|
TWI329105B
(en)
|
2002-02-01 |
2010-08-21 |
Rigel Pharmaceuticals Inc |
2,4-pyrimidinediamine compounds and their uses
|
|
AR042052A1
(es)
*
|
2002-11-15 |
2005-06-08 |
Vertex Pharma |
Diaminotriazoles utiles como inhibidores de proteinquinasas
|
|
EP1628666B1
(de)
|
2003-05-14 |
2015-09-23 |
NeuroGenetic Pharmaceuticals, Inc. |
Verbindungen und ihre verwendungen zur modulierung von amyloid beta
|
|
DK1636215T3
(da)
|
2003-05-23 |
2008-06-02 |
Basilea Pharmaceutica Ag |
Furazanobenzimidazoler
|
|
CN102358738A
(zh)
|
2003-07-30 |
2012-02-22 |
里格尔药品股份有限公司 |
2,4-嘧啶二胺化合物及其预防和治疗自体免疫疾病的用途
|
|
BRPI0507634A
(pt)
*
|
2004-02-11 |
2007-07-03 |
Janssen Pharmaceutica Nv |
processo para preparação de compostos triazóis substituìdos
|
|
US20070167505A1
(en)
*
|
2004-02-11 |
2007-07-19 |
Basilea Pharmaceutica Ag |
Substituted benzimidazoles and their use for inducing apoptosis
|
|
MX2007003154A
(es)
*
|
2004-09-17 |
2007-05-15 |
Vertex Pharma |
Compuestos de diaminotriazol de utilidad como inhibidores de proteina quinasa.
|
|
AU2012205127B2
(en)
*
|
2004-09-17 |
2014-10-30 |
Vertex Pharmaceuticals Incorporated |
Diaminotriazole Compounds Useful as Protein Kinase Inhibitors
|
|
JP2008515925A
(ja)
|
2004-10-08 |
2008-05-15 |
ジヤンセン・フアーマシユーチカ・ナームローゼ・フエンノートシヤツプ |
1,2,4−トリアゾリルアミノアリール(ヘテロアリール)スルホンアミド誘導体
|
|
CN101389335A
(zh)
|
2004-10-18 |
2009-03-18 |
安姆根有限公司 |
噻二唑化合物和使用方法
|
|
ATE485042T1
(de)
|
2004-10-21 |
2010-11-15 |
Vertex Pharma |
Triazole als hemmer von proteinkinasen
|
|
KR20070085433A
(ko)
*
|
2004-11-24 |
2007-08-27 |
노파르티스 아게 |
Jak 저해제들과 bcr-abl, flt-3, fak 또는raf 키나제 저해제들 중 하나 이상의 조합물
|
|
PL2559690T3
(pl)
|
2005-05-10 |
2016-09-30 |
|
Modulatory 2,3-dioksygenazy indoloaminy i sposoby ich zastosowania
|
|
US20070203161A1
(en)
*
|
2006-02-24 |
2007-08-30 |
Rigel Pharmaceuticals, Inc. |
Compositions and methods for inhibition of the jak pathway
|
|
EP1904457B1
(de)
|
2005-06-08 |
2017-09-06 |
Rigel Pharmaceuticals, Inc. |
Zusammensetzungen und verfahren zur inhibierung des jak-pfades
|
|
US8071768B2
(en)
|
2005-06-10 |
2011-12-06 |
Janssen Pharmaceutica, N.V. |
Alkylquinoline and alkylquinazoline kinase modulators
|
|
US20060281788A1
(en)
|
2005-06-10 |
2006-12-14 |
Baumann Christian A |
Synergistic modulation of flt3 kinase using a flt3 inhibitor and a farnesyl transferase inhibitor
|
|
US7825244B2
(en)
|
2005-06-10 |
2010-11-02 |
Janssen Pharmaceutica Nv |
Intermediates useful in the synthesis of alkylquinoline and alkylquinazoline kinase modulators, and related methods of synthesis
|
|
CA2607901C
(en)
|
2005-06-13 |
2016-08-16 |
Rigel Pharmaceuticals, Inc. |
Methods and compositions for treating degenerative bone disorders using a syk inhibitory 2,4-pyrimidinediamine
|
|
DE602005000514T2
(de)
*
|
2005-06-17 |
2007-10-25 |
Magneti Marelli Powertrain S.P.A. |
Brennstoffeinspritzventil
|
|
JP5255438B2
(ja)
*
|
2005-07-26 |
2013-08-07 |
バーテックス ファーマシューティカルズ インコーポレイテッド |
プロテインキナーゼ阻害薬として有用なベンズイミダゾール
|
|
US7884119B2
(en)
|
2005-09-07 |
2011-02-08 |
Rigel Pharmaceuticals, Inc. |
Triazole derivatives useful as Axl inhibitors
|
|
EP2270014A1
(de)
|
2005-09-22 |
2011-01-05 |
Incyte Corporation |
Azepinhemmer von Janus-Kinasen
|
|
EP1951234A2
(de)
|
2005-10-18 |
2008-08-06 |
Janssen Pharmaceutica N.V. |
Verfahren zur hemmung von flt3-kinase
|
|
CN103214484B
(zh)
|
2005-12-13 |
2016-07-06 |
因塞特控股公司 |
作为两面神激酶抑制剂的杂芳基取代的吡咯并[2,3-b]吡啶和吡咯并[2,3-b]嘧啶
|
|
CN101421265A
(zh)
|
2006-01-18 |
2009-04-29 |
安姆根有限公司 |
作为蛋白激酶b(pkb)抑制剂的噻唑化合物
|
|
JP2009528295A
(ja)
|
2006-02-24 |
2009-08-06 |
ライジェル ファーマシューティカルズ, インコーポレイテッド |
Jak経路の阻害のための組成物および方法
|
|
MX2008013533A
(es)
|
2006-04-20 |
2009-01-15 |
Janssen Pharmaceutica Nv |
Compuestos heterociclicos como inhibidores de c-fms cinasa.
|
|
EP2016070B1
(de)
|
2006-04-20 |
2016-01-13 |
Janssen Pharmaceutica N.V. |
Inhibitoren von c-fms-kinase
|
|
US8697716B2
(en)
|
2006-04-20 |
2014-04-15 |
Janssen Pharmaceutica Nv |
Method of inhibiting C-KIT kinase
|
|
CA2658764A1
(en)
*
|
2006-07-20 |
2008-01-24 |
Mehmet Kahraman |
Benzothiophene inhibitors of rho kinase
|
|
MX2009003456A
(es)
|
2006-10-02 |
2009-04-14 |
Irm Llc |
Compuestos y composiciones como inhibidores de proteina cinasa.
