ATE473730T1 - Verwendung von 3-positions-cyclosporin-derivaten für haarwachstum - Google Patents

Verwendung von 3-positions-cyclosporin-derivaten für haarwachstum

Info

Publication number: ATE473730T1
Authority: AT; Austria
Prior art keywords: hair growth; cyclosporine derivatives; active ingredient; cyclosporin; cyclosporine
Prior art date: 2001-05-11

Application number

AT02728237T

Other languages

English (en)

Inventor

Sang-Nyun Kim

Ho-Jeong Ahn

Chang-Woo Lee

Min-Ho Lee

Jung-Hun Kim

Jong-Il Kim

Seung-Jin Kim

Ho-Song Cho

Heon-Sik Lee

Hyung-Jin Kim

Original Assignee

Lg Household & Health Care Ltd

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2001-05-11

Filing date

2002-05-11

Publication date

2010-07-15

2002-05-11 Application filed by Lg Household & Health Care Ltd filed Critical Lg Household & Health Care Ltd

2010-07-15 Application granted granted Critical

2010-07-15 Publication of ATE473730T1 publication Critical patent/ATE473730T1/de

Links

PMATZTZNYRCHOR-CGLBZJNRSA-N Cyclosporin A Chemical class CC[C@@H]1NC(=O)[C@H]([C@H](O)[C@H](C)C\C=C\C)N(C)C(=O)[C@H](C(C)C)N(C)C(=O)[C@H](CC(C)C)N(C)C(=O)[C@H](CC(C)C)N(C)C(=O)[C@@H](C)NC(=O)[C@H](C)NC(=O)[C@H](CC(C)C)N(C)C(=O)[C@H](C(C)C)NC(=O)[C@H](CC(C)C)N(C)C(=O)CN(C)C1=O PMATZTZNYRCHOR-CGLBZJNRSA-N 0.000 title abstract 3
230000003779 hair growth Effects 0.000 title abstract 3
239000004480 active ingredient Substances 0.000 abstract 2
230000001737 promoting effect Effects 0.000 abstract 2

Classifications

- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K8/00—Cosmetics or similar toiletry preparations
- A61K8/18—Cosmetics or similar toiletry preparations characterised by the composition
- A61K8/30—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds
- A61K8/40—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing nitrogen
- A61K8/44—Aminocarboxylic acids or derivatives thereof, e.g. aminocarboxylic acids containing sulfur; Salts; Esters or N-acylated derivatives thereof
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
- A61K38/04—Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
- A61K38/12—Cyclic peptides, e.g. bacitracins; Polymyxins; Gramicidins S, C; Tyrocidins A, B or C
- A61K38/13—Cyclosporins
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K8/00—Cosmetics or similar toiletry preparations
- A61K8/18—Cosmetics or similar toiletry preparations characterised by the composition
- A61K8/30—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds
- A61K8/64—Proteins; Peptides; Derivatives or degradation products thereof
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A61P17/14—Drugs for dermatological disorders for baldness or alopecia
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/10—Antimycotics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A61P33/02—Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/02—Immunomodulators
- A61P37/06—Immunosuppressants, e.g. drugs for graft rejection
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61Q—SPECIFIC USE OF COSMETICS OR SIMILAR TOILETRY PREPARATIONS
- A61Q5/00—Preparations for care of the hair
- A61Q5/12—Preparations containing hair conditioners
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61Q—SPECIFIC USE OF COSMETICS OR SIMILAR TOILETRY PREPARATIONS
- A61Q7/00—Preparations for affecting hair growth
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K7/00—Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
- C07K7/64—Cyclic peptides containing only normal peptide links
- C07K7/645—Cyclosporins; Related peptides

