ATE459621T1 - Benzisoxazolpiperidinverbindungen und verfahren zu deren anwendung - Google Patents

Benzisoxazolpiperidinverbindungen und verfahren zu deren anwendung

Info

Publication number
ATE459621T1
ATE459621T1 AT06751665T AT06751665T ATE459621T1 AT E459621 T1 ATE459621 T1 AT E459621T1 AT 06751665 T AT06751665 T AT 06751665T AT 06751665 T AT06751665 T AT 06751665T AT E459621 T1 ATE459621 T1 AT E459621T1
Authority
AT
Austria
Prior art keywords
benzisoxazolepiperidine
compounds
compositions
methods
invention includes
Prior art date
Application number
AT06751665T
Other languages
English (en)
Inventor
Daniel Coughlin
James White
Kazumi Shiosaki
David Hangauer
Michael Solomon
Dale Edgar
Original Assignee
Hypnion Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hypnion Inc filed Critical Hypnion Inc
Application granted granted Critical
Publication of ATE459621T1 publication Critical patent/ATE459621T1/de

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/20—Hypnotics; Sedatives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D261/00—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings
    • C07D261/20—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings condensed with carbocyclic rings or ring systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Anesthesiology (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Plural Heterocyclic Compounds (AREA)
AT06751665T 2005-04-26 2006-04-26 Benzisoxazolpiperidinverbindungen und verfahren zu deren anwendung ATE459621T1 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US67520205P 2005-04-26 2005-04-26
PCT/US2006/016057 WO2006116614A1 (en) 2005-04-26 2006-04-26 Benzisoxazole piperidine compounds and methods of use thereof

Publications (1)

Publication Number Publication Date
ATE459621T1 true ATE459621T1 (de) 2010-03-15

Family

ID=36754209

Family Applications (2)

Application Number Title Priority Date Filing Date
AT06751667T ATE461925T1 (de) 2005-04-26 2006-04-26 Benzisoxazolpiperidinverbindungen und verfahren zu deren anwendung
AT06751665T ATE459621T1 (de) 2005-04-26 2006-04-26 Benzisoxazolpiperidinverbindungen und verfahren zu deren anwendung

Family Applications Before (1)

Application Number Title Priority Date Filing Date
AT06751667T ATE461925T1 (de) 2005-04-26 2006-04-26 Benzisoxazolpiperidinverbindungen und verfahren zu deren anwendung

Country Status (15)

Country Link
US (3) US7494998B2 (de)
EP (2) EP1877405B1 (de)
JP (2) JP5049267B2 (de)
CN (1) CN101208314B (de)
AT (2) ATE461925T1 (de)
AU (1) AU2006239302B2 (de)
CA (2) CA2606473C (de)
CY (1) CY1110026T1 (de)
DE (2) DE602006013115D1 (de)
DK (1) DK1877390T3 (de)
ES (2) ES2341127T3 (de)
MX (1) MX2007013352A (de)
PL (1) PL1877390T3 (de)
PT (1) PT1877390E (de)
WO (1) WO2006116614A1 (de)

