) *	2004-11-03	2009-07-28	Xenoport, Inc.	Acyloxyalkyl carbamate prodrugs of sulfinic acids, methods of synthesis, and use
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MX2007005306A (es) *	2004-11-04	2007-06-11	Xenoport Inc	Formas de dosis oral de liberacion sostenida de la prodroga gabapentina.
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ZA200711123B (en)	2005-06-27	2009-08-26	Biovail Lab Int Srl	Modified-release formulations of a bupropion salt
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US20080075768A1 (en) *	2006-07-21	2008-03-27	Vaughn Jason M	Hydrophobic opioid abuse deterrent delivery system using opioid antagonists
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US20080161393A1 (en) *	2006-12-08	2008-07-03	Barrett Ronald W	Use of prodrugs of GABA analogs for treating disease
US20090246276A1 (en)	2008-01-28	2009-10-01	Graham Jackson	Pharmaceutical Compositions
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DK2621282T3 (da)	2010-09-28	2020-05-04	Univ California	Gaba-agonister i behandlingen af forstyrrelser forbundet med metabolisk syndrom og gaba-kombinationer i behandling eller profylakse af type i diabetes
AU2016332071B2 (en)	2015-10-01	2019-04-18	Elysium Therapeutics, Inc.	Polysubunit opioid prodrugs resistant to overdose and abuse
US10335406B2 (en)	2015-10-01	2019-07-02	Elysium Therapeutics, Inc.	Opioid compositions resistant to overdose and abuse
EP3595663A4 (de)	2017-03-17	2021-01-13	Elysium Therapeutics, Inc.	Mehrfachuntereinheit-opioid-prodrugs mit resistenz gegen überdosierung und missbrauch
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1982
- 1982-05-20 US US06/379,848 patent/US4421736A/en not_active Expired - Lifetime
1983
- 1983-05-16 ZA ZA833489A patent/ZA833489B/xx unknown
- 1983-05-16 IL IL68703A patent/IL68703A/xx not_active IP Right Cessation
- 1983-05-16 JP JP58084292A patent/JPS58210008A/ja active Pending
- 1983-05-16 PH PH28908A patent/PH19295A/en unknown
- 1983-05-17 NZ NZ204263A patent/NZ204263A/en unknown
- 1983-05-17 AT AT83104832T patent/ATE29215T1/de not_active IP Right Cessation
- 1983-05-17 EP EP83104832A patent/EP0095123B1/de not_active Expired
- 1983-05-17 DE DE8383104832T patent/DE3373272D1/de not_active Expired
- 1983-05-17 AU AU14617/83A patent/AU550992B2/en not_active Expired
- 1983-05-18 IE IE1172/83A patent/IE55115B1/en not_active IP Right Cessation

Also Published As

Publication number	Publication date
AU550992B2 (en)	1986-04-10
EP0095123B1 (de)	1987-09-02
JPS58210008A (ja)	1983-12-07
ZA833489B (en)	1984-02-29
IL68703A (en)	1986-09-30
DE3373272D1 (en)	1987-10-08
PH19295A (en)	1986-03-05
IE55115B1 (en)	1990-06-06
EP0095123A2 (de)	1983-11-30
US4421736A (en)	1983-12-20
IE831172L (en)	1983-11-20
AU1461783A (en)	1983-11-24
EP0095123A3 (en)	1984-12-12
NZ204263A (en)	1986-02-21
IL68703A0 (en)	1983-09-30

Legal Events

Date	Code	Title	Description
1988-01-15	UEP	Publication of translation of european patent specification
2003-08-15	EELA	Cancelled due to lapse of time

Publication	Publication Date	Title
ATE29215T1 (de)	1987-09-15	Diaethylpropionpraeparate mit verzoegerter wirkung.
ES519423A0 (es)	1985-04-16	Procedimiento para preparar 9-(1 o 3-monoaciloxi-o 1,3-diaciloxi-2-propoximetil)-purinas substituidas en calidad de agentes antiviricos.
MX9203428A (es)	1992-07-01	Bifosfonatos activos farmacologicamente, procedimiento para su preparacion y composiciones farmaceuticas de los mismos.
DE69007650D1 (de)	1994-05-05	Ionomer-Zusammensetzung.
DE69014519D1 (de)	1995-01-12	Ionomer-Zusammensetzung.
TR199800077T1 (xx)	1998-05-21	Kontroll� ��z�len paroksetin terkipleri.
SE421412B (sv)	1981-12-21	2',4-diklor-4'-bensoylureido-difenyletrar till anvendning som insekticider
DE3887839D1 (de)	1994-03-24	Trennmittelzusammensetzung.
TR21983A (tr)	1987-02-06	N-fenilpirazol muestaklari,bunlari ihtiva eden terkipler ve bunlarin herbisid olarak kullanilmasi
FI802488A7 (fi)	1981-01-01	Antimykotiska aineita, jotka vapauttavat enemmän vaikutusaineita.
ES523243A0 (es)	1985-04-01	"procedimiento para preparar derivados de 1,4-dihidropiridina".
FI891364A0 (fi)	1989-03-22	Fast, vattenfri raney-katalysatordispersion.
DE59000222D1 (de)	1992-09-03	Vorderbacken.
ATE36455T1 (de)	1988-09-15	Pharmazeutische zusammensetzungen.
IT8323378A0 (it)	1983-10-20	Sedia da lavoro.
TR21806A (tr)	1985-07-19	Feniluereler,hazirlanmalarina mahsus usueller ve bunlarin herbisidler olarak kullanimi
SE7713700L (sv)	1978-06-07	2-substituerade-1-(omega-aminoalkoxi)bensener
DE69017678D1 (de)	1995-04-13	Verbesserte lösbare schnellkupplung.
ES532109A0 (es)	1985-06-16	Procedimiento para preparar 9-(1 o 3-monoaciloxi-o 1,3-diaciloxi-2-propoximetil)-purinas substituidas en calidad de agentes antiviricos.
ES1015137Y (es)	1992-01-01	Repeladora perfeccionada para pepita de almendra.
MA19859A1 (fr)	1984-04-01	Formulations fongicides .
IT7920991A0 (it)	1979-03-15	Derivato isoindolinico, processo per la sua preparazione e composizioni terapeutiche che lo comprendono come principio attivo.
FI834194L (fi)	1984-05-18	Preparat foer munvaord.
ES264088Y (es)	1983-05-16	"conjunto bastidor-colgador desplazable, multiexpositor, perfeccionado".
ES264458Y (es)	1983-05-16	"trituradora desbrozadora perfeccionada".