Landscapes

Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
General Health & Medical Sciences (AREA)
Veterinary Medicine (AREA)
Animal Behavior & Ethology (AREA)
Public Health (AREA)
Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Organic Chemistry (AREA)
Dermatology (AREA)
Pharmacology & Pharmacy (AREA)
Epidemiology (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Immunology (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
General Chemical & Material Sciences (AREA)
Chemical Kinetics & Catalysis (AREA)
Proteomics, Peptides & Aminoacids (AREA)
Birds (AREA)
Gastroenterology & Hepatology (AREA)
Oncology (AREA)
Communicable Diseases (AREA)
Biochemistry (AREA)
Biophysics (AREA)
Genetics & Genomics (AREA)
Molecular Biology (AREA)
Virology (AREA)
Tropical Medicine & Parasitology (AREA)
Transplantation (AREA)
Cosmetics (AREA)
Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Peptides Or Proteins (AREA)

AT02728237T 2001-05-11 2002-05-11 Verwendung von 3-positions-cyclosporin-derivaten für haarwachstum ATE473730T1 (de)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
KR10-2001-0025682A KR100465012B1 (ko)	2001-05-11	2001-05-11	모발 성장 효과를 갖는 사이클로스포린 3 위치 유도체를유효성분으로 하는 모발 성장 촉진제
PCT/KR2002/000879 WO2002092032A1 (en)	2001-05-11	2002-05-11	Use of 3-position cyclosporin derivatives for hair growth

Publications (1)

Publication Number	Publication Date
ATE473730T1 true ATE473730T1 (de)	2010-07-15

Family

ID=19709334

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
AT02728237T ATE473730T1 (de)	2001-05-11	2002-05-11	Verwendung von 3-positions-cyclosporin-derivaten für haarwachstum

Country Status (17)

Country	Link
US (2)	US6790830B2 (de)
EP (1)	EP1387660B1 (de)
JP (1)	JP4214181B2 (de)
KR (1)	KR100465012B1 (de)
CN (1)	CN1248671C (de)
AT (1)	ATE473730T1 (de)
AU (1)	AU2002258271B2 (de)
BR (1)	BRPI0209619B8 (de)
CA (1)	CA2446971C (de)
DE (1)	DE60237003D1 (de)
ES (1)	ES2348225T3 (de)
MX (1)	MXPA03010027A (de)
PL (1)	PL208536B1 (de)
RU (1)	RU2291682C2 (de)
TR (1)	TR200301931T2 (de)
WO (1)	WO2002092032A1 (de)
ZA (1)	ZA200308532B (de)

Families Citing this family (18)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
KR20020039528A (ko) *	2000-11-22	2002-05-27	조명재	사이클로스포린 7- 티오아미드 유도체를 유효성분으로하는 모발성장촉진제
KR100865211B1 (ko) *	2001-10-26	2008-10-23	주식회사 엘지생활건강	비면역 [감마 히드록시 엔-메틸 엘-루신4] 사이클로스포린 유도체를 유효성분으로 하는 항암 화학요법 기인 탈모증상 억제제
US6987090B2 (en) *	2002-05-09	2006-01-17	Lg Household & Health Care Ltd.	Use of 3-position cyclosporin derivatives for hair growth
US7538084B2 (en)	2003-03-17	2009-05-26	Amr Technology, Inc.	Cyclosporins
JP2008514701A (ja)	2004-09-29	2008-05-08	エーエムアールテクノロジーインコーポレイテッド	シクロスポリンアルキン類似体およびそれらの薬学的使用
JP2008514702A (ja)	2004-09-29	2008-05-08	エーエムアールテクノロジーインコーポレイテッド	新規シクロスポリン類似体およびそれらの薬学的使用
JP2008515886A (ja)	2004-10-06	2008-05-15	エーエムアールテクノロジーインコーポレイテッド	シクロスポリンアルキンおよびそれらの医用薬剤としての有用性
WO2007103311A2 (en) *	2006-03-06	2007-09-13	Rouse Martin D Jr	Thermal vaporizer apparatus
US7696165B2 (en)	2006-03-28	2010-04-13	Albany Molecular Research, Inc.	Use of cyclosporin alkyne analogues for preventing or treating viral-induced disorders
US7696166B2 (en)	2006-03-28	2010-04-13	Albany Molecular Research, Inc.	Use of cyclosporin alkyne/alkene analogues for preventing or treating viral-induced disorders
DE102008060549A1 (de)	2008-12-04	2010-06-10	MAX-PLANCK-Gesellschaft zur Förderung der Wissenschaften e.V.	Wirkstoff-Peptid-Konstrukt zur extrazellulären Anreicherung
WO2010138422A1 (en) *	2009-05-27	2010-12-02	Allergan, Inc.	Cyclosporin derivatives for enhancing the growth of hair
WO2010146622A1 (ja)	2009-06-15	2010-12-23	花王株式会社	Nfatシグナル阻害剤及びカルシニューリン阻害剤
BR112013014890B1 (pt)	2010-12-15	2023-10-24	Contravir Pharmaceuticals, Inc	Composto análogo de moléculas pertencentes à família ciclosporina, composição farmacêutica compreendendo o mesmo, uso terapêutico ou profilático do referido composto e processos para a preparação dos mesmos
RU2479872C1 (ru) *	2012-01-11	2013-04-20	Государственное бюджетное образовательное учреждение высшего профессионального образования "Курский государственный медицинский университет" Министерства здравоохранения и социального развития Российской Федерации	Способ коррекции ишемических нарушений, возникших в результате реперфузионной травмы печени
EP2705856A1 (de)	2012-09-07	2014-03-12	Deutsches Zentrum für Neurodegenerative Erkrankungen e.V.	Verbindungen zur Behandlung von neurodegenerativen Erkrankungen
KR102469342B1 (ko) *	2021-06-14	2022-11-21	주식회사 오리엔트바이오	환형 펩타이드를 포함하는 방출조절형 국소주사용 조성물 및 이의 제조방법
FR3162624A1 (fr) *	2024-05-31	2025-12-05	L'oreal	Composition comprenant au moins un actif antipelliculaire, au moins un agent antioxydant et au moins 35% en poids d’un monoalcool en C1 à C6

