ATE392899T1 - (androst-5-en-17beta-yl)alkyl sulfoxide und sulfone und deren verwendung zur kontrolle der fruchtbarkeit - Google Patents

(androst-5-en-17beta-yl)alkyl sulfoxide und sulfone und deren verwendung zur kontrolle der fruchtbarkeit

Info

Publication number
ATE392899T1
ATE392899T1 AT00907626T AT00907626T ATE392899T1 AT E392899 T1 ATE392899 T1 AT E392899T1 AT 00907626 T AT00907626 T AT 00907626T AT 00907626 T AT00907626 T AT 00907626T AT E392899 T1 ATE392899 T1 AT E392899T1
Authority
AT
Austria
Prior art keywords
17beta
androst
sulfones
fertility control
alkyl sulfoxides
Prior art date
Application number
AT00907626T
Other languages
English (en)
Inventor
Dirk Leysen
Der Louw Jaap Van
Anja Wiersma
Original Assignee
Organon Nv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Organon Nv filed Critical Organon Nv
Application granted granted Critical
Publication of ATE392899T1 publication Critical patent/ATE392899T1/de

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/57—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane or progesterone
    • A61K31/573—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane or progesterone substituted in position 21, e.g. cortisone, dexamethasone, prednisone or aldosterone
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A61P15/08—Drugs for genital or sexual disorders; Contraceptives for gonadal disorders or for enhancing fertility, e.g. inducers of ovulation or of spermatogenesis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A61P15/18—Feminine contraceptives

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Reproductive Health (AREA)
  • Gynecology & Obstetrics (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Endocrinology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Pregnancy & Childbirth (AREA)
  • Steroid Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
AT00907626T 1999-03-02 2000-02-25 (androst-5-en-17beta-yl)alkyl sulfoxide und sulfone und deren verwendung zur kontrolle der fruchtbarkeit ATE392899T1 (de)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP99200572 1999-03-02

Publications (1)

Publication Number Publication Date
ATE392899T1 true ATE392899T1 (de) 2008-05-15

Family

ID=8239933

Family Applications (1)

Application Number Title Priority Date Filing Date
AT00907626T ATE392899T1 (de) 1999-03-02 2000-02-25 (androst-5-en-17beta-yl)alkyl sulfoxide und sulfone und deren verwendung zur kontrolle der fruchtbarkeit

Country Status (9)

Country Link
US (1) US6552011B1 (de)
EP (1) EP1162977B1 (de)
JP (1) JP2002538123A (de)
AT (1) ATE392899T1 (de)
AU (1) AU2914800A (de)
DE (1) DE60038671T2 (de)
DK (1) DK1162977T3 (de)
ES (1) ES2304943T3 (de)
WO (1) WO2000051618A1 (de)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN111320664B (zh) * 2018-12-13 2023-01-24 上海医药工业研究院 一种24-胆烯烯酸乙酯的制备方法
CN111320663B (zh) * 2018-12-13 2023-01-24 上海医药工业研究院 一种24-胆烯烯酸乙酯中间体的制备方法

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE272854C (de)
DE247008C (de)
DE282230C (de)
DE3265509D1 (en) * 1981-04-29 1985-09-26 Hoffmann La Roche Process for the preparation of cholesterol derivatives, and intermediate derivatives therefor
DD247008A1 (de) * 1986-02-24 1987-06-24 Akad Wissenschaften Ddr Verfahren zur herstellung von aryl-3beta-hydroxy-23,24-bisnorchola-5,7-dien-22-yl-sulfon-derivaten
DD272854A1 (de) * 1988-06-02 1989-10-25 Jenapharm Veb Verfahren zur herstellung von 3 beta-substituierten(20s)-20-aryl-sulfonylmethyl-pregna-5,7-dienen
DD282230A5 (de) * 1989-04-13 1990-09-05 Akad Wissenschaften Ddr Verfahren zur herstellung von (3s)-3,24,25-trihydroxycholesta-5,7-dienen
EP0946584B1 (de) * 1996-12-20 2003-04-23 Novo Nordisk A/S Verbindungen zur Regulierung der Meiose
AU726016B2 (en) * 1997-05-16 2000-10-26 Akzo Nobel N.V. 20-aralkyl-5alpha-pregnane derivatives
IL132799A0 (en) 1997-06-04 2001-03-19 Akzo Nobel Nv 17Beta-allyloxy(thio)alkyl-androstane derivatives for the modulation of meiosis

Also Published As

Publication number Publication date
US6552011B1 (en) 2003-04-22
WO2000051618A1 (en) 2000-09-08
JP2002538123A (ja) 2002-11-12
ES2304943T3 (es) 2008-11-01
EP1162977B1 (de) 2008-04-23
DE60038671T2 (de) 2009-05-07
DK1162977T3 (da) 2008-07-28
AU2914800A (en) 2000-09-21
DE60038671D1 (de) 2008-06-05
EP1162977A1 (de) 2001-12-19

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Legal Events

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