ATE377599T1 - Verfahren zur herstellung von substituierten 5- aminopyrazolo(4,3-e)-1,2,4-triazolo(1,5- c)pyrimidinen - Google Patents

Verfahren zur herstellung von substituierten 5- aminopyrazolo(4,3-e)-1,2,4-triazolo(1,5- c)pyrimidinen

Info

Publication number
ATE377599T1
ATE377599T1 AT04812380T AT04812380T ATE377599T1 AT E377599 T1 ATE377599 T1 AT E377599T1 AT 04812380 T AT04812380 T AT 04812380T AT 04812380 T AT04812380 T AT 04812380T AT E377599 T1 ATE377599 T1 AT E377599T1
Authority
AT
Austria
Prior art keywords
triazolo
aminopyrazolo
pyrimidines
producing substituted
substituted
Prior art date
Application number
AT04812380T
Other languages
English (en)
Inventor
Shen-Chun Kuo
Loc Tran
Pengyi Zhang
Original Assignee
Schering Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Schering Corp filed Critical Schering Corp
Application granted granted Critical
Publication of ATE377599T1 publication Critical patent/ATE377599T1/de

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/12—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains three hetero rings
    • C07D487/14—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
    • A61P25/16—Anti-Parkinson drugs

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Psychology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
AT04812380T 2003-12-01 2004-11-29 Verfahren zur herstellung von substituierten 5- aminopyrazolo(4,3-e)-1,2,4-triazolo(1,5- c)pyrimidinen ATE377599T1 (de)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US52592503P 2003-12-01 2003-12-01

Publications (1)

Publication Number Publication Date
ATE377599T1 true ATE377599T1 (de) 2007-11-15

Family

ID=34652398

Family Applications (1)

Application Number Title Priority Date Filing Date
AT04812380T ATE377599T1 (de) 2003-12-01 2004-11-29 Verfahren zur herstellung von substituierten 5- aminopyrazolo(4,3-e)-1,2,4-triazolo(1,5- c)pyrimidinen

Country Status (8)

Country Link
US (3) US7235659B2 (de)
EP (1) EP1689749B1 (de)
JP (1) JP2007513091A (de)
AT (1) ATE377599T1 (de)
CA (1) CA2547248A1 (de)
DE (1) DE602004009962T2 (de)
ES (1) ES2293380T3 (de)
WO (1) WO2005054245A2 (de)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SI1283839T1 (de) * 2000-05-26 2005-08-31 Schering Corp
PT1678182E (pt) * 2003-10-28 2007-04-30 Schering Corp Processo para preparar 5-amino-pirazolo-[4,3-e]-1,2,4-triazolo[1,5-c]pirimidinas
EP1902716A4 (de) * 2005-06-07 2009-05-13 Kyowa Hakko Kirin Co Ltd Prophylaktisches und/oder therapeutisches mittel für motorische störungen
ES2273599B1 (es) 2005-10-14 2008-06-01 Universidad De Barcelona Compuestos para el tratamiento de la fibrilacion auricular.
US8188098B2 (en) 2008-05-19 2012-05-29 Hoffmann-La Roche Inc. GPR119 receptor agonists
WO2010114894A1 (en) 2009-03-31 2010-10-07 Arqule, Inc. Substituted heterocyclic compounds
EP2724739B1 (de) 2009-07-30 2015-07-01 Tandem Diabetes Care, Inc. Tragbares Infusionspumpensystem
WO2012129381A1 (en) 2011-03-22 2012-09-27 Concert Pharmaceuticals Inc. Deuterated preladenant
WO2012127472A1 (en) * 2011-03-22 2012-09-27 Mapi Pharma Ltd. Process and intermediates for the preparation of preladenant and related compounds
WO2013024474A1 (en) * 2011-08-18 2013-02-21 Mapi Phrarma Ltd. Polymorphs of preladenant
CR20210271A (es) 2018-11-30 2021-07-14 Merck Sharp & Dohme Derivados de amino triazolo quinazolina 9-sustituidos como antagonistas del receptor de adenosina, composiciones farmacéuticas y su uso

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IT1264901B1 (it) * 1993-06-29 1996-10-17 Schering Plough S P A Analoghi eterociclici di 1,2,4-triazolo(15-c)pirimidine ad attivita' antagonista per il recettore a2 dell'adenosina
SI1283839T1 (de) 2000-05-26 2005-08-31 Schering Corp

Also Published As

Publication number Publication date
WO2005054245A2 (en) 2005-06-16
US20090131663A1 (en) 2009-05-21
CA2547248A1 (en) 2005-06-16
US20070238874A1 (en) 2007-10-11
WO2005054245A3 (en) 2005-08-11
EP1689749B1 (de) 2007-11-07
US7507822B2 (en) 2009-03-24
JP2007513091A (ja) 2007-05-24
DE602004009962D1 (de) 2007-12-20
US7235659B2 (en) 2007-06-26
ES2293380T3 (es) 2008-03-16
EP1689749A2 (de) 2006-08-16
US20060149060A1 (en) 2006-07-06
DE602004009962T2 (de) 2008-08-28

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