ATE371645T1 - Naphthalinderivate, die sich an den ep4?rezeptor binden - Google Patents

Naphthalinderivate, die sich an den ep4?rezeptor binden

Info

Publication number: ATE371645T1
Authority: AT; Austria
Prior art keywords: bind; receptor; naphthaline derivatives; derivatives; naphthaline
Prior art date: 2000-12-21

Application number

AT01271355T

Other languages

English (en)

Inventor

Gerard Martin Paul Giblin

Haydn Terence Jones

Andrew Mason

Neil Miller

Susan Roomans

Stephen Shanahan

Ann Walker

Original Assignee

Glaxo Group Ltd

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2000-12-21

Filing date

2001-12-20

Publication date

2007-09-15

2001-12-20 Application filed by Glaxo Group Ltd filed Critical Glaxo Group Ltd

2007-09-15 Application granted granted Critical

2007-09-15 Publication of ATE371645T1 publication Critical patent/ATE371645T1/de

Links

UFWIBTONFRDIAS-UHFFFAOYSA-N Naphthalene Chemical class C1=CC=CC2=CC=CC=C21 UFWIBTONFRDIAS-UHFFFAOYSA-N 0.000 title 1
208000020084 Bone disease Diseases 0.000 abstract 1
101150109738 Ptger4 gene Proteins 0.000 abstract 1
208000027520 Somatoform disease Diseases 0.000 abstract 1
210000000988 bone and bone Anatomy 0.000 abstract 1
150000001875 compounds Chemical class 0.000 abstract 1
230000001900 immune effect Effects 0.000 abstract 1
208000026278 immune system disease Diseases 0.000 abstract 1
208000027866 inflammatory disease Diseases 0.000 abstract 1
230000002757 inflammatory effect Effects 0.000 abstract 1
208000017169 kidney disease Diseases 0.000 abstract 1
208000015122 neurodegenerative disease Diseases 0.000 abstract 1
230000000626 neurodegenerative effect Effects 0.000 abstract 1
230000036407 pain Effects 0.000 abstract 1
208000027753 pain disease Diseases 0.000 abstract 1
230000002265 prevention Effects 0.000 abstract 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
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- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D209/56—Ring systems containing three or more rings
- C07D209/58—[b]- or [c]-condensed
- C07D209/62—Naphtho [c] pyrroles; Hydrogenated naphtho [c] pyrroles
- C07D209/64—Naphtho [c] pyrroles; Hydrogenated naphtho [c] pyrroles with an oxygen atom in position 1
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Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Life Sciences & Earth Sciences (AREA)
General Health & Medical Sciences (AREA)
Pharmacology & Pharmacy (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Veterinary Medicine (AREA)
Public Health (AREA)
Animal Behavior & Ethology (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Neurology (AREA)
Biomedical Technology (AREA)
Neurosurgery (AREA)
Diabetes (AREA)
Physical Education & Sports Medicine (AREA)
Rheumatology (AREA)
Hematology (AREA)
Addiction (AREA)
Virology (AREA)
Orthopedic Medicine & Surgery (AREA)
Endocrinology (AREA)
Pulmonology (AREA)
Psychiatry (AREA)
Oncology (AREA)
Ophthalmology & Optometry (AREA)
Communicable Diseases (AREA)
Dermatology (AREA)
Obesity (AREA)
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AT01271355T 2000-12-21 2001-12-20 Naphthalinderivate, die sich an den ep4?rezeptor binden ATE371645T1 (de)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
GBGB0031302.3A GB0031302D0 (en)	2000-12-21	2000-12-21	Napthalene derivatives

Publications (1)

Publication Number	Publication Date
ATE371645T1 true ATE371645T1 (de)	2007-09-15

Family

ID=9905630

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
AT01271355T ATE371645T1 (de)	2000-12-21	2001-12-20	Naphthalinderivate, die sich an den ep4?rezeptor binden

Country Status (9)

Country	Link
US (1)	US6924297B2 (de)
EP (1)	EP1351934B1 (de)
JP (1)	JP4397586B2 (de)
AT (1)	ATE371645T1 (de)
AU (1)	AU2002216218A1 (de)
DE (1)	DE60130256T2 (de)
ES (1)	ES2290093T3 (de)
GB (1)	GB0031302D0 (de)
WO (1)	WO2002050032A1 (de)

Families Citing this family (32)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
HN2001000224A (es)	2000-10-19	2002-06-13	Pfizer	Compuestos de imidazol condensado con arilo o heteroarilo como agentes anti - inflamatorios y analgesicos.
GB0031295D0 (en) *	2000-12-21	2001-01-31	Glaxo Group Ltd	Naphthalene derivatives
WO2005102389A2 (en) *	2004-04-20	2005-11-03	Pfizer Products Inc.	Combinations comprising alpha-2-delta ligands and ep4 receptor antagonists
WO2006122403A1 (en) *	2005-05-19	2006-11-23	Merck Frosst Canada Ltd.	Quinoline derivatives as ep4 antagonists
UY30121A1 (es)	2006-02-03	2007-08-31	Glaxo Group Ltd	Nuevos compuestos
GB0615111D0 (en) *	2006-07-28	2006-09-06	Glaxo Group Ltd	Novel compounds
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2000
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2001
- 2001-12-20 DE DE60130256T patent/DE60130256T2/de not_active Expired - Lifetime
- 2001-12-20 JP JP2002551529A patent/JP4397586B2/ja not_active Expired - Fee Related
- 2001-12-20 EP EP01271355A patent/EP1351934B1/de not_active Expired - Lifetime
- 2001-12-20 AU AU2002216218A patent/AU2002216218A1/en not_active Abandoned
- 2001-12-20 AT AT01271355T patent/ATE371645T1/de not_active IP Right Cessation
- 2001-12-20 WO PCT/GB2001/005676 patent/WO2002050032A1/en not_active Ceased
- 2001-12-20 US US10/450,891 patent/US6924297B2/en not_active Expired - Fee Related
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AU2002216218A1 (en)	2002-07-01
EP1351934B1 (de)	2007-08-29
ES2290093T3 (es)	2008-02-16
EP1351934A1 (de)	2003-10-15
US6924297B2 (en)	2005-08-02
DE60130256T2 (de)	2008-05-21
JP4397586B2 (ja)	2010-01-13
GB0031302D0 (en)	2001-01-31
JP2004517099A (ja)	2004-06-10
DE60130256D1 (de)	2007-10-11
WO2002050032A1 (en)	2002-06-27
US20040102508A1 (en)	2004-05-27

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