Family Cites Families (23)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
JPS60243008A (ja)	1984-05-17	1985-12-03	Wakamoto Pharmaceut Co Ltd	発毛養毛剤
EP0194972B1 (de) *	1985-03-11	1992-07-29	Sandoz Ag	Cyclosporine
JPS6219512A (ja)	1985-07-17	1987-01-28	Shiseido Co Ltd	養毛剤
JPS6219513A (ja)	1985-07-17	1987-01-28	Shiseido Co Ltd	養毛剤
CH679119A5 (de)	1988-05-13	1991-12-31	Sandoz Ag
GB8916901D0 (en) *	1989-07-24	1989-09-06	Sandoz Ltd	Improvements in or relating to organic compounds
US5284826A (en) *	1989-07-24	1994-02-08	Sandoz Ltd.	0-hydroxyethyl and acyloxyethyl derivatives of [ser]8 cyclosporins
GB9203886D0 (en) *	1992-02-24	1992-04-08	Sandoz Ltd	Improvements in or relating to organic compounds
SE517678C2 (sv) *	1994-07-12	2002-07-02	Lipocore Holding Ab	Lipofila bärarpreparat med en kontinuerlig lipidfas
JPH07316023A (ja) *	1994-05-26	1995-12-05	Shiseido Co Ltd	育毛料
PL324531A1 (en) *	1995-07-17	1998-06-08	Chem Ag C	Derivatives of cyclosporin effective against hiv virus
FR2757521B1 (fr) *	1996-12-24	1999-01-29	Rhone Poulenc Rorer Sa	Nouveaux derives de cyclosporine, leur preparation et les compositions pharmaceutiques qui les contiennent
CN1205220C (zh) *	1998-06-12	2005-06-08	斯－凯穆公司	新颖的环孢菌素
FR2780061B1 (fr) *	1998-06-22	2001-09-07	Rhone Poulenc Rorer Sa	Nouveau procede de preparation de derives de cyclosporine
AU3861900A (en)	1999-03-05	2000-09-21	University Of Texas Southwestern Medical Center, The	Method of treating hair loss using non-immunosuppressive compounds
US6521595B1 (en) *	1999-11-19	2003-02-18	Lg Chemical, Ltd.	Nonimmunosuppressive [γ-hydroxy-methylleucine4] cyclosporin A, hair growth stimulator and external composition for skin using the same
JP2003514000A (ja) *	1999-11-19	2003-04-15	エル・ジーハウスホールドアンドヘルスケアリミティッド	シクロスポリン誘導体含有毛髪成長促進剤
KR100316604B1 (ko) *	1999-11-19	2001-12-12	성재갑	모발 성장 효과를 갖는 비면역억제 사이클로스포린 에이유도체
KR20020039528A (ko) *	2000-11-22	2002-05-27	조명재	사이클로스포린 7- 티오아미드 유도체를 유효성분으로하는 모발성장촉진제
KR100360716B1 (ko) *	2000-11-22	2002-11-13	주식회사 엘지생활건강	사이클로스포린 에이 7- 티오아미드 유도체를유효성분으로 하는 모발성장촉진제
KR100681670B1 (ko) *	2001-02-14	2007-02-09	주식회사 엘지생활건강	[감마 히드록시 엔- 메틸-엘-루신9]사이클로스포린 에이를유효성분으로 하는 모발 성장 촉진제
KR100695610B1 (ko) *	2001-05-15	2007-03-14	주식회사 엘지생활건강	비면역성 발모성분인 [감마 히드록시 엔-메틸 엘-루신4] 사이클로스포린 유도체를 함유한 두피 및 경피용 제제 조성물
KR100695611B1 (ko) *	2001-05-17	2007-03-14	주식회사 엘지생활건강	[감마 히드록시 엔-메틸 엘-루신4] 사이클로스포린유도체를 유효성분으로 하는 모발 성장 촉진제

