ATE293101T1 - Piperidine zur verwendung als orexin rezeptor antagonisten - Google Patents

Piperidine zur verwendung als orexin rezeptor antagonisten

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Publication number
ATE293101T1
ATE293101T1 AT01951591T AT01951591T ATE293101T1 AT E293101 T1 ATE293101 T1 AT E293101T1 AT 01951591 T AT01951591 T AT 01951591T AT 01951591 T AT01951591 T AT 01951591T AT E293101 T1 ATE293101 T1 AT E293101T1
Authority
AT
Austria
Prior art keywords
optionally substituted
phenyl
heteroatoms selected
heteroaryl group
group containing
Prior art date
Application number
AT01951591T
Other languages
English (en)
Inventor
Clive Leslie Branch
Christopher Norbert Johnson
Geoffrey Stemp
Kevin Thewlis
Original Assignee
Smithkline Beecham Plc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GB0014823A external-priority patent/GB0014823D0/en
Priority claimed from GB0027704A external-priority patent/GB0027704D0/en
Application filed by Smithkline Beecham Plc filed Critical Smithkline Beecham Plc
Application granted granted Critical
Publication of ATE293101T1 publication Critical patent/ATE293101T1/de

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    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
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    • C07D211/18—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms
    • C07D211/26—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms with hydrocarbon radicals, substituted by nitrogen atoms
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AT01951591T 2000-06-16 2001-06-13 Piperidine zur verwendung als orexin rezeptor antagonisten ATE293101T1 (de)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GB0014823A GB0014823D0 (en) 2000-06-16 2000-06-16 Compounds
GB0027704A GB0027704D0 (en) 2000-11-11 2000-11-11 Compounds
PCT/EP2001/006752 WO2001096302A1 (en) 2000-06-16 2001-06-13 Piperidines for use as orexin receptor antagonists

Publications (1)

Publication Number Publication Date
ATE293101T1 true ATE293101T1 (de) 2005-04-15

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Family Applications (1)

Application Number Title Priority Date Filing Date
AT01951591T ATE293101T1 (de) 2000-06-16 2001-06-13 Piperidine zur verwendung als orexin rezeptor antagonisten

Country Status (10)

Country Link
US (1) US6677354B2 (de)
EP (1) EP1289955B1 (de)
JP (1) JP4611608B2 (de)
AT (1) ATE293101T1 (de)
AU (1) AU2001272476A1 (de)
CA (1) CA2450922C (de)
DE (1) DE60110066T2 (de)
ES (1) ES2238458T3 (de)
PT (1) PT1289955E (de)
WO (1) WO2001096302A1 (de)

Families Citing this family (139)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU2002224885A1 (en) * 2000-11-28 2002-06-11 Smithkline Beecham Plc Morpholine derivatives as antagonists of orexin receptors
EP1435955A2 (de) * 2001-05-05 2004-07-14 SmithKline Beecham P.L.C. N-aroyl-zyklisches amin-derivat als orexin-rezeptor-antagonisten
MXPA03010129A (es) * 2001-05-05 2004-03-10 Smithkline Beecham Plc N-aroilaminas-ciclicas.
GB0115862D0 (en) * 2001-06-28 2001-08-22 Smithkline Beecham Plc Compounds
US7470710B2 (en) * 2001-06-28 2008-12-30 Smithkline Beecham P.L.C. N-aroyl cyclic amine derivatives as orexin receptor antagonists
GB0124463D0 (en) * 2001-10-11 2001-12-05 Smithkline Beecham Plc Compounds
GB0126292D0 (en) * 2001-11-01 2002-01-02 Smithkline Beecham Plc Compounds
GB0127145D0 (en) * 2001-11-10 2002-01-02 Smithkline Beecham Compounds
GB0130335D0 (en) * 2001-12-19 2002-02-06 Smithkline Beecham Plc Compounds
US7105526B2 (en) 2002-06-28 2006-09-12 Banyu Pharmaceuticals Co., Ltd. Benzimidazole derivatives
ES2278197T3 (es) 2002-07-09 2007-08-01 Actelion Pharmaceuticals Ltd. Derivados de 7,8,9,10-tetrahidro-6h-azepino, 6,7,8,9-tetrahidro-pirido y 2,3-dihidro-2h-pirrolo(1,2-b)-quinazolinona.
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