|
|
ATE497496T1
(de)
|
2006-10-19 |
2011-02-15 |
Rigel Pharmaceuticals Inc |
2,4-pyridimediamon-derivate als hemmer von jak- kinasen zur behandlung von autoimmunerkrankungen
|
|
ES2415863T3
(es)
|
2006-12-22 |
2013-07-29 |
Incyte Corporation |
Heterociclos sustituidos como inhibidores de Janus Quinasas
|
|
AU2007342005A1
(en)
*
|
2006-12-29 |
2008-07-10 |
Rigel Pharmaceuticals, Inc. |
N3-heteroaryl substituted triazoles and N5-heteroaryl substituted triazoles useful as Axl inhibitors
|
|
ES2404668T3
(es)
|
2006-12-29 |
2013-05-28 |
Rigel Pharmaceuticals, Inc. |
Triazoles sustituidos con arilo bicíclico puenteado y heteroarilo bicíclico puenteado, útiles como agentes inhibidores del axl
|
|
PT2078010E
(pt)
|
2006-12-29 |
2014-05-07 |
Rigel Pharmaceuticals Inc |
Triazoles substituídos com heteroarilos policíclicos úteis como inibidores de axl
|
|
EP2114954B1
(de)
|
2006-12-29 |
2013-02-13 |
Rigel Pharmaceuticals, Inc. |
Durch bicyclisches aryl bzw. bicyclisches heteroaryl substituierte triazole, die sich als axl-inihibitoren eignen
|
|
AU2014200825B2
(en)
*
|
2006-12-29 |
2016-05-26 |
Rigel Pharmaceuticals, Inc. |
N3-heteroaryl substituted triazoles and N5-heteroaryl substituted triazoles useful as Axl inhibitors
|
|
AU2014200824B2
(en)
*
|
2006-12-29 |
2016-12-15 |
Rigel Pharmaceuticals, Inc. |
Substituted triazoles useful as Axl inhibitors
|
|
AU2016259396B2
(en)
*
|
2006-12-29 |
2018-11-08 |
Rigel Pharmaceuticals, Inc. |
Substituted triazoles useful as Axl inhibitors
|
|
JP2010514810A
(ja)
|
2006-12-29 |
2010-05-06 |
ライジェル ファーマシューティカルズ, インコーポレイテッド |
Axlインヒビターとして有用な置換トリアゾール
|
|
JP5642973B2
(ja)
*
|
2007-03-22 |
2014-12-17 |
バーテックス ファーマシューティカルズ インコーポレイテッドVertex Pharmaceuticals Incorporated |
Jak阻害薬として有用なn−複素環式化合物
|
|
HUE029236T2
(en)
|
2007-06-13 |
2017-02-28 |
Incyte Holdings Corp |
(R) -3- (4- (7H-Pyrrolo [2,3-d] pyrimidin-4-yl) -1H-pyrazol-1-yl) -3-cyclopentylpropanenitrile Crystalline salts of Janus kinase inhibitor
|
|
CL2008001709A1
(es)
|
2007-06-13 |
2008-11-03 |
Incyte Corp |
Compuestos derivados de pirrolo [2,3-b]pirimidina, moduladores de quinasas jak; composicion farmaceutica; y uso en el tratamiento de enfermedades tales como cancer, psoriasis, artritis reumatoide, entre otras.
|
|
AU2008266290A1
(en)
*
|
2007-06-15 |
2008-12-24 |
Irm Llc |
Protein kinase inhibitors and methods for using thereof
|
|
WO2009011871A2
(en)
|
2007-07-17 |
2009-01-22 |
Amgen Inc. |
Thiadiazole modulators of pkb
|
|
AU2008276521B2
(en)
*
|
2007-07-17 |
2011-11-03 |
Amgen Inc. |
Heterocyclic modulators of PKB
|
|
CN104586832B
(zh)
|
2007-09-10 |
2018-02-16 |
北京强新生物科技有限公司 |
用于癌症治疗的组合物和方法
|
|
WO2009042677A2
(en)
*
|
2007-09-24 |
2009-04-02 |
Farjo Rafal A |
Stat3 inhibiting compositions and methods
|
|
JO3240B1
(ar)
|
2007-10-17 |
2018-03-08 |
Janssen Pharmaceutica Nv |
c-fms مثبطات كيناز
|
|
JP2011500625A
(ja)
*
|
2007-10-18 |
2011-01-06 |
ジヤンセン・フアーマシユーチカ・ナームローゼ・フエンノートシヤツプ |
トリ置換された1,2,4−トリアゾール
|
|
JO2784B1
(en)
*
|
2007-10-18 |
2014-03-15 |
شركة جانسين فارماسوتيكا ان. في |
5,3,1 - Triazole substitute derivative
|
|
CA2704052C
(en)
*
|
2007-10-26 |
2015-04-21 |
Rigel Pharmaceuticals, Inc. |
Polycyclic aryl substituted triazoles and polycyclic heteroaryl substituted triazoles useful as axl inhibitors
|
|
EP2217716A4
(de)
*
|
2007-11-09 |
2011-02-09 |
Salk Inst For Biological Studi |
Verwendung von tam-rezeptor-inhibitoren als antimikrobielle mittel
|
|
MX2010005300A
(es)
|
2007-11-16 |
2010-06-25 |
Incyte Corp |
4-pirazolil-n-arilpirimidin-2-aminas y 4-pirazolil-n-heteroarilpir imidin-2-aminas como inhibidores de cinasas janus.
|
|
WO2009065132A1
(en)
*
|
2007-11-16 |
2009-05-22 |
Oklahoma Medical Research Foundation |
Predicting and diagnosing patients with autoimmune disease
|
|
HUE030912T2
(en)
|
2008-02-15 |
2017-06-28 |
Rigel Pharmaceuticals Inc |
Pyrimidine-2-amine compounds and their use as inhibitors of yak kinases
|
|
TWI444382B
(zh)
|
2008-03-11 |
2014-07-11 |
Incyte Corp |
作為jak抑制劑之氮雜環丁烷及環丁烷衍生物
|
|
MX2010011463A
(es)
|
2008-04-16 |
2011-06-03 |
Portola Pharm Inc |
2,6-diamino-pirimidin-5-il-carboxamidas como inhibidores de syk o jak quinasas.
|
|
US8138339B2
(en)
*
|
2008-04-16 |
2012-03-20 |
Portola Pharmaceuticals, Inc. |
Inhibitors of protein kinases
|
|
JP2011518219A
(ja)
|
2008-04-22 |
2011-06-23 |
ポートラ ファーマシューティカルズ, インコーポレイテッド |
タンパク質キナーゼの阻害剤
|
|
CA2722326A1
(en)
|
2008-04-24 |
2009-10-29 |
Incyte Corporation |
Macrocyclic compounds and their use as kinase inhibitors
|
|
US20100035875A1
(en)
*
|
2008-06-20 |
2010-02-11 |
Bing-Yan Zhu |
Triazolopyridine jak inhibitor compounds and methods
|
|
KR20110033223A
(ko)
*
|
2008-06-20 |
2011-03-30 |
제넨테크, 인크. |
트리아졸로피리딘 jak 억제제 화합물 및 방법
|
|
ES2524266T3
(es)
|
2008-07-08 |
2014-12-04 |
Incyte Corporation |
1,2,5-Oxadiazoles como inhibidores de la indoleamina 2,3-dioxigenasa
|
|
US8431594B2
(en)
|
2008-07-09 |
2013-04-30 |
Rigel Pharmaceuticals, Inc. |
Bridged bicyclic heteroaryl substituted triazoles useful as AXL inhibitors
|
|
JP5592884B2
(ja)
|
2008-07-09 |
2014-09-17 |
ライジェル ファーマシューティカルズ, インコーポレイテッド |
Axl阻害剤として有用な多環式ヘテロアリール置換トリアゾール
|
|
US8466290B2
(en)
*
|
2008-07-10 |
2013-06-18 |
Pharma Ip General Incorporated Association |
STAT3 inhibitor containing quinolinecarboxamide derivative as active ingredient
|
|
TWI453207B
(zh)
*
|
2008-09-08 |
2014-09-21 |
Signal Pharm Llc |
胺基三唑并吡啶,其組合物及使用其之治療方法
|
|
CA2737738A1
(en)
*
|
2008-09-18 |
2010-03-25 |
Astellas Pharma Inc. |
Heterocyclic carboxamide compounds
|
|
CL2009001884A1
(es)
|
2008-10-02 |
2010-05-14 |
Incyte Holdings Corp |
Uso de 3-ciclopentil-3-[4-(7h-pirrolo[2,3-d]pirimidin-4-il)-1h-pirazol-1-il)propanonitrilo, inhibidor de janus quinasa, y uso de una composición que lo comprende para el tratamiento del ojo seco.