2001
- 2001-05-11 KR KR10-2001-0025682A patent/KR100465012B1/ko not_active Expired - Lifetime
2002
- 2002-05-09 US US10/141,723 patent/US6790830B2/en not_active Expired - Lifetime
- 2002-05-11 BR BRPI0209619A patent/BRPI0209619B8/pt not_active IP Right Cessation
- 2002-05-11 DE DE60237003T patent/DE60237003D1/de not_active Expired - Lifetime
- 2002-05-11 MX MXPA03010027A patent/MXPA03010027A/es active IP Right Grant
- 2002-05-11 JP JP2002588951A patent/JP4214181B2/ja not_active Expired - Lifetime
- 2002-05-11 RU RU2003135846/15A patent/RU2291682C2/ru active
- 2002-05-11 AT AT02728237T patent/ATE473730T1/de not_active IP Right Cessation
- 2002-05-11 TR TR2003/01931T patent/TR200301931T2/xx unknown
- 2002-05-11 WO PCT/KR2002/000879 patent/WO2002092032A1/en not_active Ceased
- 2002-05-11 CN CNB028096754A patent/CN1248671C/zh not_active Expired - Lifetime
- 2002-05-11 EP EP02728237A patent/EP1387660B1/de not_active Expired - Lifetime
- 2002-05-11 AU AU2002258271A patent/AU2002258271B2/en not_active Expired
- 2002-05-11 PL PL366407A patent/PL208536B1/pl unknown
- 2002-05-11 ES ES02728237T patent/ES2348225T3/es not_active Expired - Lifetime
- 2002-05-11 CA CA2446971A patent/CA2446971C/en not_active Expired - Lifetime
- 2002-11-25 US US10/303,281 patent/US6762164B2/en not_active Expired - Lifetime
2003
- 2003-10-31 ZA ZA200308532A patent/ZA200308532B/en unknown

