ATE353329T1 - Heteroalkylamino-substituierte bicyclische stickstoffheterocyclen - Google Patents

Heteroalkylamino-substituierte bicyclische stickstoffheterocyclen

Info

Publication number: ATE353329T1
Authority: AT; Austria
Prior art keywords: heteroalkylamino; substituted bicyclic; nitrogen heterocycles; bicyclic nitrogen; heterocycles
Prior art date: 1999-10-21

Application number

AT00967864T

Other languages

English (en)

Inventor

James Patrick Dunn

Lawrence Emerson Fisher

David Michael Goldstein

William Harris

Christopher Huw Bill

Ian Edward David Smith

Teresa Rosanne Welch

Original Assignee

Hoffmann La Roche

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1999-10-21

Filing date

2000-10-13

Publication date

2007-02-15

2000-10-13 Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche

2007-02-15 Application granted granted Critical

2007-02-15 Publication of ATE353329T1 publication Critical patent/ATE353329T1/de

Links

IJGRMHOSHXDMSA-UHFFFAOYSA-N Atomic nitrogen Chemical compound N#N IJGRMHOSHXDMSA-UHFFFAOYSA-N 0.000 title 2
229910052757 nitrogen Inorganic materials 0.000 title 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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- A—HUMAN NECESSITIES
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- A61P1/16—Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
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Health & Medical Sciences (AREA)
Organic Chemistry (AREA)
Chemical & Material Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
Veterinary Medicine (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Public Health (AREA)
Medicinal Chemistry (AREA)
General Chemical & Material Sciences (AREA)
Pharmacology & Pharmacy (AREA)
Chemical Kinetics & Catalysis (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Immunology (AREA)
Physical Education & Sports Medicine (AREA)
Virology (AREA)
Pulmonology (AREA)
Diabetes (AREA)
Rheumatology (AREA)
Oncology (AREA)
Dermatology (AREA)
Hematology (AREA)
Neurology (AREA)
Orthopedic Medicine & Surgery (AREA)
Communicable Diseases (AREA)
Cardiology (AREA)
Neurosurgery (AREA)
Biomedical Technology (AREA)
Tropical Medicine & Parasitology (AREA)
Heart & Thoracic Surgery (AREA)
Pain & Pain Management (AREA)
Ophthalmology & Optometry (AREA)
Endocrinology (AREA)
Molecular Biology (AREA)
Reproductive Health (AREA)
Urology & Nephrology (AREA)
Hospice & Palliative Care (AREA)
Transplantation (AREA)

AT00967864T 1999-10-21 2000-10-13 Heteroalkylamino-substituierte bicyclische stickstoffheterocyclen ATE353329T1 (de)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
US16080399P	1999-10-21	1999-10-21
US21374300P	2000-06-22	2000-06-22

Publications (1)

Publication Number	Publication Date
ATE353329T1 true ATE353329T1 (de)	2007-02-15

Family

ID=26857240

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
AT00967864T ATE353329T1 (de)	1999-10-21	2000-10-13	Heteroalkylamino-substituierte bicyclische stickstoffheterocyclen

Country Status (26)

Country	Link
US (1)	US6451804B1 (de)
EP (1)	EP1228070B1 (de)
JP (1)	JP3961830B2 (de)
KR (1)	KR100523120B1 (de)
CN (1)	CN1171889C (de)
AR (1)	AR026084A1 (de)
AT (1)	ATE353329T1 (de)
AU (1)	AU776250B2 (de)
BR (1)	BR0015243A (de)
CA (1)	CA2388142C (de)
CZ (1)	CZ20021744A3 (de)
DE (1)	DE60033307T2 (de)
ES (1)	ES2280247T3 (de)
HR (1)	HRP20020328A2 (de)
HU (1)	HUP0203564A3 (de)
IL (1)	IL149100A0 (de)
MA (1)	MA26837A1 (de)
MX (1)	MXPA02003950A (de)
NO (1)	NO20021781L (de)
NZ (1)	NZ518119A (de)
PE (1)	PE20010758A1 (de)
PL (1)	PL357502A1 (de)
RU (1)	RU2265606C2 (de)
TR (1)	TR200201057T2 (de)
WO (1)	WO2001029042A1 (de)
YU (1)	YU29102A (de)

