ATE394399T1 - Tetrahydropyridoindolderivate - Google Patents

Tetrahydropyridoindolderivate

Info

Publication number: ATE394399T1
Authority: AT; Austria
Prior art keywords: tetrahydropyridoindole derivatives; tetrahydropyridoindole; derivatives
Prior art date: 2004-03-11

Application number

AT05715779T

Other languages

English (en)

Inventor

Heinz Fretz

Anja Fecher

Kurt Hilpert

Markus Riederer

Original Assignee

Actelion Pharmaceuticals Ltd

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2004-03-11

Filing date

2005-03-07

Publication date

2008-05-15

Family has litigation

First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=34961211&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=ATE394399(T1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.

2005-03-07 Application filed by Actelion Pharmaceuticals Ltd filed Critical Actelion Pharmaceuticals Ltd

2008-05-15 Application granted granted Critical

2008-05-15 Publication of ATE394399T1 publication Critical patent/ATE394399T1/de

Links

UFXNNGDEYWTROW-UHFFFAOYSA-N 2,3,3a,4-tetrahydro-1h-pyrrolo[2,3-f]quinoline Chemical class C1C=C2N=CC=CC2=C2C1CCN2 UFXNNGDEYWTROW-UHFFFAOYSA-N 0.000 title 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/4353—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
- A61K31/437—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a five-membered ring having nitrogen as a ring hetero atom, e.g. indolizine, beta-carboline
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/02—Nasal agents, e.g. decongestants
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/06—Antiasthmatics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/12—Drugs for disorders of the urinary system of the kidneys
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A61P17/02—Drugs for dermatological disorders for treating wounds, ulcers, burns, scars, keloids, or the like
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A61P17/04—Antipruritics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/02—Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/16—Otologicals
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A61P35/02—Antineoplastic agents specific for leukemia
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/02—Immunomodulators
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/08—Vasodilators for multiple indications
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Veterinary Medicine (AREA)
Pharmacology & Pharmacy (AREA)
Public Health (AREA)
General Health & Medical Sciences (AREA)
Animal Behavior & Ethology (AREA)
Medicinal Chemistry (AREA)
Life Sciences & Earth Sciences (AREA)
General Chemical & Material Sciences (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Chemical Kinetics & Catalysis (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Pulmonology (AREA)
Immunology (AREA)
Dermatology (AREA)
Cardiology (AREA)
Urology & Nephrology (AREA)
Heart & Thoracic Surgery (AREA)
Rheumatology (AREA)
Vascular Medicine (AREA)
Ophthalmology & Optometry (AREA)
Pain & Pain Management (AREA)
Oncology (AREA)
Orthopedic Medicine & Surgery (AREA)
Physical Education & Sports Medicine (AREA)
Otolaryngology (AREA)
Hematology (AREA)
Epidemiology (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Indole Compounds (AREA)

AT05715779T 2004-03-11 2005-03-07 Tetrahydropyridoindolderivate ATE394399T1 (de)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
EP2004002493		2004-03-11

Publications (1)

Publication Number	Publication Date
ATE394399T1 true ATE394399T1 (de)	2008-05-15

Family

ID=34961211

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
AT05715779T ATE394399T1 (de)	2004-03-11	2005-03-07	Tetrahydropyridoindolderivate

Country Status (24)

Country	Link
US (2)	US7714132B2 (de)
EP (1)	EP1725553B1 (de)
JP (1)	JP4051398B2 (de)
KR (1)	KR100808742B1 (de)
CN (1)	CN1930162B (de)
AR (1)	AR047928A1 (de)
AT (1)	ATE394399T1 (de)
AU (1)	AU2005229356B2 (de)
BR (1)	BRPI0508540B8 (de)
CA (1)	CA2558509C (de)
DE (1)	DE602005006539D1 (de)
DK (1)	DK1725553T3 (de)
ES (1)	ES2304010T3 (de)
IL (1)	IL177968A0 (de)
MY (1)	MY143795A (de)
NO (1)	NO337996B1 (de)
NZ (1)	NZ550365A (de)
PL (1)	PL1725553T3 (de)
PT (1)	PT1725553E (de)
RU (1)	RU2387652C2 (de)
SI (1)	SI1725553T1 (de)
TW (1)	TWI369356B (de)
WO (1)	WO2005095397A1 (de)
ZA (1)	ZA200608446B (de)