|
|
CN102307997B
(zh)
*
|
2008-12-04 |
2018-03-30 |
库尔纳公司 |
通过抑制针对沉默调节蛋白1的天然反义转录物来治疗沉默调节蛋白1(sirt1)相关的疾病
|
|
TWI469979B
(zh)
*
|
2008-12-24 |
2015-01-21 |
Bial Portela & Ca Sa |
脂肪酸醯胺水解酶(faah)抑制劑、以及其藥學組成物與用途
|
|
RU2555326C2
(ru)
|
2009-01-16 |
2015-07-10 |
Риджел Фармасьютикалз, Инк. |
ИНГИБИТОРЫ Axl ДЛЯ ПРИМЕНЕНИЯ В КОМБИНИРОВАННОЙ ТЕРАПИИ ДЛЯ ПРЕДОТВРАЩЕНИЯ, УСТРАНЕНИЯ ИЛИ ЛЕЧЕНИЯ МЕТАСТAЗИРУЮЩЕГО РАКА
|
|
US8765727B2
(en)
|
2009-01-23 |
2014-07-01 |
Incyte Corporation |
Macrocyclic compounds and their use as kinase inhibitors
|
|
ES2740424T3
(es)
|
2009-03-13 |
2020-02-05 |
Agios Pharmaceuticals Inc |
Métodos y composiciones para trastornos relacionados con la proliferación celular
|
|
MY156727A
(en)
|
2009-05-22 |
2016-03-15 |
Incyte Corp |
N-(hetero)aryl-pyrrolidine derivatives of pyrazol-4-yl-pyrrolo[2,3-d]pyrimidines and pyrrol-3-yl-pyrrolo[2,3-d]pyrimidines as janus kinase inhibitors
|
|
EP2432472B1
(de)
|
2009-05-22 |
2019-10-02 |
Incyte Holdings Corporation |
3-[4-(7h-pyrrolo[2,3-d]pyrimidin-4-yl)-1h-pyrazol-1-yl]octan- oder heptannitril als jak-inhibitoren
|
|
JP5095035B2
(ja)
*
|
2009-06-09 |
2012-12-12 |
アクテリオン ファーマシューティカルズ リミテッド |
フッ素化アミノトリアゾール誘導体
|
|
EP2845856A1
(de)
|
2009-06-29 |
2015-03-11 |
Incyte Corporation |
Pyrimidone als PI3K-Hemmer
|
|
SG10201403696UA
(en)
|
2009-06-29 |
2014-10-30 |
Agios Pharmaceuticals Inc |
Therapeutic compounds and compositions
|
|
CA2768543C
(en)
*
|
2009-07-28 |
2017-06-20 |
Rigel Pharmaceuticals, Inc. |
Compositions and methods for inhibition of the jak pathway
|
|
TW201113285A
(en)
|
2009-09-01 |
2011-04-16 |
Incyte Corp |
Heterocyclic derivatives of pyrazol-4-yl-pyrrolo[2,3-d]pyrimidines as janus kinase inhibitors
|
|
MX2012004180A
(es)
|
2009-10-09 |
2012-07-17 |
Incyte Corp |
Derivados de hidroxil, ceto y glucuronido de 3-(4-7h-pirrolo[2,3-d ]pirimidin-a-il)-1h-pirazol-1-il)-3-ciclopentilpropanonitrilo.
|
|
EP3064595B1
(de)
|
2009-10-21 |
2019-02-27 |
Agios Pharmaceuticals, Inc. |
Verfahren für zellproliferationsbedingte erkrankungen
|
|
WO2011075630A1
(en)
|
2009-12-18 |
2011-06-23 |
Incyte Corporation |
Substituted fused aryl and heteroaryl derivatives as pi3k inhibitors
|
|
US8759359B2
(en)
|
2009-12-18 |
2014-06-24 |
Incyte Corporation |
Substituted heteroaryl fused derivatives as PI3K inhibitors
|
|
HUE045270T2
(hu)
|
2010-01-05 |
2019-12-30 |
Inst Nat Sante Rech Med |
FLT3 receptor anatgonisták fájdalom rendellenességek kezelésére
|
|
TWI523852B
(zh)
|
2010-01-12 |
2016-03-01 |
Ab科學公司 |
經取代之唑衍生物、含彼之組合物及其用途
|
|
CN102811620B
(zh)
*
|
2010-01-25 |
2015-03-25 |
Chdi基金会股份有限公司 |
一些犬尿氨酸-3-单加氧酶抑制剂、药物组合物及其使用方法
|
|
CA2790070C
(en)
|
2010-02-18 |
2018-03-06 |
Incyte Corporation |
Cyclobutane and methylcyclobutane derivatives as janus kinase inhibitors
|
|
EP3354652B1
(de)
|
2010-03-10 |
2020-05-06 |
Incyte Holdings Corporation |
Piperidin-4-yl azetidin-derivate als jak1-inhibitoren
|
|
CN103025159A
(zh)
*
|
2010-03-19 |
2013-04-03 |
波士顿生物医学公司 |
靶向癌症干细胞的新方法
|
|
SG10201706265PA
(en)
*
|
2010-03-19 |
2017-08-30 |
Boston Biomedical Inc |
Novel compounds and compositions for targeting cancer stem cells
|
|
MX339192B
(es)
*
|
2010-03-24 |
2016-05-13 |
Amitech Therapeutic Solutions Inc |
Compuestos heterociclicos utiles para inhibicion de cinasa.