Also Published As

Publication number	Publication date
WO2002092032A1 (en)	2002-11-21
BR0209619A (pt)	2004-03-30
AU2002258271B2 (en)	2006-06-29
EP1387660A4 (de)	2006-05-17
KR20020086041A (ko)	2002-11-18
US20030207798A1 (en)	2003-11-06
CN1507339A (zh)	2004-06-23
ES2348225T3 (es)	2010-12-01
TR200301931T2 (tr)	2004-09-21
MXPA03010027A (es)	2005-09-08
CA2446971A1 (en)	2002-11-21
EP1387660B1 (de)	2010-07-14
ZA200308532B (en)	2004-07-01
BRPI0209619B1 (pt)	2015-05-19
US20030186857A1 (en)	2003-10-02
JP4214181B2 (ja)	2009-01-28
KR100465012B1 (ko)	2005-01-13
BRPI0209619B8 (pt)	2021-05-25
PL208536B1 (pl)	2011-05-31
US6762164B2 (en)	2004-07-13
PL366407A1 (en)	2005-01-24
DE60237003D1 (de)	2010-08-26
JP2004530685A (ja)	2004-10-07
EP1387660A1 (de)	2004-02-11
CA2446971C (en)	2011-07-05
RU2003135846A (ru)	2005-03-27
RU2291682C2 (ru)	2007-01-20
CN1248671C (zh)	2006-04-05
US6790830B2 (en)	2004-09-14

Legal Events

Date	Code	Title	Description
2011-01-15	RER	Ceased as to paragraph 5 lit. 3 law introducing patent treaties

Publication	Publication Date	Title
ATE473730T1 (de)	2010-07-15	Verwendung von 3-positions-cyclosporin-derivaten für haarwachstum
YU9404A (sh)	2006-08-17	Multimerna, usmerena kontrastna sredstva na bazi peptida
DK1091975T3 (da)	2006-04-18	Ny cyclosporin med forbedret aktivitetsprofil
ECSP034859A (es)	2004-01-28	Nuevos derivados de pirrol como agentes farmacéuticos
BR0209242A (pt)	2004-06-15	Aminopolidiorganossiloxanos amido-funcionais
DE50004334D1 (de)	2003-12-11	Desodoriende zubereitungen enthaltend wasserlösliche -(1,3)-glucane
ATE288747T1 (de)	2005-02-15	Methoden und zusammensetzungen zur modulierung der aktivität von alpha-adrenergen rezeptoren
EP1435899A4 (de)	2005-03-16	Zusammensetzung zur förderung des haarwachstums
ATE275400T1 (de)	2004-09-15	Verwendung von melatonin zur behandlung der androgenetischen und diffusen alopezie vom weiblichen typ
EP1319402A4 (de)	2006-05-03	IgE-ENTSTEHUNGSHEMMSTOFFE
ATE330017T1 (de)	2006-07-15	Kallikrein gen
ATE493176T1 (de)	2011-01-15	Verwendung von 3-positions-cyclosporin-derivaten für haarwachstum
DK1204659T3 (da)	2004-04-05	Serotonerge benzofuraner
DE60131085D1 (de)	2007-12-06	Antimikrobielle sulfonamide-derivate von lipopeptidantibiotika
EP0995430A3 (de)	2001-12-19	Verwendung von Wirkstoffen, gewählt aus der Gruppe der 1,2-Diacylglycerole, zur Stärkung der Barrierefunktion der Haut
TR200102212T2 (tr)	2001-12-21	Fungisidal açıdan aktif bileşik birleşimleri.
NZ504614A (en)	2002-12-20	Echinocandin derivatives and application as anti-fungal agents
DK1189615T3 (da)	2004-06-07	Endoparasiticid synergistisk kombination indeholdende cykliske depsipeptider og piperaziner
ID26929A (id)	2001-02-22	Fungisida
EP1007032A4 (de)	2002-03-27	4-cyano-4-deformylsordarizin-derivate
DK1173065T3 (da)	2007-01-08	Anvendelse af cellulosemikrofibriller i fermenterede mælkepræparater
EP1007031A4 (de)	2001-10-24	4-cyano-4-deformylsordarinderivate
IL147223A0 (en)	2002-08-14	The use of the protein uk 114 for inhibiting organ transplant rejection
DE60203726D1 (de)	2005-05-19	Topische zusammensetzung enthaltend brucin und ihre verwendung zur behandlung von hautschäden
DE50115198D1 (de)	2009-12-10	Antihelmintika zur verhinderung von parasitären infektionen bei mensch und tier