ATE335753T1 - Glucopyranosyloxybenzylbenzol derivate und medizinische zusammensetzungen, die diese verbindungen enthalten - Google Patents

Glucopyranosyloxybenzylbenzol derivate und medizinische zusammensetzungen, die diese verbindungen enthalten

Info

Publication number
ATE335753T1
ATE335753T1 AT01970186T AT01970186T ATE335753T1 AT E335753 T1 ATE335753 T1 AT E335753T1 AT 01970186 T AT01970186 T AT 01970186T AT 01970186 T AT01970186 T AT 01970186T AT E335753 T1 ATE335753 T1 AT E335753T1
Authority
AT
Austria
Prior art keywords
compounds
compositions containing
medicinal compositions
glucopyranosyloxybenzylbenzene derivatives
glucopyranosyloxybenzylbenzene
Prior art date
Application number
AT01970186T
Other languages
English (en)
Inventor
Hideki Fujikura
Nobuhiko Fushimi
Toshihiro Nishimura
Kazuya Tatani
Masayuki Isaji
Original Assignee
Kissei Pharmaceutical
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Kissei Pharmaceutical filed Critical Kissei Pharmaceutical
Application granted granted Critical
Publication of ATE335753T1 publication Critical patent/ATE335753T1/de

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H15/00—Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
    • C07H15/20—Carbocyclic rings
    • C07H15/203—Monocyclic carbocyclic rings other than cyclohexane rings; Bicyclic carbocyclic ring systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/70—Carbohydrates; Sugars; Derivatives thereof
    • A61K31/7028—Compounds having saccharide radicals attached to non-saccharide compounds by glycosidic linkages
    • A61K31/7034—Compounds having saccharide radicals attached to non-saccharide compounds by glycosidic linkages attached to a carbocyclic compound, e.g. phloridzin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/04—Anorexiants; Antiobesity agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Diabetes (AREA)
  • Molecular Biology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Biotechnology (AREA)
  • Obesity (AREA)
  • Biochemistry (AREA)
  • Hematology (AREA)
  • Genetics & Genomics (AREA)
  • Epidemiology (AREA)
  • Endocrinology (AREA)
  • Child & Adolescent Psychology (AREA)
  • Emergency Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
AT01970186T 2000-09-29 2001-09-21 Glucopyranosyloxybenzylbenzol derivate und medizinische zusammensetzungen, die diese verbindungen enthalten ATE335753T1 (de)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP2000301523 2000-09-29

Publications (1)

Publication Number Publication Date
ATE335753T1 true ATE335753T1 (de) 2006-09-15

Family

ID=18783054

Family Applications (1)

Application Number Title Priority Date Filing Date
AT01970186T ATE335753T1 (de) 2000-09-29 2001-09-21 Glucopyranosyloxybenzylbenzol derivate und medizinische zusammensetzungen, die diese verbindungen enthalten

Country Status (32)

Country Link
US (2) US6872706B2 (de)
EP (1) EP1329456B1 (de)
JP (1) JP3798375B2 (de)
KR (1) KR100647204B1 (de)
CN (1) CN1293087C (de)
AR (1) AR030816A1 (de)
AT (1) ATE335753T1 (de)
AU (2) AU9025701A (de)
BG (1) BG66015B1 (de)
BR (1) BR0114310A (de)
CA (1) CA2423568C (de)
CY (1) CY1106076T1 (de)
CZ (1) CZ303544B6 (de)
DE (1) DE60122193T2 (de)
DK (1) DK1329456T3 (de)
EA (1) EA005994B1 (de)
ES (1) ES2269456T3 (de)
HU (1) HUP0301178A3 (de)
IL (2) IL155071A0 (de)
MX (1) MXPA03002779A (de)
MY (1) MY129023A (de)
NO (1) NO327182B1 (de)
NZ (1) NZ524917A (de)
PE (1) PE20020476A1 (de)
PL (1) PL205607B1 (de)
PT (1) PT1329456E (de)
SI (1) SI1329456T1 (de)
SK (1) SK287811B6 (de)
TW (1) TWI284641B (de)
UA (1) UA73606C2 (de)
WO (1) WO2002028872A1 (de)
ZA (1) ZA200302283B (de)

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JP5073948B2 (ja) * 2005-01-31 2012-11-14 田辺三菱製薬株式会社 医薬組成物
JP5264183B2 (ja) * 2005-02-23 2013-08-14 ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング グルコピラノシル置換（（ヘテロ）アリールエチニル−ベンジル）−ベンゼン誘導体及びナトリウム依存性グルコース共輸送体２（ｓｇｌｔ２）インヒビターとしてのそれらの使用
WO2006108842A1 (en) * 2005-04-15 2006-10-19 Boehringer Ingelheim International Gmbh Glucopyranosyl-substituted (heteroaryloxy-benzyl)-benzene derivatives as sglt inhibitors
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JP5330260B2 (ja) 2006-12-06 2013-10-30 スミスクライン ビーチャム コーポレーション 二環式化合物ならびに抗糖尿病薬としての使用
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Also Published As

Publication number Publication date
TWI284641B (en) 2007-08-01
IL155071A (en) 2010-04-15
SK3342003A3 (en) 2003-08-05
AR030816A1 (es) 2003-09-03
IL155071A0 (en) 2003-10-31
CN1466590A (zh) 2004-01-07
BR0114310A (pt) 2003-10-14
SI1329456T1 (sl) 2006-12-31
PE20020476A1 (es) 2002-07-04
SK287811B6 (sk) 2011-10-04
PT1329456E (pt) 2006-12-29
EP1329456A4 (de) 2005-03-30
EP1329456B1 (de) 2006-08-09
PL362177A1 (en) 2004-10-18
BG107674A (bg) 2004-01-30
CZ303544B6 (cs) 2012-11-28
CA2423568A1 (en) 2002-04-11
DK1329456T3 (da) 2006-12-04
MXPA03002779A (es) 2004-05-04
MY129023A (en) 2007-03-30
AU9025701A (en) 2002-04-15
BG66015B1 (bg) 2010-10-29
US20040018998A1 (en) 2004-01-29
KR20030036867A (ko) 2003-05-09
CY1106076T1 (el) 2011-06-08
DE60122193D1 (de) 2006-09-21
NO20031407D0 (no) 2003-03-27
EP1329456A1 (de) 2003-07-23
US6872706B2 (en) 2005-03-29
ES2269456T3 (es) 2007-04-01
EA200300316A1 (ru) 2003-08-28
AU2001290257B2 (en) 2007-08-30
EA005994B1 (ru) 2005-08-25
US20050065098A1 (en) 2005-03-24
PL205607B1 (pl) 2010-05-31
NO327182B1 (no) 2009-05-04
NZ524917A (en) 2005-01-28
KR100647204B1 (ko) 2006-11-17
HUP0301178A2 (hu) 2003-11-28
JPWO2002028872A1 (ja) 2004-02-12
JP3798375B2 (ja) 2006-07-19
DE60122193T2 (de) 2007-07-05
CA2423568C (en) 2011-03-15
ZA200302283B (en) 2005-05-27
HK1061037A1 (en) 2004-09-03
WO2002028872A1 (fr) 2002-04-11
UA73606C2 (en) 2005-08-15
NO20031407L (no) 2003-04-30
HUP0301178A3 (en) 2009-08-28
CN1293087C (zh) 2007-01-03

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