|
|
EP2558463A1
(de)
|
2010-04-14 |
2013-02-20 |
Incyte Corporation |
Kondensierte derivate als i3-hemmer
|
|
AR084691A1
(es)
|
2010-05-21 |
2013-06-05 |
Incyte Corp |
Formulacion de uso topico para un inhibidor de jak y metodo para tratar trastorno de la piel
|
|
WO2011163195A1
(en)
|
2010-06-21 |
2011-12-29 |
Incyte Corporation |
Fused pyrrole derivatives as pi3k inhibitors
|
|
JP2012102090A
(ja)
*
|
2010-10-15 |
2012-05-31 |
Sumitomo Chemical Co Ltd |
ピリミジン化合物およびその有害生物防除用途
|
|
EP2635557A2
(de)
|
2010-11-01 |
2013-09-11 |
Portola Pharmaceuticals, Inc. |
Nicotinamide als jak-kinasemodulatoren
|
|
CA2818542A1
(en)
|
2010-11-19 |
2012-05-24 |
Incyte Corporation |
Cyclobutyl substituted pyrrolopyridine and pyrrolopyrimidine derivatives as jak inhibitors
|
|
WO2012068440A1
(en)
|
2010-11-19 |
2012-05-24 |
Incyte Corporation |
Heterocyclic-substituted pyrrolopyridines and pyrrolopyrimidines as jak inhibitors
|
|
TW201249844A
(en)
|
2010-12-20 |
2012-12-16 |
Incyte Corp |
N-(1-(substituted-phenyl)ethyl)-9H-purin-6-amines as PI3K inhibitors
|
|
WO2012112847A1
(en)
|
2011-02-18 |
2012-08-23 |
Novartis Pharma Ag |
mTOR/JAK INHIBITOR COMBINATION THERAPY
|
|
EP2680846A4
(de)
*
|
2011-03-01 |
2014-08-06 |
Npharmakon Llc |
Verwendung von n-(4-methoxyphenyl)-1-phenyl-1h-pyrazol-3-amin und verbindungen in zusammenhang damit
|
|
WO2012125629A1
(en)
|
2011-03-14 |
2012-09-20 |
Incyte Corporation |
Substituted diamino-pyrimidine and diamino-pyridine derivatives as pi3k inhibitors
|
|
US9126948B2
(en)
|
2011-03-25 |
2015-09-08 |
Incyte Holdings Corporation |
Pyrimidine-4,6-diamine derivatives as PI3K inhibitors
|
|
JP6272754B2
(ja)
|
2011-05-03 |
2018-01-31 |
アジオス ファーマシューティカルズ, インコーポレイテッド |
ピルビン酸キナーゼ活性化剤の使用方法
|
|
CN102827170A
(zh)
|
2011-06-17 |
2012-12-19 |
安吉奥斯医药品有限公司 |
治疗活性组合物和它们的使用方法
|
|
CN102827073A
(zh)
|
2011-06-17 |
2012-12-19 |
安吉奥斯医药品有限公司 |
治疗活性组合物和它们的使用方法
|
|
MY165963A
(en)
|
2011-06-20 |
2018-05-18 |
Incyte Holdings Corp |
Azetidinyl phenyl, pyridyl or pyrazinyl carboxamide derivatives as jak inhibitors
|
|
CA2844507A1
(en)
|
2011-08-10 |
2013-02-14 |
Novartis Pharma Ag |
Jak pi3k/mtor combination therapy
|
|
TW201313721A
(zh)
|
2011-08-18 |
2013-04-01 |
Incyte Corp |
作為jak抑制劑之環己基氮雜環丁烷衍生物
|
|
BR112014004741B1
(pt)
|
2011-08-30 |
2021-10-13 |
Chdi Foundation, Inc |
Entidade química, seu uso e composição farmacêutica compreendendo a mesma
|
|
AU2012300246A1
(en)
|
2011-08-30 |
2014-03-06 |
Chdi Foundation, Inc. |
Kynurenine-3-monooxygenase inhibitors, pharmaceutical compositions, and methods of use thereof
|
|
UA121539C2
(uk)
|
2011-09-02 |
2020-06-25 |
Інсайт Холдинґс Корпорейшн |
Гетероцикліламіни як інгібітори рі3к
|
|
UA111854C2
(uk)
|
2011-09-07 |
2016-06-24 |
Інсайт Холдінгс Корпорейшн |
Способи і проміжні сполуки для отримання інгібіторів jak
|
|
WO2013049591A2
(en)
*
|
2011-09-29 |
2013-04-04 |
Verseon Corporation |
Dual inhibitor compounds and methods of use thereof
|
|
SG11201402570QA
(en)
|
2011-11-23 |
2014-06-27 |
Portola Pharm Inc |
Pyrazine kinase inhibitors
|
|
LT2800743T
(lt)
|
2012-01-06 |
2018-06-25 |
Agios Pharmaceuticals, Inc. |
Terapiškai aktyvūs junginiai ir jų panaudojimo būdai
|
|
US9474779B2
(en)
|
2012-01-19 |
2016-10-25 |
Agios Pharmaceuticals, Inc. |
Therapeutically active compositions and their methods of use
|
|
JP2015507007A
(ja)
*
|
2012-02-14 |
2015-03-05 |
ジーアールエル |
抗ウイルス性の特性を有する小分子
|
|
AR090548A1
(es)
|
2012-04-02 |
2014-11-19 |
Incyte Corp |
Azaheterociclobencilaminas biciclicas como inhibidores de pi3k
|
|
AU2013258107B2
(en)
|
2012-05-08 |
2017-06-22 |
Bayer Pharma Aktiengesellschaft |
Method for the preparation of triazole compounds
|
|
TW201406761A
(zh)
|
2012-05-18 |
2014-02-16 |
Incyte Corp |
做爲jak抑制劑之哌啶基環丁基取代之吡咯并吡啶及吡咯并嘧啶衍生物
|
|
LT3495367T
(lt)
|
2012-06-13 |
2021-02-25 |
Incyte Holdings Corporation |
Pakeistieji tricikliniai junginiai, kaip fgfr inhibitoriai
|
|
US20140010783A1
(en)
*
|
2012-07-06 |
2014-01-09 |
Hoffmann-La Roche Inc. |
Antiviral compounds
|
|
US20150148292A1
(en)
*
|
2012-07-09 |
2015-05-28 |
Emory University |
Bone morphogenetic protein pathway activation, compositions for ossification, and methods related thereto
|
|
CN104870454B
(zh)
|
2012-08-07 |
2020-03-03 |
詹森药业有限公司 |
用于制备杂环酯衍生物的方法
|
|
CN107266405A
(zh)
|
2012-08-07 |
2017-10-20 |
詹森药业有限公司 |
用于制备c‑fms激酶抑制剂的方法
|
|
JP6407504B2
(ja)
|
2012-09-21 |
2018-10-17 |
アログ・ファーマシューティカルズ・インコーポレイテッドArog Pharmaceuticals,Inc. |
恒常的に活性であるリン酸化型flt3キナーゼの阻害方法
|
|
US9676756B2
(en)
|
2012-10-08 |
2017-06-13 |
Portola Pharmaceuticals, Inc. |
Substituted pyrimidinyl kinase inhibitors
|
|
NZ706999A
(en)
|
2012-10-15 |
2018-12-21 |
Agios Pharmaceuticals Inc |
Inhibitors of mutant isocitrate dehydrogenase and therapeutical uses thereof
|
|
JP6359546B2
(ja)
|
2012-11-01 |
2018-07-18 |
インサイト・ホールディングス・コーポレイションIncyte Holdings Corporation |
Jak阻害薬としての三環式縮合チオフェン誘導体
|
|
TWI761825B
(zh)
|
2012-11-15 |
2022-04-21 |
美商英塞特控股公司 |
盧梭利替尼之緩釋性劑型
|
|
BR112015016282A2
(en)
|
2013-01-07 |
2017-07-11 |
Arog Pharmaceuticals, Inc. |
crenolanib for treatment of mutated flt3 proliferative disorders
|
|
TWI841376B
(zh)
|
2013-03-01 |
2024-05-01 |
美商英塞特控股公司 |
吡唑并嘧啶衍生物治療PI3Kδ相關病症之用途
|
|
CA2900892A1
(en)
|
2013-03-05 |
2014-09-12 |
F. Hoffmann-La Roche Ag |
Antiviral compounds
|
|
WO2014135483A1
(en)
*
|
2013-03-05 |
2014-09-12 |
F. Hoffmann-La Roche Ag |
Antiviral compounds
|
|
MX384910B
(es)
|
2013-03-06 |
2025-03-14 |
Incyte Holdings Corp |
Procesos e intermedios para hacer un inhibidor de jak.