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WO2017019858A1 (en)	2015-07-30	2017-02-02	The Trustees Of The University Of Pennsylvania	Single nucleotide polymorphic alleles of human dp-2 gene for detection of susceptibility to hair growth inhibition by pgd2
CN108026093B (zh)	2015-09-15	2021-11-16	爱杜西亚药品有限公司	结晶形式
WO2019170848A1 (en) *	2018-03-09	2019-09-12	Panoptes Pharma Ges.M.B.H.	Ophthalmic formulation
TWI915239B (zh)	2018-06-21	2026-02-11	瑞士商赫孚孟拉羅股份公司	3-((1r,3r)-1-(2,6-二氟-4-((1-(3-氟丙基)氮雜環丁-3-基)胺基)苯基)-3-甲基-1,3,4,9-四氫-2h-吡啶并[3,4-b]吲哚-2-基)-2,2-二氟丙-1-醇之固體形式及用於製備包含經取代苯基或吡啶基部分之稠合三環化合物之製程，包括其使用方法
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- 2005-03-07 AT AT05715779T patent/ATE394399T1/de active
- 2005-03-07 DE DE602005006539T patent/DE602005006539D1/de active Active
- 2005-03-07 RU RU2006135651/04A patent/RU2387652C2/ru not_active IP Right Cessation
- 2005-03-07 JP JP2007501238A patent/JP4051398B2/ja not_active Expired - Fee Related
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- 2005-03-07 ES ES05715779T patent/ES2304010T3/es not_active Expired - Lifetime
- 2005-03-07 DK DK05715779T patent/DK1725553T3/da active
- 2005-03-07 CN CN2005800076993A patent/CN1930162B/zh not_active Expired - Fee Related
- 2005-03-07 SI SI200530281T patent/SI1725553T1/sl unknown
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- 2005-03-07 WO PCT/EP2005/002362 patent/WO2005095397A1/en not_active Ceased
- 2005-03-07 EP EP05715779A patent/EP1725553B1/de not_active Expired - Lifetime
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2006
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- 2006-10-10 NO NO20064584A patent/NO337996B1/no not_active IP Right Cessation
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Also Published As

Publication number	Publication date
IL177968A0 (en)	2006-12-31
DE602005006539D1 (de)	2008-06-19
CA2558509A1 (en)	2005-10-13
MY143795A (en)	2011-07-15
NO337996B1 (no)	2016-07-18
JP4051398B2 (ja)	2008-02-20
AU2005229356A1 (en)	2005-10-13
DK1725553T3 (da)	2008-08-18
RU2006135651A (ru)	2008-04-20
PT1725553E (pt)	2008-07-16
KR100808742B1 (ko)	2008-02-29
BRPI0508540A (pt)	2007-09-18
JP2007526276A (ja)	2007-09-13
NO20064584L (no)	2006-10-10
EP1725553A1 (de)	2006-11-29
TWI369356B (en)	2012-08-01
CN1930162A (zh)	2007-03-14
CA2558509C (en)	2011-11-22
US7714132B2 (en)	2010-05-11
ZA200608446B (en)	2008-06-25
US20070191416A1 (en)	2007-08-16
AR047928A1 (es)	2006-03-01
BRPI0508540B8 (pt)	2021-05-25
AU2005229356B2 (en)	2011-06-09
KR20070029670A (ko)	2007-03-14
NZ550365A (en)	2010-09-30
CN1930162B (zh)	2010-06-16
EP1725553B1 (de)	2008-05-07
BRPI0508540A8 (pt)	2017-12-26
WO2005095397A1 (en)	2005-10-13
BRPI0508540B1 (pt)	2019-04-02
TW200538434A (en)	2005-12-01
US20100234396A1 (en)	2010-09-16
PL1725553T3 (pl)	2008-10-31
SI1725553T1 (sl)	2008-08-31
ES2304010T3 (es)	2008-09-01
RU2387652C2 (ru)	2010-04-27

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