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US7762006B2 (en) * 2006-06-14 2010-07-27 Siestamed, Technologies Medical equipment drying device
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CN104069567A (zh) * 2007-03-19 2014-10-01 茵苏莱恩医药有限公司 药物输送设备
US9220837B2 (en) * 2007-03-19 2015-12-29 Insuline Medical Ltd. Method and device for drug delivery
US8622991B2 (en) 2007-03-19 2014-01-07 Insuline Medical Ltd. Method and device for drug delivery
EP2136863A2 (de) * 2007-03-19 2009-12-30 Insuline Medical Ltd. Vorrichtung zur abgabe von arzneimitteln und relevante verbindungen
JP5393677B2 (ja) 2007-08-15 2014-01-22 アリーナ ファーマシューティカルズ， インコーポレイテッド ５−ＨＴ２Ａセロトニン受容体に関連した障害の治療のための５−ＨＴ２Ａセロトニン受容体のモジュレーターとしてのイミダゾ［１，２−ａ］ピリジン誘導体
EP2231229A1 (de) 2007-12-18 2010-09-29 Insuline Medical Ltd. Wirkstofffreisetzungsvorrichtung mit sensor für geschlossenen kreislauf
US20110021538A1 (en) 2008-04-02 2011-01-27 Arena Pharmaceuticals, Inc. Processes for the preparation of pyrazole derivatives useful as modulators of the 5-ht2a serotonin receptor
US20090263449A1 (en) * 2008-04-09 2009-10-22 Surmodics, Inc. Delivery of nucleic acid complexes from materials including negatively charged groups
JP2010043063A (ja) 2008-05-09 2010-02-25 Agency For Science Technology & Research 川崎病の診断及び治療
HRP20180589T1 (hr) 2008-10-28 2018-05-18 Arena Pharmaceuticals, Inc. Pripravci modulatora serotoninskog receptora 5-ht2a koji su korisni za liječenje s njim povezanih poremećaja
WO2010062321A1 (en) 2008-10-28 2010-06-03 Arena Pharmaceuticals, Inc. Processes useful for the preparation of 1-[3-(4-bromo-2-methyl-2h-pyrazol-3-yl)-4-methoxy-phenyl]-3-(2,4-difluoro-phenyl)-urea and crystalline forms related thereto
KR20110086132A (ko) 2008-11-07 2011-07-27 인슐린 메디컬 엘티디 약물 전달 장치 및 방법
WO2010074753A1 (en) 2008-12-23 2010-07-01 Map Pharmaceuticals, Inc. Inhalation devices and related methods for administration of sedative hypnotic compounds
US8980891B2 (en) 2009-12-18 2015-03-17 Arena Pharmaceuticals, Inc. Crystalline forms of certain 3-phenyl-pyrazole derivatives as modulators of the 5-HT2A serotonin receptor useful for the treatment of disorders related thereto
US8565107B2 (en) 2010-09-24 2013-10-22 Hand Held Products, Inc. Terminal configurable for use within an unknown regulatory domain
RU2017145976A (ru) 2015-06-12 2019-07-15 Аксовант Сайенсиз Гмбх Производные диарил- и арилгетероарилмочевины, применимые для профилактики и лечения нарушения поведения во время REM-фазы сна
TW201720439A (zh) 2015-07-15 2017-06-16 Axovant Sciences Gmbh 用於預防及治療與神經退化性疾病相關的幻覺之作為５－ｈｔ２ａ血清素受體的二芳基及芳基雜芳基脲衍生物
GB201810092D0 (en) 2018-06-20 2018-08-08 Ctxt Pty Ltd Compounds
LT4299135T (lt) 2019-06-18 2025-09-10 Pfizer Inc. Benzizoksazolo sulfonamido dariniai
PT4082616T (pt) * 2019-12-24 2025-12-02 Sumitomo Pharma Co Ltd Derivado de amida ácida alifática
JP7655885B2 (ja) * 2021-06-30 2025-04-02 住友ファーマ株式会社 脂肪族酸アミド誘導体を含有する医薬組成物

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CN101208314B (zh) * 2005-04-26 2010-12-08 海普尼昂公司 苯并异*唑哌嗪化合物及其使用方法

Also Published As

Publication number Publication date
DE602006012650D1 (de) 2010-04-15
EP1877390A1 (de) 2008-01-16
DE602006013115D1 (de) 2010-05-06
DK1877390T3 (da) 2010-05-31
AU2006239302A1 (en) 2006-11-02
ES2340066T3 (es) 2010-05-28
CN101208314A (zh) 2008-06-25
EP1877405B1 (de) 2010-03-03
EP1877390B1 (de) 2010-03-24
US20090163514A1 (en) 2009-06-25
EP1877405A1 (de) 2008-01-16
MX2007013352A (es) 2008-03-26
AU2006239302B2 (en) 2011-07-07
CA2606471C (en) 2014-02-11
ES2341127T3 (es) 2010-06-15
PT1877390E (pt) 2010-05-31
WO2006116614A1 (en) 2006-11-02
JP5049267B2 (ja) 2012-10-17
US8129410B2 (en) 2012-03-06
PL1877390T3 (pl) 2010-08-31
ATE461925T1 (de) 2010-04-15
US8088778B2 (en) 2012-01-03
CA2606473C (en) 2013-08-13
JP2008539268A (ja) 2008-11-13
US7494998B2 (en) 2009-02-24
US20080214539A1 (en) 2008-09-04
US20070004752A1 (en) 2007-01-04
CY1110026T1 (el) 2015-01-14
JP2008539267A (ja) 2008-11-13
CA2606471A1 (en) 2006-11-02
CA2606473A1 (en) 2006-11-02
CN101208314B (zh) 2010-12-08

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