ATE462711T1 - Kristalline komplexe von fluticasone 2-furoat - Google Patents

Kristalline komplexe von fluticasone 2-furoat

Info

Publication number
ATE462711T1
ATE462711T1 AT03704759T AT03704759T ATE462711T1 AT E462711 T1 ATE462711 T1 AT E462711T1 AT 03704759 T AT03704759 T AT 03704759T AT 03704759 T AT03704759 T AT 03704759T AT E462711 T1 ATE462711 T1 AT E462711T1
Authority
AT
Austria
Prior art keywords
furoate
fluticasone
crystalline complexes
crystalline complex
crystalline
Prior art date
Application number
AT03704759T
Other languages
English (en)
Inventor
Keith Biggadike
Steven John Coote
Andrew Craig
David Malcolm Crowe
Victor Witold Jacewicz
Michael John Millan
Rosalyn Kay Nice
Brian Noga
John Frederick Seager
Andrew Lewis Theophilus
Original Assignee
Glaxo Group Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Glaxo Group Ltd filed Critical Glaxo Group Ltd
Application granted granted Critical
Publication of ATE462711T1 publication Critical patent/ATE462711T1/de

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J31/00—Normal steroids containing one or more sulfur atoms not belonging to a hetero ring
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/08—Antiallergic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A61P5/38—Drugs for disorders of the endocrine system of the suprarenal hormones
    • A61P5/44—Glucocorticosteroids; Drugs increasing or potentiating the activity of glucocorticosteroids
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J17/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, having an oxygen-containing hetero ring not condensed with the cyclopenta(a)hydrophenanthrene skeleton

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Diabetes (AREA)
  • Endocrinology (AREA)
  • Pulmonology (AREA)
  • Immunology (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Steroid Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Medicinal Preparation (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
AT03704759T 2002-02-04 2003-02-04 Kristalline komplexe von fluticasone 2-furoat ATE462711T1 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US10/067,010 US6777399B2 (en) 2000-08-05 2002-02-04 Anti-inflammatory androstane derivative compositions
PCT/GB2003/000478 WO2003066656A1 (en) 2002-02-04 2003-02-04 Crystalline complexes of fluticasone 2-furoate

Publications (1)

Publication Number Publication Date
ATE462711T1 true ATE462711T1 (de) 2010-04-15

Family

ID=27732223

Family Applications (1)

Application Number Title Priority Date Filing Date
AT03704759T ATE462711T1 (de) 2002-02-04 2003-02-04 Kristalline komplexe von fluticasone 2-furoat

Country Status (8)

Country Link
US (3) US6777399B2 (de)
EP (1) EP1472272B1 (de)
JP (1) JP4508651B2 (de)
AT (1) ATE462711T1 (de)
AU (1) AU2003207019A1 (de)
DE (1) DE60331891D1 (de)
ES (1) ES2343315T3 (de)
WO (1) WO2003066656A1 (de)

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GB0615108D0 (en) * 2006-07-28 2006-09-06 Glaxo Group Ltd Novel formulations
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WO2010016931A2 (en) * 2008-08-07 2010-02-11 Plus Chemicals Sa Polymorphs of fluticasone furoate and process for preparation thereof
WO2010108107A1 (en) 2009-03-19 2010-09-23 Plus Chemicals Sa Polymorphs of fluticasone furoate and processes for preparation thereof
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EP1472272B1 (de) 2010-03-31
JP4508651B2 (ja) 2010-07-21
AU2003207019A1 (en) 2003-09-02
US20050043284A1 (en) 2005-02-24
EP1472272A1 (de) 2004-11-03
WO2003066656A1 (en) 2003-08-14
US6777399B2 (en) 2004-08-17
ES2343315T3 (es) 2010-07-28
US20030153542A1 (en) 2003-08-14
JP2005527497A (ja) 2005-09-15
US20040224932A1 (en) 2004-11-11
US7592329B2 (en) 2009-09-22
DE60331891D1 (de) 2010-05-12

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