ATE360818T1 - Festphasensynthese von n,n-disubstituierten diazacycloalkylcarboxy-derivaten - Google Patents
Festphasensynthese von n,n-disubstituierten diazacycloalkylcarboxy-derivatenInfo
- Publication number
- ATE360818T1 ATE360818T1 AT00939847T AT00939847T ATE360818T1 AT E360818 T1 ATE360818 T1 AT E360818T1 AT 00939847 T AT00939847 T AT 00939847T AT 00939847 T AT00939847 T AT 00939847T AT E360818 T1 ATE360818 T1 AT E360818T1
- Authority
- AT
- Austria
- Prior art keywords
- diazacycloalkylcarboxy
- disubstituted
- derivatives
- solid phase
- phase synthesis
- Prior art date
Links
- 238000010532 solid phase synthesis reaction Methods 0.000 title abstract 2
- 238000000034 method Methods 0.000 abstract 2
- 230000015572 biosynthetic process Effects 0.000 abstract 1
- BRYCUMKDWMEGMK-UHFFFAOYSA-N piperazine-2-carboxamide Chemical compound NC(=O)C1CNCCN1 BRYCUMKDWMEGMK-UHFFFAOYSA-N 0.000 abstract 1
- 238000003786 synthesis reaction Methods 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D241/00—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings
- C07D241/02—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings
- C07D241/10—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members
- C07D241/14—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D241/24—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
- C07B2200/00—Indexing scheme relating to specific properties of organic compounds
- C07B2200/11—Compounds covalently bound to a solid support
-
- C—CHEMISTRY; METALLURGY
- C40—COMBINATORIAL TECHNOLOGY
- C40B—COMBINATORIAL CHEMISTRY; LIBRARIES, e.g. CHEMICAL LIBRARIES
- C40B40/00—Libraries per se, e.g. arrays, mixtures
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US13930199P | 1999-06-15 | 1999-06-15 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ATE360818T1 true ATE360818T1 (de) | 2007-05-15 |
Family
ID=22486002
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AT00939847T ATE360818T1 (de) | 1999-06-15 | 2000-06-13 | Festphasensynthese von n,n-disubstituierten diazacycloalkylcarboxy-derivaten |
Country Status (6)
| Country | Link |
|---|---|
| US (1) | US7138526B1 (de) |
| EP (1) | EP1200824B1 (de) |
| AT (1) | ATE360818T1 (de) |
| AU (1) | AU5486600A (de) |
| DE (1) | DE60034571T2 (de) |
| WO (1) | WO2000077519A1 (de) |
Families Citing this family (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| ATE261959T1 (de) | 1999-12-30 | 2004-04-15 | Lundbeck & Co As H | Substituierte phenyl-piperazin-derivate, deren herstellung und verwendung |
| EP1246819A1 (de) * | 1999-12-30 | 2002-10-09 | H. Lundbeck A/S | Verfahren zur herstellung substituierter benzenderivate |
| WO2001054503A1 (en) * | 2000-01-28 | 2001-08-02 | Akkadix Corporation | Methods for killing nematodes and nematode eggs using 4-phenoxy-6-aminopyrimidine derivatives |
| WO2002008227A2 (en) * | 2000-07-21 | 2002-01-31 | Lion Bioscience Ag | Bicyclic hydantoin derivatives and combinatorial libraries thereof |
| CA2513716A1 (en) | 2003-02-14 | 2004-08-26 | Applied Research Systems Ars Holding N.V. | Piperazine-2-carboxamide derivatives |
| US8017612B2 (en) * | 2006-04-18 | 2011-09-13 | Japan Tobacco Inc. | Piperazine compound and use thereof as a HCV polymerase inhibitor |
| RU2012114770A (ru) | 2009-09-04 | 2013-10-10 | Вандербилт Юниверсити | АЛЛОСТЕРИЧЕСКИЕ СРЕДСТВА ПОТЕНЦИРОВАНИЯ mGluR4, КОМПОЗИЦИИ И СПОСОБЫ ЛЕЧЕНИЯ НЕВРОЛОГИЧЕСКИХ ДИСФУНКЦИЙ |
Family Cites Families (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| KR100310939B1 (ko) * | 1992-10-01 | 2002-06-20 | 추후제출 | 태그로암호화한복합조합화학라이브러리 |
| US5324483B1 (en) * | 1992-10-08 | 1996-09-24 | Warner Lambert Co | Apparatus for multiple simultaneous synthesis |
| US5880128A (en) * | 1996-05-08 | 1999-03-09 | Schering Corporation | Carbonyl piperazinyl and piperidinyl compounds |
| US5734054A (en) | 1996-11-05 | 1998-03-31 | Pharmacopeia, Inc. | Hydroxy-amino acid amides |
| US5972719A (en) * | 1996-11-05 | 1999-10-26 | Pharmacopeia, Inc. | Combinatorial hydroxy-amino acid amide libraries |
| WO1998058947A1 (en) | 1997-06-25 | 1998-12-30 | Pfizer Inc. | Dipeptide derivatives as growth hormone secretagogues |
-
2000
- 2000-06-13 DE DE60034571T patent/DE60034571T2/de not_active Expired - Lifetime
- 2000-06-13 AT AT00939847T patent/ATE360818T1/de not_active IP Right Cessation
- 2000-06-13 EP EP00939847A patent/EP1200824B1/de not_active Expired - Lifetime
- 2000-06-13 WO PCT/US2000/016243 patent/WO2000077519A1/en not_active Ceased
- 2000-06-13 US US10/009,621 patent/US7138526B1/en not_active Expired - Fee Related
- 2000-06-13 AU AU54866/00A patent/AU5486600A/en not_active Abandoned
Also Published As
| Publication number | Publication date |
|---|---|
| US7138526B1 (en) | 2006-11-21 |
| WO2000077519A1 (en) | 2000-12-21 |
| EP1200824B1 (de) | 2007-04-25 |
| DE60034571T2 (de) | 2007-12-27 |
| EP1200824A4 (de) | 2003-03-12 |
| DE60034571D1 (de) | 2007-06-06 |
| AU5486600A (en) | 2001-01-02 |
| EP1200824A1 (de) | 2002-05-02 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| RER | Ceased as to paragraph 5 lit. 3 law introducing patent treaties |