|
|
JP6163214B2
(ja)
|
2013-03-06 |
2017-07-12 |
エフ.ホフマン−ラ ロシュ アーゲーF. Hoffmann−La Roche Aktiengesellschaft |
抗ウイルス化合物
|
|
KR20150139955A
(ko)
|
2013-04-09 |
2015-12-14 |
보스톤 바이오메디칼, 인크. |
암 치료에 사용하기 위한 2-아세틸나프토[2,3-b]푸란-4,9-디온
|
|
LT2986610T
(lt)
|
2013-04-19 |
2018-04-10 |
Incyte Holdings Corporation |
Bicikliniai heterociklai, kaip fgfr inhibitoriai
|
|
PE20200527A1
(es)
|
2013-05-17 |
2020-03-09 |
Incyte Corp |
Derivados del bipirazol como inhibidores jak
|
|
US10376510B2
(en)
|
2013-07-11 |
2019-08-13 |
Agios Pharmaceuticals, Inc. |
2,4- or 4,6-diaminopyrimidine compounds as IDH2 mutants inhibitors for the treatment of cancer
|
|
ES2807582T3
(es)
|
2013-07-11 |
2021-02-23 |
Agios Pharmaceuticals Inc |
Compuestos N,6-bis(aril o heteroaril)-1,3,5-triazina-2,4-diamina como inhibidores de mutantes IDH2 para el tratamiento del cáncer
|
|
WO2015003360A2
(en)
|
2013-07-11 |
2015-01-15 |
Agios Pharmaceuticals, Inc. |
Therapeutically active compounds and their methods of use
|
|
WO2015003355A2
(en)
|
2013-07-11 |
2015-01-15 |
Agios Pharmaceuticals, Inc. |
Therapeutically active compounds and their methods of use
|
|
WO2015010297A1
(en)
|
2013-07-25 |
2015-01-29 |
Agios Pharmaceuticals, Inc. |
Therapeutically active compounds and their methods of use
|
|
SG11201600815WA
(en)
|
2013-08-07 |
2016-03-30 |
Incyte Corp |
Sustained release dosage forms for a jak1 inhibitor
|
|
WO2015026818A1
(en)
|
2013-08-20 |
2015-02-26 |
Incyte Corporation |
Survival benefit in patients with solid tumors with elevated c-reactive protein levels
|
|
US10463658B2
(en)
|
2013-10-25 |
2019-11-05 |
Videra Pharmaceuticals, Llc |
Method of inhibiting FLT3 kinase
|
|
SG10201807952PA
(en)
|
2014-02-28 |
2018-10-30 |
Incyte Corp |
Jak1 inhibitors for the treatment of myelodysplastic syndromes
|
|
US9968595B2
(en)
|
2014-03-14 |
2018-05-15 |
Agios Pharmaceuticals, Inc. |
Pharmaceutical compositions of therapeutically active compounds
|
|
CN106413716B
(zh)
|
2014-04-08 |
2020-03-27 |
因赛特公司 |
通过jak和pi3k抑制剂组合治疗b细胞恶性肿瘤
|
|
BR112016025427A2
(pt)
|
2014-04-30 |
2017-08-15 |
Incyte Corp |
processos de preparação de um inibidor de jak1 e formas do mesmo
|
|
WO2015184305A1
(en)
|
2014-05-30 |
2015-12-03 |
Incyte Corporation |
TREATMENT OF CHRONIC NEUTROPHILIC LEUKEMIA (CNL) AND ATYPICAL CHRONIC MYELOID LEUKEMIA (aCML) BY INHIBITORS OF JAK1
|
|
US10077277B2
(en)
|
2014-06-11 |
2018-09-18 |
Incyte Corporation |
Bicyclic heteroarylaminoalkyl phenyl derivatives as PI3K inhibitors
|
|
AU2015289492B2
(en)
|
2014-07-17 |
2020-02-20 |
Chdi Foundation, Inc. |
Methods and compositions for treating HIV-related disorders
|
|
BR112017002001B1
(pt)
|
2014-07-31 |
2022-10-25 |
INSERM (Institut National de la Santé et de la Recherche Médicale) |
Compostos e composição farmacêutica
|
|
WO2016130501A1
(en)
|
2015-02-09 |
2016-08-18 |
Incyte Corporation |
Aza-heteroaryl compounds as pi3k-gamma inhibitors
|
|
SG11201706287PA
(en)
|
2015-02-20 |
2017-09-28 |
Incyte Corp |
Bicyclic heterocycles as fgfr inhibitors
|
|
MA41551A
(fr)
|
2015-02-20 |
2017-12-26 |
Incyte Corp |
Hétérocycles bicycliques utilisés en tant qu'inhibiteurs de fgfr4
|
|
UA122332C2
(uk)
|
2015-02-27 |
2020-10-26 |
Інсайт Корпорейшн |
Солі інгібітора pi3k і способи їх отримання
|
|
US20160362424A1
(en)
|
2015-05-11 |
2016-12-15 |
Incyte Corporation |
Salts of (s)-7-(1-(9h-purin-6-ylamino)ethyl)-6-(3-fluorophenyl)-3-methyl-5h-thiazolo[3,2-a]pyrimidin-5-one
|
|
WO2016183063A1
(en)
|
2015-05-11 |
2016-11-17 |
Incyte Corporation |
Crystalline forms of a pi3k inhibitor
|
|
WO2016183060A1
(en)
|
2015-05-11 |
2016-11-17 |
Incyte Corporation |
Process for the synthesis of a phosphoinositide 3-kinase inhibitor
|
|
RS64777B1
(sr)
|
2015-06-11 |
2023-11-30 |
Agios Pharmaceuticals Inc |
Postupci upotrebe aktivatora piruvat kinaze
|
|
UA123401C2
(uk)
|
2015-10-15 |
2021-03-31 |
Аджиос Фармасьютікалз, Інк. |
Комбінована терапія для лікування злоякісних пухлин
|
|
DK3362066T3
(da)
|
2015-10-15 |
2021-11-22 |
Les Laboratoires Servier Sas |
Kombinationsterapi til behandling af maligniteter
|
|
TWI744256B
(zh)
|
2015-11-06 |
2021-11-01 |
美商英塞特公司 |
作為PI3K-γ抑制劑之雜環化合物
|
|
TW201734003A
(zh)
|
2016-01-05 |
2017-10-01 |
英塞特公司 |
作為PI3K-γ抑制劑之吡啶及嘧啶化合物
|
|
EP3241830A1
(de)
|
2016-05-04 |