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PA8577501A1 (es)	2002-07-25	2004-02-07	Warner Lambert Co	Inhibidores de quinasas
RU2324695C2 (ru) *	2002-08-06	2008-05-20	Ф.Хоффманн-Ля Рош Аг	6-АЛКОКСИПИРИДОПИРИМИДИНЫ И ФАРМАЦЕВТИЧЕСКАЯ КОМПОЗИЦИЯ, ОБЛАДАЮЩАЯ АКТИВНОСТЬЮ ИНГИБИТОРОВ КИНАЗЫ МАР р38
US7084270B2 (en) *	2002-08-14	2006-08-01	Hoffman-La Roche Inc.	Pyrimido compounds having antiproliferative activity
US7112676B2 (en)	2002-11-04	2006-09-26	Hoffmann-La Roche Inc.	Pyrimido compounds having antiproliferative activity
TW200413381A (en)	2002-11-04	2004-08-01	Hoffmann La Roche	Novel amino-substituted dihydropyrimido [4,5-d]pyrimidinone derivatives, their manufacture and use as pharmaceutical agents
ATE427951T1 (de) *	2002-11-18	2009-04-15	Hoffmann La Roche	Diazinopyrimidine und ihre verwendung als proteinkinaseinhibitoren
CN100497339C (zh) *	2003-04-10	2009-06-10	霍夫曼-拉罗奇有限公司	嘧啶并化合物
BRPI0413005A (pt)	2003-07-29	2006-09-26	Irm Llc	compostos e composições como inibidores da proteìna cinase
US20060035893A1 (en)	2004-08-07	2006-02-16	Boehringer Ingelheim International Gmbh	Pharmaceutical compositions for treatment of respiratory and gastrointestinal disorders
CN1984914A (zh)	2004-08-31	2007-06-20	霍夫曼-拉罗奇有限公司	7－氨基－3－苯基－二氢嘧啶并[4,5－d]嘧啶酮的酰胺衍生物、其制备和作为蛋白激酶抑制剂的应用
WO2006024486A2 (en)	2004-08-31	2006-03-09	F. Hoffmann-La Roche Ag	Amide derivatives of 3-phenyl dihydropyrimido[4,5-d]pyrimidinones, their manufacture and use as pharmaceutical agents
WO2006038112A1 (en) *	2004-10-01	2006-04-13	Warner-Lambert Company Llc	Use of kinase inhibitors to promote neochondrogenesis
EP1831215A1 (de) *	2004-11-23	2007-09-12	Ranbaxy Laboratories Limited	Pyrido[2,3-d]pyrimidine als entzüngungshemmende mittel
PE20060777A1 (es)	2004-12-24	2006-10-06	Boehringer Ingelheim Int	Derivados de indolinona para el tratamiento o la prevencion de enfermedades fibroticas
EP1846403A1 (de) *	2005-02-02	2007-10-24	Ranbaxy Laboratories Limited	Azabicycloderivate als entzündungshemmende mittel
CN101341116A (zh) *	2005-12-22	2009-01-07	巴斯夫欧洲公司	制备o-烷基化环状氨基醇的方法
ES2329419T3 (es)	2006-01-31	2009-11-25	F. Hoffmann-La Roche Ag	7h-pirido(3,4-d)pirimidin-8-onas, su preparacion y uso como inhibidores de proteinas cinasas.
ES2301380B1 (es)	2006-08-09	2009-06-08	Laboratorios Almirall S.A.	Nuevos derivados de 1,7-naftiridina.
ES2320955B1 (es)	2007-03-02	2010-03-16	Laboratorios Almirall S.A.	Nuevos derivados de 3-((1,2,4)triazolo(4,3-a)piridin-7-il)benzamida.
ES2329639B1 (es)	2007-04-26	2010-09-23	Laboratorios Almirall S.A.	Nuevos derivados de 4,8-difenilpoliazanaftaleno.
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EP1992344A1 (de)	2007-05-18	2008-11-19	Institut Curie	P38 Alpha als therapeutisches Target für Erkrankungen, die mit einer FGFR3- Mutation assoziiert sind
GB2452696B (en) *	2007-08-02	2009-09-23	Cambridge Entpr Ltd	3-(2',2'-dimethylpropanoylamino)-tetrahydropyridin-2-one and its use in pharmaceutical compositions
EP2108641A1 (de) *	2008-04-11	2009-10-14	Laboratorios Almirall, S.A.	Neue substituierte Spiro[Cycloalkyl-1,3'-indo]-2'(1'H)-on-Derivate und ihre Verwendung als p38 mitogen-activated Kinase Inhibitoren
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2000
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Publication number	Publication date
AU776250B2 (en)	2004-09-02
CA2388142C (en)	2008-12-09
NO20021781D0 (no)	2002-04-16
PL357502A1 (en)	2004-07-26
HUP0203564A3 (en)	2004-07-28
HRP20020328A2 (en)	2004-02-29
WO2001029042A1 (en)	2001-04-26
EP1228070A1 (de)	2002-08-07
AU7787300A (en)	2001-04-30
HUP0203564A2 (hu)	2003-02-28
JP3961830B2 (ja)	2007-08-22
NZ518119A (en)	2004-02-27
HK1051039A1 (en)	2003-07-18
US6451804B1 (en)	2002-09-17
CZ20021744A3 (cs)	2002-08-14
MXPA02003950A (es)	2002-10-23
PE20010758A1 (es)	2001-07-21
BR0015243A (pt)	2002-07-16
RU2265606C2 (ru)	2005-12-10
CN1171889C (zh)	2004-10-20
MA26837A1 (fr)	2004-12-20
JP2003512378A (ja)	2003-04-02
CN1382144A (zh)	2002-11-27
TR200201057T2 (tr)	2002-09-23
RU2002112753A (ru)	2004-01-20
DE60033307D1 (en)	2007-03-22
YU29102A (sh)	2004-12-31
IL149100A0 (en)	2002-11-10
KR20020038963A (ko)	2002-05-24
AR026084A1 (es)	2002-12-26
NO20021781L (no)	2002-04-18
EP1228070B1 (de)	2007-02-07
ES2280247T3 (es)	2007-09-16
DE60033307T2 (de)	2007-07-12
KR100523120B1 (ko)	2005-10-20
CA2388142A1 (en)	2001-04-26

