ATE381333T1 - Glucocorticoid-mimetika, deren herstellung, pharmazeutische zusammensetzungen und verwendung - Google Patents

Glucocorticoid-mimetika, deren herstellung, pharmazeutische zusammensetzungen und verwendung

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Publication number
ATE381333T1
ATE381333T1 AT03714339T AT03714339T ATE381333T1 AT E381333 T1 ATE381333 T1 AT E381333T1 AT 03714339 T AT03714339 T AT 03714339T AT 03714339 T AT03714339 T AT 03714339T AT E381333 T1 ATE381333 T1 AT E381333T1
Authority
AT
Austria
Prior art keywords
preparation
pharmaceutical compositions
glucocorticoid mimetics
glucocorticoid
mimetics
Prior art date
Application number
AT03714339T
Other languages
English (en)
Inventor
Y Bekkali
R Betageri
Thomas Gilmore
Mario Cardozo
T M Kirrane
D Kuzmich
J Proudfoot
H Takahashi
D Thomson
Ji Wang
R Zindell
C Harcken
D Riether
Hossein Razavi
Original Assignee
Boehringer Ingelheim Pharma
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Publication of ATE381333T1 publication Critical patent/ATE381333T1/de

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    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D209/00Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/04Indoles; Hydrogenated indoles
    • C07D209/10Indoles; Hydrogenated indoles with substituted hydrocarbon radicals attached to carbon atoms of the hetero ring
    • C07D209/12Radicals substituted by oxygen atoms
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    • C07DHETEROCYCLIC COMPOUNDS
    • C07D213/00Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/24Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with substituted hydrocarbon radicals attached to ring carbon atoms
    • C07D213/28Radicals substituted by singly-bound oxygen or sulphur atoms
    • C07D213/30Oxygen atoms
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    • C07D231/10Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
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AT03714339T 2002-03-26 2003-03-21 Glucocorticoid-mimetika, deren herstellung, pharmazeutische zusammensetzungen und verwendung ATE381333T1 (de)

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US36775802P 2002-03-26 2002-03-26
US43181702P 2002-12-09 2002-12-09
US44240403P 2003-01-24 2003-01-24

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ATE381333T1 true ATE381333T1 (de) 2008-01-15

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