2017-11-08 |
Bayer CropScience Aktiengesellschaft |
Kondensierte bicyclische heterocyclen-derivate als schädlingsbekämpfungsmittel
|
|
EP3254698A1
(de)
|
2016-06-08 |
2017-12-13 |
Universite De Montpellier |
Flt3-rezeptor-inhibitoren bei niedriger dosierung zur behandlung von neuropathischem schmerz
|
|
AR108875A1
(es)
|
2016-06-24 |
2018-10-03 |
Incyte Corp |
COMPUESTOS HETEROCÍCLICOS COMO INHIBIDORES DE PI3K-g
|
|
WO2018014802A1
(en)
|
2016-07-18 |
2018-01-25 |
National Institute Of Biological Sciences, Beijing |
Apoptosis inhibitors
|
|
EP3359155A4
(de)
|
2016-11-02 |
2019-05-22 |
Arog Pharmaceuticals, Inc. |
Crenolanib zur behandlung von mutationen im zusammenhang mit flt3-mutierten proliferativen erkrankungen
|
|
US12534764B2
(en)
|
2016-11-02 |
2026-01-27 |
Arog Pharmaceuticals, Inc. |
Crenolanib for treating FLT3 mutated proliferative disorders associated mutations
|
|
JP7106563B2
(ja)
|
2016-11-29 |
2022-07-26 |
スミトモ ファーマ オンコロジー, インコーポレイテッド |
ナフトフラン誘導体、その調製、および使用方法
|
|
RU2629360C1
(ru)
*
|
2016-12-08 |
2017-08-29 |
Федеральное государственное бюджетное образовательное учреждение высшего образования "Московский технологический университет" |
НОВЫЕ 1-β-D-РИБОФУРАНОЗИЛ-3-(5-ЗАМЕЩЕННЫЕ-1,2,4-ОКСАДИАЗОЛ-3-ИЛ)-1,2,4-ТРИАЗОЛЫ, ОБЛАДАЮЩИЕ ПРОТИВОВИРУСНЫМИ СВОЙСТВАМИ, И СПОСОБ ИХ ПОЛУЧЕНИЯ
|
|
JP2020519665A
(ja)
|
2017-05-17 |
2020-07-02 |
アンセルム(アンスティテュト ナショナル ド ラ サンテ エ ド ラ ルシェルシュ メディカル) |
オピオイドによる痛みの処置を改善する為のflt3阻害剤
|
|
WO2018213424A1
(en)
|
2017-05-17 |
2018-11-22 |
Boston Biomedical, Inc. |
Methods for treating cancer
|
|
AR111960A1
(es)
|
2017-05-26 |
2019-09-04 |
Incyte Corp |
Formas cristalinas de un inhibidor de fgfr y procesos para su preparación
|
|
WO2019057649A1
(en)
|
2017-09-19 |
2019-03-28 |
INSERM (Institut National de la Santé et de la Recherche Médicale) |
METHODS AND PHARMACEUTICAL COMPOSITIONS FOR THE TREATMENT OF ACUTE MYELOID LEUKEMIA
|
|
AU2018350980C1
(en)
|
2017-10-18 |
2024-12-12 |
Incyte Corporation |
Condensed imidazole derivatives substituted by tertiary hydroxy groups as pi3k-y gamma inhibitors
|
|
US10596161B2
(en)
|
2017-12-08 |
2020-03-24 |
Incyte Corporation |
Low dose combination therapy for treatment of myeloproliferative neoplasms
|
|
US11306079B2
(en)
|
2017-12-21 |
2022-04-19 |
Incyte Corporation |
3-(5-amino-pyrazin-2-yl)-benzenesulfonamide derivatives and related compounds as PI3K-gamma kinase inhibitors
|
|
GB201801226D0
(en)
*
|
2018-01-25 |
2018-03-14 |
Redx Pharma Plc |
Modulators of Rho-associated protein kinase
|
|
JP7393348B2
(ja)
|
2018-01-30 |
2023-12-06 |
インサイト・コーポレイション |
(1-(3-フルオロ-2(トリフルオロメチル)イソニコチニル)ピぺリジン―4-オン)を作製するためのプロセス及び中間体
|
|
UA127519C2
(uk)
|
2018-02-16 |
2023-09-20 |
Інсайт Корпорейшн |
Інгібітори шляху jak1, призначені для лікування порушень, пов'язаних із цитокінами
|
|
BR122023024273A2
(pt)
|
2018-02-27 |
2024-02-20 |
Incyte Corporation |
Compostos imidazopirimidinas e triazolopirimidinas, seus usos, método para inibir uma atividade de um receptor de adenosina e composição farmacêutica dos mesmos
|
|
MD3762368T2
(ro)
|
2018-03-08 |
2022-07-31 |
Incyte Corp |
Compuși diol aminopirazină ca inhibitori ai PI3K-Y
|
|
CN113768934A
(zh)
|
2018-03-30 |
2021-12-10 |
因赛特公司 |
使用jak抑制剂治疗化脓性汗腺炎
|
|
JP7565798B2
(ja)
|
2018-03-30 |
2024-10-11 |
インサイト・コーポレイション |
炎症性皮膚疾患のバイオマーカー
|
|
US11220510B2
(en)
|
2018-04-09 |
2022-01-11 |
Incyte Corporation |
Pyrrole tricyclic compounds as A2A / A2B inhibitors
|
|
SG11202010068VA
(en)
|
2018-04-25 |
2020-11-27 |
Bayer Ag |
Novel heteroaryl-triazole and heteroaryl-tetrazole compounds as pesticides
|
|
MX2020011718A
(es)
|
2018-05-04 |
2021-02-15 |
Incyte Corp |
Formas solidas de un inhibidor de receptores del factor de crecimiento de fibroblastos (fgfr) y procesos para prepararlas.
|
|
ES3061844T3
(en)
|
2018-05-04 |
2026-04-07 |
Incyte Corp |
Salts of an fgfr inhibitor
|
|
EP3810610A1
(de)
|
2018-05-18 |
2021-04-28 |
Incyte Corporation |
Kondensierte pyrimidinderivate als a2a/a2b-inhibitoren
|
|
ES2929415T3
(es)
|
2018-05-25 |
2022-11-29 |
Incyte Corp |
Compuestos heterocíclicos tricíclicos como activadores de STING
|
|
MX2020012826A
(es)
|
2018-06-01 |
2021-03-09 |
Incyte Corp |
Regimen de dosificacion para el tratamiento de trastornos relacionados con fosfatidilinositol 3-cinasas (pi3k).