Legal Events

Date	Code	Title	Description
2007-08-15	RER	Ceased as to paragraph 5 lit. 3 law introducing patent treaties

Publication	Publication Date	Title
ATE353329T1 (de)	2007-02-15	Heteroalkylamino-substituierte bicyclische stickstoffheterocyclen
DK1218382T3 (da)	2004-03-22	Bicykliske imidazo-3-ylaminderivater
DK1224174T3 (da)	2004-01-26	Benzodiazepinderivater
NO20021691D0 (no)	2002-04-10	Benzodiazepinderivater
DE60025791D1 (de)	2006-04-13	Ellipsometer
EP1120205A4 (de)	2004-05-12	Roboter
DE60044873D1 (de)	2010-10-07	Orientierte biopolymermembrane
DE60026169D1 (de)	2006-04-27	Selektive neurokinin-antagonisten
DE50015443D1 (de)	2008-12-18	Bicyclische imidazo-5-yl-aminderivate
DE60022893D1 (de)	2006-02-09	Naphthyridinverbindungen
NO990431D0 (no)	1999-01-29	Golfk°llehode
DE50009640D1 (de)	2005-04-07	Drehmaschine
DE10080545D2 (de)	2002-01-31	Werktisch
DE50010263D1 (de)	2005-06-16	Arbeitsbühne
DE19945322B8 (de)	2004-07-08	Spannfutter
DK1123295T3 (da)	2005-01-31	Bicykliske nitrogenheterocykliske grupper
NO992540D0 (no)	1999-05-26	L°ftetralle
NO992248D0 (no)	1999-05-07	Rekkverk
DE50002518D1 (de)	2003-07-17	Werkstück mit Referenzelementen
NO993071D0 (no)	1999-06-22	L°vsamler
NO992685D0 (no)	1999-06-03	Stillas-l°pekatt
FI3964U1 (fi)	1999-05-19	Pylväs
NO992887D0 (no)	1999-06-14	B°lgebehandling
NO992842D0 (no)	1999-06-11	H°rselvern
NO993283D0 (no)	1999-07-02	Meiselverkt°y