|
|
US11684625B2
(en)
*
|
2018-06-04 |
2023-06-27 |
Ac Immune Sa |
Compounds for the treatment, alleviation or prevention of disorders associated with tau aggregates
|
|
US10980788B2
(en)
|
2018-06-08 |
2021-04-20 |
Agios Pharmaceuticals, Inc. |
Therapy for treating malignancies
|
|
US11046658B2
(en)
|
2018-07-02 |
2021-06-29 |
Incyte Corporation |
Aminopyrazine derivatives as PI3K-γ inhibitors
|
|
AU2019297361B2
(en)
|
2018-07-05 |
2024-06-27 |
Incyte Corporation |
Fused pyrazine derivatives as A2A / A2B inhibitors
|
|
US10875872B2
(en)
|
2018-07-31 |
2020-12-29 |
Incyte Corporation |
Heteroaryl amide compounds as sting activators
|
|
US11008344B2
(en)
|
2018-07-31 |
2021-05-18 |
Incyte Corporation |
Tricyclic heteroaryl compounds as STING activators
|
|
WO2020036133A1
(ja)
*
|
2018-08-17 |
2020-02-20 |
クミアイ化学工業株式会社 |
3-(1h-1,2,4-トリアゾール-1-イル)安息香酸アミド誘導体及び有害生物防除剤
|
|
CR20250050A
(es)
|
2018-09-05 |
2025-03-19 |
Incyte Corp |
Formas cristalinas de un inhibidor de fosfoinositida 3–quinasa (pi3k) (divisional 2021-0165)
|
|
US11066404B2
(en)
|
2018-10-11 |
2021-07-20 |
Incyte Corporation |
Dihydropyrido[2,3-d]pyrimidinone compounds as CDK2 inhibitors
|
|
US11078204B2
(en)
|
2018-11-13 |
2021-08-03 |
Incyte Corporation |
Heterocyclic derivatives as PI3K inhibitors
|
|
WO2020102216A1
(en)
|
2018-11-13 |
2020-05-22 |
Incyte Corporation |
Substituted heterocyclic derivatives as pi3k inhibitors
|
|
US11161838B2
(en)
|
2018-11-13 |
2021-11-02 |
Incyte Corporation |
Heterocyclic derivatives as PI3K inhibitors
|
|
US11596692B1
(en)
|
2018-11-21 |
2023-03-07 |
Incyte Corporation |
PD-L1/STING conjugates and methods of use
|
|
WO2020146237A1
(en)
|
2019-01-07 |
2020-07-16 |
Incyte Corporation |
Heteroaryl amide compounds as sting activators
|
|
TWI829857B
(zh)
|
2019-01-29 |
2024-01-21 |
美商英塞特公司 |
作為a2a / a2b抑制劑之吡唑并吡啶及三唑并吡啶
|
|
US11384083B2
(en)
|
2019-02-15 |
2022-07-12 |
Incyte Corporation |
Substituted spiro[cyclopropane-1,5′-pyrrolo[2,3-d]pyrimidin]-6′(7′h)-ones as CDK2 inhibitors
|
|
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(de)
|
2019-02-15 |
2021-12-22 |
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Cyclinabhängige kinase-2-biomarker und deren verwendungen
|
|
TW202100520A
(zh)
|
2019-03-05 |
2021-01-01 |
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作為cdk2 抑制劑之吡唑基嘧啶基胺化合物
|
|
US11628162B2
(en)
|
2019-03-08 |
2023-04-18 |
Incyte Corporation |
Methods of treating cancer with an FGFR inhibitor
|
|
WO2020205560A1
(en)
|
2019-03-29 |
2020-10-08 |
Incyte Corporation |
Sulfonylamide compounds as cdk2 inhibitors
|
|
US11440914B2
(en)
|
2019-05-01 |
2022-09-13 |
Incyte Corporation |
Tricyclic amine compounds as CDK2 inhibitors
|
|
US11447494B2
(en)
|
2019-05-01 |
2022-09-20 |
Incyte Corporation |
Tricyclic amine compounds as CDK2 inhibitors
|
|
JP7532511B2
(ja)
|
2019-06-10 |
2024-08-13 |
インサイト・コーポレイション |
Jak阻害剤による尋常性白斑の局所治療
|
|
US11591329B2
(en)
|
2019-07-09 |
2023-02-28 |
Incyte Corporation |
Bicyclic heterocycles as FGFR inhibitors
|
|
US12610949B2
(en)
|
2019-07-23 |
2026-04-28 |
Bayer Aktiengesellschaft |
Heteroaryl-triazole compounds as pesticides
|
|
PH12022550166A1
(en)
|
2019-07-23 |
2022-11-14 |
Bayer Ag |
Novel heteroaryl-triazole compounds as pesticides
|
|
EP4007602A1
(de)
|
2019-08-01 |
2022-06-08 |
Incyte Corporation |
Dosierungsschema für einen ido-inhibitor
|
|
CN116348458A
(zh)
|
2019-08-14 |
2023-06-27 |
因赛特公司 |
作为cdk2抑制剂的咪唑基嘧啶基胺化合物
|
|
MX2022002219A
(es)
|
2019-08-26 |
2022-06-14 |
Incyte Corp |
Triazolopirimidinas como inhibidores de a2a/a2b.
|
|
US12122767B2
(en)
|
2019-10-01 |
2024-10-22 |
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Bicyclic heterocycles as FGFR inhibitors
|
|
CN119930611A
(zh)
|
2019-10-11 |
2025-05-06 |
因赛特公司 |
作为cdk2抑制剂的双环胺
|
|
TWI891666B
(zh)
|
2019-10-14 |
2025-08-01 |
美商英塞特公司 |
作為fgfr抑制劑之雙環雜環
|
|
US11992490B2
(en)
|
2019-10-16 |
2024-05-28 |
Incyte Corporation |
Use of JAK1 inhibitors for the treatment of cutaneous lupus erythematosus and Lichen planus (LP)
|
|
US11566028B2
(en)
|
2019-10-16 |
2023-01-31 |
Incyte Corporation |
Bicyclic heterocycles as FGFR inhibitors
|
|
JP7518900B2
(ja)
|
2019-10-16 |
2024-07-18 |
インサイト・コーポレイション |
皮膚エリテマトーデス及び扁平苔癬(lp)の治療のためのjak1阻害剤の使用
|
|
WO2021113462A1
(en)
|
2019-12-04 |
2021-06-10 |
Incyte Corporation |
Derivatives of an fgfr inhibitor
|
|
CA3163875A1
(en)
|
2019-12-04 |
2021-06-10 |
Incyte Corporation |
Tricyclic heterocycles as fgfr inhibitors
|
|
US12012409B2
(en)
|
2020-01-15 |
2024-06-18 |
Incyte Corporation |
Bicyclic heterocycles as FGFR inhibitors
|
|
PH12022552347A1
(en)
|
2020-03-06 |
2024-01-29 |
Incyte Corp |
Combination therapy comprising axl/mer and pd-1/pd-l1 inhibitors
|
|
CA3179692A1
(en)
|
2020-04-16 |
2021-10-21 |
Incyte Corporation |
Fused tricyclic kras inhibitors
|
|
GB202006382D0
(en)
|
2020-04-30 |
2020-06-17 |
Spermatech As |
Use
|
|
WO2021231526A1
(en)
|
2020-05-13 |
2021-11-18 |
Incyte Corporation |
Fused pyrimidine compounds as kras inhibitors
|
|
JP7802696B2
(ja)
|
2020-06-02 |
2026-01-20 |
インサイト・コーポレイション |
Jak1阻害剤の調製プロセス
|
|
US11833155B2
(en)
|
2020-06-03 |
2023-12-05 |
Incyte Corporation |
Combination therapy for treatment of myeloproliferative neoplasms
|
|
WO2022019998A1
(en)
|
2020-07-20 |
2022-01-27 |
Arog Pharmaceuticals, Inc. |
Crystal forms of crenolanib and methods of use thereof
|
|
US11999752B2
(en)
|
2020-08-28 |
2024-06-04 |
Incyte Corporation |
Vinyl imidazole compounds as inhibitors of KRAS
|
|
US20230364095A1
(en)
|
2020-09-16 |
2023-11-16 |
Incyte Corporation |
Topical treatment of vitiligo
|
|
WO2022072783A1
(en)
|
2020-10-02 |
2022-04-07 |
Incyte Corporation |
Bicyclic dione compounds as inhibitors of kras
|
|
WO2022090547A1
(en)
|
2020-10-30 |
2022-05-05 |
Dsm Ip Assets B.V. |
Production of carotenoids by fermentation
|
|
US11969420B2
(en)
|
2020-10-30 |
2024-04-30 |
Arog Pharmaceuticals, Inc. |
Combination therapy of crenolanib and apoptosis pathway agents for the treatment of proliferative disorders
|
|
JP2023552452A
(ja)
|
2020-12-08 |
2023-12-15 |
インサイト・コーポレイション |
白斑治療用のjak1経路阻害薬
|
|
WO2022155941A1
(en)
|
2021-01-25 |
2022-07-28 |
Qilu Regor Therapeutics Inc. |
Cdk2 inhibitors
|
|
WO2022206888A1
(en)
|
2021-03-31 |
2022-10-06 |
Qilu Regor Therapeutics Inc. |
Cdk2 inhibitors and use thereof
|
|
TW202304459A
(zh)
|
2021-04-12 |
2023-02-01 |
美商英塞特公司 |
包含fgfr抑制劑及nectin-4靶向劑之組合療法
|
|
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(de)
|
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2026-05-06 |
Incyte Corporation |
Jak1-pfad-hemmer zur behandlung von prurigo nodularis
|
|
JP2024522189A
(ja)
|
2021-06-09 |
2024-06-11 |
インサイト・コーポレイション |
Fgfr阻害剤としての三環式ヘテロ環
|
|
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(de)
|
2021-06-09 |
2024-04-17 |
Incyte Corporation |
Tricyclische heterocyclen als fgfr-inhibitoren
|
|
US11981671B2
(en)
|
2021-06-21 |
2024-05-14 |
Incyte Corporation |
Bicyclic pyrazolyl amines as CDK2 inhibitors
|
|
AU2022306671A1
(en)
|
2021-07-07 |
2024-01-25 |
Incyte Corporation |
Tricyclic compounds as inhibitors of kras
|
|
JP2024529347A
(ja)
|
2021-07-14 |
2024-08-06 |
インサイト・コーポレイション |
Krasの阻害剤としての三環式化合物
|
|
JP2024534187A
(ja)
|
2021-08-31 |
2024-09-18 |
インサイト・コーポレイション |
Krasの阻害剤としてのナフチリジン化合物
|
|
WO2023049697A1
(en)
|
2021-09-21 |
2023-03-30 |
Incyte Corporation |
Hetero-tricyclic compounds as inhibitors of kras
|
|
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(de)
|
2021-10-01 |
2024-08-07 |
Incyte Corporation |
Pyrazolochinolin-kras-hemmer
|
|
US20250034112A1
(en)
*
|
2021-10-13 |
2025-01-30 |
Yale University |
Improved selective jak2 inhibitors and methods of use
|
|
KR20240101561A
(ko)
|
2021-10-14 |
2024-07-02 |
인사이트 코포레이션 |
Kras의 저해제로서의 퀴놀린 화합물
|
|
WO2023091746A1
(en)
|
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2023-05-25 |
Incyte Corporation |
Combination therapy comprising an fgfr inhibitor and a kras inhibitor
|
|
US20230203010A1
(en)
|
2021-12-03 |
2023-06-29 |
Incyte Corporation |
Bicyclic amine cdk12 inhibitors
|
|
US11976073B2
(en)
|
2021-12-10 |
2024-05-07 |
Incyte Corporation |
Bicyclic amines as CDK2 inhibitors
|
|
US12084453B2
(en)
|
2021-12-10 |
2024-09-10 |
Incyte Corporation |
Bicyclic amines as CDK12 inhibitors
|
|
AR128043A1
(es)
|
2021-12-22 |
2024-03-20 |
Incyte Corp |
Sales y formas sólidas de un inhibidor de fgfr y procesos para su preparación
|
|
WO2023168686A1
(en)
|
2022-03-11 |
2023-09-14 |
Qilu Regor Therapeutics Inc. |
Substituted cyclopentanes as cdk2 inhibitors
|
|
TW202341982A
(zh)
|
2021-12-24 |
2023-11-01 |
大陸商上海齊魯銳格醫藥研發有限公司 |
Cdk2抑制劑及其用途
|
|
CR20240408A
(es)
|
2022-03-07 |
2024-11-22 |
Incyte Corp |
Formas sólidas, sales y procesos de preparación de un inhibidor de cdk2.
|
|
EP4540252A1
(de)
|
2022-06-14 |
2025-04-23 |
Incyte Corporation |
Feste formen eines jak-hemmers und verfahren zur herstellung davon
|
|
WO2023250430A1
(en)
|
2022-06-22 |
2023-12-28 |
Incyte Corporation |
Bicyclic amine cdk12 inhibitors
|
|
US20240101557A1
(en)
|
2022-07-11 |
2024-03-28 |
Incyte Corporation |
Fused tricyclic compounds as inhibitors of kras g12v mutants
|
|
WO2024030600A1
(en)
|
2022-08-05 |
2024-02-08 |
Incyte Corporation |
Treatment of urticaria using jak inhibitors
|
|
WO2024051667A1
(zh)
*
|
2022-09-05 |
2024-03-14 |
南京正大天晴制药有限公司 |
具有axl抑制活性的取代三唑化合物
|
|
WO2024218236A1
(en)
*
|
2023-04-18 |
2024-10-24 |
Centre National De La Recherche Scientifique |
3,5-diaminotriazole derivatives and uses thereof for treating ocular diseases
|
|
US20240390340A1
(en)
|
2023-04-18 |
2024-11-28 |
Incyte Corporation |
Pyrrolidine kras inhibitors
|
|
EP4698542A1
(de)
|
2023-04-18 |
2026-02-25 |
Incyte Corporation |
2-azabicyclo[2.2.1 heptan kras-inhibitoren
|
|
WO2024254245A1
(en)
|
2023-06-09 |
2024-12-12 |
Incyte Corporation |
Bicyclic amines as cdk2 inhibitors
|
|
WO2025080695A1
(en)
*
|
2023-10-10 |
2025-04-17 |
Collaborations Pharmaceuticals, Inc. |
1-sulfonyl-3-amino-1h-1,2,4-triazoles as yellow fever virus inhibitors
|
|
US20250163079A1
(en)
|
2023-11-01 |
2025-05-22 |
Incyte Corporation |
Kras inhibitors
|
|
US20250195536A1
(en)
|
2023-12-13 |
2025-06-19 |
Incyte Corporation |
Bicyclooctane kras inhibitors
|
|
AU2025271553A1
(en)
|
2024-08-26 |
2026-03-12 |
Incyte Corporation |
Topical skin formulations of a pharmaceutically acceptable salt of ruxolitinib
|
|
WO2026060143A1
(en)
|
2024-09-11 |
2026-03-19 |
Incyte Corporation |
Kras inhibitors
|
|
WO2026076207A1
(en)
|
2024-10-04 |
2026-04-09 |
Incyte Corporation |
Tricyclic heteroaryl compounds as inhibitors of tyk2 and/or jak1
|
|
US20260125391A1
(en)
|
2024-11-04 |
2026-05-07 |
Incyte Corporation |
Pyrimidine indoles as cdk4 inhibitors
|